Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 39 件

2X01
DownloadVisualize
BU of 2x01 by Molmil
CRYSTAL STRUCTURE OF THE OXA-10 S67A MUTANT AT PH 7
分子名称: BETA-LACTAMASE OXA-10, DIMETHYL SULFOXIDE, SULFATE ION, ...
著者Vercheval, L, Kerff, F, Bauvois, C, Sauvage, E, Guiet, R, Galleni, M, Charlier, P.
登録日2009-12-04
公開日2010-12-08
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Evidence of Chloride Inhibition and Impact of the Hydrophobic Core on the Lysine Carboxylated in Class D Beta-Lactamase
To be Published
1FOF
DownloadVisualize
BU of 1fof by Molmil
CRYSTAL STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-10
分子名称: BETA LACTAMASE OXA-10, COBALT (II) ION, SULFATE ION
著者Paetzel, M, Danel, F, de Castro, L, Mosimann, S.C, Page, M.G.P, Strynadka, N.C.J.
登録日2000-08-28
公開日2000-10-09
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the class D beta-lactamase OXA-10.
Nat.Struct.Biol., 7, 2000
1K4E
DownloadVisualize
BU of 1k4e by Molmil
CRYSTAL STRUCTURE OF THE CLASS D BETA-LACTAMASES OXA-10 DETERMINED BY MAD PHASING WITH SELENOMETHIONINE
分子名称: Beta-lactamase PSE-2, SULFATE ION
著者Kerff, F, Fonze, E, Bouillene, F, Frere, J.M, Charlier, P.
登録日2001-10-08
公開日2001-10-31
最終更新日2022-12-21
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献STRUCTURE OF CLASS D BETA-LACTAMASE OXA-2
To be Published
3LCE
DownloadVisualize
BU of 3lce by Molmil
Crystal Structure of Oxa-10 Beta-Lactamase Covalently Bound to Cyclobutanone Beta-Lactam Mimic
分子名称: (1S,3S,4S,5S)-7,7-dichloro-3-methoxy-2-thiabicyclo[3.2.0]heptan-6-one-4-carboxylic acid, Beta-lactamase OXA-10, GLYCEROL, ...
著者Gretes, M, Strynadka, N.C.J.
登録日2010-01-10
公開日2010-03-09
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Cyclobutanone Analogues of beta-Lactams Revisited: Insights into Conformational Requirements for Inhibition of Serine- and Metallo-beta-Lactamases.
J.Am.Chem.Soc., 132, 2010
1K6S
DownloadVisualize
BU of 1k6s by Molmil
STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-10 IN COMPLEX WITH A PHENYLBORONIC ACID
分子名称: 4-IODO-ACETAMIDO PHENYLBORONIC ACID, Beta-lactamase PSE-2, CALCIUM ION, ...
著者Kerff, F, Fonze, E, Sauvage, E, Frere, J.M, Charlier, P.
登録日2001-10-17
公開日2003-06-24
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献CRYSTAL STRUCTURE OF CLASS D BETA-LACTAMASE OXA-10 IN COMPLEX WITH DIFFERENT SUBSTRATES AND ONE INHIBITOR.
To be Published
2HPB
DownloadVisualize
BU of 2hpb by Molmil
Crystal structure of the OXA-10 W154A mutant at pH 9.0
分子名称: Beta-lactamase PSE-2, SULFATE ION
著者Kerff, F, Falzone, C, Herman, R, Sauvage, E, Charlier, P.
登録日2006-07-17
公開日2007-07-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Critical role of tryptophan 154 for the activity and stability of class D beta-lactamases.
Biochemistry, 48, 2009
2WKI
DownloadVisualize
BU of 2wki by Molmil
Crystal structure of the OXA-10 K70C mutant at pH 7.0
分子名称: 1,2-ETHANEDIOL, BETA-LACTAMASE OXA-10, GLYCEROL, ...
著者Vercheval, L, Bauvois, C, Kerff, F, Sauvage, E, Guiet, R, Charlier, P, Galleni, M.
登録日2009-06-11
公開日2010-08-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Three Factors that Modulate the Activity of Class D Beta-Lactamases and Interfere with the Post-Translational Carboxylation of Lys70.
Biochem.J., 432, 2010
6RTN
