3CL0
| N1 Neuraminidase H274Y + oseltamivir | 分子名称: | (3R,4R,5S)-4-(acetylamino)-5-amino-3-(pentan-3-yloxy)cyclohex-1-ene-1-carboxylic acid, CALCIUM ION, Neuraminidase | 著者 | Collins, P, Haire, L.F, Lin, Y.P, Liu, J, Russell, R.J, Walker, P.A, Skehel, J.J, Martin, S.R, Hay, A.J, Gamblin, S.J. | 登録日 | 2008-03-18 | 公開日 | 2008-05-20 | 最終更新日 | 2018-08-22 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structures of oseltamivir-resistant influenza virus neuraminidase mutants. Nature, 453, 2008
|
|
3CKZ
| N1 Neuraminidase H274Y + Zanamivir | 分子名称: | CALCIUM ION, Neuraminidase, ZANAMIVIR | 著者 | Colllins, P, Haire, L.F, Lin, Y.P, Liu, J, Russell, R.J, Walker, P.A, Skehel, J.J, Martin, S.R, Hay, A.J, Gamblin, S.J. | 登録日 | 2008-03-18 | 公開日 | 2008-05-20 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of oseltamivir-resistant influenza virus neuraminidase mutants. Nature, 453, 2008
|
|
3CL2
| N1 Neuraminidase N294S + Oseltamivir | 分子名称: | (3R,4R,5S)-4-(acetylamino)-5-amino-3-(pentan-3-yloxy)cyclohex-1-ene-1-carboxylic acid, Neuraminidase | 著者 | Collins, P, Haire, L.F, Lin, Y.P, Liu, J, Russell, R.J, Walker, P.A, Skehel, J.J, Martin, S.R, Hay, A.J, Gamblin, S.J. | 登録日 | 2008-03-18 | 公開日 | 2008-05-20 | 最終更新日 | 2018-08-22 | 実験手法 | X-RAY DIFFRACTION (2.538 Å) | 主引用文献 | Crystal structures of oseltamivir-resistant influenza virus neuraminidase mutants. Nature, 453, 2008
|
|
4CR0
| Crystal Structure of H5 (VN1194) Asn186Lys/Gly143Arg Mutant Haemagglutinin | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Hemagglutinin HA1, Hemagglutinin HA2 | 著者 | Collins, P.J, Vachieri, S.G, Xiong, X, Xiao, H, Martin, S.R, Coombs, P.J, Liu, J, Walker, P.A, Lin, Y.P, McCauley, J.W, Gamblin, S.J, Skehel, J.J. | 登録日 | 2014-02-21 | 公開日 | 2014-05-28 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Enhanced Human Receptor Binding by H5 Haemagglutinins. Virology, 456, 2014
|
|
5X4G
| Crystal structure of Fab fragment of anti-CD147 monoclonal antibody 6H8 | 分子名称: | 6H8 Fab heavy chain, 6H8 Fab light chain | 著者 | Lin, P, Zhang, M.-Y, Chen, X, Ye, S, Yu, X.-L, Zhang, R.-G, Zhu, P, Chen, Z.-N. | 登録日 | 2017-02-13 | 公開日 | 2018-01-24 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Crystal structure of CD147 C2 domain in complex with Fab of its monoclonal antibody To Be Published
|
|
5X0T
| Crystal structure of CD147 C2 domain in complex with Fab of its monoclonal antibody 6H8 | 分子名称: | 6H8 Fab fragment heavy chain, 6H8 Fab fragment light chain, Basigin | 著者 | Lin, P, Zhang, M.-Y, Ye, S, Chen, X, Yu, X.-L, Zhang, R.-G, Zhu, P, Chen, Z.-N. | 登録日 | 2017-01-23 | 公開日 | 2018-01-24 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of CD147 C2 domain in complex with Fab of its monoclonal antibody To Be Published
|
|
4DGW
| |
417D
| A THYMINE-LIKE BASE ANALOGUE FORMS WOBBLE PAIRS WITH ADENINE | 分子名称: | DNA (5'-D(*CP*AP*CP*GP*(C46)P*G)-3') | 著者 | Lin, P.K.T, Schuerman, M.H, Moore, G.S, Van Meervelt, L, Loakes, D, Brown, D.M, Moore, M.H. | 登録日 | 1998-07-15 | 公開日 | 1998-09-30 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | A thymine-like base analogue forms wobble pairs with adenine in a Z-DNA duplex. J.Mol.Biol., 282, 1998
|
|
3QHQ
| Structure of CRISPR-associated protein Csn2 | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, Sag0897 family CRISPR-associated protein | 著者 | Ellinger, P, Arslan, Z, Wurm, R, Tschapek, B, Pfeffer, K, Wagner, R, Schmitt, L, Pul, U, Smits, S.H. | 登録日 | 2011-01-26 | 公開日 | 2012-02-01 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of CRISPR-associated protein Csn2 To be Published
|
|
5JW3
| Structure of MEDI8852 Fab Fragment in Complex with H7 HA | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Hemagglutinin, ... | 著者 | Collins, P.J, Neu, U, Walker, P.A, Vorlaender, M.K, Ogrodowicz, R.W, Martin, S.R, Gamblin, S.J, Skehel, J.J. | 登録日 | 2016-05-11 | 公開日 | 2016-08-03 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (3.75 Å) | 主引用文献 | Structure and Function Analysis of an Antibody Recognizing All Influenza A Subtypes. Cell, 166, 2016
|
|
3G5F
| Crystallographic analysis of cytochrome P450 cyp121 | 分子名称: | Cytochrome P450 121, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION | 著者 | Belin, P, Le Du, M.H, Gondry, M. | 登録日 | 2009-02-05 | 公開日 | 2009-04-21 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Identification and structural basis of the reaction catalyzed by CYP121, an essential cytochrome P450 in Mycobacterium tuberculosis. Proc.Natl.Acad.Sci.USA, 106, 2009
|
|
2GLQ
