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1SKF
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BU of 1skf by Molmil
CRYSTAL STRUCTURE OF THE STREPTOMYCES K15 DD-TRANSPEPTIDASE
分子名称: D-ALANYL-D-ALANINE TRANSPEPTIDASE
著者Fonze, E, Charlier, P.
登録日1998-08-20
公開日1999-08-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The crystal structure of a penicilloyl-serine transferase of intermediate penicillin sensitivity. The DD-transpeptidase of streptomyces K15.
J.Biol.Chem., 274, 1999
1ESI
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BU of 1esi by Molmil
R248L MUTANT OF STREPTOMYCES K15 DD-TRANSPEPTIDASE
分子名称: DD-TRANSPEPTIDASE
著者Fonze, E, Charlier, P.
登録日2000-04-10
公開日2000-05-03
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献DD-TRANSPEPTIDASE
To be Published
1ES5
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BU of 1es5 by Molmil
S216A MUTANT OF STREPTOMYCES K15 DD-TRANSPEPTIDASE
分子名称: DD-TRANSPEPTIDASE
著者Fonze, E, Charlier, P.
登録日2000-04-07
公開日2000-05-03
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献DD-TRANSPEPTIDASE
To be Published
1I2S
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BU of 1i2s by Molmil
BETA-LACTAMASE FROM BACILLUS LICHENIFORMIS BS3
分子名称: BETA-LACTAMASE, CITRIC ACID, SODIUM ION
著者Fonze, E, Vanhove, M, Dive, G, Sauvage, E, Frere, J.M, Charlier, P.
登録日2001-02-12
公開日2002-03-13
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of the Bacillus licheniformis BS3 class A beta-lactamase and of the acyl-enzyme adduct formed with cefoxitin
Biochemistry, 41, 2002
1I2W
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BU of 1i2w by Molmil
BETA-LACTAMASE FROM BACILLUS LICHENIFORMIS BS3 COMPLEXED WITH CEFOXITIN
分子名称: (2R)-5-[(carbamoyloxy)methyl]-2-{(1S)-1-methoxy-2-oxo-1-[(thiophen-2-ylacetyl)amino]ethyl}-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid, BETA-LACTAMASE, CARBAMIC ACID
著者Fonze, E, Vanhove, M, Dive, G, Sauvage, E, Frere, J.M, Charlier, P.
登録日2001-02-12
公開日2002-03-13
最終更新日2018-09-12
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structures of the Bacillus licheniformis BS3 class A beta-lactamase and of the acyl-enzyme adduct formed with cefoxitin
Biochemistry, 41, 2002
1XPB
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BU of 1xpb by Molmil
STRUCTURE OF BETA-LACTAMASE TEM1
分子名称: BETA-LACTAMASE, SULFATE ION
著者Fonze, E, Charlier, P.
登録日1997-01-10
公開日1997-04-01
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献TEM1 beta-lactamase structure solved by molecular replacement and refined structure of the S235A mutant.
Acta Crystallogr.,Sect.D, 51, 1995
1ESU
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BU of 1esu by Molmil
S235A MUTANT OF TEM1 BETA-LACTAMASE
分子名称: BETA-LACTAMASE, SULFATE ION
著者Fonze, E, Charlier, P.
登録日2000-04-11
公開日2000-05-03
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献TEM1 beta-lactamase structure solved by molecular replacement and refined structure of the S235A mutant.
Acta Crystallogr.,Sect.D, 51, 1995
1ES2
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BU of 1es2 by Molmil
S96A mutant of streptomyces K15 DD-transpeptidase
分子名称: DD-TRANSPEPTIDASE
著者Fonze, E, Charlier, P.
登録日2000-04-07
公開日2000-05-03
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Catalytic mechanism of the Streptomyces K15 DD-transpeptidase/penicillin-binding protein probed by site-directed mutagenesis and structural analysis.
