1JL5
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![BU of 1jl5 by Molmil](/molmil-images/mine/1jl5) | Novel Molecular Architecture of YopM-a Leucine-rich Effector Protein from Yersinia pestis | 分子名称: | CALCIUM ION, outer protein YopM | 著者 | Evdokimov, A.G, Anderson, D.E, Routzahn, K.M, Waugh, D.S. | 登録日 | 2001-07-15 | 公開日 | 2001-10-10 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Unusual molecular architecture of the Yersinia pestis cytotoxin YopM: a leucine-rich repeat protein with the shortest repeating unit. J.Mol.Biol., 312, 2001
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2I3R
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![BU of 2i3r by Molmil](/molmil-images/mine/2i3r) | Engineered catalytic domain of protein tyrosine phosphatase HPTPbeta | 分子名称: | CHLORIDE ION, Receptor-type tyrosine-protein phosphatase beta | 著者 | Evdokimov, A.G, Pokross, M.E, Walter, R.L, Mekel, M. | 登録日 | 2006-08-20 | 公開日 | 2006-08-29 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Engineering the catalytic domain of human protein tyrosine phosphatase beta for structure-based drug discovery. Acta Crystallogr.,Sect.D, 62, 2006
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2I4E
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![BU of 2i4e by Molmil](/molmil-images/mine/2i4e) | Structural studies of protein tyrosine phosphatase beta catalytic domain in complex with inhibitors | 分子名称: | Receptor-type tyrosine-protein phosphatase beta, VANADATE ION | 著者 | Evdokimov, A.G, Pokross, M.E, Walter, R.L, Mekel, M. | 登録日 | 2006-08-21 | 公開日 | 2006-08-29 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Engineering the catalytic domain of human protein tyrosine phosphatase beta for structure-based drug discovery. Acta Crystallogr.,Sect.D, 62, 2006
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2I4G
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![BU of 2i4g by Molmil](/molmil-images/mine/2i4g) | Structural studies of protein tyrosine phosphatase beta catalytic domain in complex with a sulfamic acid (soaking experiment) | 分子名称: | CHLORIDE ION, N-(TERT-BUTOXYCARBONYL)-L-TYROSYL-N-METHYL-4-(SULFOAMINO)-L-PHENYLALANINAMIDE, Receptor-type tyrosine-protein phosphatase beta | 著者 | Evdokimov, A.G, Pokross, M.E, Walter, R.L, Mekel, M. | 登録日 | 2006-08-21 | 公開日 | 2006-08-29 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Engineering the catalytic domain of human protein tyrosine phosphatase beta for structure-based drug discovery. Acta Crystallogr.,Sect.D, 62, 2006
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2I5X
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![BU of 2i5x by Molmil](/molmil-images/mine/2i5x) | Engineering the PTPbeta catalytic domain with improved crystallization properties | 分子名称: | (4-ETHYLPHENYL)SULFAMIC ACID, CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Evdokimov, A.G, Pokross, M.E, Walter, R.L, Mekel, M, Klopfenstein, S. | 登録日 | 2006-08-26 | 公開日 | 2006-09-05 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Engineering the catalytic domain of human protein tyrosine phosphatase beta for structure-based drug discovery. Acta Crystallogr.,Sect.D, 62, 2006
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2I3U
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![BU of 2i3u by Molmil](/molmil-images/mine/2i3u) | Structural studies of protein tyrosine phosphatase beta catalytic domain in complex with inhibitors | 分子名称: | Receptor-type tyrosine-protein phosphatase beta | 著者 | Evdokimov, A.G, Pokross, M.E, Walter, R.L, Mekel, M. | 登録日 | 2006-08-20 | 公開日 | 2006-08-29 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Engineering the catalytic domain of human protein tyrosine phosphatase beta for structure-based drug discovery. Acta Crystallogr.,Sect.D, 62, 2006
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4W8J
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![BU of 4w8j by Molmil](/molmil-images/mine/4w8j) | Structure of the full-length insecticidal protein Cry1Ac reveals intriguing details of toxin packaging into in vivo formed crystals | 分子名称: | CALCIUM ION, POTASSIUM ION, Pesticidal crystal protein cry1Ac | 著者 | Evdokimov, A.G, Moshiri, F, Sturman, E.J, Rydel, T.J, Zheng, M, Seale, J.W, Franklin, S. | 登録日 | 2014-08-25 | 公開日 | 2014-09-17 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.78 Å) | 主引用文献 | Structure of the full-length insecticidal protein Cry1Ac reveals intriguing details of toxin packaging into in vivo formed crystals. Protein Sci., 23, 2014
