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PDB: 8 results

4U5L
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BU of 4u5l by Molmil
IMPORTIN-ALPHA MINOR NLS SITE INHIBITOR
Descriptor: Importin subunit alpha-1, N~2~-[4-(pyridin-3-yl)benzyl]-L-lysinamide
Authors:Stewart, M, Valkov, E, Holvey, R.S.
Deposit date:2014-07-25
Release date:2015-05-13
Last modified:2015-07-08
Method:X-RAY DIFFRACTION (2.53 Å)
Cite:Selective Targeting of the TPX2 Site of Importin-alpha Using Fragment-Based Ligand Design.
Chemmedchem, 10, 2015
4U5V
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BU of 4u5v by Molmil
IMPORTIN-ALPHA MINOR NLS SITE INHIBITOR
Descriptor: Importin subunit alpha-1, N~2~-{[5-(pyridin-3-yl)thiophen-2-yl]methyl}-L-lysinamide
Authors:Stewart, M, Valkov, E, Holvey, R.S.
Deposit date:2014-07-25
Release date:2015-05-13
Last modified:2015-07-08
Method:X-RAY DIFFRACTION (1.968 Å)
Cite:Selective Targeting of the TPX2 Site of Importin-alpha Using Fragment-Based Ligand Design.
Chemmedchem, 10, 2015
4U5N
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BU of 4u5n by Molmil
IMPORTIN-ALPHA MINOR NLS SITE INHIBITOR
Descriptor: Importin subunit alpha-1, N~2~-[4-(pyridin-3-yl)benzyl]-L-lysyl-N-[(1R,2S,3R)-1-{[(2R)-1-amino-1-oxo-3-phenylpropan-2-yl]amino}-1,3-dihydroxybutan-2-yl]glycinamide
Authors:Stewart, M, Valkov, E, Holvey, R.S.
Deposit date:2014-07-25
Release date:2015-05-13
Last modified:2015-07-08
Method:X-RAY DIFFRACTION (2.31 Å)
Cite:Selective Targeting of the TPX2 Site of Importin-alpha Using Fragment-Based Ligand Design.
Chemmedchem, 10, 2015
4U5S
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BU of 4u5s by Molmil
IMPORTIN-ALPHA MINOR NLS SITE INHIBITOR
Descriptor: Importin subunit alpha-1, N-[(2S)-2-[(N~2~-acetyl-D-lysyl)amino]-3-(pyridin-3-ylmethoxy)propyl]-L-allothreonyl-D-phenylalaninamide
Authors:Stewart, M, Valkov, E, Holvey, R.S.
Deposit date:2014-07-25
Release date:2015-05-13
Last modified:2017-06-21
Method:X-RAY DIFFRACTION (2.12 Å)
Cite:Selective Targeting of the TPX2 Site of Importin-alpha Using Fragment-Based Ligand Design.
Chemmedchem, 10, 2015
4U54
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BU of 4u54 by Molmil
IMPORTIN-ALPHA MINOR NLS SITE INHIBITOR
Descriptor: Importin subunit alpha-1, N-methyl-1-[3-(pyridin-3-yl)phenyl]methanamine
Authors:Stewart, M, Valkov, E, Holvey, R.S.
Deposit date:2014-07-24
Release date:2015-05-13
Last modified:2015-07-08
Method:X-RAY DIFFRACTION (2.41 Å)
Cite:Selective Targeting of the TPX2 Site of Importin-alpha Using Fragment-Based Ligand Design.
Chemmedchem, 10, 2015
4U58
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BU of 4u58 by Molmil
IMPORTIN-ALPHA MINOR NLS SITE INHIBITOR
Descriptor: Importin subunit alpha-1, N~2~-[4-(pyridin-3-yl)benzoyl]-L-lysinamide
Authors:Stewart, M, Valkov, E, Holvey, R.S.
Deposit date:2014-07-24
Release date:2015-05-13
Last modified:2015-07-08
Method:X-RAY DIFFRACTION (2.56 Å)
Cite:Selective Targeting of the TPX2 Site of Importin-alpha Using Fragment-Based Ligand Design.
Chemmedchem, 10, 2015
4U5O
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BU of 4u5o by Molmil
IMPORTIN-ALPHA MINOR NLS SITE INHIBITOR
Descriptor: Importin subunit alpha-1, N~2~-[4-(pyridin-3-yl)benzyl]-D-lysinamide
Authors:Stewart, M, Valkov, E, Holvey, R.S.
Deposit date:2014-07-25
Release date:2015-05-13
Last modified:2015-07-08
Method:X-RAY DIFFRACTION (2 Å)
Cite:Selective Targeting of the TPX2 Site of Importin-alpha Using Fragment-Based Ligand Design.
Chemmedchem, 10, 2015
4U5U
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BU of 4u5u by Molmil
IMPORTIN-ALPHA MINOR NLS SITE INHIBITOR
Descriptor: Importin subunit alpha-1, N~2~-[3-(pyridin-3-yl)benzyl]-L-lysinamide
Authors:Stewart, M, Valkov, E, Holvey, R.S.
Deposit date:2014-07-25
Release date:2015-05-13
Last modified:2015-07-08
Method:X-RAY DIFFRACTION (1.96 Å)
Cite:Selective Targeting of the TPX2 Site of Importin-alpha Using Fragment-Based Ligand Design.
Chemmedchem, 10, 2015

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