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PDB: 175 件

1SXH
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apo structure of B. megaterium transcription regulator
分子名称: Glucose-resistance amylase regulator
著者Schumacher, M.A, Allen, G.S, Diel, M, Seidel, G, Hillen, W, Brennan, R.G.
登録日2004-03-30
公開日2004-10-19
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Structural studies on the apo transcription factor form B. megaterium
Cell(Cambridge,Mass.), 118, 2004
1UPF
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STRUCTURE OF THE URACIL PHOSPHORIBOSYLTRANSFERASE, MUTANT C128V BOUND TO THE DRUG 5-FLUOROURACIL
分子名称: 5-FLUOROURACIL, SULFATE ION, URACIL PHOSPHORIBOSYLTRANSFERASE
著者Schumacher, M.A, Carter, D, Scott, D, Roos, D, Ullman, B, Brennan, R.G.
登録日1998-06-17
公開日1999-06-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structures of Toxoplasma gondii uracil phosphoribosyltransferase reveal the atomic basis of pyrimidine discrimination and prodrug binding.
EMBO J., 17, 1998
1UPU
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STRUCTURE OF THE URACIL PHOSPHORIBOSYLTRANSFERASE, MUTANT C128V, BOUND TO PRODUCT URIDINE-1-MONOPHOSPHATE (UMP)
分子名称: PHOSPHATE ION, URACIL PHOSPHORIBOSYLTRANSFERASE, URIDINE-5'-MONOPHOSPHATE
著者Schumacher, M.A, Carter, D, Scott, D, Roos, D, Ullman, B, Brennan, R.G.
登録日1998-04-16
公開日1999-05-11
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structures of Toxoplasma gondii uracil phosphoribosyltransferase reveal the atomic basis of pyrimidine discrimination and prodrug binding.
EMBO J., 17, 1998
1VPW
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STRUCTURE OF THE PURR MUTANT, L54M, BOUND TO HYPOXANTHINE AND PURF OPERATOR DNA
分子名称: DNA (5'-D(*TP*AP*CP*GP*CP*AP*AP*AP*CP*GP*TP*TP*TP*GP*CP*GP*T )-3'), HYPOXANTHINE, PURINE REPRESSOR
著者Arvidson, D.N, Lu, F, Faber, C, Zalkin, H, Brennan, R.G.
登録日1998-02-27
公開日1998-06-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The structure of PurR mutant L54M shows an alternative route to DNA kinking.
Nat.Struct.Biol., 5, 1998
1SDL
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BU of 1sdl by Molmil
CROSS-LINKED, CARBONMONOXY HEMOGLOBIN A
分子名称: 1,3,5-BENZENETRICARBOXYLIC ACID, CARBON MONOXIDE, HEMOGLOBIN A, ...
著者Schumacher, M.A, Dixon, M.M, Kluger, R, Jones, R.T, Brennan, R.G.
登録日1996-02-26
公開日1996-08-01
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Allosteric transition intermediates modelled by crosslinked haemoglobins.
Nature, 375, 1995
1BOW
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BU of 1bow by Molmil
MULTIDRUG-BINDING DOMAIN OF TRANSCRIPTION ACTIVATOR BMRR (APO FORM)
分子名称: MANGANESE (II) ION, MULTIDRUG-EFFLUX TRANSPORTER 1 REGULATOR BMRR
著者Zheleznova, E.E, Markham, P.N, Neyfakh, A.A, Brennan, R.G.
登録日1998-08-06
公開日1999-08-06
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural basis of multidrug recognition by BmrR, a transcription activator of a multidrug transporter.
Cell(Cambridge,Mass.), 96, 1999
1BD4
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UPRT-URACIL COMPLEX
分子名称: PHOSPHATE ION, URACIL, URACIL PHOSPHORIBOSYLTRANSFERASE
著者Schumacher, M.A, Carter, D, Scott, D, Roos, D, Ullman, B, Brennan, R.G.
登録日1998-05-12
公開日1999-05-18
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structures of Toxoplasma gondii uracil phosphoribosyltransferase reveal the atomic basis of pyrimidine discrimination and prodrug binding.
EMBO J., 17, 1998
1DH3
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BU of 1dh3 by Molmil
CRYSTAL STRUCTURE OF A CREB BZIP-CRE COMPLEX REVEALS THE BASIS FOR CREB FAIMLY SELECTIVE DIMERIZATION AND DNA BINDING
分子名称: DNA (5'-D(*CP*CP*TP*TP*GP*GP*CP*TP*GP*AP*CP*GP*TP*CP*AP*GP*CP*CP*AP*AP*G)-3'), MAGNESIUM ION, TRANSCRIPTION FACTOR CREB
著者Schumacher, M.A, Goodman, R.H, Brennan, R.G.