| X-ray structure of human alkaline phosphatase in complex with strontium | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Alkaline phosphatase, placental type, ... | 著者 | Llinas, P, Masella, M, Stigbrand, T, Menez, A, Stura, E.A, Le Du, M.H. | 登録日 | 2006-04-05 | 公開日 | 2006-04-25 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structural studies of human alkaline phosphatase in complex with strontium: Implication for its secondary effect in bones. Protein Sci., 15, 2006
|
|
3G5H
| Crystallographic analysis of cytochrome P450 cyp121 | 分子名称: | (3S,6S)-3,6-bis(4-hydroxybenzyl)piperazine-2,5-dione, Cytochrome P450 121, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Belin, P, Le Du, M.H, Gondry, M. | 登録日 | 2009-02-05 | 公開日 | 2009-04-21 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Identification and structural basis of the reaction catalyzed by CYP121, an essential cytochrome P450 in Mycobacterium tuberculosis. Proc.Natl.Acad.Sci.USA, 106, 2009
|
|
4PXJ
| |
5EXO
| Crystal structure of Human galectin-3 CRD in complex with methyl 2-O-acetyl-3-O-(2H-chromene-3-yl-methyl)-a-D-galactopyranoside inhibitor | 分子名称: | CHLORIDE ION, Galectin-3, [(2~{S},3~{R},4~{S},5~{S},6~{R})-6-(hydroxymethyl)-2-methoxy-5-oxidanyl-4-[(2-oxidanylidenechromen-3-yl)methoxy]oxan-3-yl] ethanoate | 著者 | Collins, P.M, Blanchard, H. | 登録日 | 2015-11-23 | 公開日 | 2016-10-05 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.502 Å) | 主引用文献 | A Selective Galactose-Coumarin-Derived Galectin-3 Inhibitor Demonstrates Involvement of Galectin-3-glycan Interactions in a Pulmonary Fibrosis Model. J.Med.Chem., 59, 2016
|
|
1ZEF
| structure of alkaline phosphatase from human placenta in complex with its uncompetitive inhibitor L-Phe | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Alkaline phosphatase, CALCIUM ION, ... | 著者 | Llinas, P, Stura, E.A, Menez, A, Kiss, Z, Stigbrand, T, Millan, J.L, Le Du, M.H. | 登録日 | 2005-04-18 | 公開日 | 2005-06-28 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural Studies of Human Placental Alkaline Phosphatase in Complex with Functional Ligands. J.Mol.Biol., 350, 2005
|
|
4LBM
| |
4LBO
| |
4LBN
| |
1YWH
| crystal structure of urokinase plasminogen activator receptor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Llinas, P, Le Du, M.H, Gardsvoll, H, Dano, K, Ploug, M, Gilquin, B, Stura, E.A, Menez, A. | 登録日 | 2005-02-18 | 公開日 | 2005-05-10 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal structure of the human urokinase plasminogen activator receptor bound to an antagonist peptide EMBO J., 24, 2005
|
|
1ZED
| Alkaline phosphatase from human placenta in complex with p-nitrophenyl-phosphonate | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Alkaline phosphatase, CALCIUM ION, ... | 著者 | Llinas, P, Stura, E.A, Menez, A, Kiss, Z, Stigbrand, T, Millan, J.L, Le Du, M.H. | 登録日 | 2005-04-18 | 公開日 | 2005-06-28 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Structural Studies of Human Placental Alkaline Phosphatase in Complex with Functional Ligands. J.Mol.Biol., 350, 2005
|
|
5E88
| Crystal structure of Human galectin-3 CRD in complex with thienyl-1,2,3-triazolyl thiodigalactoside inhibitor | 分子名称: | 3-deoxy-3-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]-beta-D-galactopyranosyl 3-deoxy-1-thio-3-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]-beta-D-galactopyranoside, CHLORIDE ION, Galectin-3 | 著者 | Collins, P.M, Blanchard, H. | 登録日 | 2015-10-13 | 公開日 | 2016-08-24 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Galectin-3-Binding Glycomimetics that Strongly Reduce Bleomycin-Induced Lung Fibrosis and Modulate Intracellular Glycan Recognition. Chembiochem, 17, 2016
|
|
4JC1
| |
5Y5N
| Crystal structure of human Sirtuin 2 in complex with a selective inhibitor | 分子名称: | 2-[[3-(2-phenylethoxy)phenyl]amino]benzamide, NAD-dependent protein deacetylase sirtuin-2, ZINC ION | 著者 | Mellini, P, Itoh, Y, Tsumoto, H, Li, Y, Suzuki, M, Tokuda, N, Kakizawa, T, Miura, Y, Takeuchi, J, Lahtela-Kakkonen, M, Suzuki, T. | 登録日 | 2017-08-09 | 公開日 | 2017-09-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Potent mechanism-based sirtuin-2-selective inhibition by anin situ-generated occupant of the substrate-binding site, "selectivity pocket" and NAD+-binding site. Chem Sci, 8, 2017
|
|
1EQY
| COMPLEX BETWEEN RABBIT MUSCLE ALPHA-ACTIN: HUMAN GELSOLIN DOMAIN 1 | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, ALPHA ACTIN, CALCIUM ION, ... | 著者 | McLaughlin, P.J, Gooch, J.T, Mannherz, H.G, Weeds, A.G. | 登録日 | 2000-04-06 | 公開日 | 2000-05-03 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure of gelsolin segment 1-actin complex and the mechanism of filament severing. Nature, 364, 1993
|
|