8QB5
| Crystal structure of apo-GltTk obtained with in meso crystallization (P6322 space group) | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, OLEIC ACID, Proton/glutamate symporter, ... | 著者 | Marin, E, Guskov, A, Borshchevskiy, V, Kovalev, K. | 登録日 | 2023-08-24 | 公開日 | 2024-09-11 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Crystal structure of apo-GltTk obtained with in meso crystallization (P6322 space group) To Be Published
|
|
8AZ0
| IAPP S20G growth-phase fibril polymorph 2PF-L | 分子名称: | Islet amyloid polypeptide | 著者 | Wilkinson, M, Xu, Y, Gallardo, R, Radford, S.E, Ranson, N.A. | 登録日 | 2022-09-05 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Structural evolution of fibril polymorphs during amyloid assembly. Cell, 186, 2023
|
|
7H0X
| Crystal structure of SARS-CoV-2 NSP3 Macrodomain in complex with ASAP-0013255-001 | 分子名称: | (4M)-1-methyl-4-(4-{[(1S)-2-methyl-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)propyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-6-yl)-1H-pyrazole-5-carbonitrile, Papain-like protease nsp3 | 著者 | Aschenbrenner, J.C, Fearon, D, Tomlinson, C.W.E, Marples, P.G, Fairhead, M, Balcomb, B.H, Chandran, A.V, Godoy, A.S, Koekemoer, L, Lithgo, R.M, Ni, X, Thompson, W, Wang, S, Wild, C, Williams, E.P, Winokan, M, Walsh, M.A, von Delft, F. | 登録日 | 2024-01-23 | 公開日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Group deposition of SARS-CoV-2 NSP3 Macrodomain in complex with inhibitors from the ASAP AViDD centre To Be Published
|
|
6XQ7
| Receptor for Advanced Glycation End Products VC1 domain in complex with Fragment 5 | 分子名称: | 5-bromo-3-methyl-1H-indole-2-carboxylic acid, ACETATE ION, Advanced glycosylation end product-specific receptor, ... | 著者 | Salay, L.E, Kozlyuk, N, Gilston, B.A, Gogliotti, R.D, Christov, P.P, Kim, K, Ovee, M, Waterson, A.G, Chazin, W.J. | 登録日 | 2020-07-09 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | A fragment-based approach to discovery of Receptor for Advanced Glycation End products inhibitors. Proteins, 89, 2021
|
|
8AZ6
| IAPP S20G plateau-phase fibril polymorph 4PF-LU | 分子名称: | Islet amyloid polypeptide | 著者 | Wilkinson, M, Xu, Y, Gallardo, R, Radford, S.E, Ranson, N.A. | 登録日 | 2022-09-05 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structural evolution of fibril polymorphs during amyloid assembly. Cell, 186, 2023
|
|
8AZ1
| IAPP S20G growth-phase fibril polymorph 2PF-C | 分子名称: | Islet amyloid polypeptide | 著者 | Wilkinson, M, Xu, Y, Gallardo, R, Radford, S.E, Ranson, N.A. | 登録日 | 2022-09-05 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structural evolution of fibril polymorphs during amyloid assembly. Cell, 186, 2023
|
|
2J1K
| CAV-2 fibre head in complex with CAR D1 | 分子名称: | COXSACKIEVIRUS AND ADENOVIRUS RECEPTOR, FIBER PROTEIN | 著者 | Seiradake, E, Lortat-Jacob, H, Billet, O, Kremer, E.J, Cusack, S. | 登録日 | 2006-08-14 | 公開日 | 2006-09-05 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural and Mutational Analysis of Human Ad37 and Canine Adenovirus 2 Fiber Heads in Complex with the D1 Domain of Coxsackie and Adenovirus Receptor. J.Biol.Chem., 281, 2006
|
|
8AZ2
