1EJM
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![BU of 1ejm by Molmil](/molmil-images/mine/1ejm) | CRYSTAL STRUCTURE OF THE BPTI ALA16LEU MUTANT IN COMPLEX WITH BOVINE TRYPSIN | 分子名称: | BETA-TRYPSIN, PANCREATIC TRYPSIN INHIBITOR, SULFATE ION | 著者 | Otlewski, J, Smalas, A, Helland, R, Grzesiak, A, Krowarsch, D. | 登録日 | 2000-03-03 | 公開日 | 2001-03-03 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Substitutions at the P(1) position in BPTI strongly affect the association energy with serine proteinases. J.Mol.Biol., 301, 2000
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7Z13
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![BU of 7z13 by Molmil](/molmil-images/mine/7z13) | S. cerevisiae CMGE dimer nucleating origin DNA melting | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Cell division control protein 45, ... | 著者 | Lewis, J.S, Sousa, J.S, Costa, A. | 登録日 | 2022-02-24 | 公開日 | 2022-06-15 | 最終更新日 | 2024-07-17 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Mechanism of replication origin melting nucleated by CMG helicase assembly. Nature, 606, 2022
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8P1O
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![BU of 8p1o by Molmil](/molmil-images/mine/8p1o) | Solubilizer tag effect on PD-L1/inhibitor binding properties for m-terphenyl derivatives | 分子名称: | (3~{R})-1-[[4-[2-chloranyl-3-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]-2-methoxy-phenyl]methyl]-~{N}-(2-hydroxyethyl)pyrrolidine-3-carboxamide, CHLORIDE ION, Programmed cell death 1 ligand 1, ... | 著者 | Plewka, J, Magiera-Mularz, K, Surmiak, E, Kalinowska-Tluscik, J, Holak, T.A. | 登録日 | 2023-05-12 | 公開日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | Solubilizer Tag Effect on PD-L1/Inhibitor Binding Properties for m -Terphenyl Derivatives. Acs Med.Chem.Lett., 15, 2024
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7QHS
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![BU of 7qhs by Molmil](/molmil-images/mine/7qhs) | S. cerevisiae CMGE nucleating origin DNA melting | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Cell division control protein 45, ... | 著者 | Lewis, J.S, Sousa, J.S, Costa, A. | 登録日 | 2021-12-14 | 公開日 | 2022-06-15 | 最終更新日 | 2024-07-17 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Mechanism of replication origin melting nucleated by CMG helicase assembly. Nature, 606, 2022
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8P61
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![BU of 8p61 by Molmil](/molmil-images/mine/8p61) | Crystal structure of O'nyong'nyong virus capsid protease (106-256) | 分子名称: | Capsid protein, GLYCEROL, SULFATE ION | 著者 | Plewka, J, Chykunova, Y, Wilk, P, Sienczyk, M, Dubin, G, Pyrc, K. | 登録日 | 2023-05-24 | 公開日 | 2024-03-06 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Autoinhibition of suicidal capsid protease from O'nyong'nyong virus. Int.J.Biol.Macromol., 262, 2024
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8FEM
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![BU of 8fem by Molmil](/molmil-images/mine/8fem) | Panicum vigratum Dihydroflavonol 4-reductase complexed with NADP | 分子名称: | Dihydroflavonol 4-Reductase, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE | 著者 | Lewis, J.A, Kang, C. | 登録日 | 2022-12-06 | 公開日 | 2023-09-20 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.34 Å) | 主引用文献 | Structural Similarities and Overlapping Activities among Dihydroflavonol 4-Reductase, Flavanone 4-Reductase, and Anthocyanidin Reductase Offer Metabolic Flexibility in the Flavonoid Pathway. Int J Mol Sci, 24, 2023
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8FEN
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![BU of 8fen by Molmil](/molmil-images/mine/8fen) | Panicum vigratum Dihydroflavonol 4-reductase complexed with NADP and DHQ | 分子名称: | (2R,3R)-2-(3,4-DIHYDROXYPHENYL)-3,5,7-TRIHYDROXY-2,3-DIHYDRO-4H-CHROMEN-4-ONE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, Panicum virgatum Dihydroflavonol 4-Reductase | 著者 | Lewis, J.A, Kang, C. | 登録日 | 2022-12-06 | 公開日 | 2023-09-20 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Structural Similarities and Overlapping Activities among Dihydroflavonol 4-Reductase, Flavanone 4-Reductase, and Anthocyanidin Reductase Offer Metabolic Flexibility in the Flavonoid Pathway. Int J Mol Sci, 24, 2023
