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PDB: 42289 件

7RHD
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darkmRuby M94T/F96Y mutant at pH 7.5
分子名称: 1,2-ETHANEDIOL, darkmRuby M94T/F96Y mutant
著者Huang, M, Ng, H.L, Zhang, S, Deng, M, Chu, J.
登録日2021-07-16
公開日2022-07-27
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A Long-range Interaction Affects Brightness and pH Stability of a Dark Fluorescent Protein
To Be Published
3ONL
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BU of 3onl by Molmil
yeast Ent3_ENTH-Vti1p_Habc complex structure
分子名称: Epsin-3, t-SNARE VTI1
著者Wang, J, Fang, P, Niu, L, Teng, M.
登録日2010-08-29
公開日2011-07-20
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Epsin N-terminal homology domains bind on opposite sides of two SNAREs
Proc.Natl.Acad.Sci.USA, 108, 2011
8BE9
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BU of 8be9 by Molmil
Crystal structure of SOS1-HRas-peptidomimetic5
分子名称: CHLORIDE ION, FORMIC ACID, GTPase HRas, ...
著者Fischer, B, Wohlkonig, A, Steyaert, J.
登録日2022-10-21
公開日2023-04-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Nanobody Loop Mimetics Enhance Son of Sevenless 1-Catalyzed Nucleotide Exchange on RAS.
Angew.Chem.Int.Ed.Engl., 62, 2023
2O9K
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BU of 2o9k by Molmil
WDR5 in Complex with Dimethylated H3K4 Peptide
分子名称: H3 HISTONE, WD repeat protein 5
著者Min, J.R, Schuetz, A, Allali-Hassani, A, Martin, F, Loppnau, P, Vedadi, M, Weigelt, J, Sundstrom, M, Edwards, A.M, Arrowsmith, C.H, Bochkarev, A, Plotnikov, A.N, Structural Genomics Consortium (SGC)
登録日2006-12-13
公開日2006-12-19
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Basis for Molecular Recognition and Presentation of Histone H3 by Wdr5.
Embo J., 25, 2006
7RDV
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BU of 7rdv by Molmil
TFH TCR bound to MHC Class II IAd presenting aggrecan epitope
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Aggrecan core peptide, H-2 class II histocompatibility antigen, ...
著者Lim, J.J, Rossjohn, J, Reid, H.
登録日2021-07-11
公開日2022-07-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.90006614 Å)
主引用文献TFH TCR bound to MHC Class II IAd presenting aggrecan epitope
To Be Published
8BEA
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BU of 8bea by Molmil
Crystal structure of SOS1-HRas-peptidomimetic10
分子名称: GTPase HRas, SOS1-HRas-peptidomimetic10, Son of sevenless homolog 1
著者Fischer, B, Wohlkonig, A, Steyaert, J.
登録日2022-10-21
公開日2023-04-26
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.47 Å)
主引用文献Nanobody Loop Mimetics Enhance Son of Sevenless 1-Catalyzed Nucleotide Exchange on RAS.
Angew.Chem.Int.Ed.Engl., 62, 2023
8BE6
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BU of 8be6 by Molmil
Crystal structure of SOS1-HRas-peptidomimetic2
分子名称: GTPase HRas, SOS1-HRas-peptidomimetic2, Son of sevenless homolog 1
著者Fischer, B, Wohlkonig, A, Steyaert, J.
登録日2022-10-21
公開日2023-04-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.89880252 Å)
主引用文献Nanobody Loop Mimetics Enhance Son of Sevenless 1-Catalyzed Nucleotide Exchange on RAS.
Angew.Chem.Int.Ed.Engl., 62, 2023
6WRX
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BU of 6wrx by Molmil
Crystal structure of computationally designed protein 2DS25.1 in complex with the human Transferrin receptor ectodomain
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Abraham, J, Coscia, A, Olal, D, Sahtoe, D.D, Baker, D, Clark, L.
登録日2020-04-30
公開日2021-04-28
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.07 Å)
主引用文献Transferrin receptor targeting by de novo sheet extension.
Proc.Natl.Acad.Sci.USA, 118, 2021
7RHC
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BU of 7rhc by Molmil
A new fluorescent protein darkmRuby at pH 9.0
分子名称: 1,2-ETHANEDIOL, darkmRuby
著者Huang, M, Ng, H.L, Zhang, S, Deng, M, Chu, J.
