3DL8
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![BU of 3dl8 by Molmil](/molmil-images/mine/3dl8) | Structure of the complex of aquifex aeolicus SecYEG and bacillus subtilis SecA | 分子名称: | Preprotein translocase subunit secY, Protein translocase subunit secA, Protein-export membrane protein secG, ... | 著者 | Nam, Y, Zimmer, J, Rapoport, T.A. | 登録日 | 2008-06-26 | 公開日 | 2008-12-02 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (7.5 Å) | 主引用文献 | Structure of a complex of the ATPase SecA and the protein-translocation channel. Nature, 455, 2008
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5UDZ
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3TS0
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![BU of 3ts0 by Molmil](/molmil-images/mine/3ts0) | Mouse Lin28A in complex with let-7f-1 microRNA pre-element | 分子名称: | Protein lin-28 homolog A, RNA (5'-R(*GP*GP*GP*GP*UP*AP*GP*UP*GP*AP*UP*UP*UP*UP*AP*CP*CP*CP*UP*GP*GP*AP*G)-3'), ZINC ION | 著者 | Nam, Y, Sliz, P. | 登録日 | 2011-09-11 | 公開日 | 2011-11-16 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.763 Å) | 主引用文献 | Molecular Basis for Interaction of let-7 MicroRNAs with Lin28. Cell(Cambridge,Mass.), 147, 2011
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3TRZ
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![BU of 3trz by Molmil](/molmil-images/mine/3trz) | Mouse Lin28A in complex with let-7d microRNA pre-element | 分子名称: | Protein lin-28 homolog A, RNA (5'-R(*GP*GP*GP*CP*AP*GP*GP*GP*AP*UP*UP*UP*UP*GP*CP*CP*CP*GP*GP*AP*G)-3'), ZINC ION | 著者 | Nam, Y, Sliz, P. | 登録日 | 2011-09-11 | 公開日 | 2011-11-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Molecular Basis for Interaction of let-7 MicroRNAs with Lin28. Cell(Cambridge,Mass.), 147, 2011
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3TS2
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![BU of 3ts2 by Molmil](/molmil-images/mine/3ts2) | Mouse Lin28A in complex with let-7g microRNA pre-element | 分子名称: | Protein lin-28 homolog A, RNA (5'-R(*GP*GP*GP*GP*UP*CP*UP*AP*UP*GP*AP*UP*AP*CP*CP*AP*CP*CP*CP*CP*GP*GP*AP*G)-3'), ZINC ION | 著者 | Nam, Y, Sliz, P. | 登録日 | 2011-09-11 | 公開日 | 2011-11-16 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Molecular Basis for Interaction of let-7 MicroRNAs with Lin28. Cell(Cambridge,Mass.), 147, 2011
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3V79
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![BU of 3v79 by Molmil](/molmil-images/mine/3v79) | Structure of human Notch1 transcription complex including CSL, RAM, ANK, and MAML-1 on HES-1 promoter DNA sequence | 分子名称: | DNA 5'-D(*GP*TP*TP*AP*CP*TP*GP*TP*GP*GP*GP*AP*AP*AP*GP*AP*AP*A)-3', DNA 5'-D(*TP*TP*TP*CP*TP*TP*TP*CP*CP*CP*AP*CP*AP*GP*TP*AP*AP*C)-3', Mastermind-like protein 1, ... | 著者 | Nam, Y, Sliz, P, Blacklow, S. | 登録日 | 2011-12-20 | 公開日 | 2012-02-15 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.85 Å) | 主引用文献 | Conformational Locking upon Cooperative Assembly of Notch Transcription Complexes. Structure, 20, 2012
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2F8Y
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![BU of 2f8y by Molmil](/molmil-images/mine/2f8y) | Crystal structure of human Notch1 ankyrin repeats to 1.55A resolution. | 分子名称: | Notch homolog 1, translocation-associated (Drosophila), SULFATE ION | 著者 | Nam, Y, Sliz, P, Blacklow, S.C. | 登録日 | 2005-12-04 | 公開日 | 2006-04-04 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structural basis for cooperativity in recruitment of MAML coactivators to Notch transcription complexes. Cell(Cambridge,Mass.), 124, 2006
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2F8X
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![BU of 2f8x by Molmil](/molmil-images/mine/2f8x) | Crystal structure of activated Notch, CSL and MAML on HES-1 promoter DNA sequence | 分子名称: | 5'-D(*GP*TP*TP*AP*CP*TP*GP*TP*GP*GP*GP*AP*AP*AP*GP*AP*AP*A)-3', 5'-D(*TP*TP*TP*CP*TP*TP*TP*CP*CP*CP*AP*CP*AP*GP*TP*AP*AP*C)-3', Mastermind-like protein 1, ... | 著者 | Nam, Y, Sliz, P, Blacklow, S.C. | 登録日 | 2005-12-04 | 公開日 | 2006-04-04 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | Structural basis for cooperativity in recruitment of MAML coactivators to Notch transcription complexes. Cell(Cambridge,Mass.), 124, 2006
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5AWJ
