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PDB: 22 件
3D27
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E. coli methionine aminopeptidase with Fe inhibitor W29
分子名称: 4-(3-ethylthiophen-2-yl)benzene-1,2-diol, MANGANESE (II) ION, Methionine aminopeptidase
著者Ye, Q.Z, Chai, S, He, H.Z.
登録日2008-05-07
公開日2008-08-19
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Discovery of inhibitors of Escherichia coli methionine aminopeptidase with the Fe(II)-form selectivity and antibacterial activity.
J.Med.Chem., 51, 2008
4JUQ
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Pseudomonas aeruginosa MetAP T2N mutant, in Mn form
分子名称: MANGANESE (II) ION, Methionine aminopeptidase
著者Ye, Q.Z, Lu, J.P.
登録日2013-03-25
公開日2014-04-30
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Methionine excision captured by the structures of a methionine aminopeptidase
To be published
4FLL
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Human MetAP1 with bengamide analog YZ6, in Mn form
分子名称: (E,2R,3R,4S,5R)-N-[(3R)-3-(furan-2-yl)-3-phenyl-propyl]-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, MANGANESE (II) ION, Methionine aminopeptidase 1, ...
著者Ye, Q.Z, Xu, W.
登録日2012-06-14
公開日2012-09-19
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structural analysis of bengamide derivatives as inhibitors of methionine aminopeptidases.
J.Med.Chem., 55, 2012
4FO7
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Pseudomonas aeruginosa MetAP, in Mn form
分子名称: MANGANESE (II) ION, Methionine aminopeptidase
著者Ye, Q.Z, Lu, J.P.
登録日2012-06-20
公開日2013-07-03
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Methionine excision captured by the structures of a methionine aminopeptidase
To be published
4FLK
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Human MetAP1 with bengamide analog Y10, in Mn form
分子名称: (E,2R,3R,4S,5R)-N-(2,3-dihydro-1H-inden-2-yl)-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, MANGANESE (II) ION, Methionine aminopeptidase 1, ...
著者Ye, Q.Z, Xu, W.
登録日2012-06-14
公開日2012-09-19
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.47 Å)
主引用文献Structural analysis of bengamide derivatives as inhibitors of methionine aminopeptidases.
J.Med.Chem., 55, 2012
4FO8
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Pseudomonas aeruginosa MetAP with Met, in Mn form
分子名称: MANGANESE (II) ION, METHIONINE, Methionine aminopeptidase
著者Ye, Q.Z, Lu, J.P.
登録日2012-06-20
公開日2013-07-03
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Methionine excision captured by the structures of a methionine aminopeptidase
To be published
3PKE
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M. tuberculosis MetAP with bengamide analog Y10, in Ni form
分子名称: (E,2R,3R,4S,5R)-N-(2,3-dihydro-1H-inden-2-yl)-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, CHLORIDE ION, Methionine aminopeptidase, ...
著者Ye, Q.Z, Lu, J.P.
登録日2010-11-11
公開日2011-04-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidases by Bengamide Derivatives.
Chemmedchem, 6, 2011
3PKB
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M. tuberculosis MetAP with bengamide analog Y16, in Mn form
分子名称: (E,2R,3R,4S,5R)-N-(2-azanyl-2-oxidanylidene-ethyl)-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, CHLORIDE ION, MANGANESE (II) ION, ...
著者Ye, Q.Z, Lu, J.P.
登録日2010-11-11
公開日2011-04-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidases by Bengamide Derivatives.
Chemmedchem, 6, 2011
4FLI
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Human MetAP1 with bengamide analog Y16, in Mn form
分子名称: (E,2R,3R,4S,5R)-N-(2-azanyl-2-oxidanylidene-ethyl)-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, MANGANESE (II) ION, Methionine aminopeptidase 1, ...
著者Ye, Q.Z, Xu, W.
登録日2012-06-14
公開日2012-09-19
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structural analysis of bengamide derivatives as inhibitors of methionine aminopeptidases.
J.Med.Chem., 55, 2012
4FLJ
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Human MetAP1 with bengamide analog Y08, in Mn form
分子名称: (E,2R,3R,4S,5R)-N-[[(3S)-1-cyclopropylcarbonylpiperidin-3-yl]methyl]-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, MANGANESE (II) ION, Methionine aminopeptidase 1, ...
著者Ye, Q.Z, Xu, W.
登録日2012-06-14
公開日2012-09-19
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献Structural analysis of bengamide derivatives as inhibitors of methionine aminopeptidases.
J.Med.Chem., 55, 2012
3PKD
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M. tuberculosis MetAP with bengamide analog Y10, in Mn form
分子名称: (E,2R,3R,4S,5R)-N-(2,3-dihydro-1H-inden-2-yl)-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, MANGANESE (II) ION, Methionine aminopeptidase
著者Ye, Q.Z, Lu, J.P.
