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3WT5

A mixed population of antagonist and agonist binding conformers in a single crystal explains partial agonism against vitamin D receptor: Active vitamin D analogues with 22R-alkyl group

Summary for 3WT5
Entry DOI10.2210/pdb3wt5/pdb
Related3WT6 3WT7
DescriptorVitamin D3 receptor, Mediator of RNA polymerase II transcription subunit 1, (1R,3R,7E,17beta)-17-[(2R,3R)-3-butyl-6-hydroxy-6-methylheptan-2-yl]-2-methylidene-9,10-secoestra-5,7-diene-1,3-diol, ... (4 entities in total)
Functional Keywordstranscription, vitamin d3, vdre, rxr, co-factors, nuclear
Biological sourceRattus norvegicus (rats)
More
Cellular locationNucleus: P13053 Q15648
Total number of polymer chains2
Total formula weight32638.68
Authors
Anami, Y.,Itoh, T.,Yamamoto, K. (deposition date: 2014-04-08, release date: 2014-06-11, Last modification date: 2024-03-20)
Primary citationAnami, Y.,Itoh, T.,Egawa, D.,Yoshimoto, N.,Yamamoto, K.
A Mixed Population of Antagonist and Agonist Binding Conformers in a Single Crystal Explains Partial Agonism against Vitamin D Receptor: Active Vitamin D Analogues with 22R-Alkyl Group.
J.Med.Chem., 57:4351-4367, 2014
Cited by
PubMed: 24742174
DOI: 10.1021/jm500392t
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.9 Å)
Structure validation

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