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PDB: 1542 件

2OZL
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Human pyruvate dehydrogenase S264E variant
分子名称: MAGNESIUM ION, POTASSIUM ION, Pyruvate dehydrogenase E1 component alpha subunit, ...
著者Ciszak, E.M, Dominiak, P.M, Patel, M.S, Korotchkina, L.G.
登録日2007-02-26
公開日2007-05-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Phosphorylation of Serine 264 Impedes Active Site Accessibility in the E1 Component of the Human Pyruvate Dehydrogenase Multienzyme Complex
Biochemistry, 46, 2007
2OW4
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Crystal structure of a lectin from Canavalia maritima seeds (ConM) in complex with man1-2man-OMe
分子名称: CALCIUM ION, Canavalia maritima lectin, MANGANESE (II) ION, ...
著者Moreno, F.B.M.B, Bezerra, G.A, de Oliveira, T.M, de Souza, E.M, da Rocha, B.A.M, Benevides, R.G, Delatorre, P, Cavada, B.S, de Azevedo Jr, W.F.
登録日2007-02-15
公開日2007-10-23
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural analysis of Canavalia maritima and Canavalia gladiata lectins complexed with different dimannosides: New insights into the understanding of the structure-biological activity relationship in legume lectins.
J.Struct.Biol., 160, 2007
1OUM
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M64V PNP +Talo
分子名称: 9-(6-DEOXY-ALPHA-L-TALOFURANOSYL)-6-METHYLPURINE, PHOSPHATE ION, Purine nucleoside phosphorylase
著者Ealick, S.E, Bennett, E.M, Anand, R, Secrist, J.A, Parker, W.B, Hassan, A.E, Allan, P.W, McPherson, D.T, Sorscher, E.J.
登録日2003-03-24
公開日2004-02-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Designer gene therapy using an Escherichia coli purine nucleoside phosphorylase/prodrug system.
Chem.Biol., 10, 2003
1W8C
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CO-CRYSTAL STRUCTURE OF 6-CYCLOHEXYLMETHOXY-8-ISOPROPYL-9H-PURIN-2- YLAMINE AND MONOMERIC CDK2
分子名称: 6-(CYCLOHEXYLMETHOXY)-8-ISOPROPYL-9H-PURIN-2-AMINE, CELL DIVISION PROTEIN KINASE 2
著者Pratt, D.J, Endicott, J.A, Noble, M.E.M.
登録日2004-09-20
公開日2006-08-30
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献8-Substituted O6-Cyclohexylmethylguanine Cdk2 Inhibitors; Using Structure-Based Inhibitor Design to Optimise an Alternative Binding Mode.
J.Med.Chem., 57, 2014
1QKO
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HIGH RESOLUTION X-RAY STRUCTURE OF AN EARLY INTERMEDIATE IN THE BACTERIORHODOPSIN PHOTOCYCLE
分子名称: BACTERIORHODOPSIN, RETINAL
著者Edman, K, Nollert, P, Royant, A, Belrhali, H, Pebay-Peyroula, E, Hajdu, J, Neutze, R, Landau, E.M.
登録日1999-07-30
公開日1999-10-24
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献High Resolution X-Ray Structure of an Early Intermediate in the Bacteriorhodopsin Photocycle
Nature, 401, 1999
1QMZ
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PHOSPHORYLATED CDK2-CYCLYIN A-SUBSTRATE PEPTIDE COMPLEX
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CELL DIVISION PROTEIN KINASE 2, G2/MITOTIC-SPECIFIC CYCLIN A, ...
著者Brown, N.R, Noble, M.E.M, Endicott, J.A, Johnson, L.N.
登録日1999-10-11
公開日1999-12-14
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Structural Basis for Specificity of Substrate and Recruitment Peptides for Cyclin-Dependent Kinases
Nat.Cell Biol., 1, 1999
1OVG
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M64V PNP +MePdr
分子名称: 9-(2-DEOXY-BETA-D-RIBOFURANOSYL)-6-METHYLPURINE, PHOSPHATE ION, Purine nucleoside phosphorylase
著者Ealick, S.E, Bennett, E.M, Anand, R, Secrist, J.A, Parker, P.W, Hassan, A.E, Allan, P.W, McPherson, D.T, Sorscher, E.J.
登録日2003-03-26
公開日2004-02-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Designer gene therapy using an Escherichia coli purine nucleoside phosphorylase/prodrug system.
Chem.Biol., 10, 2003
1OW6
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Paxillin LD4 motif bound to the Focal Adhesion Targeting (FAT) domain of the Focal Adhesion Kinase
分子名称: Focal adhesion kinase 1, Paxillin
著者Hoellerer, M.K, Noble, M.E.M, Labesse, G, Campbell, I.D, Werner, J.M, Arold, S.T.
