8IYX
| Cryo-EM structure of the GPR34 receptor in complex with the antagonist YL-365 | 分子名称: | 1-[4-(3-chlorophenyl)phenyl]carbonyl-4-[2-(4-phenylmethoxyphenyl)ethanoylamino]piperidine-4-carboxylic acid, Probable G-protein coupled receptor 34,YL-365 | 著者 | Jia, G.W, Wang, X, Zhang, C.B, Dong, H.H, Su, Z.M. | 登録日 | 2023-04-06 | 公開日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.34 Å) | 主引用文献 | Cryo-EM structures of human GPR34 enable the identification of selective antagonists. Proc.Natl.Acad.Sci.USA, 120, 2023
|
|
5YUD
| Flagellin derivative in complex with the NLR protein NAIP5 | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Baculoviral IAP repeat-containing protein 1e, Phase 2 flagellin,Flagellin | 著者 | Yang, X.R, Yang, F, Wang, W.G, Lin, G.Z. | 登録日 | 2017-11-21 | 公開日 | 2018-01-03 | 最終更新日 | 2024-03-27 | 実験手法 | ELECTRON MICROSCOPY (4.28 Å) | 主引用文献 | Structural basis for specific flagellin recognition by the NLR protein NAIP5. Cell Res., 28, 2018
|
|
3FP9
| |
4Z62
| The plant peptide hormone free receptor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Phytosulfokine receptor 1 | 著者 | Chai, J, Wang, J, Han, Z. | 登録日 | 2015-04-03 | 公開日 | 2016-03-02 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Allosteric receptor activation by the plant peptide hormone phytosulfokine Nature, 525, 2015
|
|
4Z5W
| The plant peptide hormone receptor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Phytosulfokine, ... | 著者 | Chai, J, Wang, J, Han, Z. | 登録日 | 2015-04-03 | 公開日 | 2016-03-02 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Allosteric receptor activation by the plant peptide hormone phytosulfokine Nature, 525, 2015
|
|
4Z61
| The plant peptide hormone receptor complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, PTR-ILE-PTR-THR-GLN, Phytosulfokine receptor 1, ... | 著者 | Chai, J, Wang, J. | 登録日 | 2015-04-03 | 公開日 | 2016-03-02 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Allosteric receptor activation by the plant peptide hormone phytosulfokine Nature, 525, 2015
|
|
4Z64
| the plant peptide hormone receptor complex in arabidopsis | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Phytosulfokine, ... | 著者 | Chai, J, Wang, J, Han, Z. | 登録日 | 2015-04-03 | 公開日 | 2016-03-02 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.659 Å) | 主引用文献 | Allosteric receptor activation by the plant peptide hormone phytosulfokine Nature, 525, 2015
|
|
4Z63
| |
5BOC
| |
3PDF
| Discovery of Novel Cyanamide-Based Inhibitors of Cathepsin C | 分子名称: | 2,5-dibromo-N-{(3R,5S)-1-[(Z)-iminomethyl]-5-methylpyrrolidin-3-yl}benzenesulfonamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Zhao, B, Laine, D. | 登録日 | 2010-10-22 | 公開日 | 2011-10-26 | 最終更新日 | 2023-07-26 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Discovery of novel cyanamide-based inhibitors of cathepsin C. Acs Med.Chem.Lett., 2, 2011
|
|
3MFE
| |
3MKA
| |
3MI0
| Crystal Structure of Mycobacterium Tuberculosis Proteasome at 2.2 A | 分子名称: | (2R,3S,4R)-2-[(S)-(1S)-cyclohex-2-en-1-yl(hydroxy)methyl]-4-ethyl-3-hydroxy-3-methyl-5-oxopyrrolidine-2-carbaldehyde, DIMETHYLFORMAMIDE, Proteasome subunit alpha, ... | 著者 | Li, D, Li, H. | 登録日 | 2010-04-09 | 公開日 | 2010-06-23 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural basis for the assembly and gate closure mechanisms of the Mycobacterium tuberculosis 20S proteasome. Embo J., 2010
