1GJU
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![BU of 1gju by Molmil](/molmil-images/mine/1gju) | Maltosyltransferase from Thermotoga maritima | 分子名称: | MALTODEXTRIN GLYCOSYLTRANSFERASE, PHOSPHATE ION | 著者 | Roujeinikova, A, Raasch, C, Burke, J, Baker, P.J, Liebl, W, Rice, D.W. | 登録日 | 2001-08-02 | 公開日 | 2001-09-06 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | The Crystal Structure of Thermotoga Maritima Maltosyltransferase and its Implications for the Molecular Basis of the Novel Transfer Specificity J.Mol.Biol., 312, 2001
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1GM1
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![BU of 1gm1 by Molmil](/molmil-images/mine/1gm1) | Second PDZ Domain (PDZ2) of PTP-BL | 分子名称: | PROTEIN TYROSINE PHOSPHATASE | 著者 | Walma, T, Tessari, M, Aelen, J, Schepens, J, Hendriks, W, Vuister, G.W. | 登録日 | 2001-09-06 | 公開日 | 2002-03-08 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure, dynamics and binding characteristics of the second PDZ domain of PTP-BL. J. Mol. Biol., 316, 2002
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1GMY
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![BU of 1gmy by Molmil](/molmil-images/mine/1gmy) | Cathepsin B complexed with dipeptidyl nitrile inhibitor | 分子名称: | 2-AMINOETHANIMIDIC ACID, 3-METHYLPHENYLALANINE, CATHEPSIN B, ... | 著者 | Greenspan, P.D, Clark, K.L, Tommasi, R.A, Cowen, S.D, McQuire, L.W, Farley, D.L, van Duzer, J.H, Goldberg, R.L, Zhou, H, Du, Z, Fitt, J.J, Coppa, D.E, Fang, Z, Macchia, W, Zhu, L, Capparelli, M.P, Goldstein, R, Wigg, A.M, Doughty, J.R, Bohacek, R.S, Knap, A.K. | 登録日 | 2001-09-25 | 公開日 | 2002-09-19 | 最終更新日 | 2017-07-05 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Identification of Dipeptidyl Nitriles as Potent and Selective Inhibitors of Cathepsin B Through Structure-Based Drug Design J.Med.Chem., 44, 2001
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3TI7
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8H9Z
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![BU of 8h9z by Molmil](/molmil-images/mine/8h9z) | Annexin A5 protein mutant | 分子名称: | Annexin A5, CALCIUM ION | 著者 | Hua, Z.C, Tang, W. | 登録日 | 2022-10-26 | 公開日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | structure dissection of the membrane aggregation mechanism induced by Annexin A5 mutation To Be Published
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1HLA
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![BU of 1hla by Molmil](/molmil-images/mine/1hla) | STRUCTURE OF THE HUMAN CLASS I HISTOCOMPATIBILITY ANTIGEN, HLA-A2 | 分子名称: | BETA 2-MICROGLOBULIN, CLASS I HISTOCOMPATIBILITY ANTIGEN (HLA-A2) (ALPHA CHAIN) | 著者 | Bjorkman, P.J, Saper, M.A, Samraoui, B, Bennett, W.S, Strominger, J.L, Wiley, D.C. | 登録日 | 1987-10-15 | 公開日 | 1988-01-16 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Structure of the human class I histocompatibility antigen, HLA-A2. Nature, 329, 1987
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8H4F
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![BU of 8h4f by Molmil](/molmil-images/mine/8h4f) | Blasnase-T13A/P55F with D-asn | 分子名称: | D-ASPARAGINE, FORMIC ACID, L-asparaginase, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
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4I5M
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![BU of 4i5m by Molmil](/molmil-images/mine/4i5m) | Selective & Brain-Permeable Polo-like Kinase-2 (Plk-2) Inhibitors that Reduce -Synuclein Phosphorylation in Rat Brain | 分子名称: | 4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide, Serine/threonine-protein kinase PLK2 | 著者 | Aubele, D.L, Hom, R.K, Adler, M, Galemmo Jr, R.A, Bowers, S, Truong, A.P, Pan, H, Beroza, P, Neitz, R.J, Yao, N, Lin, M, Tonn, G, Zhang, H, Bova, M.P, Ren, Z, Tam, D, Ruslim, L, Baker, J, Diep, L, Fitzgerald, K, Hoffman, J, Motter, R, Fauss, D, Tanaka, P, Dappen, M, Jagodzinski, J, Chan, W, Konradi, A.W, Latimer, L, Zhu, Y.L, Artis, D.R, Sham, H.L, Anderson, J.P, Bergeron, M. | 登録日 | 2012-11-28 | 公開日 | 2013-12-25 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.801 Å) | 主引用文献 | Selective and brain-permeable polo-like kinase-2 (Plk-2) inhibitors that reduce alpha-synuclein phosphorylation in rat brain. Chemmedchem, 8, 2013