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![BU of 5awj by Molmil](/molmil-images/mine/5awj) | Crystal structure of VDR-LBD/partial agonist complex: 22S-hexyl analogue | 分子名称: | (1R,3R)-5-[(2E)-2-[(1R,3aS,7aR)-1-[(2R,3S)-3-(2-hydroxyethyl)nonan-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-2-methylidene-cyclohexane-1,3-diol, Mediator of RNA polymerase II transcription subunit 1, Vitamin D3 receptor,Vitamin D3 receptor | 著者 | Anami, Y, Itoh, T, Inaba, Y, Nakabayashi, M, Ikura, T, Ito, N, Yamamoto, K. | 登録日 | 2015-07-04 | 公開日 | 2015-11-18 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Fine tuning of agonistic/antagonistic activity for vitamin D receptor by 22-alkyl chain length of ligands: 22S-Hexyl compound unexpectedly restored agonistic activity. Bioorg.Med.Chem., 23, 2015
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5AWK
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![BU of 5awk by Molmil](/molmil-images/mine/5awk) | Crystal structure of VDR-LBD/partial agonist complex: 22S-ethyl analogue | 分子名称: | (1R,3R)-5-[(2E)-2-[(1R,3aS,7aR)-1-[(2R,3S)-3-ethyl-5-oxidanyl-pentan-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-2-methylidene-cyclohexane-1,3-diol, Mediator of RNA polymerase II transcription subunit 1, Vitamin D3 receptor,Vitamin D3 receptor | 著者 | Anami, Y, Itoh, T, Yamamoto, K. | 登録日 | 2015-07-04 | 公開日 | 2015-11-18 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Fine tuning of agonistic/antagonistic activity for vitamin D receptor by 22-alkyl chain length of ligands: 22S-Hexyl compound unexpectedly restored agonistic activity. Bioorg.Med.Chem., 23, 2015
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5B41
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![BU of 5b41 by Molmil](/molmil-images/mine/5b41) | Crystal structure of VDR-LBD complexed with 2-methylidene-19-nor-1a,25-dihydroxyvitamin D3 | 分子名称: | (1R,3R)-5-(2-((1R,3aS,7aR,E)-1-((R)-6-hydroxy-6-methylheptan-2-yl)-7a-methyloctahydro-4H-inden-4-ylidene)ethylidene)-2- methylenecyclohexane-1,3-diol, Mediator of RNA polymerase II transcription subunit 1, Vitamin D3 receptor | 著者 | Anami, Y, Itoh, T, Yamamoto, K. | 登録日 | 2016-03-23 | 公開日 | 2016-12-07 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Apo- and Antagonist-Binding Structures of Vitamin D Receptor Ligand-Binding Domain Revealed by Hybrid Approach Combining Small-Angle X-ray Scattering and Molecular Dynamics J.Med.Chem., 59, 2016
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3WT5
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![BU of 3wt5 by Molmil](/molmil-images/mine/3wt5) | A mixed population of antagonist and agonist binding conformers in a single crystal explains partial agonism against vitamin D receptor: Active vitamin D analogues with 22R-alkyl group | 分子名称: | (1R,3R,7E,17beta)-17-[(2R,3R)-3-butyl-6-hydroxy-6-methylheptan-2-yl]-2-methylidene-9,10-secoestra-5,7-diene-1,3-diol, Mediator of RNA polymerase II transcription subunit 1, Vitamin D3 receptor | 著者 | Anami, Y, Itoh, T, Yamamoto, K. | 登録日 | 2014-04-08 | 公開日 | 2014-06-11 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | A Mixed Population of Antagonist and Agonist Binding Conformers in a Single Crystal Explains Partial Agonism against Vitamin D Receptor: Active Vitamin D Analogues with 22R-Alkyl Group. J.Med.Chem., 57, 2014
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3WT7
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![BU of 3wt7 by Molmil](/molmil-images/mine/3wt7) | Crystal structure of VDR-LBD complexed with 22R-Butyl-2-methylidene-26,27-dimethyl-19,24-dinor-1 ,25-dihydroxyvitamin D3 | 分子名称: | (1R,3R,7E,17beta)-17-[(2R,3R)-3-butyl-5-ethyl-5-hydroxyheptan-2-yl]-2-methylidene-9,10-secoestra-5,7-diene-1,3-diol, Mediator of RNA polymerase II transcription subunit 1, Vitamin D3 receptor | 著者 | Anami, Y, Itoh, T, Yamamoto, K. | 登録日 | 2014-04-08 | 公開日 | 2014-06-11 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | A Mixed Population of Antagonist and Agonist Binding Conformers in a Single Crystal Explains Partial Agonism against Vitamin D Receptor: Active Vitamin D Analogues with 22R-Alkyl Group. J.Med.Chem., 57, 2014
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3WT6
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![BU of 3wt6 by Molmil](/molmil-images/mine/3wt6) | A mixed population of antagonist and agonist binding conformers in a single crystal explains partial agonism against vitamin D receptor: Active vitamin D analogues with 22R-alkyl group | 分子名称: | (1R,3R,7E,17beta)-17-[(2R,3R)-3-butyl-6-hydroxy-6-methylheptan-2-yl]-2-methylidene-9,10-secoestra-5,7-diene-1,3-diol, Mediator of RNA polymerase II transcription subunit 1, Vitamin D3 receptor | 著者 | Anami, Y, Itoh, T, Yamamoto, K. | 登録日 | 2014-04-08 | 公開日 | 2014-06-11 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | A Mixed Population of Antagonist and Agonist Binding Conformers in a Single Crystal Explains Partial Agonism against Vitamin D Receptor: Active Vitamin D Analogues with 22R-Alkyl Group. J.Med.Chem., 57, 2014
