Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 289 results

4V84
DownloadVisualize
BU of 4v84 by Molmil
Crystal structure of a complex containing domain 3 of CrPV IGR IRES RNA bound to the 70S ribosome.
Descriptor: 23S ribosomal RNA, 30S ribosomal protein S10, 30S ribosomal protein S11, ...
Authors:Zhu, J, Korostelev, A, Costantino, D, Noller, H.F, Kieft, J.S.
Deposit date:2010-12-13
Release date:2014-07-09
Last modified:2019-07-17
Method:X-RAY DIFFRACTION (3.4 Å)
Cite:Crystal structures of complexes containing domains from two viral internal ribosome entry site (IRES) RNAs bound to the 70S ribosome.
Proc.Natl.Acad.Sci.USA, 108, 2011
2QVO
DownloadVisualize
BU of 2qvo by Molmil
Crystal structure of AF1382 from Archaeoglobus fulgidus
Descriptor: Uncharacterized protein AF_1382
Authors:Zhu, J, Zhao, M, Fu, Z.-Q, Yang, H, Chang, J, Hao, X, Chen, L, Liu, Z.J, Rose, J.P, Wang, B.C, Southeast Collaboratory for Structural Genomics (SECSG)
Deposit date:2007-08-08
Release date:2007-09-04
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Crystal structure of AF1382 from Archaeoglobus fulgidus.
To be Published
7TCT
DownloadVisualize
BU of 7tct by Molmil
Integrin alaphIIBbeta3 complex with UR2922
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Zhu, J, Lin, F.-Y, Zhu, J, Springer, T.A.
Deposit date:2021-12-28
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.501 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7TD8
DownloadVisualize
BU of 7td8 by Molmil
Integrin alaphIIBbeta3 complex with Tirofiban
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Zhu, J, Lin, F.-Y, Zhu, J, Springer, T.A.
Deposit date:2021-12-30
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
5OWK
DownloadVisualize
BU of 5owk by Molmil
Crystal structure of CREBBP bromodomain complexed with DSPB2A002
Descriptor: CREB-binding protein, ethyl 4-chloranyl-1-methyl-6-oxidanylidene-pyridine-3-carboxylate
Authors:Zhu, J, Spiliotopoulos, D, Caflisch, A.
Deposit date:2017-09-01
Release date:2018-08-29
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.25 Å)
Cite:Binding Motifs in the CBP Bromodomain: An Analysis of 20 Crystal Structures of Complexes with Small Molecules.
ACS Med Chem Lett, 9, 2018
4XEJ
DownloadVisualize
BU of 4xej by Molmil
IRES bound to bacterial Ribosome
Descriptor: 16S ribosomal RNA, 23S ribosomal RNA, 30S ribosomal protein S10, ...
Authors:Zhu, J, Korostelev, A, Noller, H.F, Donohue, J.P.
Deposit date:2014-12-23
Release date:2015-02-25
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (3.8 Å)
Cite:Initiation of translation in bacteria by a structured eukaryotic IRES RNA.
Nature, 519, 2015
4UIM
DownloadVisualize
BU of 4uim by Molmil
crystal structure of quinine-dependent Fab 314.3
Descriptor: FAB 314.3, SULFATE ION
Authors:Zhu, J, Zhu, J, Bougie, D.W, Aster, R.H, Springer, T.A.
Deposit date:2015-03-30
Release date:2015-09-02
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Structural Basis for Quinine-Dependent Antibody Binding to Platelet Integrin Alphaiib Beta3
Blood, 126, 2015
4UIK
DownloadVisualize
BU of 4uik by Molmil
crystal structure of quinine-dependent Fab 314.1
Descriptor: FAB 314.1
Authors:Zhu, J, Zhu, J, Bougie, D.W, Aster, R.H, Springer, T.A.
Deposit date:2015-03-30
Release date:2015-09-02
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2 Å)
Cite:Structural Basis for Quinine-Dependent Antibody Binding to Platelet Integrin Alphaiib Beta3
Blood, 126, 2015
4UIN
DownloadVisualize
BU of 4uin by Molmil
crystal structure of quinine-dependent Fab 314.3 with quinine
Descriptor: FAB 314.3, Quinine
Authors:Zhu, J, Zhu, J, Bougie, D.W, Aster, R.H, Springer, T.A.
