1CL7
| ANTI HIV1 PROTEASE FAB | 分子名称: | PROTEIN (IGG1 ANTIBODY 1696 (constant heavy chain)), PROTEIN (IGG1 ANTIBODY 1696 (light chain)), PROTEIN (IGG1 ANTIBODY 1696 (variable heavy chain)) | 著者 | Lescar, J, Bentley, G.A. | 登録日 | 1999-05-06 | 公開日 | 2000-01-12 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Inhibition of the HIV-1 and HIV-2 proteases by a monoclonal antibody. Protein Sci., 8, 1999
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5JJR
| Dengue 3 NS5 protein with compound 29 | 分子名称: | 1,2-ETHANEDIOL, 5-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-4-methoxy-2-methyl-N-[(quinolin-8-yl)sulfonyl]benzamide, DI(HYDROXYETHYL)ETHER, ... | 著者 | Lescar, J, El Sahili, A. | 登録日 | 2016-04-25 | 公開日 | 2016-07-06 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.99 Å) | 主引用文献 | Potent Allosteric Dengue Virus NS5 Polymerase Inhibitors: Mechanism of Action and Resistance Profiling Plos Pathog., 12, 2016
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5JJS
| Dengue 3 NS5 protein with compound 27 | 分子名称: | 1,2-ETHANEDIOL, 5-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-2,4-dimethoxy-N-{[(1R,3R)-3-methoxycyclohexyl]sulfonyl}benzamide, DI(HYDROXYETHYL)ETHER, ... | 著者 | Lescar, J, El Sahili, A. | 登録日 | 2016-04-25 | 公開日 | 2016-07-06 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Potent Allosteric Dengue Virus NS5 Polymerase Inhibitors: Mechanism of Action and Resistance Profiling Plos Pathog., 12, 2016
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1FBI
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1GNZ
| LECTIN I-B4 FROM GRIFFONIA SIMPLICIFOLIA (GS I-B4)METAL FREE FORM | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, GSI-B4 ISOLECTIN, PHOSPHATE ION | 著者 | Lescar, J, Loris, R, Mitchell, E, Gautier, C, Imberty, A. | 登録日 | 2001-10-11 | 公開日 | 2001-11-29 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Isolectins I-A and I-B of Griffonia (Bandeiraea) Simplicifolia. Crystal Structure of Metal-Free Gs I-B(4) and Molecular Basis for Metal Binding and Monosaccharide Specificity. J.Biol.Chem., 277, 2002
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1MF2
| ANTI HIV1 PROTEASE FAB COMPLEX | 分子名称: | MONOCLONAL ANTIBODY F11.2.32 | 著者 | Lescar, J, Bentley, G.A. | 登録日 | 1996-12-27 | 公開日 | 1997-12-31 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Three-dimensional structure of an Fab-peptide complex: structural basis of HIV-1 protease inhibition by a monoclonal antibody. J.Mol.Biol., 267, 1997
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1I9W
| CRYSTAL STRUCTURE OF THE FUSION GLYCOPROTEIN E1 FROM SEMLIKI FOREST VIRUS | 分子名称: | FUSION PROTEIN E1 | 著者 | Lescar, J, Roussel, A, Wien, M.W, Navaza, J, Fuller, S.D, Wengler, G, Wengler, G, Rey, F.A. | 登録日 | 2001-03-21 | 公開日 | 2002-04-06 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | The Fusion glycoprotein shell of Semliki Forest virus: an icosahedral assembly primed for fusogenic activation at endosomal pH. Cell(Cambridge,Mass.), 105, 2001
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6ID4
| Defining the structural basis for human alloantibody binding to human leukocyte antigen allele HLA-A*11:01 | 分子名称: | Beta-2-microglobulin, DI(HYDROXYETHYL)ETHER, GLYCEROL, ... | 著者 | Lescar, J, Wong, Y.H, Liew, C.W, Gu, Y, MacAry, P.A. | 登録日 | 2018-09-08 | 公開日 | 2019-02-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Defining the structural basis for human alloantibody binding to human leukocyte antigen allele HLA-A*11:01. Nat Commun, 10, 2019
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1N4X
