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4U6G
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BU of 4u6g by Molmil
Crystal structure of 10E8 Fab in complex with a hydrocarbon-stapled HIV-1 gp41 MPER peptide
分子名称: 10E8 Fab Heavy Chain, 10E8 Fab Light Chain, SAH-MPER(662-683KKK)(B,q)
著者Ofek, G, Bird, G.H, Walensky, L.D, Kwong, P.D.
登録日2014-07-28
公開日2014-12-03
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (4.2012 Å)
主引用文献Structural Fidelity and Neutralizing Antibody Binding Capacity of Hydrocarbon-Stapled HIV-1 Antigens
To be published
2K7W
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BU of 2k7w by Molmil
BAX Activation is Initiated at a Novel Interaction Site
分子名称: Apoptosis regulator BAX, Bcl-2-like protein 11
著者Gavathiotis, E, Suzuki, M, Davis, M.L, Pitter, K, Bird, G.H, Katz, S.G, Tu, H.C, Kim, H, Cheng, E.H, Tjandra, N, Walensky, L.D.
登録日2008-08-27
公開日2008-10-21
最終更新日2022-03-16
実験手法SOLUTION NMR
主引用文献BAX activation is initiated at a novel interaction site.
Nature, 455, 2008
4NGH
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BU of 4ngh by Molmil
Crystal structure of the HIV-1 neutralizing antibody 4E10 Fab fragment in complex with a hydrocarbon-stapled peptide containing the 4e10 epitope on gp41 and a tethered phosphate moiety.
分子名称: FAB HEAVY CHAIN, FAB LIGHT CHAIN, MODIFIED FRAGMENT OF HIV GLYCOPROTEIN (GP41)
著者Irimia, A, Wilson, I.A.
登録日2013-11-01
公開日2014-12-03
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.68 Å)
主引用文献Stapled HIV-1 peptides recapitulate antigenic structures and engage broadly neutralizing antibodies.
Nat.Struct.Mol.Biol., 21, 2014
4NHC
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BU of 4nhc by Molmil
Crystal structure of the HIV-1 neutralizing antibody 4E10 Fab fragment in complex with a hydrocarbon-stapled peptide containing the 4e10 epitope on gp41.
分子名称: FAB HEAVY CHAIN, FAB LIGHT CHAIN, MODIFIED FRAGMENT OF HIV GLYCOPROTEIN (GP41), ...
著者Irimia, A, Wilson, I.A.
登録日2013-11-04
公開日2014-12-03
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.912 Å)
主引用文献Stapled HIV-1 peptides recapitulate antigenic structures and engage broadly neutralizing antibodies.
Nat.Struct.Mol.Biol., 21, 2014
5W89
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BU of 5w89 by Molmil
Crystal structure of human Mcl-1 in complex with modified Bim BH3 peptide SAH-MS1-18
分子名称: Induced myeloid leukemia cell differentiation protein Mcl-1, ZINC ION, modified Bim BH3 peptide SAH-MS1-18
著者Rezaei Araghi, R, Jenson, J.M, Grant, R.A, Keating, A.E.
登録日2017-06-21
公開日2018-01-17
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Iterative optimization yields Mcl-1-targeting stapled peptides with selective cytotoxicity to Mcl-1-dependent cancer cells.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
5WHI
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BU of 5whi by Molmil
Crystal Structure of Bcl-2-related protein A1
分子名称: Bcl-2-related protein A1, CACODYLIC ACID
著者Seo, H.-S, Dhe-Paganon, S.
登録日2017-07-17
公開日2018-01-17
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Crystal Structures of Anti-apoptotic BFL-1 and Its Complex with a Covalent Stapled Peptide Inhibitor.
Structure, 26, 2018
5W8F
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BU of 5w8f by Molmil
Crystal structure of human Mcl-1 in complex with modified Bim BH3 peptide SAH-MS1-14
分子名称: Induced myeloid leukemia cell differentiation protein Mcl-1, ZINC ION, modified Bim BH3 peptide SAH-MS1-14
著者Rezaei Araghi, R, Jenson, J.M, Grant, R.A, Keating, A.E.
登録日2017-06-21
公開日2018-01-17
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Iterative optimization yields Mcl-1-targeting stapled peptides with selective cytotoxicity to Mcl-1-dependent cancer cells.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
5WHH
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BU of 5whh by Molmil
Crystal Structure of Bcl-2-related protein A1 in complex with stapled peptide (AQ7)T(0EH)LRRFGD(MK8)INFRQ(NH2)
分子名称: (AQ7)T(0EH)LRRFGD(MK8)INFRQ(NH2), Bcl-2-related protein A1, CHLORIDE ION
著者Seo, H.-S, Dhe-Paganon, S.
登録日2017-07-17
公開日2018-01-17
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Crystal Structures of Anti-apoptotic BFL-1 and Its Complex with a Covalent Stapled Peptide Inhibitor.
Structure, 26, 2018
6VO4
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BU of 6vo4 by Molmil
Crystal Structure Analysis of BFL1
分子名称: Bcl-2-related protein A1
著者Seo, H.-S, Dhe-Paganon, S.
登録日2020-01-29
公開日2020-06-03
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献Identification of a Covalent Molecular Inhibitor of Anti-apoptotic BFL-1 by Disulfide Tethering.
Cell Chem Biol, 27, 2020

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件を2024-05-01に公開中

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