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5F5P
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![BU of 5f5p by Molmil](/molmil-images/mine/5f5p) | |
8R6Q
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![BU of 8r6q by Molmil](/molmil-images/mine/8r6q) | Co-crystal structure of PD-L1 with low molecular weight inhibitor | 分子名称: | (3~{R})-1-[[4-[2-chloranyl-3-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]-2-methoxy-phenyl]methyl]-~{N}-(2-hydroxyethyl)pyrrolidine-3-carboxamide, CHLORIDE ION, Programmed cell death 1 ligand 1, ... | 著者 | Plewka, J, Surmiak, E, Magiera-Mularz, K, Kalinowska-Tluscik, J. | 登録日 | 2023-11-22 | 公開日 | 2024-01-17 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | Solubilizer Tag Effect on PD-L1/Inhibitor Binding Properties for m -Terphenyl Derivatives. Acs Med.Chem.Lett., 15, 2024
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8V8P
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![BU of 8v8p by Molmil](/molmil-images/mine/8v8p) | Sorghum Chalcone Isomerase | 分子名称: | 7-HYDROXY-2-(4-HYDROXY-PHENYL)-CHROMAN-4-ONE, Chalcone-flavonone isomerase family protein | 著者 | Lewis, J.A, Kang, C. | 登録日 | 2023-12-05 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (3.18 Å) | 主引用文献 | Structural and Interactional Analysis of the Flavonoid Pathway Proteins: Chalcone Synthase, Chalcone Isomerase and Chalcone Isomerase-like Protein. Int J Mol Sci, 25, 2024
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8V8M
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![BU of 8v8m by Molmil](/molmil-images/mine/8v8m) | Switchgrass Chalcone Synthase | 分子名称: | COENZYME A, Chalcone synthase, NARINGENIN | 著者 | Lewis, J.A, Kang, C. | 登録日 | 2023-12-05 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | Structural and Interactional Analysis of the Flavonoid Pathway Proteins: Chalcone Synthase, Chalcone Isomerase and Chalcone Isomerase-like Protein. Int J Mol Sci, 25, 2024
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8TSI
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![BU of 8tsi by Molmil](/molmil-images/mine/8tsi) | |
8TSW
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![BU of 8tsw by Molmil](/molmil-images/mine/8tsw) | S. thermodepolymerans KpsMT-KpsE Apo 1 | 分子名称: | ABC transporter ATP-binding protein, Capsular biosynthesis protein, Transport permease protein | 著者 | Kuklewicz, J, Zimmer, J. | 登録日 | 2023-08-12 | 公開日 | 2024-04-17 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Molecular insights into capsular polysaccharide secretion. Nature, 628, 2024
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8TSL
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![BU of 8tsl by Molmil](/molmil-images/mine/8tsl) | |
8TT3
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![BU of 8tt3 by Molmil](/molmil-images/mine/8tt3) | S. thermodepolymerans KpsM-KpsE in Glycolipid 2 state with rigid body fitted KpsT | 分子名称: | (2R,5S,8S)-2,5-dihydroxy-5,10-dioxo-8-[(undecanoyloxy)methyl]-4,6,9-trioxa-5lambda~5~-phosphahenicosan-1-yl 3-deoxy-alpha-L-altro-oct-2-ulopyranosidonic acid, ABC transporter ATP-binding protein, Capsular biosynthesis protein, ... | 著者 | Kuklewicz, J, Zimmer, J. | 登録日 | 2023-08-12 | 公開日 | 2024-04-17 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Molecular insights into capsular polysaccharide secretion. Nature, 628, 2024
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8TSH
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![BU of 8tsh by Molmil](/molmil-images/mine/8tsh) | |
8TUN
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![BU of 8tun by Molmil](/molmil-images/mine/8tun) | S. thermodepolymerans KpsM-KpsE in Glycolipid 1 state with rigid body fitted KpsT | 分子名称: | (2R,5S,8S)-2,5-dihydroxy-5,10-dioxo-8-[(undecanoyloxy)methyl]-4,6,9-trioxa-5lambda~5~-phosphahenicosan-1-yl 3-deoxy-alpha-L-altro-oct-2-ulopyranosidonic acid, ABC transporter ATP-binding protein, Capsular biosynthesis protein, ... | 著者 | Kuklewicz, J, Zimmer, J. | 登録日 | 2023-08-16 | 公開日 | 2024-04-17 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Molecular insights into capsular polysaccharide secretion. Nature, 628, 2024
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9EO0