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6DU4
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![BU of 6du4 by Molmil](/molmil-images/mine/6du4) | Crystal structure of hMettl16 catalytic domain in complex with MAT2A 3'UTR hairpin 1 | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, U6 small nuclear RNA (adenine-(43)-N(6))-methyltransferase, ... | 著者 | Doxtader, K, Wang, P, Nam, Y. | 登録日 | 2018-06-19 | 公開日 | 2018-09-26 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural Basis for Regulation of METTL16, an S-Adenosylmethionine Homeostasis Factor. Mol. Cell, 71, 2018
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6V5C
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![BU of 6v5c by Molmil](/molmil-images/mine/6v5c) | Human Drosha and DGCR8 in complex with Primary MicroRNA (MP/RNA complex) - partially docked state | 分子名称: | Microprocessor complex subunit DGCR8, Pri-miR-16-2 (66-MER), Ribonuclease 3 | 著者 | Partin, A, Zhang, K, Jeong, B, Herrell, E, Li, S, Chiu, W, Nam, Y. | 登録日 | 2019-12-04 | 公開日 | 2020-04-08 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (4.4 Å) | 主引用文献 | Cryo-EM Structures of Human Drosha and DGCR8 in Complex with Primary MicroRNA. Mol.Cell, 78, 2020
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6UV4
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![BU of 6uv4 by Molmil](/molmil-images/mine/6uv4) | Crystal structure of the core domain of RNA helicase DDX17 with RNA pri-18a-oligo1 | 分子名称: | 18a_oligo1, ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, ... | 著者 | Ngo, T.D, Partin, A.C, Nam, Y. | 登録日 | 2019-11-01 | 公開日 | 2020-01-01 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | RNA Specificity and Autoregulation of DDX17, a Modulator of MicroRNA Biogenesis. Cell Rep, 29, 2019
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6UV3
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![BU of 6uv3 by Molmil](/molmil-images/mine/6uv3) | Crystal structure of the core domain of RNA helicase DDX17 with RNA pri-125a-oligo2 | 分子名称: | 125a-oligo2, ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, ... | 著者 | Ngo, T.D, Partin, A.C, Nam, Y. | 登録日 | 2019-11-01 | 公開日 | 2020-01-01 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.597 Å) | 主引用文献 | RNA Specificity and Autoregulation of DDX17, a Modulator of MicroRNA Biogenesis. Cell Rep, 29, 2019
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6UV0
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6UV1
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![BU of 6uv1 by Molmil](/molmil-images/mine/6uv1) | Crystal structure of RNA helicase DDX17 in complex of rU10 RNA | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, MAGNESIUM ION, ... | 著者 | Ngo, T.D, Partin, A.C, Nam, Y. | 登録日 | 2019-11-01 | 公開日 | 2020-01-01 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.307 Å) | 主引用文献 | RNA Specificity and Autoregulation of DDX17, a Modulator of MicroRNA Biogenesis. Cell Rep, 29, 2019
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6UV2
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![BU of 6uv2 by Molmil](/molmil-images/mine/6uv2) | Crystal structure of the core domain of RNA helicase DDX17 with RNA pri-125a-oligo1 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, MAGNESIUM ION, ... | 著者 | Ngo, T.D, Partin, A.C, Nam, Y. | 登録日 | 2019-11-01 | 公開日 | 2020-01-01 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.894 Å) | 主引用文献 | RNA Specificity and Autoregulation of DDX17, a Modulator of MicroRNA Biogenesis. Cell Rep, 29, 2019
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6V5B
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![BU of 6v5b by Molmil](/molmil-images/mine/6v5b) | Human Drosha and DGCR8 in complex with Primary MicroRNA (MP/RNA complex) - Active state | 分子名称: | CALCIUM ION, Microprocessor complex subunit DGCR8, Pri-miR-16-2 (78-MER), ... | 著者 | Partin, A, Zhang, K, Jeong, B, Herrell, E, Li, S, Chiu, W, Nam, Y. | 登録日 | 2019-12-04 | 公開日 | 2020-04-08 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Cryo-EM Structures of Human Drosha and DGCR8 in Complex with Primary MicroRNA. Mol.Cell, 78, 2020
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7RX6
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7RX8
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5K7U
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![BU of 5k7u by Molmil](/molmil-images/mine/5k7u) | |