1ZS4
| Structure of bacteriophage lambda cII protein in complex with DNA | 分子名称: | DNA - 27mer, Regulatory protein CII | 著者 | Jain, D, Kim, Y, Maxwell, K.L, Beasley, S, Gussin, G.N, Edwards, A.M, Darst, S.A. | 登録日 | 2005-05-23 | 公開日 | 2005-08-23 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal Structure of Bacteriophage lambdacII and Its DNA Complex. Mol.Cell, 19, 2005
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1ZS5
| Structure-based evaluation of selective and non-selective small molecules that block HIV-1 TAT and PCAF association | 分子名称: | (3E)-4-(1-METHYL-1H-INDOL-3-YL)BUT-3-EN-2-ONE, Histone acetyltransferase PCAF | 著者 | Zeng, L, Godbole, S, Muller, M, Yan, S, Sanchez, R, Zhou, M. | 登録日 | 2005-05-23 | 公開日 | 2006-05-23 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure-based evaluation of selective nad non-selective small molecules that block hiv-1 tat and pcaf association TO BE PUBLISHED
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1ZS6
| structure of human nucleoside-diphosphate kinase 3 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Nucleoside diphosphate kinase 3 | 著者 | Choe, J, Dimov, S, Arrowsmith, C, Edwards, A, Sundstrom, M, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2005-05-23 | 公開日 | 2005-06-07 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure of human nucleoside-diphosphate kinase 3 To be Published
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1ZS7
| The structure of gene product APE0525 from Aeropyrum pernix | 分子名称: | PHOSPHATE ION, POTASSIUM ION, hypothetical protein APE0525 | 著者 | Cuff, M.E, Skarina, T, Edwards, A, Savchenko, A, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2005-05-23 | 公開日 | 2005-07-05 | 最終更新日 | 2014-04-16 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | The structure of gene product APE0525 from Aeropyrum pernix To be Published
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1ZS8
| Crystal Structure of the Murine MHC Class Ib Molecule M10.5 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-2-microglobulin, histocompatibility 2, ... | 著者 | Olson, R, Huey-Tubman, K.E, Dulac, C, Bjorkman, P.J. | 登録日 | 2005-07-22 | 公開日 | 2005-07-26 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structure of a pheromone receptor-associated MHC molecule with an open and empty groove. Plos Biol., 3, 2005
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1ZS9
| Crystal structure of human enolase-phosphatase E1 | 分子名称: | E-1 ENZYME, MAGNESIUM ION | 著者 | Wang, H, Pang, H, Bartlam, M, Rao, Z. | 登録日 | 2005-05-23 | 公開日 | 2005-06-21 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal Structure of Human E1 Enzyme and its Complex with a Substrate Analog Reveals the Mechanism of its Phosphatase/Enolase J.Mol.Biol., 348, 2005
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1ZSA
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1ZSB
| CARBONIC ANHYDRASE II MUTANT E117Q, TRANSITION STATE ANALOGUE ACETAZOLAMIDE | 分子名称: | 5-ACETAMIDO-1,3,4-THIADIAZOLE-2-SULFONAMIDE, CARBONIC ANHYDRASE II, ZINC ION | 著者 | Lesburg, C.A, Christianson, D.W. | 登録日 | 1996-01-09 | 公開日 | 1996-07-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Reversal of the hydrogen bond to zinc ligand histidine-119 dramatically diminishes catalysis and enhances metal equilibration kinetics in carbonic anhydrase II. Biochemistry, 35, 1996
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1ZSC
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1ZSD
| Crystal Structure Of HLA-B*3501 Presenting an 11-Mer EBV Antigen EPLPQGQLTAY | 分子名称: | BZLF1 trans-activator protein, Beta-2-microglobulin, HLA class I histocompatibility antigen, ... | 著者 | Miles, J.J, Elhassen, D, Borg, N.A, Silins, S.L, Tynan, F.E, Burrows, J.M, Purcell, A.W, Kjer-Nielsen, L, Rossjohn, J, Burrows, S.R, McCluskey, J. | 登録日 | 2005-05-24 | 公開日 | 2005-06-07 | 最終更新日 | 2024-10-09 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | CTL Recognition of a Bulged Viral Peptide Involves Biased TCR Selection. J.Immunol., 175, 2005
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1ZSE