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6V1V
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![BU of 6v1v by Molmil](/molmil-images/mine/6v1v) | VIP3B (VIP3B_2160) adapted for crystallization | 分子名称: | Vegetative insecticidal protein | 著者 | Evdokimov, A.G, Zheng, M, Moshiri, F, Haas, J, Lowder, C. | 登録日 | 2019-11-21 | 公開日 | 2019-12-18 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (3.189 Å) | 主引用文献 | Crystal structure of a Vip3B family insecticidal protein reveals a new fold and a unique tetrameric assembly. Protein Sci., 29, 2020
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1ELJ
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![BU of 1elj by Molmil](/molmil-images/mine/1elj) | THE CRYSTAL STRUCTURE OF LIGANDED MALTODEXTRIN-BINDING PROTEIN FROM PYROCOCCUS FURIOSUS | 分子名称: | MALTODEXTRIN-BINDING PROTEIN, SULFATE ION, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose | 著者 | Evdokimov, A.G, Anderson, E.D, Routzahn, K.M, Waugh, D.S. | 登録日 | 2000-03-13 | 公開日 | 2001-01-19 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structural basis for oligosaccharide recognition by Pyrococcus furiosus maltodextrin-binding protein. J.Mol.Biol., 305, 2001
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1G9U
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![BU of 1g9u by Molmil](/molmil-images/mine/1g9u) | CRYSTAL STRUCTURE OF YOPM-LEUCINE RICH EFFECTOR PROTEIN FROM YERSINIA PESTIS | 分子名称: | ACETATE ION, CALCIUM ION, MERCURY (II) ION, ... | 著者 | Evdokimov, A.G, Anderson, D.E, Routzahn, K.M, Waugh, D.S. | 登録日 | 2000-11-28 | 公開日 | 2001-10-10 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Unusual molecular architecture of the Yersinia pestis cytotoxin YopM: a leucine-rich repeat protein with the shortest repeating unit. J.Mol.Biol., 312, 2001
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2WIU
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![BU of 2wiu by Molmil](/molmil-images/mine/2wiu) | Mercury-modified bacterial persistence regulator hipBA | 分子名称: | CHLORIDE ION, HTH-TYPE TRANSCRIPTIONAL REGULATOR HIPB, MERCURY (II) ION, ... | 著者 | Evdokimov, A, Voznesensky, I, Fennell, K, Anderson, M, Smith, J.F, Fisher, D.A. | 登録日 | 2009-05-17 | 公開日 | 2009-07-28 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | New Kinase Regulation Mechanism Found in Hipba: A Bacterial Persistence Switch. Acta Crystallogr.,Sect.D, 65, 2009
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1HUF
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![BU of 1huf by Molmil](/molmil-images/mine/1huf) | |
1HY5
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![BU of 1hy5 by Molmil](/molmil-images/mine/1hy5) | |
1ORY
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![BU of 1ory by Molmil](/molmil-images/mine/1ory) | FLAGELLAR EXPORT CHAPERONE IN COMPLEX WITH ITS COGNATE BINDING PARTNER | 分子名称: | Flagellin, PHOSPHATE ION, flagellar protein FliS | 著者 | Evdokimov, A.G, Phan, J, Tropea, J.E, Routzahn, K.M, Peters III, H.K, Pokross, M, Waugh, D.S. | 登録日 | 2003-03-17 | 公開日 | 2003-09-16 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Similar modes of polypeptide recognition by export chaperones in flagellar biosynthesis and type III secretion Nat.Struct.Biol., 10, 2003
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1ORJ
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![BU of 1orj by Molmil](/molmil-images/mine/1orj) | FLAGELLAR EXPORT CHAPERONE | 分子名称: | flagellar protein FliS | 著者 | Evdokimov, A.G, Phan, J, Tropea, J.E, Routzahn, K.M, Peters III, H.K, Pokross, M, Waugh, D.S. | 登録日 | 2003-03-13 | 公開日 | 2003-09-16 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Similar modes of polypeptide recognition by export chaperones in flagellar biosynthesis and type III secretion Nat.Struct.Biol., 10, 2003
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1K6Z
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![BU of 1k6z by Molmil](/molmil-images/mine/1k6z) | Crystal Structure of the Yersinia Secretion Chaperone SycE | 分子名称: | IMIDAZOLE, Type III secretion chaperone SycE | 著者 | Evdokimov, A.G, Tropea, J.E, Routzahn, K.M, Waugh, D.S. | 登録日 | 2001-10-17 | 公開日 | 2001-10-31 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Three-dimensional structure of the type III secretion chaperone SycE from Yersinia pestis. Acta Crystallogr.,Sect.D, 58, 2002