登録日2003-03-28
公開日2003-10-21
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Molecular Recognition of Paxillin LD motifs by the Focal Adhesion Targeting Domain
Structure, 11, 2003
1OGV
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Lipidic cubic phase crystal structure of the photosynthetic reaction centre from Rhodobacter sphaeroides
分子名称: BACTERIOCHLOROPHYLL A, BACTERIOPHEOPHYTIN A, CARDIOLIPIN, ...
著者Katona, G, Andreasson, U, Landau, E.M, Andreasson, L.-E, Neutze, R.
登録日2003-05-13
公開日2003-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Lipidic Cubic Phase Crystal Structure of the Photosynthetic Reaction Centre from Rhodobacter Sphaeroides at 2.35 A Resolution
J.Mol.Biol., 331, 2003
1OGU
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STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH A 2-ARYLAMINO-4-CYCLOHEXYLMETHYL-5-NITROSO-6-AMINOPYRIMIDINE INHIBITOR
分子名称: 4-{[4-AMINO-6-(CYCLOHEXYLMETHOXY)-5-NITROSOPYRIMIDIN-2-YL]AMINO}BENZAMIDE, CELL DIVISION PROTEIN KINASE 2, CYCLIN A2, ...
著者Pratt, D.J, Endicott, J.A, Noble, M.E.M.
登録日2003-05-13
公開日2003-09-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure-Based Design of 2-Arylamino-4-Cyclohexyl Methyl-5-Nitroso-6-Aminopyrimidine Inhibitors of Cyclin-Dependent Kinases 1 and 2
Bioorg.Med.Chem.Lett., 13, 2003
1W6C
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AGAO holoenzyme in a small cell, at 2.2 angstroms
分子名称: COPPER (II) ION, PHENYLETHYLAMINE OXIDASE, SODIUM ION
著者Duff, A.P, Langley, D.B, Juda, G.A, Shepard, E.M, Dooley, D.M, Freeman, H.C, Guss, J.M.
登録日2004-08-17
公開日2005-12-08
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Copper Containing Amine Oxidase from Arthrobacter Globiformis: Refinement at 1.55 And 2.20 A Resolution in Two Crystal Forms.
Acta Crystallogr.,Sect.F, 62, 2006
1W5R
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X-ray crystallographic structure of a C70Q Mycobacterium smegmatis N- arylamine Acetyltransferase
分子名称: ARYLAMINE N-ACETYLTRANSFERASE
著者Holton, S.J, Sandy, J, Rodrigues-Lima, F, Dupret, J.-M, Bhakta, S, Noble, M.E.M, Sim, E.
登録日2004-08-09
公開日2005-05-11
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Investigation of the Catalytic Triad of Arylamine N-Acetyltransferases: Essential Residues Required for Acetyl Transfer to Arylamines.
Biochem.J., 390, 2005
1OW7
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Paxillin LD4 motif bound to the Focal Adhesion Targeting (FAT) domain of the Focal Adhesion Kinase
分子名称: Focal adhesion kinase 1, Paxillin
著者Hoellerer, M.K, Noble, M.E.M, Labesse, G, Werner, J.M, Arold, S.T.
登録日2003-03-28
公開日2003-10-21
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Molecular Recognition of Paxillin LD Motifs by the Focal Adhesion Targeting Domain
Structure, 11, 2003
1NTF
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Crystal Structure of Cimex Nitrophorin
分子名称: PROTOPORPHYRIN IX CONTAINING FE, salivary nitrophorin
著者Weichsel, A, Maes, E.M, Andersen, J.F, Valenzuela, J.G, Walker, F.A, Montfort, W.R.
登録日2003-01-29
公開日2004-03-16
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Heme-assisted S-nitrosation of a proximal thiolate in a nitric oxide transport protein.
Proc.Natl.Acad.Sci.USA, 102, 2005
1ODB
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THE CRYSTAL STRUCTURE OF HUMAN S100A12 - COPPER COMPLEX
分子名称: CALCIUM ION, CALGRANULIN C, COPPER (II) ION
著者Moroz, O.V, Antson, A.A, Grist, S.J, Maitland, N.J, Dodson, G.G, Wilson, K.S, Lukanidin, E.M, Bronstein, I.B.
登録日2003-02-15
公開日2003-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Structure of the Human S100A12-Copper Complex: Implications for Host-Parasite Defence
Acta Crystallogr.,Sect.D, 59, 2003
1W6F
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Arylamine N-acetyltransferase from Mycobacterium smegmatis with the anti-tubercular drug isoniazid bound in the active site.
分子名称: 4-(DIAZENYLCARBONYL)PYRIDINE, ARYLAMINE N-ACETYLTRANSFERASE
著者Sandy, J, Holton, S, Fullham, E, Sim, E, Noble, M.E.M.
登録日2004-08-17
公開日2005-02-23
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Binding of the Anti-Tubercular Drug Isoniazid to the Arylamine N-Acetyltransferase Protein from Mycobacterium Smegmatis
Protein Sci., 14, 2005
1W4N
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AGAO covalent complex with Tranylcypromine
分子名称: COPPER (II) ION, GLYCEROL, PHENYLETHYLAMINE OXIDASE, ...
