7AJL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ajl by Molmil](/molmil-images/mine/7ajl) | Cyrstal structure of CYRI-B/Fam49B | 分子名称: | CYFIP-related Rac1 interactor B | 著者 | Yelland, T, Anh, H, Insall, R, Machesky, L, Ismail, S. | 登録日 | 2020-09-29 | 公開日 | 2020-11-18 | 最終更新日 | 2021-06-02 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Structural Basis of CYRI-B Direct Competition with Scar/WAVE Complex for Rac1. Structure, 29, 2021
|
|
7AJK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ajk by Molmil](/molmil-images/mine/7ajk) | Crystal structure of CRYI-B Rac1 complex | 分子名称: | CYFIP-related Rac1 interactor B, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, ... | 著者 | Yelland, T, Anh, L, Insall, R, Machesky, L, Ismail, S. | 登録日 | 2020-09-29 | 公開日 | 2020-11-18 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structural Basis of CYRI-B Direct Competition with Scar/WAVE Complex for Rac1. Structure, 29, 2021
|
|
6FMC
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6fmc by Molmil](/molmil-images/mine/6fmc) | Neuropilin1-b1 domain in complex with EG01377, 0.9 Angstrom structure | 分子名称: | (2~{S})-2-[[3-[[5-[4-(aminomethyl)phenyl]-1-benzofuran-7-yl]sulfonylamino]thiophen-2-yl]carbonylamino]-5-carbamimidamido-pentanoic acid, Neuropilin-1 | 著者 | Yelland, T, Djordjevic, S, Fotinou, K, Selwood, D, Zachary, I, Frankel, P. | 登録日 | 2018-01-30 | 公開日 | 2018-10-17 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (0.9 Å) | 主引用文献 | Small Molecule Neuropilin-1 Antagonists Combine Antiangiogenic and Antitumor Activity with Immune Modulation through Reduction of Transforming Growth Factor Beta (TGF beta ) Production in Regulatory T-Cells. J. Med. Chem., 61, 2018
|
|
6FMF
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6fmf by Molmil](/molmil-images/mine/6fmf) | Neuropilin-1 b1 domain in complex with EG01377; 2.8 Angstrom structure | 分子名称: | (2~{S})-2-[[3-[[5-[4-(aminomethyl)phenyl]-1-benzofuran-7-yl]sulfonylamino]thiophen-2-yl]carbonylamino]-5-carbamimidamido-pentanoic acid, Neuropilin-1, trifluoroacetic acid | 著者 | Yelland, T, Djordjevic, S, Selwood, D, Zachary, I, Frankel, P. | 登録日 | 2018-01-31 | 公開日 | 2018-10-17 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.811 Å) | 主引用文献 | Small Molecule Neuropilin-1 Antagonists Combine Antiangiogenic and Antitumor Activity with Immune Modulation through Reduction of Transforming Growth Factor Beta (TGF beta ) Production in Regulatory T-Cells. J. Med. Chem., 61, 2018
|
|
7OK6
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ok6 by Molmil](/molmil-images/mine/7ok6) | |
7OK7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ok7 by Molmil](/molmil-images/mine/7ok7) | Crystal structure of the UNC119B ARL3 complex | 分子名称: | 1,2-ETHANEDIOL, ADP-ribosylation factor-like protein 3, GLYCEROL, ... | 著者 | Yelland, T, Ismail, S. | 登録日 | 2021-05-17 | 公開日 | 2021-06-09 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (3.15 Å) | 主引用文献 | The Structural and Biochemical Characterization of UNC119B Cargo Binding and Release Mechanisms. Biochemistry, 60, 2021
|
|
6H6A
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6h6a by Molmil](/molmil-images/mine/6h6a) | Crystal structure of UNC119 in complex with LCK peptide | 分子名称: | GLY-CYS-GLY-CYS-SER-SER, GLYCEROL, MYRISTIC ACID, ... | 著者 | Yelland, T, ElMaghloob, Y, McIlwraith, M, Stephen, L, Ismail, S. | 登録日 | 2018-07-26 | 公開日 | 2018-09-26 | 最終更新日 | 2019-11-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The Ciliary Machinery Is Repurposed for T Cell Immune Synapse Trafficking of LCK. Dev.Cell, 47, 2018