登録日2021-07-16
公開日2022-07-27
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献A Long-range Interaction Affects Brightness and pH Stability of a Dark Fluorescent Protein
To Be Published
6QWK
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BU of 6qwk by Molmil
The Transcriptional Regulator PrfA-L140F mutant from Listeria Monocytogenes in complex with a 30-bp operator PrfA-box motif
分子名称: DNA (30-MER), GLYCEROL, Listeriolysin positive regulatory factor A
著者Hall, M, Grundstrom, C, Hansen, S, Brannstrom, K, Johansson, J, Sauer-Eriksson, A.E.
登録日2019-03-05
公開日2020-04-01
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献A Novel Growth-Based Selection Strategy Identifies New Constitutively Active Variants of the Major Virulence Regulator PrfA in Listeria monocytogenes.
J.Bacteriol., 202, 2020
6WRV
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BU of 6wrv by Molmil
Crystal structure of computationally designed protein 3DS18 in complex with the human Transferrin receptor ectodomain
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Computationally designed protein 3DS18, ...
著者Abraham, J, Baker, D, Sahtoe, D.D, Coscia, A, Clark, L, Olal, D.
登録日2020-04-30
公開日2021-04-28
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.47 Å)
主引用文献Transferrin receptor targeting by de novo sheet extension.
Proc.Natl.Acad.Sci.USA, 118, 2021
8BNU
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BU of 8bnu by Molmil
Escherichia coli anaerobic fatty acid beta oxidation trifunctional enzyme (anEcTFE) tetrameric complex
分子名称: 3-ketoacyl-CoA thiolase FadI, Fatty acid oxidation complex subunit alpha
著者Sah-Teli, S.K, Pinkas, M, Novacek, J, Venkatesan, R.
登録日2022-11-14
公開日2023-05-17
最終更新日2023-07-19
実験手法ELECTRON MICROSCOPY (3.55 Å)
主引用文献Structural basis for different membrane-binding properties of E. coli anaerobic and human mitochondrial beta-oxidation trifunctional enzymes.
Structure, 31, 2023
6WJZ
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BU of 6wjz by Molmil
Crystal structure of human ribokinase in complex with AMPCP
分子名称: GLYCEROL, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER, ...
著者Park, J.
登録日2020-04-15
公開日2021-04-21
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structures of human ribokinase
To Be Published
6WRW
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BU of 6wrw by Molmil
Crystal structure of computationally designed protein 2DS25.5 in complex with the human Transferrin receptor ectodomain
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Computationally designed protein 2DS25.5, ...
著者Abraham, J, Coscia, A, Olal, D, Sahtoe, D.D, Baker, D, Clark, L.
登録日2020-04-30
公開日2021-04-28
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.84 Å)
主引用文献Transferrin receptor targeting by de novo sheet extension.
Proc.Natl.Acad.Sci.USA, 118, 2021
8BRJ
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BU of 8brj by Molmil
Escherichia coli anaerobic fatty acid beta oxidation trifunctional enzyme (anEcTFE) trimeric complex
分子名称: 3-ketoacyl-CoA thiolase FadI, Fatty acid oxidation complex subunit alpha
著者Sah-Teli, S.K, Pinkas, M, Novacek, J, Venkatesan, R.
登録日2022-11-23
公開日2023-05-17
最終更新日2023-07-19
実験手法ELECTRON MICROSCOPY (4.08 Å)
主引用文献Structural basis for different membrane-binding properties of E. coli anaerobic and human mitochondrial beta-oxidation trifunctional enzymes.
Structure, 31, 2023
6QMT
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BU of 6qmt by Molmil
Complement factor D in complex with the inhibitor 2-(2-(3'-(aminomethyl)-[1,1'-biphenyl]-3-carboxamido)phenyl)acetic acid
分子名称: 2-[2-[[3-[3-(aminomethyl)phenyl]phenyl]carbonylamino]phenyl]ethanoic acid, Complement factor D
著者Karki, R, Powers, J, Mainolfi, N, Anderson, K, Belanger, D, Liu, D, Jendza, K, Gelin, C.F, Solovay, C, Mac Sweeeny, A, Delgado, O, Crowley, M, Liao, S.-M, Argikar, U.A, Flohr, S, La Bonte, L.R, Lorthiois, E.L, Vulpetti, A, Cumin, F, Brown, A, Adams, C, Jaffee, B, Mogi, M.
登録日2019-02-08
公開日2019-04-24
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Design, Synthesis, and Preclinical Characterization of Selective Factor D Inhibitors Targeting the Alternative Complement Pathway.