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4I6Z
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![BU of 4i6z by Molmil](/molmil-images/mine/4i6z) | Crystal structure of the transcriptional regulator TM1030 with 24bp DNA oligonucleotide | 分子名称: | DNA OLIGONUCLEOTIDE, Transcriptional regulator, TetR family | 著者 | Koclega, K.D, Chruszcz, M, Cooper, D.R, Petkowski, J.J, Tkaczuk, K.L, Joachimiak, A, Minor, W, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2012-11-30 | 公開日 | 2013-01-02 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Crystal structure of the transcriptional regulator TM1030 with 24bp DNA oligonucleotide To be Published
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8HIG
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8U45
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![BU of 8u45 by Molmil](/molmil-images/mine/8u45) | Crystal Structure Analysis of Aspergillus fumigatus alkaline protease | 分子名称: | Alkaline protease 1, CALCIUM ION, CHLORIDE ION, ... | 著者 | Fernandez, D, Diec, D.D.L, Guo, W, Russi, S. | 登録日 | 2023-09-08 | 公開日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Targeting Aspergillus allergen oryzin with a chemical probe at atomic precision. Sci Rep, 13, 2023
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4IAR
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![BU of 4iar by Molmil](/molmil-images/mine/4iar) | Crystal structure of the chimeric protein of 5-HT1B-BRIL in complex with ergotamine (PSI Community Target) | 分子名称: | (2S)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Chimera protein of human 5-hydroxytryptamine receptor 1B and E. Coli soluble cytochrome b562, Ergotamine | 著者 | Wang, C, Jiang, Y, Ma, J, Wu, H, Wacker, D, Katritch, V, Han, G.W, Liu, W, Huang, X, Vardy, E, McCorvy, J.D, Gao, X, Zhou, E.X, Melcher, K, Zhang, C, Bai, F, Yang, H, Yang, L, Jiang, H, Roth, B.L, Cherezov, V, Stevens, R.C, Xu, H.E, GPCR Network (GPCR) | 登録日 | 2012-12-07 | 公開日 | 2013-03-13 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural basis for molecular recognition at serotonin receptors. Science, 340, 2013
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8TWI
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![BU of 8twi by Molmil](/molmil-images/mine/8twi) | Cryo-EM structure of the PP2A:B55-FAM122A complex, PP2Ac body | 分子名称: | FE (III) ION, PPP2R1A-PPP2R2A-interacting phosphatase regulator 1, Serine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform, ... | 著者 | Fuller, J.R, Padi, S.K.R, Peti, W, Page, R. | 登録日 | 2023-08-21 | 公開日 | 2023-11-01 | 最終更新日 | 2024-01-17 | 実験手法 | ELECTRON MICROSCOPY (2.69 Å) | 主引用文献 | Cryo-EM structures of PP2A:B55-FAM122A and PP2A:B55-ARPP19. Nature, 625, 2024
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8TWE
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![BU of 8twe by Molmil](/molmil-images/mine/8twe) | Cryo-EM structure of the PP2A:B55-FAM122A complex, B55 body | 分子名称: | PPP2R1A-PPP2R2A-interacting phosphatase regulator 1, Serine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B alpha isoform, Serine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform, ... | 著者 | Fuller, J.R, Padi, S.K.R, Peti, W, Page, R. | 登録日 | 2023-08-21 | 公開日 | 2023-11-01 | 最終更新日 | 2024-01-17 | 実験手法 | ELECTRON MICROSCOPY (2.55 Å) | 主引用文献 | Cryo-EM structures of PP2A:B55-FAM122A and PP2A:B55-ARPP19. Nature, 625, 2024
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8TTB