|
|
7Q9S
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7q9s by Molmil](/molmil-images/mine/7q9s) | Crystal structure of PDE6D KRas peptide complex with Compound-1 | 分子名称: | 1,2-ETHANEDIOL, 2-methyl-3-(1~{H}-pyrazol-5-yl)imidazo[1,2-a]pyridine, DIMETHYL SULFOXIDE, ... | 著者 | Yelland, T, Ismail, S. | 登録日 | 2021-11-14 | 公開日 | 2022-01-19 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Stabilization of the RAS:PDE6D Complex Is a Novel Strategy to Inhibit RAS Signaling. J.Med.Chem., 65, 2022
|
|
7Q9Q
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7q9q by Molmil](/molmil-images/mine/7q9q) | |
7Q9R
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7q9r by Molmil](/molmil-images/mine/7q9r) | Cocrystal structure of PDE6D bound to NRAS peptide | 分子名称: | 1,2-ETHANEDIOL, FARNESYL, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta, ... | 著者 | Yelland, T, Ismail, S. | 登録日 | 2021-11-14 | 公開日 | 2022-01-19 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Stabilization of the RAS:PDE6D Complex Is a Novel Strategy to Inhibit RAS Signaling. J.Med.Chem., 65, 2022
|
|
7QF9
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7qf9 by Molmil](/molmil-images/mine/7qf9) | |
7Q9U
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7q9u by Molmil](/molmil-images/mine/7q9u) | |
7QJK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7qjk by Molmil](/molmil-images/mine/7qjk) | Crystal structure of PDE6D in complex with Compound-2 | 分子名称: | 1,2-ETHANEDIOL, N-(phenylmethyl)pyridin-2-amine, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta, ... | 著者 | Yelland, T, Ismail, S. | 登録日 | 2021-12-16 | 公開日 | 2022-01-26 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Stabilization of the RAS:PDE6D Complex Is a Novel Strategy to Inhibit RAS Signaling. J.Med.Chem., 65, 2022
|
|
5L73
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5l73 by Molmil](/molmil-images/mine/5l73) | MAM domain of human neuropilin-1 | 分子名称: | BICINE, CALCIUM ION, Neuropilin-1, ... | 著者 | Yelland, T, Djordjevic, S. | 登録日 | 2016-06-01 | 公開日 | 2016-10-26 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.24 Å) | 主引用文献 | Crystal Structure of the Neuropilin-1 MAM Domain: Completing the Neuropilin-1 Ectodomain Picture. Structure, 24, 2016
|
|
3ZIX
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3zix by Molmil](/molmil-images/mine/3zix) | Clostridium perfringens Enterotoxin with the N-terminal 37 residues deleted | 分子名称: | HEAT-LABILE ENTEROTOXIN B CHAIN, HEXAETHYLENE GLYCOL | 著者 | Yelland, T, Naylor, C.E, Savva, C.G, Basak, A.K. | 登録日 | 2013-01-14 | 公開日 | 2014-01-29 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure of a C. Perfringens Enterotoxin Mutant in Complex with a Modified Claudin-2 Extracellular Loop 2 J.Mol.Biol., 426, 2014
|
|
3ZIW
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ziw by Molmil](/molmil-images/mine/3ziw) | Clostridium perfringens enterotoxin, D48A mutation and N-terminal 37 residues deleted | 分子名称: | HEAT-LABILE ENTEROTOXIN B CHAIN, HEXAETHYLENE GLYCOL | 著者 | Yelland, T, Naylor, C.E, Savva, C.G, Basak, A.K. | 登録日 | 2013-01-14 | 公開日 | 2014-01-29 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure of a C. Perfringens Enterotoxin Mutant in Complex with a Modified Claudin-2 Extracellular Loop 2 J.Mol.Biol., 426, 2014