登録日2010-11-11
公開日2011-04-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.47 Å)
主引用文献Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidases by Bengamide Derivatives.
Chemmedchem, 6, 2011
3PKC
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BU of 3pkc by Molmil
M. tuberculosis MetAP with bengamide analog Y08, in Mn form
分子名称: (E,2R,3R,4S,5R)-N-[[(3S)-1-cyclopropylcarbonylpiperidin-3-yl]methyl]-2-methoxy-8,8-dimethyl-3,4,5-tris(oxidanyl)non-6-enamide, MANGANESE (II) ION, Methionine aminopeptidase
著者Ye, Q.Z, Lu, J.P.
登録日2010-11-11
公開日2011-04-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.47 Å)
主引用文献Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidases by Bengamide Derivatives.
Chemmedchem, 6, 2011
3PKA
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BU of 3pka by Molmil
M. tuberculosis MetAP with bengamide analog Y02, in Mn form
分子名称: (2R,3R,4S,5R,6E)-3,4,5-trihydroxy-2-methoxy-8,8-dimethyl-N-[2-(2,4,6-trimethylphenoxy)ethyl]non-6-enamide, CHLORIDE ION, MANGANESE (II) ION, ...
著者Ye, Q.Z, Lu, J.P.
登録日2010-11-11
公開日2011-04-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidases by Bengamide Derivatives.
Chemmedchem, 6, 2011
3IU7
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BU of 3iu7 by Molmil
M. tuberculosis methionine aminopeptidase with Mn inhibitor A02
分子名称: 5-(2-CHLOROPHENYL)FURAN-2-CARBOXYLIC ACID, CHLORIDE ION, MANGANESE (II) ION, ...
著者Ye, Q.Z, Lu, J.P.
登録日2009-08-30
公開日2010-01-12
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Catalysis and Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidase
J.Med.Chem., 53, 2010
3IU9
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M. tuberculosis methionine aminopeptidase with Ni inhibitor T07
分子名称: 5-[(2,4-dichlorobenzyl)sulfanyl]-4H-1,2,4-triazol-3-amine, CHLORIDE ION, Methionine aminopeptidase, ...
著者Ye, Q.Z, Lu, J.P.
登録日2009-08-30
公開日2010-01-12
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Catalysis and Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidase
J.Med.Chem., 53, 2010
3IU8
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M. tuberculosis methionine aminopeptidase with Ni inhibitor T03
分子名称: 3-[(4-fluorobenzyl)sulfanyl]-4H-1,2,4-triazole, CHLORIDE ION, Methionine aminopeptidase, ...
著者Ye, Q.Z, Lu, J.P.
登録日2009-08-30
公開日2010-01-12
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Catalysis and Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidase
J.Med.Chem., 53, 2010
2BB7
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BU of 2bb7 by Molmil
Mn Form Of E. coli Methionine Aminopeptidase In Complex With a quinolinyl sulfonamide inhibitor
分子名称: MANGANESE (II) ION, Methionine aminopeptidase, N-(QUINOLIN-8-YL)METHANESULFONAMIDE, ...
著者Ye, Q.Z.
登録日2005-10-17
公開日2006-01-24
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Metal mediated inhibition of methionine aminopeptidase by quinolinyl sulfonamides
Biochem.Biophys.Res.Commun., 339, 2006
2GTX
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Structural Basis of Catalysis by Mononuclear Methionine Aminopeptidase
分子名称: (1-AMINO-PENTYL)-PHOSPHONIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.Z.
登録日2006-04-28
公開日2006-07-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis of catalysis by monometalated methionine aminopeptidase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2GU4
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E. coli methionine aminopeptidase in complex with NleP, 1: 0.5, di-metalated
分子名称: (1-AMINO-PENTYL)-PHOSPHONIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.Z.
登録日2006-04-28
公開日2006-07-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural basis of catalysis by monometalated methionine aminopeptidase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2GU5
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E. coli methionine aminopeptidase in complex with NleP, 1: 1, di-metalated
分子名称: (1-AMINO-PENTYL)-PHOSPHONIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.Z.
登録日2006-04-28
公開日2006-07-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural basis of catalysis by monometalated methionine aminopeptidase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2GU6
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E. coli methionine aminopeptidase in complex with NleP, 1: 2, di-metalated
分子名称: (1-AMINO-PENTYL)-PHOSPHONIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.Z.
登録日2006-04-28
公開日2006-07-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural basis of catalysis by monometalated methionine aminopeptidase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2GU7
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E. coli methionine aminopeptidase unliganded, 1:0.5
分子名称: MANGANESE (II) ION, Methionine aminopeptidase, SODIUM ION
著者Ye, Q.Z.
登録日2006-04-28
公開日2006-07-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis of catalysis by monometalated methionine aminopeptidase.
Proc.Natl.Acad.Sci.Usa, 103, 2006

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