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PDB: 48 results
3T9H
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BU of 3t9h by Molmil
Kainate bound to a double cysteine mutant (A452C/S652C) of the ligand binding domain of GluA2
Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor 2, ZINC ION
Authors:Ahmed, A.H, Wang, S, Chuang, H.H, Oswald, R.E.
Deposit date:2011-08-02
Release date:2011-08-17
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.015 Å)
Cite:Mechanism of AMPA Receptor Activation by Partial Agonists: DISULFIDE TRAPPING OF CLOSED LOBE CONFORMATIONS.
J.Biol.Chem., 286, 2011
3T9V
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BU of 3t9v by Molmil
CNQX bound to a reduced double cysteine mutant (A452C/S652C) of the ligand binding domain of GluA2
Descriptor: 7-nitro-2,3-dioxo-2,3-dihydroquinoxaline-6-carbonitrile, Glutamate receptor 2, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2011-08-03
Release date:2011-08-17
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.975 Å)
Cite:Mechanism of AMPA Receptor Activation by Partial Agonists: DISULFIDE TRAPPING OF CLOSED LOBE CONFORMATIONS.
J.Biol.Chem., 286, 2011
3T9X
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BU of 3t9x by Molmil
Glutamate bound to a double cysteine mutant (V484C/E657C) of the ligand binding domain of GluA2
Descriptor: GLUTAMIC ACID, Glutamate receptor 2, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2011-08-03
Release date:2011-08-17
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.823 Å)
Cite:Mechanism of AMPA Receptor Activation by Partial Agonists: DISULFIDE TRAPPING OF CLOSED LOBE CONFORMATIONS.
J.Biol.Chem., 286, 2011
3T93
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BU of 3t93 by Molmil
Glutamate bound to a double cysteine mutant (A452C/S652C) of the ligand binding domain of GluA2
Descriptor: GLUTAMIC ACID, Glutamate receptor 2, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2011-08-02
Release date:2011-08-17
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.907 Å)
Cite:Mechanism of AMPA Receptor Activation by Partial Agonists: DISULFIDE TRAPPING OF CLOSED LOBE CONFORMATIONS.
J.Biol.Chem., 286, 2011
3DP6
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BU of 3dp6 by Molmil
Crystal structure of the binding domain of the AMPA subunit GluR2 bound to glutamate
Descriptor: GLUTAMIC ACID, Glutamate receptor 2, ZINC ION
Authors:Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E.
Deposit date:2008-07-07
Release date:2008-11-25
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:Structure of the S1S2 glutamate binding domain of GLuR3.
Proteins, 75, 2008
3DLN
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BU of 3dln by Molmil
Crystal structure of the binding domain of the AMPA subunit GluR3 bound to glutamate
Descriptor: GLUTAMIC ACID, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E.
Deposit date:2008-06-27
Release date:2008-11-25
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (1.91 Å)
Cite:Structure of the S1S2 glutamate binding domain of GLuR3.
Proteins, 75, 2008
3DP4
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BU of 3dp4 by Molmil
Crystal structure of the binding domain of the AMPA subunit GluR3 bound to AMPA
Descriptor: (S)-ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E.
Deposit date:2008-07-07
Release date:2008-11-25
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2.11 Å)
Cite:Structure of the S1S2 glutamate binding domain of GLuR3.
Proteins, 75, 2008
3H06
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BU of 3h06 by Molmil
Crystal structure of the binding domain of the AMPA subunit GluR2 bound to the willardiine antagonist, UBP282
Descriptor: 4-({3-[(2R)-2-amino-2-carboxyethyl]-2,6-dioxo-3,6-dihydropyrimidin-1(2H)-yl}methyl)benzoic acid, Glutamate receptor 2
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2009-04-08
Release date:2009-05-05
Last modified:2017-08-23
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Mechanisms of antagonism of the GluR2 AMPA receptor: structure and dynamics of the complex of two willardiine antagonists with the glutamate binding domain.
Biochemistry, 48, 2009
3H03
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BU of 3h03 by Molmil
Crystal structure of the binding domain of the AMPA subunit GluR2 bound to UBP277
Descriptor: 3-[3-(2-carboxyethyl)-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl]-L-alanine, Glutamate receptor 2, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2009-04-08
Release date:2009-05-05
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Mechanisms of antagonism of the GluR2 AMPA receptor: structure and dynamics of the complex of two willardiine antagonists with the glutamate binding domain.
Biochemistry, 48, 2009
3IL1
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BU of 3il1 by Molmil
Crystal structure of the AMPA subunit GluR2 bound to the allosteric modulator, IDRA-21
Descriptor: (3S)-7-chloro-3-methyl-3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxide, GLUTAMIC ACID, Glutamate receptor 2, ...
Authors:Ahmed, A.H, Ptak, C.P, Oswald, R.E.
Deposit date:2009-08-06
Release date:2009-09-15
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.998 Å)
Cite:Probing the allosteric modulator binding site of GluR2 with thiazide derivatives
Biochemistry, 48, 2009
3ILT
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BU of 3ilt by Molmil
Crystal structure of the AMPA subunit GluR2 bound to the allosteric modulator, trichlormethiazide
Descriptor: 6-CHLORO-3-(DICHLOROMETHYL)-3,4-DIHYDRO-2H-1,2,4-BENZOTHIADIAZINE-7-SULFONAMIDE 1,1-DIOXIDE, GLUTAMIC ACID, Glutamate receptor 2, ...
Authors:Ahmed, A.H, Ptak, C.P, Oswald, R.E.
