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7RZ3
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BU of 7rz3 by Molmil
The solution structure of remipede double-ICK toxin phi-Xibalbin3-Xt3a
Descriptor: Xt3a
Authors:Maxwell, M, Chin, Y.K, Mobli, M.
Deposit date:2021-08-27
Release date:2022-08-31
Last modified:2023-03-08
Method:SOLUTION NMR
Cite:A bivalent remipede toxin promotes calcium release via ryanodine receptor activation.
Nat Commun, 14, 2023
5V37
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BU of 5v37 by Molmil
Crystal structure of SMYD3 with SAM and EPZ028862
Descriptor: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, ...
Authors:Boriack-Sjodin, P.A.
Deposit date:2017-03-06
Release date:2018-03-07
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.42 Å)
Cite:Small molecule inhibitors and CRISPR/Cas9 mutagenesis demonstrate that SMYD2 and SMYD3 activity are dispensable for autonomous cancer cell proliferation.
Plos One, 13, 2018
5V3H
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BU of 5v3h by Molmil
Crystal structure of SMYD2 with SAM and EPZ033294
Descriptor: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, GLYCEROL, ...
Authors:Boriack-Sjodin, P.A.
Deposit date:2017-03-07
Release date:2018-04-25
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.69 Å)
Cite:Small molecule inhibitors and CRISPR/Cas9 mutagenesis demonstrate that SMYD2 and SMYD3 activity are dispensable for autonomous cancer cell proliferation.
Plos One, 13, 2018
5EML
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BU of 5eml by Molmil
Crystal structure of PRMT5:MEP50 with Compound 10 and SAM
Descriptor: GLYCEROL, Methylosome protein 50, Protein arginine N-methyltransferase 5, ...
Authors:Boriack-Sjodin, P.A, Jin, L.
Deposit date:2015-11-06
Release date:2016-02-24
Last modified:2018-04-18
Method:X-RAY DIFFRACTION (2.39 Å)
Cite:Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666.
ACS Med Chem Lett, 7, 2016
5EMK
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BU of 5emk by Molmil
Crystal structure of PRMT5:MEP50 with Compound 9 and sinefungin
Descriptor: GLYCEROL, Methylosome protein 50, Protein arginine N-methyltransferase 5, ...
Authors:Boriack-Sjodin, P.A, Jin, L.
Deposit date:2015-11-06
Release date:2016-02-24
Last modified:2018-04-18
Method:X-RAY DIFFRACTION (2.52 Å)
Cite:Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666.
ACS Med Chem Lett, 7, 2016
5EMJ
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Crystal structure of PRMT5:MEP50 with Compound 8 and sinefungin
Descriptor: (2~{S})-1-(3,4-dihydro-1~{H}-isoquinolin-2-yl)-3-[[4-(3-methylbenzimidazol-5-yl)pyridin-2-yl]amino]propan-2-ol, GLYCEROL, Methylosome protein 50, ...
Authors:Boriack-Sjodin, P.A, Jin, L.
Deposit date:2015-11-06
Release date:2016-02-24
Last modified:2018-04-18
Method:X-RAY DIFFRACTION (2.273 Å)
Cite:Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666.
ACS Med Chem Lett, 7, 2016
5EMM
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BU of 5emm by Molmil
Crystal structure of PRMT5:MEP50 with Compound 15 and sinefungin
Descriptor: GLYCEROL, Methylosome protein 50, Protein arginine N-methyltransferase 5, ...
Authors:Boriack-Sjodin, P.A, Jin, L.
Deposit date:2015-11-06
Release date:2016-02-24
Last modified:2018-04-18
Method:X-RAY DIFFRACTION (2.37 Å)
Cite:Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666.
ACS Med Chem Lett, 7, 2016
5T4R
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BU of 5t4r by Molmil
NMR solution structure of the Nav1.7 selective spider venom-derived peptide Pn3a
Descriptor: Mu-theraphotoxin-Pn3a
Authors:Rosengren, K.J, Armstrong, D.A, Vetter, I.
Deposit date:2016-08-30
Release date:2017-09-06
Last modified:2023-06-14
Method:SOLUTION NMR
Cite:Pharmacological characterisation of the highly Na V 1.7 selective spider venom peptide Pn3a.
Sci Rep, 7, 2017
2MPQ
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BU of 2mpq by Molmil
Solution structure of the sodium channel toxin Hd1a
Descriptor: Hd1a
Authors:Klint, J.K, Mobli, M, King, G.F.
Deposit date:2014-06-01
Release date:2015-03-25
Last modified:2023-06-14
Method:SOLUTION NMR
Cite:Seven novel modulators of the analgesic target NaV 1.7 uncovered using a high-throughput venom-based discovery approach.
Br.J.Pharmacol., 172, 2015
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