1GME
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![BU of 1gme by Molmil](/molmil-images/mine/1gme) | Crystal structure and assembly of an eukaryotic small heat shock protein | 分子名称: | HEAT SHOCK PROTEIN 16.9B | 著者 | Van Montfort, R.L.M, Basha, E, Friedrich, K.L, Slingsby, C, Vierling, E. | 登録日 | 2001-09-13 | 公開日 | 2001-11-29 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal Structure and Assembly of an Eukaryotic Small Heat Shock Protein Nat.Struct.Biol., 8, 2001
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4ALO
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![BU of 4alo by Molmil](/molmil-images/mine/4alo) | STRUCTURE AND PROPERTIES OF H1 CRUSTACYANIN FROM LOBSTER HOMARUS AMERICANUS | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, H1 APOCRUSTACYANIN, SODIUM ION, ... | 著者 | Ferrari, M, Folli, C, Pincolini, E, Mcclintock, T.S, Roessle, M, Berni, R, Cianci, M. | 登録日 | 2012-03-05 | 公開日 | 2012-08-08 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Structural Characterization of Recombinant Crustacyanin Subunits from the Lobster Homarus Americanus. Acta Crystallogr.,Sect.F, 68, 2012
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2C86
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![BU of 2c86 by Molmil](/molmil-images/mine/2c86) | x-ray structure of the N and C-terminal domain of coronavirus nucleocapsid protein. | 分子名称: | NUCLEOCAPSID PROTEIN | 著者 | Jayaram, H, Fan, H, Bowman, B.R, Ooi, A, Jayaram, J, Collinson, E.W, Lescar, J, Prasad, B.V.V. | 登録日 | 2005-12-02 | 公開日 | 2006-06-21 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | X-Ray Structures of the N- and C-Terminal Domains of a Coronavirus Nucleocapsid Protein: Implications for Nucleocapsid Formation. J.Virol., 80, 2006
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2N34
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![BU of 2n34 by Molmil](/molmil-images/mine/2n34) | NMR assignments and solution structure of the JAK interaction region of SOCS5 | 分子名称: | Suppressor of cytokine signaling 5 | 著者 | Chandrashekaran, I.R, Mohanty, B, Linossi, E.M, Nicholson, S.E, Babon, J, Norton, R.S, Dagley, L.F, Leung, E.W.W, Murphy, J.M. | 登録日 | 2015-05-21 | 公開日 | 2015-07-29 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure and Functional Characterization of the Conserved JAK Interaction Region in the Intrinsically Disordered N-Terminus of SOCS5. Biochemistry, 54, 2015
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4BTX
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![BU of 4btx by Molmil](/molmil-images/mine/4btx) | Crystal structure of human vascular adhesion protein-1 in complex with pyridazinone inhibitors | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 5-isopropylamino-2-phenyl-6-(1H-1,2,4-triazol-5-yl)-3(2H)-pyridazinone, CALCIUM ION, ... | 著者 | Bligt-Linden, E, Pihlavisto, M, Szatmari, I, Otwinowski, Z, Smith, D.J, Lazar, L, Fulop, F, Salminen, T.A. | 登録日 | 2013-06-19 | 公開日 | 2013-12-18 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.78 Å) | 主引用文献 | Novel Pyridazinone Inhibitors for Vascular Adhesion Protein- 1 (Vap-1): Old Target - New Inhibition Mode. J.Med.Chem., 56, 2013
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4E4K
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![BU of 4e4k by Molmil](/molmil-images/mine/4e4k) | Crystal Structure of PPARgamma with the ligand JO21 | 分子名称: | (2S)-3-phenyl-2-{[2'-(propan-2-yl)biphenyl-4-yl]oxy}propanoic acid, Peroxisome proliferator-activated receptor gamma | 著者 | Pochetti, G, Montanari, R, Loiodice, F, Fracchiolla, G, Laghezza, A, Carbonara, G, Piemontese, L, Lavecchia, A, Novellino, E. | 登録日 | 2012-03-13 | 公開日 | 2013-01-23 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | New 2-(Aryloxy)-3-phenylpropanoic Acids as Peroxisome Proliferator-Activated Receptor alpha/gamma Dual Agonists Able To Upregulate Mitochondrial Carnitine Shuttle System Gene Expression. J.Med.Chem., 56, 2013
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4E4Q