著者Duff, A.P, Trambaiolo, D.M, Langley, D.B, Juda, G.A, Shepard, E.M, Dooley, D.M, Freeman, H.C, Guss, J.M.
登録日2004-07-27
公開日2005-12-08
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Complexes of the Copper-Containing Amine Oxidase from Arthrobacter Globiformis with the Inhibitors Benzylhydrazine and Tranylcypromine.
Acta Crystallogr.,Sect.F, 64, 2008
1VIN
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BOVINE CYCLIN A3
分子名称: CYCLIN A
著者Noble, M.E.M, Endicott, J.A.E, Brown, N.R.
登録日1996-03-15
公開日1996-08-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The crystal structure of cyclin A.
Structure, 3, 1995
1QA7
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CRYSTAL COMPLEX OF THE 3C PROTEINASE FROM HEPATITIS A VIRUS WITH ITS INHIBITOR AND IMPLICATIONS FOR THE POLYPROTEIN PROCESSING IN HAV
分子名称: DIMETHYL SULFOXIDE, GLYCEROL, HAV 3C PROTEINASE, ...
著者Bergmann, E.M, Cherney, M.M, Mckendrick, J, Vederas, J.C, James, M.N.G.
登録日1999-04-15
公開日1999-04-20
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of an inhibitor complex of the 3C proteinase from hepatitis A virus (HAV) and implications for the polyprotein processing in HAV.
Virology, 265, 1999
1VUB
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CCDB, A TOPOISOMERASE POISON FROM E. COLI
分子名称: CCDB, CHLORIDE ION
著者Loris, R, Dao-Thi, M.-H, Bahasi, E.M, Van Melderen, L, Poortmans, F, Liddington, R, Couturier, M, Wyns, L.
登録日1998-04-17
公開日1998-07-15
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystal structure of CcdB, a topoisomerase poison from E. coli.
J.Mol.Biol., 285, 1999
1W5Z
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AGAO covalent complex with Benzylhydrazine
分子名称: COPPER (II) ION, GLYCEROL, PHENYLETHYLAMINE OXIDASE, ...
著者Duff, A.P, Trambaiolo, D.M, Langley, D.B, Juda, G.A, Shepard, E.M, Dooley, D.M, Freeman, H.C, Guss, J.M.
登録日2004-08-11
公開日2005-12-08
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Complexes of the Copper-Containing Amine Oxidase from Arthrobacter Globiformis with the Inhibitors Benzylhydrazine and Tranylcypromine.
Acta Crystallogr.,Sect.F, 64, 2008
1PR5
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Escherichia coli Purine Nucleoside Phosphorylase Complexed with 7-deazaadenosine and Phosphate/Sulfate
分子名称: '2-(4-AMINO-PYRROLO[2,3-D]PYRIMIDIN-7-YL)-5-HYDROXYMETHYL-TETRAHYDRO-FURAN-3,4-DIOL, PHOSPHATE ION, Purine nucleoside phosphorylase DeoD-type
著者Bennett, E.M, Li, C, Allan, P.W, Parker, W.B, Ealick, S.E.
登録日2003-06-19
公開日2003-11-25
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis for substrate specificity of Escherichia coli purine nucleoside phosphorylase.
J.Biol.Chem., 278, 2003
1W6G
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AGAO holoenzyme at 1.55 angstroms
分子名称: COPPER (II) ION, GLYCEROL, PHENYLETHYLAMINE OXIDASE, ...
著者Langley, D.B, Duff, A.P, Juda, G.A, Shepard, E.M, Dooley, D.M, Freeman, H.C, Guss, J.M.
登録日2004-08-18
公開日2005-12-08
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献The Copper Containing Amine Oxidase from Arthrobacter Globiformis: Refinement at 1.55 And 2.20 A Resolution in Two Crystal Forms.
Acta Crystallogr.,Sect.F, 62, 2006
1PR0
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Escherichia coli Purine Nucleoside Phosphorylase Complexed with Inosine and Phosphate/Sulfate
分子名称: INOSINE, PHOSPHATE ION, Purine nucleoside phosphorylase DeoD-type
著者Bennett, E.M, Li, C, Allan, P.W, Parker, W.B, Ealick, S.E.
登録日2003-06-19
公開日2003-11-25
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural basis for substrate specificity of Escherichia coli purine nucleoside phosphorylase.
J.Biol.Chem., 278, 2003
2PF5
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Crystal Structure of the Human TSG-6 Link Module
分子名称: NONAETHYLENE GLYCOL, SULFATE ION, Tumor necrosis factor-inducible protein TSG-6
著者Higman, V.A, Mahoney, D.J, Noble, M.E.M, Day, A.J.
登録日2007-04-04
公開日2007-06-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Plasticity of the TSG-6 HA-binding loop and mobility in the TSG-6-HA complex revealed by NMR and X-ray crystallography
J.Mol.Biol., 371, 2007

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