Biochemistry, 42, 2003
1ES3
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BU of 1es3 by Molmil
C98A mutant of streptomyces K15 DD-transpeptidase
分子名称: DD-TRANSPEPTIDASE, SODIUM ION
著者Fonze, E, Charlier, P.
登録日2000-04-07
公開日2000-05-03
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Catalytic mechanism of the Streptomyces K15 DD-transpeptidase/penicillin-binding protein probed by site-directed mutagenesis and structural analysis.
Biochemistry, 42, 2003
1ES4
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C98N mutant of streptomyces K15 DD-transpeptidase
分子名称: DD-TRANSPEPTIDASE
著者Fonze, E, Charlier, P.
登録日2000-04-07
公開日2000-05-03
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Catalytic mechanism of the Streptomyces K15 DD-transpeptidase/penicillin-binding protein probed by site-directed mutagenesis and structural analysis.
Biochemistry, 42, 2003
1J9M
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BU of 1j9m by Molmil
K38H mutant of Streptomyces K15 DD-transpeptidase
分子名称: CHLORIDE ION, DD-transpeptidase, SODIUM ION
著者Fonze, E, Rhazi, N, Nguyen-Disteche, M, Charlier, P.
登録日2001-05-28
公開日2001-06-13
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Catalytic mechanism of the Streptomyces K15 DD-transpeptidase/penicillin-binding protein probed by site-directed mutagenesis and structural analysis.
Biochemistry, 42, 2003
2CC1
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Crystal structure of the class A beta-lactamase from Mycobacterium fortuitum
分子名称: Beta-lactamase
著者Sauvage, E, Fonze, E, Charlier, P.
登録日2006-01-11
公開日2006-01-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.13 Å)
主引用文献Crystal structure of the Mycobacterium fortuitum class A beta-lactamase: structural basis for broad substrate specificity.
Antimicrob. Agents Chemother., 50, 2006
2WK0
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BU of 2wk0 by Molmil
Crystal structure of the class A beta-lactamase BS3 inhibited by 6- beta-iodopenicillanate.
分子名称: (3S)-2,2-dimethyl-3,4-dihydro-2H-1,4-thiazine-3,6-dicarboxylic acid, BETA-LACTAMASE, CHLORIDE ION, ...
著者Sauvage, E, Zervosen, A, Dive, G, Herman, R, Kerff, F, Amoroso, A, Fonze, E, Pratt, R.F, Luxen, A, Charlier, P.
登録日2009-06-03
公開日2009-12-01
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Structural Basis of the Inhibition of Class a Beta-Lactamases and Penicillin-Binding Proteins by 6-Beta-Iodopenicillanate.
J.Am.Chem.Soc., 131, 2009
1NRF
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BU of 1nrf by Molmil
C-terminal domain of the Bacillus licheniformis BlaR penicillin-receptor
分子名称: REGULATORY PROTEIN BLAR1
著者Kerff, F, Charlier, P, Columbo, M.L, Sauvage, E, Brans, A, Frere, J.M, Joris, B, Fonze, E.
登録日2003-01-24
公開日2004-01-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of the sensor domain of the BlaR penicillin receptor from Bacillus licheniformis.
Biochemistry, 42, 2003
1K6R
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BU of 1k6r by Molmil
STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-10 IN COMPLEX WITH MOXALACTAM
分子名称: (2R)-2-((R)-CARBOXY{[CARBOXY(4-HYDROXYPHENYL)ACETYL]AMINO}METHOXYMETHYL)-5-METHYLENE-5,6-DIHYDRO-2H-1,3-OXAZINE-4-CARBO XYLIC ACID, Beta-lactamase PSE-2
著者Kerff, F, Fonze, E, Sauvage, E, Frere, J.M, Charlier, P.
登録日2001-10-17
公開日2003-06-24
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献CRYSTAL STRUCTURE OF CLASS D BETA-LACTAMASE OXA-10 IN COMPLEX WITH DIFFERENT SUBSTRATES AND ONE INHIBITOR.