|
|
5IJR
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ijr by Molmil](/molmil-images/mine/5ijr) | X-ray structure of neuropilin-1 b1 domain complexed with Arg-1 ligand. | 分子名称: | DIMETHYL SULFOXIDE, L-HOMOARGININE, Neuropilin-1 | 著者 | Fotinou, C, Rana, R, Djordjevic, S, Yelland, T. | 登録日 | 2016-03-02 | 公開日 | 2017-03-29 | 最終更新日 | 2018-07-11 | 実験手法 | X-RAY DIFFRACTION (1.52 Å) | 主引用文献 | Architecture and hydration of the arginine-binding site of neuropilin-1. FEBS J., 285, 2018
|
|
7ZC8
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7zc8 by Molmil](/molmil-images/mine/7zc8) | |
4RN5
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4rn5 by Molmil](/molmil-images/mine/4rn5) | B1 domain of human Neuropilin-1 with acetate ion in a ligand-binding site | 分子名称: | ACETATE ION, GLYCEROL, Neuropilin-1, ... | 著者 | Allerston, C.K, Yelland, T.S, Jarvis, A, Jenkins, K, Winfield, N, Cheng, L, Jia, H, Zachary, I, Selwood, D.L, Djordjevic, S. | 登録日 | 2014-10-23 | 公開日 | 2015-10-28 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Conserved water molecules in a ligand-binding site of neuropilin-1 To be Published
|
|
4P5H
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4p5h by Molmil](/molmil-images/mine/4p5h) | |
7P5U
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7p5u by Molmil](/molmil-images/mine/7p5u) | |
6TDB
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6tdb by Molmil](/molmil-images/mine/6tdb) | Neuropilin2-b1 domain in a complex with the C-terminal VEGFB167 peptide | 分子名称: | 1,2-ETHANEDIOL, ACETYL GROUP, C-terminal VEGFB167 peptide, ... | 著者 | Eldrid, C, Yu, L, Yelland, T, Fotinou, C, Djordjevic, S. | 登録日 | 2019-11-08 | 公開日 | 2020-11-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | NRP2-b1 domain in a complex with the C-terminal VEGFB167 peptide To Be Published
|
|
6TJT
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6tjt by Molmil](/molmil-images/mine/6tjt) | Neuropilin2-b1 domain in a complex with the C-terminal VEGFC peptide | 分子名称: | 1,2-ETHANEDIOL, Neuropilin-2, SULFATE ION, ... | 著者 | Eldrid, C, Yu, L, Yelland, T, Fotinou, C, Djordjevic, S. | 登録日 | 2019-11-26 | 公開日 | 2020-12-16 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.31 Å) | 主引用文献 | NRP2-b1 domain in a complex with the C-terminal VEGFC peptide To Be Published
|
|
6TKK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6tkk by Molmil](/molmil-images/mine/6tkk) | Neuropilin 1-b1 domain in a complex with the C-terminal VEGFB186 peptide | 分子名称: | 1,2-ETHANEDIOL, ACE-ARG-PRO-GLN-PRO-ARG, Neuropilin-1 | 著者 | Eldrid, C, Yu, L, Yelland, T, Fotinou, C, Djordjevic, S. | 登録日 | 2019-11-28 | 公開日 | 2020-12-16 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.06 Å) | 主引用文献 | Neuropilin 1-b1 domain in a complex with the C-terminal VEGFB186 peptide To Be Published
|
|
5JHK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5jhk by Molmil](/molmil-images/mine/5jhk) | X-ray structure of neuropilin-1 b1 domain complexed with Arg-6 ligand. | 分子名称: | N-(benzenecarbonyl)glycyl-L-arginine, Neuropilin-1 | 著者 | Fotinou, C, Rana, R, Djordjevic, S, Yelland, T. | 登録日 | 2016-04-21 | 公開日 | 2017-05-24 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Architecture and hydration of the arginine-binding site of neuropilin-1. FEBS J., 285, 2018
|
|