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![BU of 8ttb by Molmil](/molmil-images/mine/8ttb) | Cryo-EM structure of the PP2A:B55-ARPP19 complex | 分子名称: | FE (III) ION, Serine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B alpha isoform, Serine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform, ... | 著者 | Fuller, J.R, Padi, S.K.R, Peti, W, Page, R. | 登録日 | 2023-08-13 | 公開日 | 2023-10-25 | 最終更新日 | 2024-01-17 | 実験手法 | ELECTRON MICROSCOPY (2.77 Å) | 主引用文献 | Cryo-EM structures of PP2A:B55-FAM122A and PP2A:B55-ARPP19. Nature, 625, 2024
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3TY0
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![BU of 3ty0 by Molmil](/molmil-images/mine/3ty0) | Structure of PPARgamma ligand binding domain in complex with (R)-5-(3-((3-(6-methoxybenzo[d]isoxazol-3-yl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)phenyl)-5-methyloxazolidine-2,4-dione | 分子名称: | (5R)-5-(3-{[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-2,3-dihydro-1H-benzimidazol-1-yl]methyl}phenyl)-5-methyl-1,3-oxazolidine-2,4-dione, Peroxisome proliferator-activated receptor gamma | 著者 | Soisson, S.M, Meinke, P.M, McKeever, B, Liu, W. | 登録日 | 2011-09-23 | 公開日 | 2011-11-23 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Benzimidazolones: a new class of selective peroxisome proliferator-activated receptor gamma (PPAR-gamma) modulators. J.Med.Chem., 54, 2011
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4HXB
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![BU of 4hxb by Molmil](/molmil-images/mine/4hxb) | Crystal structure of 6B9 FAB | 分子名称: | 6B9 FAB HEAVY CHAIN, 6B9 FAB LIGHT CHAIN, CALCIUM ION | 著者 | Johal, A.R, Jarrell, H.C, Khieu, N.H, Letts, J.A, Landry, R.C, Jachymek, W, Yang, Q, Jennings, H.J, Brisson, J.R, Evans, S.V. | 登録日 | 2012-11-09 | 公開日 | 2013-07-24 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | The antigen-binding site of an N-propionylated polysialic acid-specific antibody protective against group B meningococci is consistent with extended epitopes. Glycobiology, 23, 2013
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3U48
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![BU of 3u48 by Molmil](/molmil-images/mine/3u48) | From soil to structure: a novel dimeric family 3-beta-glucosidase isolated from compost using metagenomic analysis | 分子名称: | CALCIUM ION, JMB19063, beta-D-glucopyranose | 著者 | McAndrew, R.P, Park, J.I, Reindl, W, Friedland, G.D, D'haeseleer, P, Northen, T, Sale, K.L, Simmons, B.A, Adams, P.D. | 登録日 | 2011-10-07 | 公開日 | 2013-04-10 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | From soil to structure: a novel dimeric family 3-beta-glucosidase isolated from compost using metagenomic analysis To be Published
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8HPI
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3U1U
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![BU of 3u1u by Molmil](/molmil-images/mine/3u1u) | Crystal structure of RNA polymerase-associated protein RTF1 homolog Plus-3 domain | 分子名称: | GLYCEROL, RNA polymerase-associated protein RTF1 homolog, SULFATE ION, ... | 著者 | Guo, Y, Tempel, W, Bian, C, Wernimont, A.K, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Min, J, Structural Genomics Consortium (SGC) | 登録日 | 2011-09-30 | 公開日 | 2012-04-04 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of RNA polymerase-associated protein RTF1 homolog Plus-3 domain to be published
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5YCL
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![BU of 5ycl by Molmil](/molmil-images/mine/5ycl) | |
8H70
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8HRZ
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![BU of 8hrz by Molmil](/molmil-images/mine/8hrz) | |
8HPC
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8HPG
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