|
|
1YO6
| |
1YQ1
| |
5HYX
| Plant peptide hormone receptor RGFR1 in complex with RGF1 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, PTR-SER-ASN-PRO-GLY-HIS-HIS-PRO-HYP-ARG-HIS-ASN, ... | 著者 | Song, W, Han, Z, Chai, J. | 登録日 | 2016-02-02 | 公開日 | 2017-01-11 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.596 Å) | 主引用文献 | Signature motif-guided identification of receptors for peptide hormones essential for root meristem growth Cell Res., 26, 2016
|
|
8IQ1
| Crystal structure of hydrogen sulfide-bound superoxide dismutase in reduced state | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, COPPER (II) ION, ... | 著者 | Zhou, J.H, Huang, W.X, Cheng, R.X, Zhang, P.J, Zhu, Y.C. | 登録日 | 2023-03-15 | 公開日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Hydrogen sulfide functions as a micro-modulator bound at the copper active site of Cu/Zn-SOD to regulate the catalytic activity of the enzyme. Cell Rep, 42, 2023
|
|
8IQ0
| Crystal structure of hydrogen sulfide-bound superoxide dismutase in oxidized state | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, COPPER (II) ION, ... | 著者 | Zhou, J.H, Huang, W.X, Cheng, R.X, Zhang, P.J, Zhu, Y.C. | 登録日 | 2023-03-15 | 公開日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | Hydrogen sulfide functions as a micro-modulator bound at the copper active site of Cu/Zn-SOD to regulate the catalytic activity of the enzyme. Cell Rep, 42, 2023
|
|
5ZMA
| |
6AVO
| Cryo-EM structure of human immunoproteasome with a novel noncompetitive inhibitor that selectively inhibits activated lymphocytes | 分子名称: | N~1~-{2-[([1,1'-biphenyl]-3-carbonyl)amino]ethyl}-N~4~-tert-butyl-N~2~-(3-phenylpropanoyl)-L-aspartamide, Proteasome subunit alpha type-1, Proteasome subunit alpha type-2, ... | 著者 | Li, H, Santos, R, Bai, L. | 登録日 | 2017-09-04 | 公開日 | 2017-12-06 | 最終更新日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Structure of human immunoproteasome with a reversible and noncompetitive inhibitor that selectively inhibits activated lymphocytes. Nat Commun, 8, 2017
|
|
6OCZ
| Crystal Structure of Mycobacterium tuberculosis Proteasome in Complex with Phenylimidazole-based Inhibitor A86 | 分子名称: | CITRIC ACID, DIMETHYLFORMAMIDE, N-{(2S)-1-({(2S)-1-[(2,4-difluorobenzyl)amino]-1-oxopropan-2-yl}amino)-1,4-dioxo-4-[(2R)-2-phenylpyrrolidin-1-yl]butan-2-yl}-5-methyl-1,2-oxazole-3-carboxamide (non-preferred name), ... | 著者 | Hsu, H.C, Li, H. | 登録日 | 2019-03-25 | 公開日 | 2019-10-09 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Selective Phenylimidazole-Based Inhibitors of theMycobacterium tuberculosisProteasome. J.Med.Chem., 62, 2019
|
|
6OCW
| Crystal Structure of Mycobacterium tuberculosis Proteasome in Complex with Phenylimidazole-based Inhibitor A85 | 分子名称: | CITRIC ACID, DIMETHYLFORMAMIDE, N-{(2S)-1-({(2S)-1-[(2,4-difluorobenzyl)amino]-1-oxopropan-2-yl}amino)-4-[(2S)-2-methylpiperidin-1-yl]-1,4-dioxobutan-2-yl}-5-methyl-1,2-oxazole-3-carboxamide (non-preferred name), ... | 著者 | Hsu, H.C, Li, H. | 登録日 | 2019-03-25 | 公開日 | 2019-10-09 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Selective Phenylimidazole-Based Inhibitors of theMycobacterium tuberculosisProteasome. J.Med.Chem., 62, 2019
|
|
6ODE
| |
7F8G
| |
7F8H
| |