2XU6
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![BU of 2xu6 by Molmil](/molmil-images/mine/2xu6) | MDV1 coiled coil domain | 分子名称: | MDV1 COILED COIL | 著者 | Koirala, S, Bui, H.T, Schubert, H.L, Eckert, D.M, Hill, C.P, Kay, M.S, Shaw, J.M. | 登録日 | 2010-10-14 | 公開日 | 2010-10-27 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Molecular Architecture of a Dynamin Adaptor: Implications for Assembly of Mitochondrial Fission Complexes J.Cell Biol., 191, 2010
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3MGN
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![BU of 3mgn by Molmil](/molmil-images/mine/3mgn) | D-Peptide inhibitor PIE71 in complex with IQN17 | 分子名称: | D-PEPTIDE INHIBITOR PIE71, IQN17 | 著者 | Hill, C.P, Whitby, F.G, Kay, M, Francis, N. | 登録日 | 2010-04-07 | 公開日 | 2011-03-02 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Design of a potent D-peptide HIV-1 entry inhibitor with a strong barrier to resistance. J.Virol., 84, 2010
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3L37
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![BU of 3l37 by Molmil](/molmil-images/mine/3l37) | PIE12 D-peptide against HIV entry | 分子名称: | GP41 N-PEPTIDE, HIV ENTRY INHIBITOR PIE12 | 著者 | Welch, B.D, Redman, J.S, Paul, S, Whitby, F.G, Weinstock, M.T, Reeves, J.D, Lie, Y.S, Eckert, D.M, Hill, C.P, Root, M.J, Kay, M.S. | 登録日 | 2009-12-16 | 公開日 | 2010-11-03 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Design of a potent D-peptide HIV-1 entry inhibitor with a strong barrier to resistance. J.Virol., 84, 2010
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3L35
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![BU of 3l35 by Molmil](/molmil-images/mine/3l35) | PIE12 D-peptide against HIV entry | 分子名称: | GP41 N-PEPTIDE, HIV ENTRY INHIBITOR PIE12 | 著者 | Welch, B.D, Redman, J.S, Paul, S, Whitby, F.G, Weinstock, M.T, Reeves, J.D, Lie, Y.S, Eckert, D.M, Hill, C.P, Root, M.J, Kay, M.S. | 登録日 | 2009-12-16 | 公開日 | 2010-11-03 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Design of a potent D-peptide HIV-1 entry inhibitor with a strong barrier to resistance. J.Virol., 84, 2010
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3L36
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![BU of 3l36 by Molmil](/molmil-images/mine/3l36) | PIE12 D-peptide against HIV entry | 分子名称: | 3-CYCLOHEXYL-1-PROPYLSULFONIC ACID, GP41 N-PEPTIDE, HIV ENTRY INHIBITOR PIE12 | 著者 | Welch, B.D, Redman, J.S, Paul, S, Whitby, F.G, Weinstock, M.T, Reeves, J.D, Lie, Y.S, Eckert, D.M, Hill, C.P, Root, M.J, Kay, M.S. | 登録日 | 2009-12-16 | 公開日 | 2010-11-03 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Design of a potent D-peptide HIV-1 entry inhibitor with a strong barrier to resistance. J.Virol., 84, 2010
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6OO2
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![BU of 6oo2 by Molmil](/molmil-images/mine/6oo2) | Vps4 with Cyclic Peptide Bound in the Central Pore | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, Designed Cyclic Peptide, ... | 著者 | Han, H, Fulcher, J.M, Dandey, V.P, Sundquist, W.I, Kay, M.S, Shen, P, Hill, C.P. | 登録日 | 2019-04-22 | 公開日 | 2019-08-21 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.4 Å) | 主引用文献 | Structure of Vps4 with circular peptides and implications for translocation of two polypeptide chains by AAA+ ATPases. Elife, 8, 2019
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6NDY
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![BU of 6ndy by Molmil](/molmil-images/mine/6ndy) | Vps4 with Cyclic Peptide Bound in the Central Pore | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, Designed Cyclic Peptide, ... | 著者 | Han, H, Fulcher, J.M, Dandey, V.P, Sundquist, W.I, Kay, M.S, Shen, P, Hill, C.P. | 登録日 | 2018-12-14 | 公開日 | 2019-08-21 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Structure of Vps4 with circular peptides and implications for translocation of two polypeptide chains by AAA+ ATPases. Elife, 8, 2019