| Structure of scFv 1696 at acidic pH | 分子名称: | CHLORIDE ION, immunoglobulin heavy chain variable region, immunoglobulin kappa chain variable region | 著者 | Lescar, J, Brynda, J, Fabry, M, Horejsi, M, Rezacova, P, Sedlacek, J, Bentley, G.A. | 登録日 | 2002-11-02 | 公開日 | 2003-06-10 | 最終更新日 | 2022-12-21 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structure of a single-chain Fv fragment of an antibody that inhibits the HIV-1 and HIV-2 proteases. Acta Crystallogr.,Sect.D, 59, 2003
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2HRP
| ANTIGEN-ANTIBODY COMPLEX | 分子名称: | HIV-1 PROTEASE PEPTIDE, MONOCLONAL ANTIBODY F11.2.32 | 著者 | Lescar, J, Bentley, G.A. | 登録日 | 1996-12-27 | 公開日 | 1997-12-31 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Three-dimensional structure of an Fab-peptide complex: structural basis of HIV-1 protease inhibition by a monoclonal antibody. J.Mol.Biol., 267, 1997
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8HO4
| Falcilysin in complex with MMV000848 | 分子名称: | (2R)-1-(9H-carbazol-9-yl)-3-(cyclopentylamino)propan-2-ol, 1,2-ETHANEDIOL, Falcilysin, ... | 著者 | Lin, J.Q, Chung, Z, Lescar, J. | 登録日 | 2022-12-09 | 公開日 | 2023-12-20 | 最終更新日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development. Cell Chem Biol, 31, 2024
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8HO5
| Falcilysin in complex with MMV665806 | 分子名称: | (2S)-1-(2,3-dimethyl-1H-indol-1-yl)-3-{[(1S,2S)-2-methylcyclohexyl]amino}propan-2-ol, 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, ... | 著者 | Lin, J.Q, Chung, Z, Lescar, J. | 登録日 | 2022-12-09 | 公開日 | 2023-12-20 | 最終更新日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (2.003 Å) | 主引用文献 | Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development. Cell Chem Biol, 31, 2024
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2C3S
| Structure Of Sars Cov Main Proteinase At 1.9 A (Ph6.5) | 分子名称: | SARS COV 3C-LIKE PROTEINASE | 著者 | Xu, T, Ooi, A, Lee, H.-C, Lescar, J. | 登録日 | 2005-10-12 | 公開日 | 2005-10-18 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure of the Sars Coronavirus Main Proteinase as an Active C2 Crystallographic Dimer. Acta Crystallogr.,Sect.F, 61, 2005
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4C11
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4S2Q
| Crystal Structure of HMG domain of the chondrogenesis master regulator, Sox9 in complex with ChIP-Seq identified DNA element | 分子名称: | DNA (5'-D(P*AP*GP*GP*AP*GP*AP*AP*CP*AP*AP*AP*GP*CP*CP*TP*G)-3'), DNA (5'-D(P*AP*GP*GP*CP*TP*TP*TP*GP*TP*TP*CP*TP*CP*CP*TP*G)-3'), Transcription factor SOX-9 | 著者 | Vivekanandan, S, Moovarkumudalvan, B, Lescar, J, Kolatkar, P.R. | 登録日 | 2015-01-21 | 公開日 | 2016-02-17 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal Structure of HMG domain of the chondrogenesis master regulator, Sox9 in complex with ChIP-Seq identified DNA element To be Published
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6AFK
| Crystal structure of TrmD from Pseudomonas aeruginosa in complex with active-site inhibitor | 分子名称: | N-{(3S)-1-[3-(pyridin-4-yl)-1H-pyrazol-5-yl]piperidin-3-yl}-1H-indole-2-carboxamide, S-ADENOSYLMETHIONINE, tRNA (guanine-N(1)-)-methyltransferase | 著者 | Zhong, W, Koay, A, Wong, Y.W, Sahili, A.E, Nah, Q, Kang, C, Poulsen, A, Chionh, Y.K, McBee, M, Matter, A, Hill, J, Lescar, J, Dedon, P.C. | 登録日 | 2018-08-08 | 公開日 | 2019-08-14 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Targeting the Bacterial Epitranscriptome for Antibiotic Development: Discovery of Novel tRNA-(N1G37) Methyltransferase (TrmD) Inhibitors. Acs Infect Dis., 5, 2019
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4BFH
