3TPJ
| APO structure of BACE1 | 分子名称: | Beta-secretase 1, CHLORIDE ION, SULFATE ION, ... | 著者 | Xu, Y.C, Li, M.J, Greenblatt, H, Chen, T.T, Silman, I, Sussman, J.L. | 登録日 | 2011-09-08 | 公開日 | 2011-11-23 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.61 Å) | 主引用文献 | Flexibility of the flap in the active site of BACE1 as revealed by crystal structures and molecular dynamics simulations Acta Crystallogr.,Sect.D, 68, 2012
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3TPR
| Crystal structure of BACE1 complexed with an inhibitor | 分子名称: | Beta-secretase 1, CHLORIDE ION, N-[(1S,2R)-1-BENZYL-3-(CYCLOPROPYLAMINO)-2-HYDROXYPROPYL]-5-[METHYL(METHYLSULFONYL)AMINO]-N'-[(1R)-1-PHENYLETHYL]ISOPHTHALAMIDE | 著者 | Xu, Y.C, Li, M.J, Greenblatt, H, Chen, T.T, Silman, I, Sussman, J.L. | 登録日 | 2011-09-08 | 公開日 | 2011-11-23 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Flexibility of the flap in the active site of BACE1 as revealed by crystal structures and molecular dynamics simulations Acta Crystallogr.,Sect.D, 68, 2012
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3TPL
| APO Structure of BACE1 | 分子名称: | Beta-secretase 1, CHLORIDE ION, SULFATE ION | 著者 | Xu, Y.C, Li, M.J, Greenblatt, H, Chen, T.T, Silman, I, Sussman, J.L. | 登録日 | 2011-09-08 | 公開日 | 2011-11-23 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Flexibility of the flap in the active site of BACE1 as revealed by crystal structures and molecular dynamics simulations Acta Crystallogr.,Sect.D, 68, 2012
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7KEW
| Bundibugyo virus GP (mucin deleted) bound to antibody Fab BDBV-43 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, BDBV-43 Fab heavy chain, ... | 著者 | Murin, C.D, Ward, A.B. | 登録日 | 2020-10-13 | 公開日 | 2021-04-28 | 実験手法 | ELECTRON MICROSCOPY (4.16 Å) | 主引用文献 | Convergence of a common solution for broad ebolavirus neutralization by glycan cap-directed human antibodies. Cell Rep, 35, 2021
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7KFG
| Antibody Fab BDBV-289 | 分子名称: | Antibody Fab BDBV-289 heavy chain, Antibody Fab BDBV-289 light chain, DI(HYDROXYETHYL)ETHER | 著者 | Murin, C.D, Bruhn, J.F, Ward, A.B. | 登録日 | 2020-10-13 | 公開日 | 2021-04-28 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (3.002 Å) | 主引用文献 | Convergence of a common solution for broad ebolavirus neutralization by glycan cap-directed human antibodies. Cell Rep, 35, 2021
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7KFE
| Bundibugyo virus GP (mucin deleted) bound to antibody Fab BDBV-329 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Antibody BDBV-329 heavy chain, ... | 著者 | Murin, C.D, Ward, A.B. | 登録日 | 2020-10-13 | 公開日 | 2021-04-28 | 実験手法 | ELECTRON MICROSCOPY (6.6 Å) | 主引用文献 | Convergence of a common solution for broad ebolavirus neutralization by glycan cap-directed human antibodies. Cell Rep, 35, 2021
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7KFH
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7KEX
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7KFB
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7KF9
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7KEJ
| BDBV-289 bound to EBOV GPdMuc Makona | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Antibody Fab heavy chain (HC) BDBV-289, Antibody Fab light chain (LC) BDBV-289, ... | 著者 | Murin, C.D, Ward, A.B. | 登録日 | 2020-10-11 | 公開日 | 2021-06-23 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Convergence of a common solution for broad ebolavirus neutralization by glycan cap-directed human antibodies. Cell Rep, 35, 2021
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7LVB
| CHOLERA TOXIN B SUBUNIT WITH ATTACHED SIV EPITOPE | 分子名称: | CHLORIDE ION, Cholera enterotoxin B-subunit,Surface protein gp120, TRIETHYLENE GLYCOL, ... | 著者 | Patskovsky, Y, Cardozo, T.J. | 登録日 | 2021-02-24 | 公開日 | 2022-03-02 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Cholera toxin B scaffolded, focused SIV V2 epitope elicits antibodies that influence the risk of SIV mac251 acquisition in macaques. Front Immunol, 14, 2023
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8HQ6
| KL2 in complex with CRM1-Ran-RanBP1 | 分子名称: | CHLORIDE ION, CRM1 isoform 1, DIMETHYL SULFOXIDE, ... | 著者 | Sun, Q, Jian, L. | 登録日 | 2022-12-13 | 公開日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Discovery of Aminoratjadone Derivatives as Potent Noncovalent CRM1 Inhibitors. J.Med.Chem., 66, 2023
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8HQ3
| KL1 in complex with CRM1-Ran-RanBP1 | 分子名称: | CHLORIDE ION, CRM1 isoform 1, DIMETHYL SULFOXIDE, ... | 著者 | Sun, Q, Jian, L. | 登録日 | 2022-12-13 | 公開日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Discovery of Aminoratjadone Derivatives as Potent Noncovalent CRM1 Inhibitors. J.Med.Chem., 66, 2023
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7XUX
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6KFT
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6MNR
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6MNQ
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6MNS
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6A3A
| MVM NES mutant Nm2 in complex with CRM1-Ran-RanBP1 | 分子名称: | 1,2-ETHANEDIOL, Exportin-1, GLYCEROL, ... | 著者 | Sun, Q, Li, Y. | 登録日 | 2018-06-15 | 公開日 | 2019-06-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor. Int J Nanomedicine, 16, 2021
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6A3E
| MVM NES mutant Nm15 in complex with CRM1-Ran-RanBP1 | 分子名称: | Exportin-1, GTP-binding nuclear protein Ran, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Sun, Q, Li, Y. | 登録日 | 2018-06-15 | 公開日 | 2019-06-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor. Int J Nanomedicine, 16, 2021
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6A3C
| MVM NES mutant Nm12 in complex with CRM1-Ran-RanBP1 | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, Exportin-1, ... | 著者 | Sun, Q, Li, Y. | 登録日 | 2018-06-15 | 公開日 | 2019-06-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor. Int J Nanomedicine, 16, 2021
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6A38
| MVM NS2 NES in complex with CRM1-Ran-RanBP1 | 分子名称: | 1,2-ETHANEDIOL, Exportin-1, GLYCEROL, ... | 著者 | Sun, Q, Li, Y. | 登録日 | 2018-06-15 | 公開日 | 2019-06-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.69 Å) | 主引用文献 | Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor. Int J Nanomedicine, 16, 2021
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6A3B
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7DKL
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