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2R3C
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![BU of 2r3c by Molmil](/molmil-images/mine/2r3c) | Structure of the gp41 N-peptide in complex with the HIV entry inhibitor PIE1 | 分子名称: | CHLORIDE ION, HIV entry inhibitor PIE1, YTTRIUM (III) ION, ... | 著者 | VanDemark, A.P, Welch, B, Heroux, A, Hill, C.P, Kay, M.S. | 登録日 | 2007-08-29 | 公開日 | 2007-10-02 | 最終更新日 | 2018-08-08 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Potent D-peptide inhibitors of HIV-1 entry Proc.Natl.Acad.Sci.Usa, 104, 2007
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2R5B
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![BU of 2r5b by Molmil](/molmil-images/mine/2r5b) | Structure of the gp41 N-trimer in complex with the HIV entry inhibitor PIE7 | 分子名称: | HIV entry inhibitor PIE7, SULFATE ION, gp41 N-peptide | 著者 | VanDemark, A.P, Welch, B, Heroux, A, Hill, C.P, Kay, M.S. | 登録日 | 2007-09-03 | 公開日 | 2007-10-02 | 最終更新日 | 2017-10-25 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Potent D-peptide inhibitors of HIV-1 entry Proc.Natl.Acad.Sci.Usa, 104, 2007
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2R5D
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![BU of 2r5d by Molmil](/molmil-images/mine/2r5d) | Structure of the gp41 N-trimer in complex with the HIV entry inhibitor PIE7 | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, HIV entry inhibitor PIE7, ... | 著者 | VanDemark, A.P, Welch, B, Heroux, A, Hill, C.P, Kay, M.S. | 登録日 | 2007-09-03 | 公開日 | 2007-10-02 | 最終更新日 | 2017-10-25 | 実験手法 | X-RAY DIFFRACTION (1.66 Å) | 主引用文献 | Potent D-peptide inhibitors of HIV-1 entry Proc.Natl.Acad.Sci.Usa, 104, 2007
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4R0R
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![BU of 4r0r by Molmil](/molmil-images/mine/4r0r) | Ebolavirus GP Prehairpin Intermediate Mimic | 分子名称: | eboIZN21 | 著者 | Clinton, T.R, Weinstock, M.T, Jacobsen, M.T, Szabo-Fresnais, N, Pandya, M.J, Whitby, F.G, Herbert, A.S, Prugar, L.I, McKinnon, R, Hill, C.P, Welch, B.D, Dye, J.M, Eckert, D.M, Kay, M.S. | 登録日 | 2014-08-01 | 公開日 | 2014-10-22 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Design and characterization of ebolavirus GP prehairpin intermediate mimics as drug targets. Protein Sci., 24, 2015
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4V4Q
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![BU of 4v4q by Molmil](/molmil-images/mine/4v4q) | Crystal structure of the bacterial ribosome from Escherichia coli at 3.5 A resolution. | 分子名称: | 16S ribosomal RNA, 23S ribosomal RNA, 30S ribosomal protein S10, ... | 著者 | Schuwirth, B.S, Borovinskaya, M.A, Hau, C.W, Zhang, W, Vila-Sanjurjo, A, Holton, J.M, Cate, J.H.D. | 登録日 | 2005-08-30 | 公開日 | 2014-07-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.46 Å) | 主引用文献 | Structures of the bacterial ribosome at 3.5 A resolution. Science, 310, 2005
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5KBV
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![BU of 5kbv by Molmil](/molmil-images/mine/5kbv) | Cryo-EM structure of GluA2 bound to antagonist ZK200775 at 6.8 Angstrom resolution | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor 2, {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid | 著者 | Twomey, E.C, Yelshanskaya, M.V, Grassucci, R.G, Frank, J, Sobolevsky, A.I. | 登録日 | 2016-06-03 | 公開日 | 2016-07-13 | 最終更新日 | 2020-07-29 | 実験手法 | ELECTRON MICROSCOPY (6.8 Å) | 主引用文献 | Elucidation of AMPA receptor-stargazin complexes by cryo-electron microscopy. Science, 353, 2016
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5KBU