登録日1999-11-27
公開日2000-11-27
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献The structure of a CREB bZIP.somatostatin CRE complex reveals the basis for selective dimerization and divalent cation-enhanced DNA binding
J.Biol.Chem., 275, 2000
1DBR
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HYPOXANTHINE GUANINE XANTHINE
分子名称: HYPOXANTHINE GUANINE XANTHINE PHOSPHORIBOSYLTRANSFERASE, MAGNESIUM ION
著者Schumacher, M.A, Carter, D, Roos, D, Ullman, B, Brennan, R.G.
登録日1996-02-13
公開日1997-12-03
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structures of Toxoplasma gondii HGXPRTase reveal the catalytic role of a long flexible loop.
Nat.Struct.Biol., 3, 1996
1BD3
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STRUCTURE OF THE APO URACIL PHOSPHORIBOSYLTRANSFERASE, 2 MUTANT C128V
分子名称: PHOSPHATE ION, URACIL PHOSPHORIBOSYLTRANSFERASE
著者Schumacher, M.A, Carter, D, Scott, D, Roos, D, Ullman, B, Brennan, R.G.
登録日1998-05-12
公開日1999-05-18
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Crystal structures of Toxoplasma gondii uracil phosphoribosyltransferase reveal the atomic basis of pyrimidine discrimination and prodrug binding.
EMBO J., 17, 1998
1DBQ
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BU of 1dbq by Molmil
DNA-BINDING REGULATORY PROTEIN
分子名称: MAGNESIUM ION, PURINE REPRESSOR
著者Schumacher, M.A, Choi, K.Y, Lu, F, Zalkin, H, Brennan, R.G.
登録日1996-02-13
公開日1996-12-07
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Mechanism of corepressor-mediated specific DNA binding by the purine repressor.
Cell(Cambridge,Mass.), 83, 1995
1ON1
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BU of 1on1 by Molmil
Bacillus Subtilis Manganese Transport Regulator (Mntr) Bound To Manganese, AB Conformation.
分子名称: MANGANESE (II) ION, Transcriptional regulator mntR
著者Glasfeld, A, Guedon, E, Helmann, J.D, Brennan, R.G.
登録日2003-02-26
公開日2003-07-15
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Structure of the Manganese-Bound Manganese Transport Regulator of Bacillus subtilis
Nat.Struct.Biol., 10, 2003
1ON2
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Bacillus subtilis Manganese Transport Regulator (MntR), D8M Mutant, Bound to Manganese
分子名称: MANGANESE (II) ION, Transcriptional regulator mntR
著者Glasfeld, A, Guedon, E, Helmann, J.D, Brennan, R.G.
登録日2003-02-26
公開日2003-07-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Structure of the Manganese-Bound Manganese Transport Regulator of Bacillus subtilis
Nat.Struct.Biol., 10, 2003
1QB7
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CRYSTAL STRUCTURES OF ADENINE PHOSPHORIBOSYLTRANSFERASE FROM LEISHMANIA DONOVANI.
分子名称: ADENINE, ADENINE PHOSPHORIBOSYLTRANSFERASE, CITRIC ACID, ...
著者Phillips, C.L, Ullman, B, Brennan, R.G, Hill, C.P.
登録日1999-04-30
公開日1999-07-21
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal structures of adenine phosphoribosyltransferase from Leishmania donovani.
EMBO J., 18, 1999
1QVU
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BU of 1qvu by Molmil
Crystal structure of the multidrug binding transcriptional repressor QacR bound to two drugs: ethidium and proflavine
分子名称: ETHIDIUM, PROFLAVIN, Transcriptional regulator qacR
著者Schumacher, M.A, Miller, M.C, Brennan, R.G.
登録日2003-08-28
公開日2004-08-03
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.96 Å)
主引用文献Structural mechanism of the simultaneous binding of two drugs to a multidrug-binding protein
Embo J., 23, 2004
1QVT
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BU of 1qvt by Molmil
CRYSTAL STRUCTURE OF THE MULTIDRUG BINDING TRANSCRIPTIONAL REPRESSOR QACR BOUND TO THE DRUG PROFLAVINE
分子名称: PROFLAVIN, SULFATE ION, Transcriptional regulator qacR
著者Schumacher, M.A, Miller, M.C, Brennan, R.G.
