8UIW
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![BU of 8uiw by Molmil](/molmil-images/mine/8uiw) | yjdF riboswitch from R. gauvreauii in complex with chelerythrine bound to Fab BL3-6 S97N | 分子名称: | 1,2-dimethoxy-12-methyl[1,3]benzodioxolo[5,6-c]phenanthridin-12-ium, Fab BL3-6 S97N heavy chain, Fab BL3-6 S97N light chain, ... | 著者 | Krochmal, D, Lewicka, A, Piccirilli, J.A. | 登録日 | 2023-10-10 | 公開日 | 2024-04-10 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.77 Å) | 主引用文献 | Structural basis for promiscuity in ligand recognition by yjdF riboswitch. Cell Discov, 10, 2024
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7B7Z
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7O2X
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![BU of 7o2x by Molmil](/molmil-images/mine/7o2x) | Crystal structure of the human METTL3-METTL14 complex with compound T180 | 分子名称: | ACETATE ION, N-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-4-oxidanylidene-pyrido[1,2-a]pyrimidine-2-carboxamide, N6-adenosine-methyltransferase catalytic subunit, ... | 著者 | Bedi, R.K, Huang, D, Caflisch, A. | 登録日 | 2021-03-31 | 公開日 | 2021-04-07 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structure of the human METTL3-METTL14 complex with compound T180 To Be Published
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7B80
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![BU of 7b80 by Molmil](/molmil-images/mine/7b80) | DeAMPylation complex of monomeric FICD and AMPylated BiP (state 2) | 分子名称: | 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, ADENOSINE MONOPHOSPHATE, DI(HYDROXYETHYL)ETHER, ... | 著者 | Perera, L.A, Ron, D. | 登録日 | 2020-12-12 | 公開日 | 2021-07-07 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Structures of a deAMPylation complex rationalise the switch between antagonistic catalytic activities of FICD. Nat Commun, 12, 2021
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8D53
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7RAY
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![BU of 7ray by Molmil](/molmil-images/mine/7ray) | Crystal structure of MBD2 with DNA | 分子名称: | DNA (5'-D(*GP*CP*CP*AP*A)-R(P*(5MC))-D(P*GP*TP*TP*GP*GP*C)-3'), Methyl-CpG-binding domain protein 2, UNKNOWN ATOM OR ION | 著者 | Liu, K, Dong, A, Loppnau, P, Edwards, A.M, Arrowsmith, C.H, Min, J, Structural Genomics Consortium (SGC) | 登録日 | 2021-07-05 | 公開日 | 2021-07-21 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Crystal structure of MBD2 with DNA To Be Published
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8DP5
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![BU of 8dp5 by Molmil](/molmil-images/mine/8dp5) | Structure of the PEAK3/14-3-3 complex | 分子名称: | 14-3-3 protein beta/alpha, 14-3-3 protein epsilon, Protein PEAK3, ... | 著者 | Torosyan, H, Paul, M, Jura, N, Verba, K.A. | 登録日 | 2022-07-14 | 公開日 | 2023-06-28 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structural insights into regulation of the PEAK3 pseudokinase scaffold by 14-3-3. Nat Commun, 14, 2023
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8EEW
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![BU of 8eew by Molmil](/molmil-images/mine/8eew) | CryoEM of the soluble OPA1 dimer from the GDP-AlFx bound helical assembly on a lipid membrane | 分子名称: | Dynamin-like 120 kDa protein, form S1, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Nyenhuis, S.B, Wu, X, Stanton, A.E, Strub, M.P, Yim, Y.I, Canagarajah, B, Hinshaw, J.E. | 登録日 | 2022-09-07 | 公開日 | 2023-06-28 | 最終更新日 | 2023-09-13 | 実験手法 | ELECTRON MICROSCOPY (5.48 Å) | 主引用文献 | OPA1 helical structures give perspective to mitochondrial dysfunction. Nature, 620, 2023
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8EFF
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![BU of 8eff by Molmil](/molmil-images/mine/8eff) | CryoEM of the soluble OPA1 tetramer from the GDP-AlFx bound helical assembly on a lipid membrane | 分子名称: | Dynamin-like 120 kDa protein, form S1, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Nyenhuis, S.B, Wu, X, Stanton, A.E, Strub, M.P, Yim, Y.I, Canagarajah, B, Hinshaw, J.E. | 登録日 | 2022-09-08 | 公開日 | 2023-06-28 | 最終更新日 | 2023-09-13 | 実験手法 | ELECTRON MICROSCOPY (5.48 Å) | 主引用文献 | OPA1 helical structures give perspective to mitochondrial dysfunction. Nature, 620, 2023
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6NX7
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6NXE
