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PDB: 5 件

3D9V
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BU of 3d9v by Molmil
CRYSTAL STRUCTURE OF ROCK I BOUND TO H-1152P A DI-METHYLATED VARIANT OF FASUDIL
分子名称: (S)-2-METHYL-1-[(4-METHYL-5-ISOQUINOLINE)SULFONYL]-HOMOPIPERAZINE, Rho-associated protein kinase 1
著者Jacobs, M.
登録日2008-05-27
公開日2008-06-10
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献The structure of dimeric ROCK I reveals the mechanism for ligand selectivity.
J.Biol.Chem., 281, 2006
2ESM
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BU of 2esm by Molmil
Crystal Structure of ROCK 1 bound to fasudil
分子名称: 5-(1,4-DIAZEPAN-1-SULFONYL)ISOQUINOLINE, Rho-associated protein kinase 1
著者Jacobs, M.
登録日2005-10-26
公開日2005-11-08
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献The Structure of Dimeric ROCK I Reveals the Mechanism for Ligand Selectivity.
J.Biol.Chem., 281, 2006
2ETK
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Crystal Structure of ROCK 1 bound to hydroxyfasudil
分子名称: 1-(1-HYDROXY-5-ISOQUINOLINESULFONYL)HOMOPIPERAZINE, Rho-associated protein kinase 1
著者Jacobs, M.
登録日2005-10-27
公開日2005-11-08
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.96 Å)
主引用文献The Structure of Dimeric ROCK I Reveals the Mechanism for Ligand Selectivity.
J.Biol.Chem., 281, 2006
2ETR
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Crystal Structure of ROCK I bound to Y-27632
分子名称: (R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXANECARBOXAMIDE, Rho-associated protein kinase 1
著者Jacobs, M.
登録日2005-10-27
公開日2005-11-08
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The Structure of Dimeric ROCK I Reveals the Mechanism for Ligand Selectivity.
J.Biol.Chem., 281, 2006
2ERZ
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BU of 2erz by Molmil
Crystal Structure of c-AMP Dependent Kinase (PKA) bound to hydroxyfasudil
分子名称: 1-(1-HYDROXY-5-ISOQUINOLINESULFONYL)HOMOPIPERAZINE, cAMP-dependent protein kinase inhibitor, alpha form, ...
著者Jacobs, M.
登録日2005-10-25
公開日2005-11-08
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Structure of Dimeric ROCK I Reveals the Mechanism for Ligand Selectivity.
J.Biol.Chem., 281, 2006

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件を2024-05-22に公開中

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