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![BU of 5kbu by Molmil](/molmil-images/mine/5kbu) | Cryo-EM structure of GluA2-2xSTZ complex at 7.8 Angstrom resolution | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor 2,Voltage-dependent calcium channel gamma-2 subunit, {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid | 著者 | Twomey, E.C, Yelshanskaya, M.V, Grassucci, R.A, Frank, J, Sobolevsky, A.I. | 登録日 | 2016-06-03 | 公開日 | 2016-07-13 | 最終更新日 | 2020-07-29 | 実験手法 | ELECTRON MICROSCOPY (7.8 Å) | 主引用文献 | Elucidation of AMPA receptor-stargazin complexes by cryo-electron microscopy. Science, 353, 2016
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5KBT
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![BU of 5kbt by Molmil](/molmil-images/mine/5kbt) | Cryo-EM structure of GluA2-1xSTZ complex at 6.4 Angstrom resolution | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor 2,Voltage-dependent calcium channel gamma-2 subunit, {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid | 著者 | Twomey, E.C, Yelshanskaya, M.V, Grassucci, R.A, Frank, J, Sobolevsky, A.I. | 登録日 | 2016-06-03 | 公開日 | 2016-07-13 | 最終更新日 | 2020-07-29 | 実験手法 | ELECTRON MICROSCOPY (6.4 Å) | 主引用文献 | Elucidation of AMPA receptor-stargazin complexes by cryo-electron microscopy. Science, 353, 2016
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6F0D
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![BU of 6f0d by Molmil](/molmil-images/mine/6f0d) | Crystal structure of a llama VHH antibody BCD090-M2 against human ErbB3 in space group P1 with cadmium ions | 分子名称: | CADMIUM ION, VHH antibody BCD090-M2 | 著者 | Eliseev, I.E, Yudenko, A.N, Vysochinskaya, V.V, Svirina, A.A, Evstratyeva, A.V, Drozhzhachih, M.S, Krendeleva, E.A, Vladimirova, A.K, Nemankin, T.A, Ekimova, V.M, Ulitin, A.B, Lomovskaya, M.I, Yakovlev, P.A, Moiseenko, F.V, Chakchir, O.B. | 登録日 | 2017-11-19 | 公開日 | 2017-11-29 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.90000749 Å) | 主引用文献 | Crystal structures of a llama VHH antibody BCD090-M2 targeting human ErbB3 receptor. F1000Res, 7, 2018
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6EZW
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![BU of 6ezw by Molmil](/molmil-images/mine/6ezw) | Crystal structure of a llama VHH antibody BCD090-M2 against human ErbB3 in space group C2 | 分子名称: | VHH antibody BCD090-M2 | 著者 | Eliseev, I.E, Yudenko, A.N, Vysochinskaya, V.V, Svirina, A.A, Evstratyeva, A.V, Drozhzhachih, M.S, Krendeleva, E.A, Vladimirova, A.K, Nemankin, T.A, Ekimova, V.M, Ulitin, A.B, Lomovskaya, M.I, Yakovlev, P.A, Moiseenko, F.V, Chakchir, O.B. | 登録日 | 2017-11-16 | 公開日 | 2017-11-29 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.59842849 Å) | 主引用文献 | Crystal structures of a llama VHH antibody BCD090-M2 targeting human ErbB3 receptor. F1000Res, 7, 2018
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8FOA
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![BU of 8foa by Molmil](/molmil-images/mine/8foa) | Cryo-EM structure of human TRPV6 in complex with the natural phytoestrogen genistein | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, CALCIUM ION, CHOLESTEROL HEMISUCCINATE, ... | 著者 | Neuberger, A, Yelshanskaya, M.V, Nadezhdin, K.D, Sobolevsky, A.I. | 登録日 | 2022-12-30 | 公開日 | 2023-05-24 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.66 Å) | 主引用文献 | Structural mechanism of human oncochannel TRPV6 inhibition by the natural phytoestrogen genistein. Nat Commun, 14, 2023
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8FOB
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![BU of 8fob by Molmil](/molmil-images/mine/8fob) | Cryo-EM structure of human TRPV6 in the open state | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, ... | 著者 | Neuberger, A, Yelshanskaya, M.V, Nadezhdin, K.D, Sobolevsky, A.I. | 登録日 | 2022-12-30 | 公開日 | 2023-05-24 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.71 Å) | 主引用文献 | Structural mechanism of human oncochannel TRPV6 inhibition by the natural phytoestrogen genistein. Nat Commun, 14, 2023