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![BU of 9eo0 by Molmil](/molmil-images/mine/9eo0) | Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 | 分子名称: | Programmed cell death 1 ligand 1, SULFATE ION, ~{N}-[3-[3-[[5-[(2-hydroxyethylamino)methyl]pyridin-2-yl]carbonylamino]-2-methyl-phenyl]-2-methyl-phenyl]-5-[[3-(methylsulfonylamino)propylamino]methyl]pyridine-2-carboxamide | 著者 | Plewka, J, Hec, A, Sitar, T, Holak, T. | 登録日 | 2024-03-14 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Nonsymmetrically Substituted 1,1'-Biphenyl-Based Small Molecule Inhibitors of the PD-1/PD-L1 Interaction. Acs Med.Chem.Lett., 15, 2024
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8V8L
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![BU of 8v8l by Molmil](/molmil-images/mine/8v8l) | Switchgrass Chalcone Isomerase | 分子名称: | Chalcone-flavonone isomerase family protein, GLYCEROL | 著者 | Lewis, J.A, Kang, C. | 登録日 | 2023-12-05 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Structural and Interactional Analysis of the Flavonoid Pathway Proteins: Chalcone Synthase, Chalcone Isomerase and Chalcone Isomerase-like Protein. Int J Mol Sci, 25, 2024
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8V8N
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![BU of 8v8n by Molmil](/molmil-images/mine/8v8n) | Switchgrass Chalcone Synthase C170S | 分子名称: | Chalcone synthase, GLYCEROL | 著者 | Lewis, J.A, Kang, C. | 登録日 | 2023-12-05 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (2.12 Å) | 主引用文献 | Structural and Interactional Analysis of the Flavonoid Pathway Proteins: Chalcone Synthase, Chalcone Isomerase and Chalcone Isomerase-like Protein. Int J Mol Sci, 25, 2024
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8V8O
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![BU of 8v8o by Molmil](/molmil-images/mine/8v8o) | Switchgrass Chalcone Isomerase-Like Protein | 分子名称: | Chalcone-flavonone isomerase family protein | 著者 | Lewis, J.A, Kang, C. | 登録日 | 2023-12-05 | 公開日 | 2024-05-29 | 最終更新日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (3.21 Å) | 主引用文献 | Structural and Interactional Analysis of the Flavonoid Pathway Proteins: Chalcone Synthase, Chalcone Isomerase and Chalcone Isomerase-like Protein. Int J Mol Sci, 25, 2024
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9EPL
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![BU of 9epl by Molmil](/molmil-images/mine/9epl) | Mpro from SARS-CoV-2 with 298Q mutation | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, Non-structural protein 11, ... | 著者 | Plewka, J, Lis, K, Czarna, A, Pyrc, K, Kantyka, T, Chykunova, Y. | 登録日 | 2024-03-18 | 公開日 | 2024-04-17 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | SARS-CoV-2 M pro oligomerization as a potential target for therapy. Int.J.Biol.Macromol., 267, 2024
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9EPM
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![BU of 9epm by Molmil](/molmil-images/mine/9epm) | Mpro from SARS-CoV-2 with 4A mutation | 分子名称: | Non-structural protein 11 | 著者 | Plewka, J, Lis, K, Czarna, A, Pyrc, K, Kantyka, T, Chykunova, Y. | 登録日 | 2024-03-19 | 公開日 | 2024-04-17 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.981 Å) | 主引用文献 | SARS-CoV-2 M pro oligomerization as a potential target for therapy. Int.J.Biol.Macromol., 267, 2024
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9EWM
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![BU of 9ewm by Molmil](/molmil-images/mine/9ewm) | Mpro from SARS-CoV-2 with R4Q R298Q double mutations | 分子名称: | Non-structural protein 11 | 著者 | Plewka, J, Lis, K, Chykunova, Y, Czarna, A, Kantyka, T, Pyrc, K. | 登録日 | 2024-04-04 | 公開日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (2.63 Å) | 主引用文献 | SARS-CoV-2 M pro oligomerization as a potential target for therapy. Int.J.Biol.Macromol., 267, 2024
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9EUS
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![BU of 9eus by Molmil](/molmil-images/mine/9eus) | Mpro from SARS-CoV-2 with R298A mutation | 分子名称: | GLYCEROL, Replicase polyprotein 1a | 著者 | Plewka, J, Lis, K, Czarna, A, Pyrc, K, Kantyka, T, Chykunova, Y. | 登録日 | 2024-03-28 | 公開日 | 2024-04-17 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | SARS-CoV-2 M pro oligomerization as a potential target for therapy. Int.J.Biol.Macromol., 267, 2024
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