| RNA stemloop from bacteriophage Qbeta complexed with an N87S mutant MS2 Capsid | 分子名称: | Coat protein, RNA HAIRPIN | 著者 | Horn, W.T, Tars, K, Grahn, E, Helgstrand, C, Baron, A.J, Lago, H, Adams, C.J, Peabody, D.S, Phillips, S.E.V, Stonehouse, N.J, Liljas, L, Stockley, P.G. | 登録日 | 2005-05-24 | 公開日 | 2006-05-09 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural Basis of RNA Binding Discrimination between Bacteriophages Qbeta and MS2 Structure, 14, 2006
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1ZSF
| Crystal Structure of Complex of a Hydroxyethylamine Inhibitor with HIV-1 Protease at 2.0A Resolution | 分子名称: | N-{(2R,3S)-3-[(tert-butoxycarbonyl)amino]-2-hydroxy-4-phenylbutyl}-L-phenylalanyl-L-alpha-glutamyl-L-phenylalaninamide, PROTEASE RETROPEPSIN | 著者 | Duskova, J, Skalova, T, Dohnalek, J, Petrokova, H, Hasek, J. | 登録日 | 2005-05-24 | 公開日 | 2006-04-25 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | On the role of the R configuration of the reaction-intermediate isostere in HIV-1 protease-inhibitor binding: X-ray structure at 2.0 A resolution. Acta Crystallogr.,Sect.D, 62, 2006
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1ZSG
| beta PIX-SH3 complexed with an atypical peptide from alpha-PAK | 分子名称: | Rho guanine nucleotide exchange factor 7, Serine/threonine-protein kinase PAK 1 | 著者 | Mott, H.R, Nietlispach, D, Evetts, K.A, Owen, D. | 登録日 | 2005-05-24 | 公開日 | 2005-08-30 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural Analysis of the SH3 Domain of beta-PIX and Its Interaction with alpha-p21 Activated Kinase (PAK) Biochemistry, 44, 2005
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1ZSH
| Crystal structure of bovine arrestin-2 in complex with inositol hexakisphosphate (IP6) | 分子名称: | Beta-arrestin 1, INOSITOL HEXAKISPHOSPHATE, MAGNESIUM ION | 著者 | Milano, S.K, Kim, Y.M, Stefano, F.P, Benovic, J.L, Brenner, C. | 登録日 | 2005-05-24 | 公開日 | 2006-01-31 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Nonvisual arrestin oligomerization and cellular localization are regulated by inositol hexakisphosphate binding J.Biol.Chem., 281, 2006
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1ZSJ
| Crystal Structure of the Catalytic Domain of Coagulation Factor XI in complex with N-(7-Carbamimidoyl-naphthalen-1-yl)-3-hydroxy-2-methyl-benzamide | 分子名称: | BICARBONATE ION, Coagulation factor XI, N-(7-CARBAMIMIDOYL-NAPHTHALEN-1-YL)-3-HYDROXY-2-METHYL-BENZAMIDE, ... | 著者 | Guo, Z, Bannister, T, Noll, R, Jin, L, Rynkiewicz, M, Bibbins, F, Magee, S, Gorga, J, Babine, R.E, Strickler, J.E, Meyers, H.V, Abdel-Meguid, S.S. | 登録日 | 2005-05-24 | 公開日 | 2006-05-23 | 最終更新日 | 2024-10-09 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Synthesis and Optimization of Potent and Selective Inhibitors for Human Factor XIa: Substituted Naphthamidine Series To be Published
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1ZSK
| Crystal Structure of the Catalytic Domain of Coagulation Factor XI in Complex with 6-Carbamimidoyl-4-(3-hydroxy-2-methyl-benzoylamino)-naphthalene-2-carboxylic acid methyl ester | 分子名称: | 6-CARBAMIMIDOYL-4-(3-HYDROXY-2-METHYL-BENZOYLAMINO)-NAPHTHALENE-2-CARBOXYLIC ACID METHYL ESTER, BICARBONATE ION, Coagulation factor XI, ... | 著者 | Guo, Z, Bannister, T, Noll, R, Jin, L, Rynkiewicz, M, Bibbins, F, Magee, S, Gorga, J, Babine, R.E, Strickler, J.E, Meyers, H.V, Abdel-Meguid, S.S. | 登録日 | 2005-05-24 | 公開日 | 2006-05-23 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Synthesis and Optimization of Potent and Selective Inhibitors for Human Factor XIa: Substituted Naphthamidine Series To be Published
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1ZSL
| Factor XI complexed with a pyrimidinone inhibitor | 分子名称: | 2-(2-(3,4-DICHLOROPHENYL)-5-(ISOPROPYLAMINO)-6-OXOPYRIMIDIN-1(6H)-YL)-N-((S)-1-OXO-1-(THIAZOL-2-YL)-5-GUANIDINOPENTAN-2-YL)ACETAMIDE, Coagulation factor XI | 著者 | Nagafuji, P, Jin, L, Rynkiewicz, M, Quinn, J, Bibbins, F, Meyers, H, Babine, R, Strickler, J, Abdel-Meguid, S. | 登録日 | 2005-05-24 | 公開日 | 2006-05-09 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Pyrimidinone Inhibitors of a Thrombolytic Protease To be Published
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1ZSN