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![BU of 4e4q by Molmil](/molmil-images/mine/4e4q) | Crystal structure of PPARgamma with the ligand FS214 | 分子名称: | (2R)-3-phenyl-2-{[2'-(propan-2-yl)biphenyl-4-yl]oxy}propanoic acid, Peroxisome proliferator-activated receptor gamma | 著者 | Pochetti, G, Montanari, R, Loiodice, F, Fracchiolla, G, Laghezza, A, Carbonara, G, Piemontese, L, Lavecchia, A, Novellino, E. | 登録日 | 2012-03-13 | 公開日 | 2013-01-23 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | New 2-(Aryloxy)-3-phenylpropanoic Acids as Peroxisome Proliferator-Activated Receptor alpha/gamma Dual Agonists Able To Upregulate Mitochondrial Carnitine Shuttle System Gene Expression. J.Med.Chem., 56, 2013
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2JCC
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![BU of 2jcc by Molmil](/molmil-images/mine/2jcc) | AH3 recognition of mutant HLA-A2 W167A | 分子名称: | BETA-2-MICROGLOBULIN, HLA CLASS I HISTOCOMPATIBILITY ANTIGEN, A-2 ALPHA CHAIN, ... | 著者 | Miller, P, Benhar, Y.P, Biddison, W, Collins, E.J. | 登録日 | 2006-12-21 | 公開日 | 2007-10-09 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Single Mhc Mutation Eliminates Enthalpy Associated with T Cell Receptor Binding. J.Mol.Biol., 373, 2007
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4BTY
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![BU of 4bty by Molmil](/molmil-images/mine/4bty) | Crystal structure of human vascular adhesion protein-1 in complex with pyridazinone inhibitors | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-[4-(4-methylpiperazin-1-yl)phenylamino]-2-(4-chlorophenyl)-6-(1H-1,2,4-triazol-5-yl)-3(2H)-pyridazinone, ... | 著者 | Bligt-Linden, E, Pihlavisto, M, Szatmari, I, Otwinowski, Z, Smith, D.J, Lazar, L, Fulop, F, Salminen, T.A. | 登録日 | 2013-06-19 | 公開日 | 2013-12-18 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Novel Pyridazinone Inhibitors for Vascular Adhesion Protein- 1 (Vap-1): Old Target - New Inhibition Mode. J.Med.Chem., 56, 2013
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2N7N
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![BU of 2n7n by Molmil](/molmil-images/mine/2n7n) | NMR structure of Peptide PG-989 in DPC micelles | 分子名称: | Peptide PG-989 | 著者 | Carotenuto, A, Merlino, F, Chai, M, Brancaccio, D, Yousif, A, Novellino, E, Hruby, V, Grieco, P. | 登録日 | 2015-09-16 | 公開日 | 2015-12-16 | 最終更新日 | 2017-10-11 | 実験手法 | SOLUTION NMR | 主引用文献 | Discovery of Novel Potent and Selective Agonists at the Melanocortin-3 Receptor. J.Med.Chem., 58, 2015
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2N7T
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![BU of 2n7t by Molmil](/molmil-images/mine/2n7t) | NMR structure of Peptide PG-992 in DPC micelles | 分子名称: | Peptide PG-992 | 著者 | Carotenuto, A, Merlino, F, Chai, M, Brancaccio, D, Yousif, A, Novellino, E, Hruby, V, Grieco, P. | 登録日 | 2015-09-17 | 公開日 | 2015-12-16 | 最終更新日 | 2017-10-11 | 実験手法 | SOLUTION NMR | 主引用文献 | Discovery of Novel Potent and Selective Agonists at the Melanocortin-3 Receptor. J.Med.Chem., 58, 2015
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7KEI
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![BU of 7kei by Molmil](/molmil-images/mine/7kei) | DQA1*01:02/DQB1*06:02 in complex with a hemagglutinin peptide from the H1N1 pandemic flu virus. | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, HA peptide from 2009 H1N1 pandemic flu virus., ... | 著者 | Birtley, J.R, Stern, L.J, Mellins, E.D, Jiang, W. | 登録日 | 2020-10-10 | 公開日 | 2021-10-13 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Crystal structure of DQA1*01:02/DQB1*06:02 in complex with a flu peptide. To Be Published
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2EWF
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![BU of 2ewf by Molmil](/molmil-images/mine/2ewf) | Crystal structure of the site-specific DNA nickase N.BspD6I | 分子名称: | BROMIDE ION, Nicking endonuclease N.BspD6I | 著者 | Kachalova, G.S, Bartunik, H.D, Artyukh, R.I, Rogulin, E.A, Perevyazova, T.A, Zheleznaya, L.A, Matvienko, N.I. | 登録日 | 2005-11-03 | 公開日 | 2006-11-21 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | Structural analysis of the heterodimeric type IIS restriction endonuclease R.BspD6I acting as a complex between a monomeric site-specific nickase and a catalytic subunit. J.Mol.Biol., 384, 2008