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1LYV
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![BU of 1lyv by Molmil](/molmil-images/mine/1lyv) | High-resolution structure of the catalytically inactive yersinia tyrosine phosphatase C403A mutant in complex with phosphate. | 分子名称: | CHLORIDE ION, PHOSPHATE ION, PROTEIN-TYROSINE PHOSPHATASE YOPH | 著者 | Evdokimov, A.G, Waugh, D.S, Routzahn, K, Tropea, J, Cherry, S. | 登録日 | 2002-06-08 | 公開日 | 2002-07-03 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.363 Å) | 主引用文献 | High-resolution structure of the catalytically inactive yersinia tyrosine phosphatase C403A mutant in complex with phosphate. To be Published
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2RHS
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![BU of 2rhs by Molmil](/molmil-images/mine/2rhs) | |
2RHQ
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2VF6
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![BU of 2vf6 by Molmil](/molmil-images/mine/2vf6) | Human FDPS synthase in complex with minodronate | 分子名称: | (1-HYDROXY-2-IMIDAZO[1,2-A]PYRIDIN-3-YLETHANE-1,1-DIYL)BIS(PHOSPHONIC ACID), FARNESYL PYROPHOSPHATE SYNTHETASE, MAGNESIUM ION | 著者 | Evdokimov, A.G, Barnett, B.L, Ebetino, F.H, Pokross, M. | 登録日 | 2007-10-31 | 公開日 | 2007-11-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Human Fdps Synthase in Complex with Novel Inhibitor To be Published
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3RYE
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![BU of 3rye by Molmil](/molmil-images/mine/3rye) | Human FDPS Synthase in Complex with a N-Methyl Pyridinum Bisphosphonate | 分子名称: | 3-(2-hydroxy-2,2-diphosphonoethyl)-1-methylpyridinium, Farnesyl pyrophosphate synthase, MAGNESIUM ION, ... | 著者 | Evdokimov, A.G, Barnett, B.L, Ebetino, F.H, Pokross, M. | 登録日 | 2011-05-11 | 公開日 | 2011-06-01 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Human FDPS Synthase in Complex with a N-Methyl Pyridinum Bisphosphonate To be Published
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3S4J
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![BU of 3s4j by Molmil](/molmil-images/mine/3s4j) | Human FDPS Synthase in Complex with a Rigid Analog of Risedronate | 分子名称: | 6,7-dihydro-5H-cyclopenta[b]pyridine-6,6-diylbis(phosphonic acid), Farnesyl pyrophosphate synthase, MAGNESIUM ION, ... | 著者 | Evdokimov, A.G, Barnett, B.L, Ebetino, F.H, Pokross, M. | 登録日 | 2011-05-19 | 公開日 | 2011-06-29 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Human FDPS Synthase in Complex with a Rigid Analog of Risedronate To be Published
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2RAH
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![BU of 2rah by Molmil](/molmil-images/mine/2rah) | Human FDPS synthase in complex with novel inhibitor | 分子名称: | Farnesyl pyrophosphate synthetase, MAGNESIUM ION, SULFATE ION, ... | 著者 | Evdokimov, A.G, Barnett, B.L, Ebetino, F.H, Pokross, M. | 登録日 | 2007-09-15 | 公開日 | 2007-09-25 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Human FDPS synthase in complex with novel inhibitor To be Published
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2F6T
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![BU of 2f6t by Molmil](/molmil-images/mine/2f6t) | Protein tyrosine phosphatase 1B with sulfamic acid inhibitors | 分子名称: | 3(S)-METHYLCARBAMOYL-7-SULFOAMINO-3,4-DIHYDRO-1H-ISOQUINOLINE-2-CARBOXYLIC ACID TERT-BUTYL ESTER, CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Evdokimov, A.G, Pokross, M.E, Klopfenstein, S.R. | 登録日 | 2005-11-29 | 公開日 | 2005-12-13 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | 1,2,3,4-Tetrahydroisoquinolinyl sulfamic acids as phosphatase PTP1B inhibitors Bioorg.Med.Chem.Lett., 16, 2006
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2F6Z
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![BU of 2f6z by Molmil](/molmil-images/mine/2f6z) | Protein tyrosine phosphatase 1B with sulfamic acid inhibitors | 分子名称: | CHLORIDE ION, MAGNESIUM ION, Tyrosine-protein phosphatase, ... | 著者 | Evdokimov, A.G, Pokross, M.E, Klopfenstein, S.R. | 登録日 | 2005-11-29 | 公開日 | 2005-12-13 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | 1,2,3,4-Tetrahydroisoquinolinyl sulfamic acids as phosphatase PTP1B inhibitors Bioorg.Med.Chem.Lett., 16, 2006
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