J.Med.Chem., 62, 2019
6QN5
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BU of 6qn5 by Molmil
Three dimensional structure of human carbonic anhydrase IX in complex with benzenesulfonamide
分子名称: 4-chloranyl-~{N}-(3-oxidanylpropyl)-2-phenylsulfanyl-5-sulfamoyl-benzamide, Carbonic anhydrase 9, ZINC ION
著者Leitans, J, Tars, K.
登録日2019-02-09
公開日2020-02-26
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Halogenated and di-substituted benzenesulfonamides as selective inhibitors of carbonic anhydrase isoforms.
Eur.J.Med.Chem., 185, 2020
6QYJ
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BU of 6qyj by Molmil
The cryo-EM structure of the connector of the mature bacteriophage phi29
分子名称: Portal protein
著者Xu, J, Wang, D, Gui, M, Xiang, Y.
登録日2019-03-09
公開日2019-06-12
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural assembly of the tailed bacteriophage φ29.
Nat Commun, 10, 2019
6W0A
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BU of 6w0a by Molmil
Open-gate KcsA soaked in 1 mM BaCl2
分子名称: BARIUM ION, Fab Heavy Chain, Fab Light Chain, ...
著者Rohaim, A, Gong, L, Li, J.
登録日2020-02-29
公開日2020-07-08
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.237 Å)
主引用文献Open and Closed Structures of a Barium-Blocked Potassium Channel.
J.Mol.Biol., 432, 2020
6W0I
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Closed-gate KcsA soaked in 10mM KCl/5mM BaCl2
分子名称: Fab Heavy Chain, Fab Light Chain, POTASSIUM ION, ...
著者Rohaim, A, Gong, L, Li, J.
登録日2020-02-29
公開日2020-07-08
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.328 Å)
主引用文献Open and Closed Structures of a Barium-Blocked Potassium Channel.
J.Mol.Biol., 432, 2020
6QNL
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Three dimensional structure of human carbonic anhydrase XII in complex with benzenesulfonamide
分子名称: Carbonic anhydrase 12, ZINC ION, methyl 4-[(4-chloranyl-2-cyclohexylsulfanyl-5-sulfamoyl-phenyl)carbonylamino]butanoate
著者Dvinskis, E, Leitans, J, Tars, K.
登録日2019-02-11
公開日2020-03-04
最終更新日2021-10-06
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Halogenated and di-substituted benzenesulfonamides as selective inhibitors of carbonic anhydrase isoforms.
Eur.J.Med.Chem., 185, 2020
3ONK
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BU of 3onk by Molmil
yeast Ent3_ENTH domain
分子名称: Epsin-3
著者Wang, J, Fang, P, Niu, L, Teng, M.
登録日2010-08-29
公開日2011-07-20
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.09 Å)
主引用文献Epsin N-terminal homology domains bind on opposite sides of two SNAREs
Proc.Natl.Acad.Sci.USA, 108, 2011
8BVW
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BU of 8bvw by Molmil
RNA polymerase II pre-initiation complex with the distal +1 nucleosome (PIC-Nuc18W)
分子名称: CDK-activating kinase assembly factor MAT1, Cyclin-H, Cyclin-dependent kinase 7, ...
著者Abril-Garrido, J, Dienemann, C, Grabbe, F, Velychko, T, Lidschreiber, M, Wang, H, Cramer, P.
登録日2022-12-20
公開日2023-05-03
最終更新日2023-06-14
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Structural basis of transcription reduction by a promoter-proximal +1 nucleosome.
Mol.Cell, 83, 2023
6W9Q
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BU of 6w9q by Molmil
Peptide-bound SARS-CoV-2 Nsp9 RNA-replicase
分子名称: 3C-like proteinase peptide, Non-structural protein 9 fusion, PHOSPHATE ION
著者Littler, D.R, Gully, B.S, Riboldi-Tunnicliffe, A, Rossjohn, J.
登録日2020-03-23
公開日2020-04-08
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystal Structure of the SARS-CoV-2 Non-structural Protein 9, Nsp9.
Iscience, 23, 2020
6W66
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The structure of the F64A, S172A mutant Keap1-BTB domain in complex with SKP1-FBXL17
分子名称: F-box/LRR-repeat protein 17, Kelch-like ECH-associated protein 1, S-phase kinase-associated protein 1
著者Mena, E.L, Gee, C.L, Kuriyan, J, Rape, M.
登録日2020-03-16
公開日2020-08-19
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.21 Å)
主引用文献Structural basis for dimerization quality control.
Nature, 586, 2020

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件を2024-07-17に公開中

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