Deposit date:2015-03-30
Release date:2015-09-02
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structural Basis for Quinine-Dependent Antibody Binding to Platelet Integrin Alphaiib Beta3
Blood, 126, 2015
4UIL
DownloadVisualize
BU of 4uil by Molmil
crystal structure of quinine-dependent Fab 314.1 with quinine
Descriptor: FAB 314.1, Quinine
Authors:Zhu, J, Zhu, J, Bougie, D.W, Aster, R.H, Springer, T.A.
Deposit date:2015-03-30
Release date:2015-09-02
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.853 Å)
Cite:Structural Basis for Quinine-Dependent Antibody Binding to Platelet Integrin Alphaiib Beta3
Blood, 126, 2015
5OV8
DownloadVisualize
BU of 5ov8 by Molmil
Crystal structure of the human BRPF1 bromodomain in complex with BZ097
Descriptor: NITRATE ION, Peregrin, ~{N}-[1,4-dimethyl-2,3-bis(oxidanylidene)-7-pyrrolidin-1-yl-quinoxalin-6-yl]-4-(2-methylpropyl)benzenesulfonamide
Authors:Zhu, J, Caflisch, A.
Deposit date:2017-08-28
Release date:2018-06-27
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Structure-based discovery of selective BRPF1 bromodomain inhibitors.
Eur J Med Chem, 155, 2018
5OWB
DownloadVisualize
BU of 5owb by Molmil
Crystal structure of the human BRPF1 bromodomain in complex with DSPBP1004
Descriptor: 4-methyl-6-oxidanyl-1-benzofuran-3-one, NITRATE ION, Peregrin
Authors:Zhu, J, Spiliotopoulos, D, Caflisch, A.
Deposit date:2017-08-31
Release date:2018-07-18
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Crystal structure of the human BRPF1 bromodomain in complex with DSPBP1004
To Be Published
5OWW
DownloadVisualize
BU of 5oww by Molmil
Crystal structure of human BRD4(1) bromodomain in complex with UT22B
Descriptor: Bromodomain-containing protein 4, ~{N}-(3-methylbenzotriazol-5-yl)-1-(phenylmethyl)imidazole-2-carboxamide
Authors:Zhu, J, Caflisch, A.
Deposit date:2017-09-04
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Chemical Space Expansion of Bromodomain Ligands Guided by in Silico Virtual Couplings (AutoCouple).
Acs Cent.Sci., 4, 2018
5OVB
DownloadVisualize
BU of 5ovb by Molmil
Crystal structure of human BRD4(1) bromodomain in complex with DR46
Descriptor: Bromodomain-containing protein 4, ~{N}-[3-(5-ethanoyl-2-ethoxy-phenyl)-5-(1-methylpyrazol-3-yl)phenyl]furan-2-carboxamide
Authors:Zhu, J, Caflisch, A.
Deposit date:2017-08-28
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Chemical Space Expansion of Bromodomain Ligands Guided by in Silico Virtual Couplings (AutoCouple).
Acs Cent.Sci., 4, 2018
5OWE
DownloadVisualize
BU of 5owe by Molmil
Crystal structure of the human BRPF1 bromodomain in complex with DSPBP1010
Descriptor: 1,3-bis(oxidanyl)benzo[c]chromen-6-one, NITRATE ION, Peregrin
Authors:Zhu, J, Spiliotopoulos, D, Caflisch, A.
Deposit date:2017-08-31
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Crystal structure of the human BRPF1 bromodomain in complex with DSPBP1010
To Be Published
5OWA
DownloadVisualize
BU of 5owa by Molmil
Crystal structure of the human BRPF1 bromodomain in complex with BZ054
Descriptor: Peregrin, ~{N}-[4-[[(3~{S},5~{R})-3,5-dimethylpiperidin-1-yl]methyl]-1,3-thiazol-2-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
Authors:Zhu, J, Caflisch, A.
Deposit date:2017-08-31
Release date:2018-06-27
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Structure-based discovery of selective BRPF1 bromodomain inhibitors.
Eur J Med Chem, 155, 2018
5OWM
DownloadVisualize
BU of 5owm by Molmil
Crystal structure of human BRD4(1) bromodomain in complex with UT48
Descriptor: Bromodomain-containing protein 4, [3-[(3-methylbenzotriazol-5-yl)methyl]phenyl]methanol
Authors:Zhu, J, Caflisch, A.
