7N8E
PptT PAP(CoA) 9056 complex
Summary for 7N8E
Entry DOI | 10.2210/pdb7n8e/pdb |
Descriptor | 4'-phosphopantetheinyl transferase PptT, COENZYME A, MAGNESIUM ION, ... (6 entities in total) |
Functional Keywords | inhibitor, structural genomics, psi-2, protein structure initiative, tb structural genomics consortium, tbsgc, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Total number of polymer chains | 2 |
Total formula weight | 55748.96 |
Authors | Mosior, J.W.,Sacchettini, J.C.,TB Structural Genomics Consortium (TBSGC) (deposition date: 2021-06-14, release date: 2022-02-02, Last modification date: 2023-10-18) |
Primary citation | Ottavi, S.,Scarry, S.M.,Mosior, J.,Ling, Y.,Roberts, J.,Singh, A.,Zhang, D.,Goullieux, L.,Roubert, C.,Bacque, E.,Lagiakos, H.R.,Vendome, J.,Moraca, F.,Li, K.,Perkowski, A.J.,Ramesh, R.,Bowler, M.M.,Tracy, W.,Feher, V.A.,Sacchettini, J.C.,Gold, B.S.,Nathan, C.F.,Aube, J. In Vitro and In Vivo Inhibition of the Mycobacterium tuberculosis Phosphopantetheinyl Transferase PptT by Amidinoureas. J.Med.Chem., 65:1996-2022, 2022 Cited by PubMed: 35044775DOI: 10.1021/acs.jmedchem.1c01565 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.74 Å) |
Structure validation
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