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2N7O
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![BU of 2n7o by Molmil](/molmil-images/mine/2n7o) | NMR Structure of Peptide PG-990 in DPC micelles | 分子名称: | Peptide PG-990 | 著者 | Carotenuto, A, Merlino, F, Chai, M, Brancaccio, D, Yousif, A, Novellino, E, Hruby, V, Grieco, P. | 登録日 | 2015-09-16 | 公開日 | 2015-12-16 | 最終更新日 | 2017-10-11 | 実験手法 | SOLUTION NMR | 主引用文献 | Discovery of Novel Potent and Selective Agonists at the Melanocortin-3 Receptor. J.Med.Chem., 58, 2015
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3RWM
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![BU of 3rwm by Molmil](/molmil-images/mine/3rwm) | Crystal Structure of Ypt32 in Complex with GppNHp | 分子名称: | GTP-binding protein YPT32/YPT11, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER | 著者 | Sultana, A, Dregger, C, Jin, Y, Franklin, E, Weisman, L.S, Khan, A.R. | 登録日 | 2011-05-09 | 公開日 | 2011-10-26 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The activation cycle of Rab GTPase Ypt32 reveals structural determinants of effector recruitment and GDI binding. Febs Lett., 585, 2011
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3RWO
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![BU of 3rwo by Molmil](/molmil-images/mine/3rwo) | Crystal structure of YPT32 in complex with GDP | 分子名称: | GTP-binding protein YPT32/YPT11, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION | 著者 | Sultana, A, Jin, Y, Dregger, C, Franklin, E, Weisman, L.S, Khan, A.R. | 登録日 | 2011-05-09 | 公開日 | 2011-10-26 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The activation cycle of Rab GTPase Ypt32 reveals structural determinants of effector recruitment and GDI binding. Febs Lett., 585, 2011
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3F5C
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![BU of 3f5c by Molmil](/molmil-images/mine/3f5c) | Structure of Dax-1:LRH-1 complex | 分子名称: | Nuclear receptor subfamily 0 group B member 1, Nuclear receptor subfamily 5 group A member 2 | 著者 | Fletterick, R.J, Sablin, E.P. | 登録日 | 2008-11-03 | 公開日 | 2008-12-23 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | The structure of corepressor Dax-1 bound to its target nuclear receptor LRH-1. Proc.Natl.Acad.Sci.USA, 105, 2008
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2KVY
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![BU of 2kvy by Molmil](/molmil-images/mine/2kvy) | NMR solution structure of the 4:1 complex between an uncharged distamycin A analogue and [d(TGGGGT)]4 | 分子名称: | 4-amino-1-methyl-N-{1-methyl-5-[(1-methyl-5-{[3-(methylamino)-3-oxopropyl]carbamoyl}-1H-pyrrol-3-yl)carbamoyl]-1H-pyrrol-3-yl}-1H-pyrrole-2-carboxamide, DNA (5'-D(*TP*GP*GP*GP*GP*T)-3') | 著者 | Cosconati, S, Marinelli, L, Trotta, R, Virno, A, De Tito, S, Romagnoli, R, Pagano, B, Limongelli, V, Giancola, C, Baraldi, P, Mayol, L, Novellino, E, Randazzo, A. | 登録日 | 2010-03-29 | 公開日 | 2010-05-26 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural and conformational requisites in DNA quadruplex groove binding: another piece to the puzzle. J.Am.Chem.Soc., 132, 2010
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3ZQT
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![BU of 3zqt by Molmil](/molmil-images/mine/3zqt) | TARGETING THE BINDING FUNCTION 3 SITE OF THE ANDROGEN RECEPTOR THROUGH IN SILICO MOLECULAR MODELING | 分子名称: | 4-[(2R,3S)-3-[(3,4-DIHYDROXYPHENYL)METHYL]-2-METHYLBUTYL]BENZENE-1,2-DIOL, ANDROGEN RECEPTOR, SULFATE ION, ... | 著者 | Lack, N.A, Axerio, P, Tavassoli, P, Kuchenbecker, K, Han, F.Q, Chan, K.H, Feau, C, LeBlanc, E, Tomlinson, E, Guy, R.K, Rennie, P.S, Cherkasov, A. | 登録日 | 2011-06-10 | 公開日 | 2011-12-07 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.29 Å) | 主引用文献 | Targeting the Binding Function 3 (Bf3) Site of the Human Androgen Receptor Through Virtual Screening. J.Med.Chem., 54, 2011