| IAPP S20G growth-phase fibril polymorph 3PF-CU | 分子名称: | Islet amyloid polypeptide | 著者 | Wilkinson, M, Xu, Y, Gallardo, R, Radford, S.E, Ranson, N.A. | 登録日 | 2022-09-05 | 公開日 | 2024-01-10 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Structural evolution of fibril polymorphs during amyloid assembly. Cell, 186, 2023
|
|
4A2H
| Crystal Structure of Laccase from Coriolopsis gallica pH 7.0 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, COPPER (II) ION, ... | 著者 | De La Mora, E, Valderrama, B, Horjales, E, Rudino-Pinera, E. | 登録日 | 2011-09-27 | 公開日 | 2011-10-12 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural Changes Caused by Radiation-Induced Reduction and Radiolysis: The Effect of X-Ray Absorbed Dose in a Fungal Multicopper Oxidase Acta Crystallogr.,Sect.D, 68, 2012
|
|
6PAZ
| OXIDIZED MUTANT P80I PSEUDOAZURIN FROM A. FAECALIS | 分子名称: | COPPER (II) ION, PSEUDOAZURIN | 著者 | Adman, E.T, Libeu, C.A.P. | 登録日 | 1997-02-21 | 公開日 | 1997-08-20 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | Site-directed mutants of pseudoazurin: explanation of increased redox potentials from X-ray structures and from calculation of redox potential differences. Biochemistry, 36, 1997
|
|
4IAR
| Crystal structure of the chimeric protein of 5-HT1B-BRIL in complex with ergotamine (PSI Community Target) | 分子名称: | (2S)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Chimera protein of human 5-hydroxytryptamine receptor 1B and E. Coli soluble cytochrome b562, Ergotamine | 著者 | Wang, C, Jiang, Y, Ma, J, Wu, H, Wacker, D, Katritch, V, Han, G.W, Liu, W, Huang, X, Vardy, E, McCorvy, J.D, Gao, X, Zhou, E.X, Melcher, K, Zhang, C, Bai, F, Yang, H, Yang, L, Jiang, H, Roth, B.L, Cherezov, V, Stevens, R.C, Xu, H.E, GPCR Network (GPCR) | 登録日 | 2012-12-07 | 公開日 | 2013-03-13 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural basis for molecular recognition at serotonin receptors. Science, 340, 2013
|
|
6XQ9
| Receptor for Advanced Glycation End Products VC1 domain in complex with Fragments 1 & 13 | 分子名称: | 4-(3-hydroxyphenoxy)benzoic acid, 7-methyl-3-phenyl-1H-indole-2-carboxylic acid, ACETATE ION, ... | 著者 | Salay, L.E, Kozlyuk, N, Gilston, B.A, Gogliotti, R.D, Christov, P.P, Kim, K, Ovee, M, Waterson, A.G, Chazin, W.J. | 登録日 | 2020-07-09 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | A fragment-based approach to discovery of Receptor for Advanced Glycation End products inhibitors. Proteins, 89, 2021
|
|
6PCL
| Crystal structure of human diphosphoinositol polyphosphate phosphohydrolase 1 in complex with 5-IP7 | 分子名称: | (1r,2R,3S,4s,5R,6S)-2,3,4,5,6-pentakis(phosphonooxy)cyclohexyl trihydrogen diphosphate, CHLORIDE ION, Diphosphoinositol polyphosphate phosphohydrolase 1, ... | 著者 | Dollins, D.E, Neubauer, J, Dong, J, York, J.D. | 登録日 | 2019-06-17 | 公開日 | 2020-04-29 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Vip1 is a kinase and pyrophosphatase switch that regulates inositol diphosphate signaling. Proc.Natl.Acad.Sci.USA, 117, 2020
|
|
7H2L
