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6CT5
PptT PAP(CoA) 8918 complex
Descriptor:
4'-phosphopantetheinyl transferase, COENZYME A, DIMETHYL SULFOXIDE, ...
Authors:
Mosior, J
,
Sacchettini, J
,
TB Structural Genomics Consortium (TBSGC)
Deposit date:
2018-03-22
Release date:
2019-02-06
Last modified:
2023-10-04
Method:
X-RAY DIFFRACTION (1.759346 Å)
Cite:
Opposing reactions in coenzyme A metabolism sensitizeMycobacterium tuberculosisto enzyme inhibition.
Science, 363, 2019
6UNC
The crystal structure of Phosphopantetheinyl Hydrolase (PptH) from Mycobacterium tuberculosis
Descriptor:
FE (III) ION, MANGANESE (II) ION, Metallophos domain-containing protein
Authors:
Mosior, J.W
,
Sacchettini, J.C
,
TB Structural Genomics Consortium (TBSGC)
Deposit date:
2019-10-11
Release date:
2020-04-22
Method:
X-RAY DIFFRACTION (2.5 Å)
Cite:
Structural insights into phosphopantetheinyl hydrolase PptH from Mycobacterium tuberculosis.
Protein Sci., 29, 2020
7N8L
PptT PAP(CoA) 9016 complex
Descriptor:
4'-phosphopantetheinyl transferase PptT, COENZYME A, DIMETHYL SULFOXIDE, ...
Authors:
Mosior, J.W
,
Sacchettini, J.C
,
TB Structural Genomics Consortium (TBSGC)
Deposit date:
2021-06-15
Release date:
2022-02-02
Last modified:
2023-10-18
Method:
X-RAY DIFFRACTION (2.26 Å)
Cite:
In Vitro and In Vivo Inhibition of the Mycobacterium tuberculosis Phosphopantetheinyl Transferase PptT by Amidinoureas.
J.Med.Chem., 65, 2022
7N8E
PptT PAP(CoA) 9056 complex
Descriptor:
4'-phosphopantetheinyl transferase PptT, COENZYME A, DIMETHYL SULFOXIDE, ...
Authors:
Mosior, J.W
,
Sacchettini, J.C
,
TB Structural Genomics Consortium (TBSGC)
Deposit date:
2021-06-14
Release date:
2022-02-02
Last modified:
2023-10-18
Method:
X-RAY DIFFRACTION (1.74 Å)
Cite:
In Vitro and In Vivo Inhibition of the Mycobacterium tuberculosis Phosphopantetheinyl Transferase PptT by Amidinoureas.
J.Med.Chem., 65, 2022
7N8M
PptT PAP(CoA) 8978B complex
Descriptor:
4'-phosphopantetheinyl transferase PptT, COENZYME A, DIMETHYL SULFOXIDE, ...
Authors:
Mosior, J.W
,
Sacchettini, J.C
,
TB Structural Genomics Consortium (TBSGC)
Deposit date:
2021-06-15
Release date:
2022-02-02
Last modified:
2023-10-18
Method:
X-RAY DIFFRACTION (1.57 Å)
Cite:
In Vitro and In Vivo Inhibition of the Mycobacterium tuberculosis Phosphopantetheinyl Transferase PptT by Amidinoureas.
J.Med.Chem., 65, 2022
8GKF
Phosphopantetheinyl transferase PptT from Mycobacterium tuberculosis in complex with Raltitrexed.
Descriptor:
4'-phosphopantetheinyl transferase PptT, TOMUDEX
Authors:
Krieger, I.V
,
Singh, A
,
Sacchettini, J.C
,
TB Structural Genomics Consortium (TBSGC)
Deposit date:
2023-03-18
Release date:
2024-03-20
Last modified:
2024-03-27
Method:
X-RAY DIFFRACTION (2.45 Å)
Cite:
Redirecting raltitrexed from cancer cell thymidylate synthase to Mycobacterium tuberculosis phosphopantetheinyl transferase.
Sci Adv, 10, 2024
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PDB entries from 2024-10-09