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7K3G
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![BU of 7k3g by Molmil](/molmil-images/mine/7k3g) | SARS-CoV-2 Envelope Protein Transmembrane Domain: Pentameric Structure Determined by Solid-State NMR | 分子名称: | Envelope small membrane protein | 著者 | Mandala, V.S, Hong, M, McKay, M.J, Shcherbakov, A.S, Dregni, A.J. | 登録日 | 2020-09-11 | 公開日 | 2020-09-30 | 最終更新日 | 2024-05-15 | 実験手法 | SOLID-STATE NMR | 主引用文献 | Structure and drug binding of the SARS-CoV-2 envelope protein transmembrane domain in lipid bilayers. Nat.Struct.Mol.Biol., 27, 2020
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6O9G
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![BU of 6o9g by Molmil](/molmil-images/mine/6o9g) | Open state GluA2 in complex with STZ and blocked by AgTx-636, after micelle signal subtraction | 分子名称: | CYCLOTHIAZIDE, GLUTAMIC ACID, Glutamate receptor 2,Voltage-dependent calcium channel gamma-2 subunit, ... | 著者 | Twomey, E.C, Yelshanskaya, M.V, Vassilevski, A.A, Sobolevsky, A.I. | 登録日 | 2019-03-13 | 公開日 | 2019-03-20 | 最終更新日 | 2019-12-18 | 実験手法 | ELECTRON MICROSCOPY (4.8 Å) | 主引用文献 | Mechanisms of Channel Block in Calcium-Permeable AMPA Receptors. Neuron, 99, 2018
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7D9X
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![BU of 7d9x by Molmil](/molmil-images/mine/7d9x) | Highly active mutant W525D of Gamma-glutamyltranspeptidase from Pseudomonas nitroreducens | 分子名称: | GAMMA-BUTYROLACTONE, GLYCEROL, GLYCINE, ... | 著者 | Hibi, T, Sano, C, Itoh, T, Wakayama, M. | 登録日 | 2020-10-14 | 公開日 | 2021-06-23 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Mutagenesis and structure-based analysis of the role of Tryptophan525 of gamma-glutamyltranspeptidase from Pseudomonas nitroreducens. Biochem.Biophys.Res.Commun., 534, 2021
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6DM0
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![BU of 6dm0 by Molmil](/molmil-images/mine/6dm0) | Open state GluA2 in complex with STZ and blocked by IEM-1460, after micelle signal subtraction | 分子名称: | CYCLOTHIAZIDE, GLUTAMIC ACID, Glutamate receptor 2,Voltage-dependent calcium channel gamma-2 subunit, ... | 著者 | Twomey, E.C, Yelshanskaya, M.V, Vassilevski, A.A, Sobolevsky, A.I. | 登録日 | 2018-06-04 | 公開日 | 2018-08-22 | 最終更新日 | 2019-12-18 | 実験手法 | ELECTRON MICROSCOPY (4.4 Å) | 主引用文献 | Mechanisms of Channel Block in Calcium-Permeable AMPA Receptors. Neuron, 99, 2018
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6DM1
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![BU of 6dm1 by Molmil](/molmil-images/mine/6dm1) | Open state GluA2 in complex with STZ and blocked by NASPM, after micelle signal subtraction | 分子名称: | CYCLOTHIAZIDE, GLUTAMIC ACID, Glutamate receptor 2,Voltage-dependent calcium channel gamma-2 subunit, ... | 著者 | Twomey, E.C, Yelshanskaya, M.V, Vassilevski, A.A, Sobolevsky, A.I. | 登録日 | 2018-06-04 | 公開日 | 2018-08-22 | 最終更新日 | 2019-12-18 | 実験手法 | ELECTRON MICROSCOPY (4.2 Å) | 主引用文献 | Mechanisms of Channel Block in Calcium-Permeable AMPA Receptors. Neuron, 99, 2018
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5ZJG
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![BU of 5zjg by Molmil](/molmil-images/mine/5zjg) | Gamma-glutamyltranspeptidase from Pseudomonas nitroreducens complexed with Gly-Gly | 分子名称: | GLYCEROL, GLYCINE, Gamma-glutamyltransferase 1 Threonine peptidase. MEROPS family T03 L-subunit, ... | 著者 | Hibi, T, Imaoka, M, Itoh, T, Wakayama, M. | 登録日 | 2018-03-20 | 公開日 | 2019-01-16 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.702 Å) | 主引用文献 | Crystal structure analysis and enzymatic characterization of gamma-glutamyltranspeptidase from Pseudomonas nitroreducens. Biosci. Biotechnol. Biochem., 83, 2019
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