| PanDDA analysis group deposition -- Crystal Structure of ZIKV NS2B-NS3 protease in complex with Z19755216 | 分子名称: | 2-(3-fluorophenoxy)-N,N-dimethylacetamide, DIMETHYL SULFOXIDE, Serine protease NS3, ... | 著者 | Ni, X, Godoy, A.S, Marples, P.G, Fairhead, M, Balcomb, B.H, Tomlinson, C.W.E, Koekemoer, L, Aschenbrenner, J.C, Lithgo, R.M, Thompson, W, Wild, C, Williams, E.P, Winokan, M, Chandran, A.V, Fearon, D, Walsh, M.A, von Delft, F. | 登録日 | 2024-04-03 | 公開日 | 2024-05-08 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.366 Å) | 主引用文献 | PanDDA analysis group deposition of ZIKV NS2B-NS3 protease To Be Published
|
|
6XST
| |
7H2E
| PanDDA analysis group deposition -- Crystal Structure of ZIKV NS2B-NS3 protease in complex with Z1428159350 | 分子名称: | (1S)-1-(1-phenyl-1H-1,2,3-triazol-4-yl)ethan-1-amine, DIMETHYL SULFOXIDE, Serine protease NS3, ... | 著者 | Ni, X, Godoy, A.S, Marples, P.G, Fairhead, M, Balcomb, B.H, Tomlinson, C.W.E, Koekemoer, L, Aschenbrenner, J.C, Lithgo, R.M, Thompson, W, Wild, C, Williams, E.P, Winokan, M, Chandran, A.V, Fearon, D, Walsh, M.A, von Delft, F. | 登録日 | 2024-04-03 | 公開日 | 2024-05-08 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.36 Å) | 主引用文献 | PanDDA analysis group deposition of ZIKV NS2B-NS3 protease To Be Published
|
|
4EB7
| A. fulgidus IscS-IscU complex structure | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, FE2/S2 (INORGANIC) CLUSTER, GLYCEROL, ... | 著者 | Marinoni, E.N, de Oliveira, J.S, Nicolet, Y, Raulfs, E.C, Amara, P, Dean, D.R, Fontecilla-Camps, J.C. | 登録日 | 2012-03-23 | 公開日 | 2012-05-02 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | (IscS-IscU)2 complex structures provide insights into Fe2S2 biogenesis and transfer. Angew.Chem.Int.Ed.Engl., 51, 2012
|
|
8AM3
| |
8AM8
| |
6XQ1
| Receptor for Advanced Glycation End Products VC1 domain in complex with 3-(3-((4-(4-carboxyphenoxy)benzyl)oxy)phenyl)-1H-indole-2-carboxylic acid | 分子名称: | 3-[3-({[3-(4-carboxyphenoxy)phenyl]methoxy}methyl)phenyl]-1H-indole-2-carboxylic acid, ACETATE ION, Advanced glycosylation end product-specific receptor, ... | 著者 | Salay, L.E, Kozlyuk, N, Gilston, B.A, Gogliotti, R.D, Christov, P.P, Kim, K, Ovee, M, Waterson, A.G, Chazin, W.J. | 登録日 | 2020-07-09 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.51 Å) | 主引用文献 | A fragment-based approach to discovery of Receptor for Advanced Glycation End products inhibitors. Proteins, 89, 2021
|
|
3GLS
| Crystal Structure of Human SIRT3 | 分子名称: | NAD-dependent deacetylase sirtuin-3, mitochondrial, SULFATE ION, ... | 著者 | Jin, L, Wei, W, Jiang, Y, Peng, H, Cai, J, Mao, C, Dai, H, Bemis, J.E, Jirousek, M.R, Milne, J.C, Westphal, C.H, Perni, R.B. | 登録日 | 2009-03-12 | 公開日 | 2009-06-16 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal Structures of Human SIRT3 Displaying Substrate-induced Conformational Changes. J.Biol.Chem., 284, 2009
|
|
6X6X
| |
8AM6
| |
4EGA
| Trypanosoma brucei methionyl-tRNA synthetase in complex with inhibitor Chem 1320 | 分子名称: | 2-({3-[(3,5-dibromo-2-methoxybenzyl)amino]propyl}amino)quinolin-4(1H)-one, DIMETHYL SULFOXIDE, GLYCEROL, ... | 著者 | Koh, C.Y, Kim, J.E, Shibata, S, Fan, E, Verlinde, C.L.M.J, Hol, W.G.J. | 登録日 | 2012-03-30 | 公開日 | 2012-09-12 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.698 Å) | 主引用文献 | Distinct States of Methionyl-tRNA Synthetase Indicate Inhibitor Binding by Conformational Selection. Structure, 20, 2012
|
|
6P42
| |