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2BXX
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8W7H
| Purine Nucleoside Phosphorylase in complex with MMV000848 | 分子名称: | (2R)-1-(9H-carbazol-9-yl)-3-(cyclopentylamino)propan-2-ol, 1,2-ETHANEDIOL, PHOSPHATE ION, ... | 著者 | Chung, Z, Lin, J.Q, Lescar, J. | 登録日 | 2023-08-30 | 公開日 | 2024-01-17 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Identification and structural validation of purine nucleoside phosphorylase from Plasmodium falciparum as a target of MMV000848. J.Biol.Chem., 300, 2023
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6JKI
| Crystal structure and catalytic mechanism of the essential m1G37 tRNA methyltransferase TrmD from Pseudomonas aeruginosa | 分子名称: | DI(HYDROXYETHYL)ETHER, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Jaroensuk, J, Liew, C.W, Atichartpongkul, S, Chionh, Y.H, Wong, Y.H, Zhong, W.H, McBee, M.E, Thongdee, N, Prestwich, E.G, DeMott, M.S, Mongkolsuk, S, Dedon, P.C, Lescar, J, Fuangthong, M. | 登録日 | 2019-03-01 | 公開日 | 2019-07-03 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.59 Å) | 主引用文献 | Crystal structure and catalytic mechanism of the essential m1G37 tRNA methyltransferase TrmD fromPseudomonas aeruginosa. Rna, 25, 2019
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5ZQK
| Dengue Virus Non Structural Protein 5 | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, MAGNESIUM ION, ... | 著者 | El Sahili, A, Soh, T.S, Schiltz, J, Gharbi-Ayachi, A, Goh, B.C, Seh, C.C, Dedon, P.C, Shi, P.Y, Lim, S.P, Lescar, J. | 登録日 | 2018-04-19 | 公開日 | 2019-06-12 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | NS5 from Dengue Virus Serotype 2 Can Adopt a Conformation Analogous to That of Its Zika Virus and Japanese Encephalitis Virus Homologues. J.Virol., 94, 2019
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6K4E
| SiaA-PP2C domain of Pseudomonas aeruginosa | 分子名称: | MAGNESIUM ION, Putative serine phosphatase | 著者 | Lin, J.Q, Lescar, J. | 登録日 | 2019-05-23 | 公開日 | 2019-06-26 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.094 Å) | 主引用文献 | The SiaABC threonine phosphorylation pathway controls biofilm formation in response to carbon availability in Pseudomonas aeruginosa. Plos One, 15, 2020
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2BHR
| Dengue virus RNA helicase | 分子名称: | RNA HELICASE, SULFATE ION | 著者 | Xu, T, Sampath, A, Chao, A, Wen, D, Nanao, M, Chene, P, Vasudevan, S.G, Lescar, J. | 登録日 | 2005-01-17 | 公開日 | 2005-08-03 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structure of the Dengue Virus Helicase/Nucleoside Triphosphatase Catalytic Domain at a Resolution of 2.4 A. J.Virol., 79, 2005
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2BMF
| Dengue virus RNA helicase at 2.4A | 分子名称: | RNA HELICASE | 著者 | Xu, T, Sampath, A, Chao, A, Wen, D, Nanao, M, Chene, P, Vasudevan, S.G, Lescar, J. | 登録日 | 2005-03-14 | 公開日 | 2005-08-03 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Structure of the Dengue Virus Helicase/Nucleoside Triphosphatase Catalytic Domain at a Resolution of 2.4 A. J.Virol., 79, 2005
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6U5O
| Structure of the Human Metapneumovirus Polymerase bound to the phosphoprotein tetramer | 分子名称: | Phosphoprotein, RNA-directed RNA polymerase L | 著者 | Pan, J, Qian, X, Lattmann, S, Sahili, A.E, Yeo, T.H, Kalocsay, M, Fearns, R, Lescar, J. | 登録日 | 2019-08-28 | 公開日 | 2019-09-25 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Structure of the human metapneumovirus polymerase phosphoprotein complex. Nature, 577, 2020
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