7U0S
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![BU of 7u0s by Molmil](/molmil-images/mine/7u0s) | Crystal Structure of FK506-binding protein 1A from Aspergillus fumigatus Bound to Ascomycin | Descriptor: | (3S,4R,5S,8R,9E,12S,14S,15R,16S,18R,19R,22R,26aS)-8-ethyl-5,19-dihydroxy-3-{(1E)-1-[(1R,3R,4R)-4-hydroxy-3-methoxycyclohexyl]prop-1-en-2-yl}-14,16-dimethoxy-4,10,12,18-tetramethyl-5,6,8,11,12,13,14,15,16,17,18,19,24,25,26,26a-hexadecahydro-3H-15,19-epoxypyrido[2,1-c][1,4]oxazacyclotricosine-1,7,20,21(4H,23H)-tetrone, ACETATE ION, FK506-binding protein 1A, ... | Authors: | DeBouver, N.D, Fox III, D, Hoy, M.J, Heitman, J, Lorimer, D.D, Horanyi, P.S, Edwards, T.E, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | Deposit date: | 2022-02-18 | Release date: | 2022-07-27 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Structure-Guided Synthesis of FK506 and FK520 Analogs with Increased Selectivity Exhibit In Vivo Therapeutic Efficacy against Cryptococcus. Mbio, 13, 2022
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7U0U
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![BU of 7u0u by Molmil](/molmil-images/mine/7u0u) | Crystal Structure of a Aspergillus fumigatus Calcineurin A - Calcineurin B fusion bound to FKBP12 and FK-506 | Descriptor: | 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN, CALCIUM ION, PHOSPHATE ION, ... | Authors: | Fox III, D, Abendroth, J, DeBouver, N.D, Hoy, M.J, Heitman, J, Lorimer, D.D, Horanyi, P.S, Edwards, T.E, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | Deposit date: | 2022-02-18 | Release date: | 2022-08-03 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Structure-Guided Synthesis of FK506 and FK520 Analogs with Increased Selectivity Exhibit In Vivo Therapeutic Efficacy against Cryptococcus. Mbio, 13, 2022
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7U0T
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![BU of 7u0t by Molmil](/molmil-images/mine/7u0t) | Crystal Structure of a human Calcineurin A - Calcineurin B fusion bound to FKBP12 and FK-520 | Descriptor: | (3S,4R,5S,8R,9E,12S,14S,15R,16S,18R,19R,22R,26aS)-8-ethyl-5,19-dihydroxy-3-{(1E)-1-[(1R,3R,4R)-4-hydroxy-3-methoxycyclohexyl]prop-1-en-2-yl}-14,16-dimethoxy-4,10,12,18-tetramethyl-5,6,8,11,12,13,14,15,16,17,18,19,24,25,26,26a-hexadecahydro-3H-15,19-epoxypyrido[2,1-c][1,4]oxazacyclotricosine-1,7,20,21(4H,23H)-tetrone, 1,2-ETHANEDIOL, CALCIUM ION, ... | Authors: | Fox III, D, Mayclin, S.J, DeBouver, N.D, Hoy, M.J, Heitman, J, Lorimer, D.D, Horanyi, P.S, Edwards, T.E, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | Deposit date: | 2022-02-18 | Release date: | 2022-08-03 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (2.45 Å) | Cite: | Structure-Guided Synthesis of FK506 and FK520 Analogs with Increased Selectivity Exhibit In Vivo Therapeutic Efficacy against Cryptococcus. Mbio, 13, 2022
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6XMY
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![BU of 6xmy by Molmil](/molmil-images/mine/6xmy) | |
8CU9
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![BU of 8cu9 by Molmil](/molmil-images/mine/8cu9) | |
8CU5
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![BU of 8cu5 by Molmil](/molmil-images/mine/8cu5) | |
8DTC
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![BU of 8dtc by Molmil](/molmil-images/mine/8dtc) | |
8DU0
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![BU of 8du0 by Molmil](/molmil-images/mine/8du0) | |
8DT6
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![BU of 8dt6 by Molmil](/molmil-images/mine/8dt6) | |
8DTE
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![BU of 8dte by Molmil](/molmil-images/mine/8dte) | |
8DU1
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![BU of 8du1 by Molmil](/molmil-images/mine/8du1) | |
7MMZ
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![BU of 7mmz by Molmil](/molmil-images/mine/7mmz) | |
7SH3
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![BU of 7sh3 by Molmil](/molmil-images/mine/7sh3) | |
7SWH
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![BU of 7swh by Molmil](/molmil-images/mine/7swh) | |
7SWK
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![BU of 7swk by Molmil](/molmil-images/mine/7swk) | |
7SYC
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![BU of 7syc by Molmil](/molmil-images/mine/7syc) | |
7SZS
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![BU of 7szs by Molmil](/molmil-images/mine/7szs) | |
7SZV
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![BU of 7szv by Molmil](/molmil-images/mine/7szv) | |
7T93
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![BU of 7t93 by Molmil](/molmil-images/mine/7t93) | |
7KQA
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![BU of 7kqa by Molmil](/molmil-images/mine/7kqa) | |
7KQ6
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![BU of 7kq6 by Molmil](/molmil-images/mine/7kq6) | |
7L9T
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![BU of 7l9t by Molmil](/molmil-images/mine/7l9t) | |
7LD8
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![BU of 7ld8 by Molmil](/molmil-images/mine/7ld8) | |
7OPB
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![BU of 7opb by Molmil](/molmil-images/mine/7opb) | IL7R in complex with an antagonist | Descriptor: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, IL7R binder, ... | Authors: | Markovic, I, Verschueren, K.H.G, Verstraete, K, Savvides, S.N. | Deposit date: | 2021-05-31 | Release date: | 2022-05-11 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.144 Å) | Cite: | Design of protein-binding proteins from the target structure alone. Nature, 605, 2022
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7TI7
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![BU of 7ti7 by Molmil](/molmil-images/mine/7ti7) | |