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5N8C
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![BU of 5n8c by Molmil](/molmil-images/mine/5n8c) | Crystal structure of Pseudomonas aeruginosa LpxC complexed with inhibitor | 分子名称: | (2~{S})-3-azanyl-2-[[(1~{R})-5-[2-[4-[[2-(hydroxymethyl)imidazol-1-yl]methyl]phenyl]ethynyl]-2,3-dihydro-1~{H}-inden-1-yl]amino]-3-methyl-~{N}-oxidanyl-butanamide, CHLORIDE ION, UDP-3-O-acyl-N-acetylglucosamine deacetylase, ... | 著者 | Cross, J.B, Ryan, M.D, Zhang, J, Cheng, R.K, Wood, M, Andersen, O.A, Brooks, M, Kwong, J, Barker, J. | 登録日 | 2017-02-23 | 公開日 | 2017-03-29 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-based discovery of LpxC inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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8EF7
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![BU of 8ef7 by Molmil](/molmil-images/mine/8ef7) | CryoEM of the soluble OPA1 dimer from the apo helical assembly on a lipid membrane | 分子名称: | Dynamin-like 120 kDa protein, form S1 | 著者 | Nyenhuis, S.B, Wu, X, Stanton, A.E, Strub, M.P, Yim, Y.I, Canagarajah, B, Hinshaw, J.E. | 登録日 | 2022-09-08 | 公開日 | 2023-06-28 | 最終更新日 | 2023-09-13 | 実験手法 | ELECTRON MICROSCOPY (9.68 Å) | 主引用文献 | OPA1 helical structures give perspective to mitochondrial dysfunction. Nature, 620, 2023
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6NWQ
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![BU of 6nwq by Molmil](/molmil-images/mine/6nwq) | Chronic traumatic encephalopathy Type II Tau filament | 分子名称: | Microtubule-associated protein tau | 著者 | Falcon, B, Zivanov, J, Zhang, W, Murzin, A.G, Garringer, H.J, Vidal, R, Crowther, R.A, Newell, K.L, Ghetti, B, Goedert, M, Scheres, H.W. | 登録日 | 2019-02-07 | 公開日 | 2019-03-27 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Novel tau filament fold in chronic traumatic encephalopathy encloses hydrophobic molecules. Nature, 568, 2019
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7BF1
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![BU of 7bf1 by Molmil](/molmil-images/mine/7bf1) | Ca2+-Calmodulin in complex with peptide from brain-type creatine kinase in extended 1:2 binding mode | 分子名称: | ACETYL GROUP, CALCIUM ION, Calmodulin-1, ... | 著者 | Sprenger, J, Akerfeldt, K.S, Bredfelt, J, Patel, N, Rowlett, R, Trifan, A, Vanderbeck, A, Lo Leggio, L, Snogerup Linse, S. | 登録日 | 2020-12-31 | 公開日 | 2021-07-21 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.24 Å) | 主引用文献 | Calmodulin complexes with brain and muscle creatine kinase peptides. Curr Res Struct Biol, 3, 2021
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6QKI
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![BU of 6qki by Molmil](/molmil-images/mine/6qki) | Native structure of EgtB from Chloracidobacterium thermophilum, a type II sulfoxide synthase | 分子名称: | FE (III) ION, Uncharacterized protein | 著者 | Stampfli, A.R, Badri, B.N, Schirmer, T, Seebeck, F.P. | 登録日 | 2019-01-29 | 公開日 | 2019-03-27 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2.04 Å) | 主引用文献 | An Alternative Active Site Architecture for O2Activation in the Ergothioneine Biosynthetic EgtB from Chloracidobacterium thermophilum. J.Am.Chem.Soc., 141, 2019
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7BF2
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![BU of 7bf2 by Molmil](/molmil-images/mine/7bf2) | Ca2+-Calmodulin in complex with human muscle form creatine kinase peptide in extended 1:2 binding mode | 分子名称: | CALCIUM ION, Calmodulin-1, Creatine kinase M-type | 著者 | Sprenger, J, Akerfeldt, K.S, Bredfelt, J, Patel, N, Rowlett, R, Trifan, A, Vanderbeck, A, Lo Leggio, L, Snogerup Linse, S. | 登録日 | 2020-12-31 | 公開日 | 2021-07-21 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.43 Å) | 主引用文献 | Calmodulin complexes with brain and muscle creatine kinase peptides. Curr Res Struct Biol, 3, 2021
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8F9Q
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![BU of 8f9q by Molmil](/molmil-images/mine/8f9q) | Guinea pig sialic acid esterase (SIAE) | 分子名称: | Sialic acid acetylesterase, alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Ide, D, Gorelik, A, Illes, K, Nagar, B. | 登録日 | 2022-11-24 | 公開日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.76 Å) | 主引用文献 | Guinea pig sialic acid esterase (SIAE) To Be Published
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7O85
