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3WT5

A mixed population of antagonist and agonist binding conformers in a single crystal explains partial agonism against vitamin D receptor: Active vitamin D analogues with 22R-alkyl group

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues19
DetailsBINDING SITE FOR RESIDUE YA1 A 501
ChainResidue
ATYR143
ACYS284
AVAL296
AHIS301
AILE306
ALEU309
AHIS393
ALEU400
APHE418
AHOH766
AHOH812
AVAL230
ASER233
AILE264
AMET268
AARG270
ASER271
ASER274
ATRP282

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBINDING: BINDING => ECO:0000269|PubMed:15065852, ECO:0000269|PubMed:17227670
ChainResidueDetails
ATYR143
AARG270
AVAL314
AVAL348

218853

PDB entries from 2024-04-24

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