登録日2003-08-28
公開日2004-08-03
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.89 Å)
主引用文献Structural mechanism of the simultaneous binding of two drugs to a multidrug-binding protein
Embo J., 23, 2004
1QCC
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BU of 1qcc by Molmil
CRYSTAL STRUCTURES OF ADENINE PHOSPHORIBOSYLTRANSFERASE FROM LEISHMANIA DONOVANI
分子名称: ADENINE PHOSPHORIBOSYLTRANSFERASE, CITRIC ACID
著者Phillips, C.L, Ullman, B, Brennan, R.G, Hill, C.P.
登録日1999-05-01
公開日1999-07-21
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献Crystal structures of adenine phosphoribosyltransferase from Leishmania donovani.
EMBO J., 18, 1999
1PNR
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PURINE REPRESSOR-HYPOXANTHINE-PURF-OPERATOR COMPLEX
分子名称: DNA (5'-D(*AP*AP*CP*GP*AP*AP*AP*AP*CP*GP*TP*TP*TP*TP*CP*GP*T )-3'), HYPOXANTHINE, PROTEIN (PURINE REPRESSOR)
著者Schumacher, M.A, Choi, K.Y, Zalkin, H, Brennan, R.G.
登録日1995-03-29
公開日1995-11-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of LacI member, PurR, bound to DNA: minor groove binding by alpha helices.
Science, 266, 1994
1QCD
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BU of 1qcd by Molmil
CRYSTAL STRUCTURES OF ADENINE PHOSPHORIBOSYLTRANSFERASE FROM LEISHMANIA DONOVANI
分子名称: ADENINE PHOSPHORIBOSYLTRANSFERASE, SULFATE ION
著者Phillips, C.L, Ullman, B, Brennan, R.G, Hill, C.P.
登録日1999-05-01
公開日1999-07-21
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.48 Å)
主引用文献Crystal structures of adenine phosphoribosyltransferase from Leishmania donovani.
EMBO J., 18, 1999
4LD5
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Crystal structure of MepR Q18P mutant from multidrug resistant S. aureus clinical isolate
分子名称: MepR, SULFATE ION
著者Birukou, I, Brennan, R.G.
登録日2013-06-24
公開日2013-09-11
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The molecular mechanisms of allosteric mutations impairing MepR repressor function in multidrug-resistant strains of Staphylococcus aureus.
MBio, 4, 2013
4L9J
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BU of 4l9j by Molmil
Crystal structure of S. aureus MepR in DNA-binding conformation
分子名称: MepR
著者Birukou, I, Brennan, R.G.
登録日2013-06-18
公開日2013-09-11
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (3.45 Å)
主引用文献The molecular mechanisms of allosteric mutations impairing MepR repressor function in multidrug-resistant strains of Staphylococcus aureus.
MBio, 4, 2013
4L9T
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Crystal structure of MepR F27L mutant from multidrug resistant S. aureus clinical isolate
分子名称: MepR, SULFATE ION
著者Birukou, I, Brennan, R.G.
登録日2013-06-18
公開日2013-09-11
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.794 Å)
主引用文献The molecular mechanisms of allosteric mutations impairing MepR repressor function in multidrug-resistant strains of Staphylococcus aureus.
MBio, 4, 2013
4LLN
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Crystal structure of S. aureus MepR-DNA complex
分子名称: MepR, Palindromized mepR operator sequence
著者Birukou, I, Brennan, R.G.
登録日2013-07-09
公開日2014-05-14
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.842 Å)
主引用文献Structural mechanism of transcription regulation of the Staphylococcus aureus multidrug efflux operon mepRA by the MarR family repressor MepR.
Nucleic Acids Res., 42, 2014
4L9N
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Crystal structure of MepR A103V mutant from multidrug resistant S. aureus clinical isolate
分子名称: MepR, SULFATE ION
著者Birukou, I, Brennan, R.G.
登録日2013-06-18
公開日2013-09-11
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献The molecular mechanisms of allosteric mutations impairing MepR repressor function in multidrug-resistant strains of Staphylococcus aureus.
MBio, 4, 2013
4LLL
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Crystal structure of S. aureus MepR-DNA complex
分子名称: MepR, Palindromized mepR operator sequence
著者Birukou, I, Brennan, R.G.
登録日2013-07-09
公開日2014-05-14
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.036 Å)
主引用文献Structural mechanism of transcription regulation of the Staphylococcus aureus multidrug efflux operon mepRA by the MarR family repressor MepR.
Nucleic Acids Res., 42, 2014

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