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![BU of 7o85 by Molmil](/molmil-images/mine/7o85) | Anthrax toxin prepore in complex with the neutralizing Fab cAb29 | 分子名称: | CALCIUM ION, Fab, Protective antigen PA-63 | 著者 | Hoelzgen, F, Zalk, R, Alcalay, R, Cohen-Schwartz, S, Garau, G, Shahar, A, Mazor, O, Frank, G.A. | 登録日 | 2021-04-14 | 公開日 | 2021-04-28 | 最終更新日 | 2021-09-29 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Neutralization of the anthrax toxin by antibody-mediated stapling of its membrane-penetrating loop. Acta Crystallogr D Struct Biol, 77, 2021
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7NSB
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![BU of 7nsb by Molmil](/molmil-images/mine/7nsb) | Supramolecular assembly module of yeast Chelator-GID SR4 E3 ubiquitin ligase | 分子名称: | Glucose-induced degradation protein 7, Glucose-induced degradation protein 8, Vacuolar import and degradation protein 30 | 著者 | Chrustowicz, J, Sherpa, D, Prabu, J.R, Schulman, B.A. | 登録日 | 2021-03-05 | 公開日 | 2021-05-05 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | GID E3 ligase supramolecular chelate assembly configures multipronged ubiquitin targeting of an oligomeric metabolic enzyme. Mol.Cell, 81, 2021
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6NY7
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![BU of 6ny7 by Molmil](/molmil-images/mine/6ny7) | Crystal Structure of NDM-1 D199N with Compound 16 | 分子名称: | Carbapenem Hydrolyzing Class B Metallo beta lactamase NDM-1, ZINC ION, [(5,7-dibromo-2-oxo-1,2-dihydroquinolin-4-yl)methyl]phosphonic acid | 著者 | Akhtar, A, Chen, Y. | 登録日 | 2019-02-11 | 公開日 | 2019-09-25 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Heteroaryl Phosphonates as Noncovalent Inhibitors of Both Serine- and Metallocarbapenemases. J.Med.Chem., 62, 2019
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7RJ1
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![BU of 7rj1 by Molmil](/molmil-images/mine/7rj1) | Crystal structure of Aro7p chorismate mutase from Candida albicans, complex with L-Trp | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Chorismate mutase, ... | 著者 | Stogios, P.J, Evdokimova, E, Tan, K, Di Leo, R, Savchenko, A, Joachimiak, A, Satchell, K.J.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2021-07-20 | 公開日 | 2021-07-28 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Crystal structure of Aro7p chorismate mutase from Candida albicans, complex with L-Trp To Be Published
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8F9R
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![BU of 8f9r by Molmil](/molmil-images/mine/8f9r) | Rabbit sialic acid esterase (SIAE) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Sialic acid acetylesterase, ... | 著者 | Ide, D, Gorelik, A, Illes, K, Nagar, B. | 登録日 | 2022-11-24 | 公開日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.97 Å) | 主引用文献 | Rabbit sialic acid esterase (SIAE) To Be Published
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7NS3
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![BU of 7ns3 by Molmil](/molmil-images/mine/7ns3) | Substrate receptor scaffolding module of yeast Chelator-GID SR4 E3 ubiquitin ligase bound to Fbp1 substrate | 分子名称: | BJ4_G0018240.mRNA.1.CDS.1, Fructose-bisphosphatase, Glucose-induced degradation protein 8, ... | 著者 | Sherpa, D, Chrustowicz, J, Prabu, J.R, Schulman, B.A. | 登録日 | 2021-03-05 | 公開日 | 2021-05-05 | 最終更新日 | 2021-07-07 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | GID E3 ligase supramolecular chelate assembly configures multipronged ubiquitin targeting of an oligomeric metabolic enzyme. Mol.Cell, 81, 2021
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6Q7B
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![BU of 6q7b by Molmil](/molmil-images/mine/6q7b) | Crystal Structure of Ephrin A2 (EphA2) Receptor Protein Kinase with the NVP-BHG712 derivative ATDL09 | 分子名称: | 3-[[4-imidazol-1-yl-6-[(3~{S})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{N}-[3-(trifluoromethyl)phenyl]benzamide, Ephrin type-A receptor 2 | 著者 | Kudlinzki, D, Troester, A, Witt, K, Linhard, V.L, Gande, S.L, Saxena, K, Schwalbe, H. | 登録日 | 2018-12-13 | 公開日 | 2020-01-15 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.009 Å) | 主引用文献 | Effects of NVP-BHG712 chemical modifications on EPHA2 binding and affinity To Be Published
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