DownloadVisualize
BU of 6rtn by Molmil
Crystal structure of OXA-10 with VNRX-5133
分子名称: (3~{R})-3-[2-[4-(2-azanylethylamino)cyclohexyl]ethanoylamino]-2-oxidanyl-3,4-dihydro-1,2-benzoxaborinine-8-carboxylic acid, Beta-lactamase OXA-10, CHLORIDE ION
著者Brem, J, Schofield, C.
登録日2019-05-24
公開日2019-09-11
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Bicyclic Boronate VNRX-5133 Inhibits Metallo- and Serine-beta-Lactamases.
J.Med.Chem., 62, 2019
2HP6
DownloadVisualize
BU of 2hp6 by Molmil
Crystal structure of the OXA-10 W154A mutant at pH 7.5
分子名称: Beta-lactamase PSE-2, SULFATE ION
著者Kerff, F, Falzone, C, Herman, R, Sauvage, E, Charlier, P.
登録日2006-07-17
公開日2007-07-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Critical role of tryptophan 154 for the activity and stability of class D beta-lactamases.
Biochemistry, 48, 2009
1K6R
DownloadVisualize
BU of 1k6r by Molmil
STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-10 IN COMPLEX WITH MOXALACTAM
分子名称: (2R)-2-((R)-CARBOXY{[CARBOXY(4-HYDROXYPHENYL)ACETYL]AMINO}METHOXYMETHYL)-5-METHYLENE-5,6-DIHYDRO-2H-1,3-OXAZINE-4-CARBO XYLIC ACID, Beta-lactamase PSE-2
著者Kerff, F, Fonze, E, Sauvage, E, Frere, J.M, Charlier, P.
登録日2001-10-17
公開日2003-06-24
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献CRYSTAL STRUCTURE OF CLASS D BETA-LACTAMASE OXA-10 IN COMPLEX WITH DIFFERENT SUBSTRATES AND ONE INHIBITOR.
To be Published
1EWZ
DownloadVisualize
BU of 1ewz by Molmil
CRYSTAL STRUCTURE OF THE OXA-10 BETA-LACTAMASE FROM PSEUDOMONAS AERUGINOSA
分子名称: BETA LACTAMASE OXA-10
著者Golemi, D, Maveyraud, L, Vakulenko, S, Tranier, S, Ishiwata, A, Kotra, L.P, Samama, J.P, Mobashery, S.
登録日2000-04-28
公開日2000-11-01
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The First Structural and Mechanistic Insights for Class D beta-Lactamases: Evidence for a Novel Catalytic Process for Turnover of beta-Lactam Antibiotics
J.Am.Chem.Soc., 122, 2000
2HP9
DownloadVisualize
BU of 2hp9 by Molmil
Crystal Structure of the OXA-10 W154A mutant at pH 6.0
分子名称: Beta-lactamase PSE-2, SULFATE ION
著者Kerff, F, Falzone, C, Herman, R, Sauvage, E, Charlier, P.
登録日2006-07-17
公開日2007-07-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Critical role of tryptophan 154 for the activity and stability of class D beta-lactamases.
Biochemistry, 48, 2009
2HP5
DownloadVisualize
BU of 2hp5 by Molmil
Crystal Structure of the OXA-10 W154G mutant at pH 7.0
分子名称: Beta-lactamase PSE-2, COBALT (II) ION, SULFATE ION
著者Kerff, F, Falzone, C, Herman, R, Sauvage, E, Charlier, P.
登録日2006-07-17
公開日2007-07-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Critical role of tryptophan 154 for the activity and stability of class D beta-lactamases.
Biochemistry, 48, 2009
2WGI
DownloadVisualize
BU of 2wgi by Molmil
Crystal structure of the acyl-enzyme OXA-10 W154A-benzylpenicillin at pH 6
分子名称: BETA-LACTAMASE OXA-10, GLYCEROL, OPEN FORM - PENICILLIN G
著者Vercheval, L, Falzone, C, Sauvage, E, Herman, R, Charlier, P, Galleni, M, Kerff, F.
登録日2009-04-20
公開日2009-11-10
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Critical Role of Tryptophan 154 for the Activity and Stability of Class D Beta-Lactamases.
Biochemistry, 48, 2009
<12

 

223790

件を2024-08-14に公開中

PDB statisticsPDBj update infoContact PDBjnumon