To be Published
1K6S
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BU of 1k6s by Molmil
STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-10 IN COMPLEX WITH A PHENYLBORONIC ACID
分子名称: 4-IODO-ACETAMIDO PHENYLBORONIC ACID, Beta-lactamase PSE-2, CALCIUM ION, ...
著者Kerff, F, Fonze, E, Sauvage, E, Frere, J.M, Charlier, P.
登録日2001-10-17
公開日2003-06-24
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献CRYSTAL STRUCTURE OF CLASS D BETA-LACTAMASE OXA-10 IN COMPLEX WITH DIFFERENT SUBSTRATES AND ONE INHIBITOR.
To be Published
1K4F
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CRYSTAL STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-10 AT 1.6 A RESOLUTION
分子名称: Beta-lactamase PSE-2, SULFATE ION
著者Kerff, F, Fonze, E, Bouillene, F, Frere, J.M, Charlier, P.
登録日2001-10-08
公開日2001-10-31
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structure of the class D beta-lactamase OXA-2
To be Published
1K38
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BU of 1k38 by Molmil
CRYSTAL STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-2
分子名称: Beta-lactamase OXA-2, FORMIC ACID
著者Kerff, F, Fonze, E, Bouillenne, F, Frere, J.M, Charlier, P.
登録日2001-10-02
公開日2003-06-24
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献CRYSTAL STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-2
To be Published
1K4E
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BU of 1k4e by Molmil
CRYSTAL STRUCTURE OF THE CLASS D BETA-LACTAMASES OXA-10 DETERMINED BY MAD PHASING WITH SELENOMETHIONINE
分子名称: Beta-lactamase PSE-2, SULFATE ION
著者Kerff, F, Fonze, E, Bouillene, F, Frere, J.M, Charlier, P.
登録日2001-10-08
公開日2001-10-31
最終更新日2022-12-21
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献STRUCTURE OF CLASS D BETA-LACTAMASE OXA-2
To be Published
1BSG
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BU of 1bsg by Molmil
BETA-LACTAMASE FROM STREPTOMYCES ALBUS G
分子名称: ACETATE ION, BETA LACTAMASE
著者Fonze, E, Charlier, P, Dideberg, O.
登録日1998-07-20
公開日1999-01-13
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献

2WKE
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Crystal structure of the Actinomadura R39 DD-peptidase inhibited by 6- beta-iodopenicillanate.
分子名称: (3S)-2,2-dimethyl-3,4-dihydro-2H-1,4-thiazine-3,6-dicarboxylic acid, COBALT (II) ION, D-ALANYL-D-ALANINE CARBOXYPEPTIDASE, ...
著者Sauvage, E, Herman, R, Kerff, F, Charlier, P.
登録日2009-06-10
公開日2009-12-01
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural Basis of the Inhibition of Class a Beta-Lactamases and Penicillin-Binding Proteins by 6-Beta-Iodopenicillanate.
J.Am.Chem.Soc., 131, 2009
1S6R
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908R class c beta-lactamase bound to iodo-acetamido-phenyl boronic acid
分子名称: 4-IODO-ACETAMIDO PHENYLBORONIC ACID, beta-lactamase
著者Wouters, J.
登録日2004-01-27
公開日2004-02-24
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.24 Å)
主引用文献Crystal structure of Enterobacter cloacae 908R class C beta-lactamase bound to iodo-acetamido-phenyl boronic acid, a transition-state analogue.
Cell.Mol.Life Sci., 60, 2003
1W7F
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Crystal structure of the class A beta-lactamase BS3 inhibited with isocitrate
分子名称: BETA-LACTAMASE, ISOCITRIC ACID
著者Petrella, S, Sauvage, E, Herman, R, Charlier, P.
登録日2004-09-01
公開日2006-05-24
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structure of the Class a Beta-Lactamase Bs3 Bs3 Inhibited with Isocitrate
To be Published

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