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1CMF
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![BU of 1cmf by Molmil](/molmil-images/mine/1cmf) | NMR SOLUTION STRUCTURE OF APO CALMODULIN CARBOXY-TERMINAL DOMAIN | 分子名称: | CALMODULIN (VERTEBRATE) | 著者 | Finn, B.E, Evenas, J, Drakenberg, T, Waltho, J.P, Thulin, E, Forsen, S. | 登録日 | 1995-07-19 | 公開日 | 1995-12-07 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Calcium-induced structural changes and domain autonomy in calmodulin. Nat.Struct.Biol., 2, 1995
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1CMG
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![BU of 1cmg by Molmil](/molmil-images/mine/1cmg) | NMR SOLUTION STRUCTURE OF CALCIUM-LOADED CALMODULIN CARBOXY-TERMINAL DOMAIN | 分子名称: | CALMODULIN (VERTEBRATE) | 著者 | Evenas, J, Finn, B.E, Drakenberg, T, Waltho, J.P, Thulin, E, Forsen, S. | 登録日 | 1995-07-19 | 公開日 | 1995-12-07 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Calcium-induced structural changes and domain autonomy in calmodulin. Nat.Struct.Biol., 2, 1995
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4KZC
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![BU of 4kzc by Molmil](/molmil-images/mine/4kzc) | Structure of PI3K gamma with Imidazopyridine inhibitors | 分子名称: | N-{6-[6-amino-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-2-yl}acetamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION | 著者 | Knapp, M.S, Elling, E.A. | 登録日 | 2013-05-29 | 公開日 | 2013-07-17 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | Structure guided optimization of a fragment hit to imidazopyridine inhibitors of PI3K. Bioorg.Med.Chem.Lett., 23, 2013
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2WBJ
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![BU of 2wbj by Molmil](/molmil-images/mine/2wbj) | TCR complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, HLA CLASS II HISTOCOMPATIBILITY ANTIGEN, DR ALPHA CHAIN, ... | 著者 | Harkiolaki, M, Holmes, S.L, Svendsen, P, Gregersen, J.W, Jensen, L.T, McMahon, R, Friese, M.A, van Boxel, G, Etzensperger, R, Tzartos, J.S, Kranc, K, Sainsbury, S, Harlos, K, Mellins, E.D, Palace, J, Esiri, M.M, van der Merwe, P.A, Jones, E.Y, Fugger, L. | 登録日 | 2009-03-02 | 公開日 | 2009-04-07 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | T Cell-Mediated Autoimmune Disease due to Low-Affinity Crossreactivity to Common Microbial Peptides. Immunity, 30, 2009
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2VRH
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![BU of 2vrh by Molmil](/molmil-images/mine/2vrh) | Structure of the E. coli trigger factor bound to a translating ribosome | 分子名称: | 50S RIBOSOMAL PROTEIN L23, 50S RIBOSOMAL PROTEIN L24, 50S RIBOSOMAL PROTEIN L29, ... | 著者 | Merz, F, Boehringer, D, Schaffitzel, C, Preissler, S, Hoffmann, A, Maier, T, Rutkowska, A, Lozza, J, Ban, N, Bukau, B, Deuerling, E. | 登録日 | 2008-04-07 | 公開日 | 2008-06-17 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (19 Å) | 主引用文献 | Molecular Mechanism and Structure of Trigger Factor Bound to the Translating Ribosome. Embo J., 27, 2008
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2P14
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![BU of 2p14 by Molmil](/molmil-images/mine/2p14) | Crystal structure of small subunit (R.BspD6I2) of the heterodimeric restriction endonuclease R.BspD6I | 分子名称: | GLYCEROL, Heterodimeric restriction endonuclease R.BspD6I small subunit, SULFATE ION | 著者 | Kachalova, G.S, Bartunik, H.D, Artyukh, R.I, Rogulin, E.A, Yunusova, A.K, Zheleznaya, L.A, Matvienko, N.I. | 登録日 | 2007-03-02 | 公開日 | 2008-03-11 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural analysis of the heterodimeric type IIS restriction endonuclease R.BspD6I acting as a complex between a monomeric site-specific nickase and a catalytic subunit. J.Mol.Biol., 384, 2008
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