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3IU8

M. tuberculosis methionine aminopeptidase with Ni inhibitor T03

Summary for 3IU8
Entry DOI10.2210/pdb3iu8/pdb
Related1XNZ 1YJ3 3IU7 3IU9
DescriptorMethionine aminopeptidase, NICKEL (II) ION, 3-[(4-fluorobenzyl)sulfanyl]-4H-1,2,4-triazole, ... (6 entities in total)
Functional Keywordsenzyme-inhibitor complex, aminopeptidase, cobalt, hydrolase, metal-binding, protease
Biological sourceMycobacterium tuberculosis
Total number of polymer chains1
Total formula weight31763.55
Authors
Ye, Q.Z.,Lu, J.P. (deposition date: 2009-08-30, release date: 2010-01-12, Last modification date: 2023-09-06)
Primary citationLu, J.P.,Chai, S.C.,Ye, Q.Z.
Catalysis and Inhibition of Mycobacterium tuberculosis Methionine Aminopeptidase
J.Med.Chem., 53:1329-1337, 2010
Cited by
PubMed: 20038112
DOI: 10.1021/jm901624n
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.85 Å)
Structure validation

219515

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