Deposit date:2017-09-01
Release date:2018-10-10
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Chemical Space Expansion of Bromodomain Ligands Guided by in Silico Virtual Couplings (AutoCouple).
Acs Cent.Sci., 4, 2018
4V83
DownloadVisualize
BU of 4v83 by Molmil
Crystal structure of a complex containing domain 3 from the PSIV IGR IRES RNA bound to the 70S ribosome.
Descriptor: 23S ribosomal RNA, 30S ribosomal protein S10, 30S ribosomal protein S11, ...
Authors:Zhu, J, Korostelev, A, Costantino, D, Noller, H.F, Kieft, J.S.
Deposit date:2010-12-13
Release date:2014-07-09
Last modified:2014-12-10
Method:X-RAY DIFFRACTION (3.5 Å)
Cite:Crystal structures of complexes containing domains from two viral internal ribosome entry site (IRES) RNAs bound to the 70S ribosome.
Proc.Natl.Acad.Sci.USA, 108, 2011
7U9V
DownloadVisualize
BU of 7u9v by Molmil
Integrin alaphIIBbeta3 complex with BMS4-1
Descriptor: (4-{[(5S)-3-(4-carbamimidoylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}piperazin-1-yl)acetic acid, 10E5 Fab heavy chain, 10E5 light chain, ...
Authors:Zhu, J, Lin, F.-Y, Zhu, J, Springer, T.A.
Deposit date:2022-03-11
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.25492167 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7TMZ
DownloadVisualize
BU of 7tmz by Molmil
Integrin alaphIIBbeta3 complex with BMS compound 4
Descriptor: (4-{[(5S)-3-{4-[(E)-imino(4-methylpiperazin-1-yl)methyl]phenyl}-4,5-dihydro-1,2-oxazol-5-yl]methyl}piperazin-1-yl)acetic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Zhu, J, Lin, F.-Y, Zhu, J, Springer, T.A.
Deposit date:2022-01-20
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.20002 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7U60
DownloadVisualize
BU of 7u60 by Molmil
Integrin alaphIIBbeta3 complex with cRGDfV
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ARG-GLY-ASP-DPN-VAL, ...
Authors:Zhu, J, Lin, F.Y, Zhu, J, Springer, T.A.
Deposit date:2022-03-03
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.55 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7THO
DownloadVisualize
BU of 7tho by Molmil
Integrin alaphIIBbeta3 complex with Eptifibatide
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Zhu, J, Lin, F.-Y, Zhu, J, Springer, T.A.
Deposit date:2022-01-11
Release date:2022-08-17
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.75 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7TPD
DownloadVisualize
BU of 7tpd by Molmil
Integrin alaphIIBbeta3 complex with EF5154
Descriptor: (4-{[2-oxo-4-(piperidin-4-yl)piperazin-1-yl]acetyl}phenoxy)acetic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Zhu, J, Lin, F.-Y, Zhu, J, Springer, T.A.
Deposit date:2022-01-25
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
5MME
DownloadVisualize
BU of 5mme by Molmil
Crystal structure of CREBBP bromodomain complexd with US46C
Descriptor: CREB-binding protein, dimethyl 5-[(5-ethanoyl-2-ethoxy-phenyl)amino]benzene-1,3-dicarboxylate
Authors:Zhu, J, Caflisch, A.
Deposit date:2016-12-09
Release date:2017-12-20
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (1.35 Å)
Cite:Binding Motifs in the CBP Bromodomain: An Analysis of 20 Crystal Structures of Complexes with Small Molecules.
ACS Med Chem Lett, 9, 2018
3T3P
DownloadVisualize
BU of 3t3p by Molmil
A Novel High Affinity Integrin alphaIIbbeta3 Receptor Antagonist That Unexpectedly Displaces Mg2+ from the beta3 MIDAS
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2011-07-25
Release date:2012-03-28
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Structure-Guided Design of a High-Affinity Platelet Integrin alphaIIbbeta3 Receptor Antagonist That Disrupts Mg2+ Binding to the MIDAS
Sci Transl Med, 4, 2012

221051

PDB entries from 2024-06-12

PDB statisticsPDBj update infoContact PDBjnumon