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PDB: 7 件

4J8N
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BU of 4j8n by Molmil
Aurora A Kinase Apo
分子名称: Aurora kinase A
著者Meyerowitz, J.G, Gustafson, W.C, Shokat, K.M, Weiss, W.A.
登録日2013-02-14
公開日2014-09-10
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.135 Å)
主引用文献Drugging MYCN through an Allosteric Transition in Aurora Kinase A.
Cancer Cell, 26, 2014
4J8M
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Aurora A in complex with CD532
分子名称: 1,2-ETHANEDIOL, 1-[4-[[4-[(5-cyclopentyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-3-[3-(trifluoromethyl)phenyl]urea, Aurora kinase A, ...
著者Meyerowitz, J.G, Gustafson, W.C, Shokat, K.M, Weiss, W.A.
登録日2013-02-14
公開日2014-09-10
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (1.853 Å)
主引用文献Drugging MYCN through an Allosteric Transition in Aurora Kinase A.
Cancer Cell, 26, 2014
7RYC
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Oxytocin receptor (OTR) bound to oxytocin in complex with a heterotrimeric Gq protein
分子名称: Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(i) subunit alpha-2,Guanine nucleotide-binding protein G(s) subunit alpha isoforms short, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, ...
著者Meyerowitz, J.G, Robertson, M.J, Skiniotis, G.
登録日2021-08-24
公開日2022-03-09
最終更新日2022-03-30
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献The oxytocin signaling complex reveals a molecular switch for cation dependence.
Nat.Struct.Mol.Biol., 29, 2022
7M3G
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Asymmetric Activation of the Calcium Sensing Receptor Homodimer
分子名称: 2-[4-[(3S)-3-[[(1R)-1-naphthalen-1-ylethyl]amino]pyrrolidin-1-yl]phenyl]ethanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Gao, Y, Robertson, M.J, Zhang, C, Meyerowitz, J.G, Panova, O, Skiniotis, G.
登録日2021-03-18
公開日2021-06-30
最終更新日2021-07-21
実験手法ELECTRON MICROSCOPY (2.5 Å)
主引用文献Asymmetric activation of the calcium-sensing receptor homodimer.
Nature, 595, 2021
7M3J
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BU of 7m3j by Molmil
Asymmetric Activation of the Calcium Sensing Receptor Homodimer
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-chloro-6-[(2R)-2-hydroxy-3-{[2-methyl-1-(naphthalen-2-yl)propan-2-yl]amino}propoxy]benzonitrile, ...
著者Gao, Y, Robertson, M.J, Zhang, C, Meyerowitz, J.G, Panova, O, Skiniotis, G.
登録日2021-03-18
公開日2021-06-30
最終更新日2021-07-21
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Asymmetric activation of the calcium-sensing receptor homodimer.
Nature, 595, 2021
7M3E
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BU of 7m3e by Molmil
Asymmetric Activation of the Calcium Sensing Receptor Homodimer
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-chloro-6-[(2R)-2-hydroxy-3-{[2-methyl-1-(naphthalen-2-yl)propan-2-yl]amino}propoxy]benzonitrile, ...
著者Gao, Y, Robertson, M.J, Zhang, C, Meyerowitz, J.G, Panova, O, Skiniotis, G.
登録日2021-03-18
公開日2021-06-30
最終更新日2021-07-21
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Asymmetric activation of the calcium-sensing receptor homodimer.
Nature, 595, 2021
7M3F
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BU of 7m3f by Molmil
Asymmetric Activation of the Calcium Sensing Receptor Homodimer
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Gao, Y, Robertson, M.J, Zhang, C, Meyerowitz, J.G, Panova, O, Skiniotis, G.
登録日2021-03-18
公開日2021-06-30
最終更新日2021-07-21
実験手法ELECTRON MICROSCOPY (2.8 Å)
主引用文献Asymmetric activation of the calcium-sensing receptor homodimer.
Nature, 595, 2021

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件を2024-07-24に公開中

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