| Synthesis, Biological Activity, and X-Ray Crystal Structural Analysis of Diaryl Ether Inhibitors of Malarial Enoyl ACP Reductase. Part 1:4'-Substituted Triclosan Derivatives | 分子名称: | 5-CHLORO-2-(2-CHLORO-4-NITROPHENOXY)PHENOL, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, enoyl-acyl carrier reductase | 著者 | Freundlich, J.S, Anderson, J.W, Sarantakis, D, Shieh, H.M, Yu, M, Lucumi, E, Kuo, M, Schiehser, G.A, Jacobus, D.P, Jacobs Jr, W.R, Fidock, D.A, Sacchettini, J.C. | 登録日 | 2005-05-24 | 公開日 | 2006-05-30 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.992 Å) | 主引用文献 | Synthesis, biological activity, and X-ray crystal structural analysis of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 1: 4'-Substituted triclosan derivatives. Bioorg.Med.Chem.Lett., 15, 2005
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1ZSO
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1ZSP
| Contribution to Structure and Catalysis of Tyrosine 34 in Human Manganese Superoxide Dismutase | 分子名称: | MANGANESE (II) ION, Superoxide dismutase [Mn], mitochondrial | 著者 | Hearn, A.S, Perry, J.J, Cabelli, D.E, Tainer, J.A, Nick, H.S, Silverman, D.S. | 登録日 | 2005-05-24 | 公開日 | 2006-05-02 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Contribution of human manganese superoxide dismutase tyrosine 34 to structure and catalysis. Biochemistry, 48, 2009
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1ZSQ
| Crystal Structure of MTMR2 in complex with phosphatidylinositol 3-phosphate | 分子名称: | 1,2-ETHANEDIOL, 2-(BUTANOYLOXY)-1-{[(HYDROXY{[2,3,4,6-TETRAHYDROXY-5-(PHOSPHONOOXY)CYCLOHEXYL]OXY}PHOSPHORYL)OXY]METHYL}ETHYL BUTANOATE, Myotubularin-related protein 2 | 著者 | Begley, M.J, Taylor, G.S, Brock, M.A, Ghosh, P, Woods, V.L, Dixon, J.E. | 登録日 | 2005-05-25 | 公開日 | 2006-01-31 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | Molecular basis for substrate recognition by MTMR2, a myotubularin family phosphoinositide phosphatase Proc.Natl.Acad.Sci.Usa, 103, 2006
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1ZSR
| Crystal structure of wild type HIV-1 protease (BRU isolate) with a hydroxyethylamine peptidomimetic inhibitor BOC-PHE-PSI[S-CH(OH)CH2NH]-PHE-GLU-PHE-NH2 | 分子名称: | N-{(2S,3S)-3-[(tert-butoxycarbonyl)amino]-2-hydroxy-4-phenylbutyl}-L-phenylalanyl-L-alpha-glutamyl-L-phenylalaninamide, PROTEASE RETROPEPSIN | 著者 | Skalova, T, Dohnalek, J, Duskova, J, Petrokova, H, Hasek, J. | 登録日 | 2005-05-24 | 公開日 | 2006-04-25 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (2.06 Å) | 主引用文献 | On the role of the R configuration of the reaction-intermediate isostere in HIV-1 protease-inhibitor binding: X-ray structure at 2.0 A resolution. Acta Crystallogr.,Sect.D, 62, 2006
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1ZSV
| Crystal structure of human NADP-dependent leukotriene B4 12-hydroxydehydrogenase | 分子名称: | CHLORIDE ION, NADP-dependent leukotriene B4 12-hydroxydehydrogenase | 著者 | Turnbull, A.P, Johansson, C, Savitsky, P, Guo, K, Edwards, A, Arrowsmith, C, Sundstrom, M, von Delft, F, Oppermann, U, Structural Genomics Consortium (SGC) | 登録日 | 2005-05-25 | 公開日 | 2005-06-21 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of human NADP-dependent leukotriene B4 12-hydroxydehydrogenase To be Published
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1ZSW
| Crystal Structure of Bacillus cereus Metallo Protein from Glyoxalase family | 分子名称: | BETA-MERCAPTOETHANOL, Glyoxalase family protein, ZINC ION | 著者 | Minasov, G, Shuvalova, L, Brunzelle, J.S, Collart, F.R, Anderson, W.F, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2005-05-25 | 公開日 | 2005-06-07 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Crystal Structure of Bacillus cereus Metallo Protein from Glyoxalase family To be Published
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1ZSX
| Crystal Structure Of Human Potassium Channel Kv Beta-subunit (KCNAB2) | 分子名称: | CHLORIDE ION, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, Voltage-gated potassium channel beta-2 subunit | 著者 | Wennerstrand, P, Johannsson, I, Ugochukwu, E, Kavanagh, K, Edwards, A, Arrowsmith, C, Williams, L, Sundstrom, M, Guo, K, von Delft, F, Oppermann, U, Structural Genomics Consortium (SGC) | 登録日 | 2005-05-25 | 公開日 | 2005-06-07 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal Structure Of Human Potassium Channel Kv Beta-subunit (KCNAB2) To be Published
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