Deposit date:2009-08-07
Release date:2009-09-15
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.107 Å)
Cite:Probing the allosteric modulator binding site of GluR2 with thiazide derivatives
Biochemistry, 48, 2009
3IK6
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BU of 3ik6 by Molmil
Crystal structure of the AMPA subunit GluR2 bound to the allosteric modulator, chlorothiazide
Descriptor: 6-chloro-3,4-dihydro-2H-1,2,4-benzothiadiazine-7-sulfonamide 1,1-dioxide, GLUTAMIC ACID, Glutamate receptor 2, ...
Authors:Ptak, C.P, Ahmed, A.H, Oswald, R.E.
Deposit date:2009-08-05
Release date:2009-09-15
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.101 Å)
Cite:Probing the allosteric modulator binding site of GluR2 with thiazide derivatives
Biochemistry, 48, 2009
3IJO
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BU of 3ijo by Molmil
Crystal structure of the AMPA subunit GluR2 bound to the allosteric modulator, althiazide
Descriptor: (3S)-6-chloro-3-[(prop-2-en-1-ylsulfanyl)methyl]-3,4-dihydro-2H-1,2,4-benzothiadiazine-7-sulfonamide 1,1-dioxide, GLUTAMIC ACID, Glutamate receptor 2, ...
Authors:Ptak, C.P, Ahmed, A.H, Oswald, R.E.
Deposit date:2009-08-04
Release date:2009-09-15
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.003 Å)
Cite:Probing the allosteric modulator binding site of GluR2 with thiazide derivatives
Biochemistry, 48, 2009
3IJX
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BU of 3ijx by Molmil
Crystal structure of the AMPA subunit GluR2 bound to the allosteric modulator, hydrochlorothiazide
Descriptor: 6-chloro-3,4-dihydro-2H-1,2,4-benzothiadiazine-7-sulfonamide 1,1-dioxide, GLUTAMIC ACID, Glutamate receptor 2, ...
Authors:Ptak, C.P, Ahmed, A.H, Oswald, R.E.
Deposit date:2009-08-05
Release date:2009-09-15
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.881 Å)
Cite:Probing the allosteric modulator binding site of GluR2 with thiazide derivatives
Biochemistry, 48, 2009
3ILU
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BU of 3ilu by Molmil
Crystal structure of the AMPA subunit GluR2 bound to the allosteric modulator, hydroflumethiazide
Descriptor: 6-(trifluoromethyl)-3,4-dihydro-2H-1,2,4-benzothiadiazine-7-sulfonamide 1,1-dioxide, GLUTAMIC ACID, Glutamate receptor 2, ...
Authors:Ahmed, A.H, Ptak, C.P, Oswald, R.E.
Deposit date:2009-08-07
Release date:2009-09-15
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.003 Å)
Cite:Probing the allosteric modulator binding site of GluR2 with thiazide derivatives
Biochemistry, 48, 2009
4F29
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BU of 4f29 by Molmil
Quisqualate bound to the ligand binding domain of GluA3i
Descriptor: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2012-05-07
Release date:2012-05-16
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.749 Å)
Cite:The loss of an electrostatic contact unique to AMPA receptor ligand binding domain 2 slows channel activation.
Biochemistry, 51, 2012
4F1Y
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BU of 4f1y by Molmil
CNQX bound to the ligand binding domain of GluA3
Descriptor: 7-nitro-2,3-dioxo-2,3-dihydroquinoxaline-6-carbonitrile, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2012-05-07
Release date:2012-05-16
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.79 Å)
Cite:The loss of an electrostatic contact unique to AMPA receptor ligand binding domain 2 slows channel activation.
Biochemistry, 51, 2012
4F2Q
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BU of 4f2q by Molmil
Quisqualate bound to the D655A mutant of the ligand binding domain of GluA3
Descriptor: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2012-05-08
Release date:2012-05-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.202 Å)
Cite:The loss of an electrostatic contact unique to AMPA receptor ligand binding domain 2 slows channel activation.
Biochemistry, 51, 2012
4F3B
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BU of 4f3b by Molmil
Glutamate bound to the D655A mutant of the ligand binding domain of GluA3
Descriptor: GLUTAMIC ACID, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2012-05-09
Release date:2012-05-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.818 Å)
Cite:The loss of an electrostatic contact unique to AMPA receptor ligand binding domain 2 slows channel activation.
Biochemistry, 51, 2012
4F31
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BU of 4f31 by Molmil
Kainate bound to the D655A mutant of the ligand binding domain of GluA3
Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2012-05-08
Release date:2012-05-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.286 Å)
Cite:The loss of an electrostatic contact unique to AMPA receptor ligand binding domain 2 slows channel activation.
Biochemistry, 51, 2012
4F39
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BU of 4f39 by Molmil
Kainate bound to the ligand binding domain of GluA3
Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2012-05-09
Release date:2012-05-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.834 Å)
Cite:The loss of an electrostatic contact unique to AMPA receptor ligand binding domain 2 slows channel activation.
Biochemistry, 51, 2012
4F2O
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BU of 4f2o by Molmil
Quisqualate bound to the D655A mutant of the ligand binding domain of GluA3
Descriptor: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2012-05-08
Release date:2012-05-23
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.912 Å)
Cite:The loss of an electrostatic contact unique to AMPA receptor ligand binding domain 2 slows channel activation.
Biochemistry, 51, 2012
4F3G
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BU of 4f3g by Molmil
Kainate bound to the ligand binding domain of GluA3i
Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor 3, ZINC ION
Authors:Ahmed, A.H, Oswald, R.E.
Deposit date:2012-05-09
Release date:2012-05-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.064 Å)
Cite:The loss of an electrostatic contact unique to AMPA receptor ligand binding domain 2 slows channel activation.
Biochemistry, 51, 2012
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