4F82
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![BU of 4f82 by Molmil](/molmil-images/mine/4f82) | |
7ULH
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![BU of 7ulh by Molmil](/molmil-images/mine/7ulh) | |
6OQE
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![BU of 6oqe by Molmil](/molmil-images/mine/6oqe) | |
5JIX
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![BU of 5jix by Molmil](/molmil-images/mine/5jix) | PKG II's Carboxyl Terminal Cyclic Nucleotide Binding Domain (CNB-B) in a complex with 8-Br-cGMP | Descriptor: | 1,2-ETHANEDIOL, 2-amino-8-bromo-9-[(2R,4aR,6R,7R,7aS)-2,7-dihydroxy-2-oxotetrahydro-2H,4H-2lambda~5~-furo[3,2-d][1,3,2]dioxaphosphinin-6-yl]-1,9-dihydro-6H-purin-6-one, 3,6,9,12,15,18,21,24-OCTAOXAHEXACOSAN-1-OL, ... | Authors: | Campbell, J.C, Kim, C.W. | Deposit date: | 2016-04-22 | Release date: | 2017-05-03 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (1.47 Å) | Cite: | Structural Basis of Analog Specificity in PKG I and II. ACS Chem. Biol., 12, 2017
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6HAR
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![BU of 6har by Molmil](/molmil-images/mine/6har) | Crystal structure of Mesotrypsin in complex with APPI-M17C/I18F/F34C | Descriptor: | 1,2-ETHANEDIOL, Amyloid-beta A4 protein, CALCIUM ION, ... | Authors: | Shahar, A, Cohen, I, Radisky, E, Papo, N. | Deposit date: | 2018-08-08 | Release date: | 2019-02-06 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.497 Å) | Cite: | Disulfide engineering of human Kunitz-type serine protease inhibitors enhances proteolytic stability and target affinity toward mesotrypsin. J.Biol.Chem., 294, 2019
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4OPH
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![BU of 4oph by Molmil](/molmil-images/mine/4oph) | X-ray structure of full-length H6N6 NS1 | Descriptor: | Nonstructural protein 1 | Authors: | Carrillo, B, Choi, J.M, Bornholdt, Z.A, Sankaran, S, Rice, A.P, Prasad, B.V.V. | Deposit date: | 2014-02-05 | Release date: | 2014-02-19 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (3.158 Å) | Cite: | The Influenza A Virus Protein NS1 Displays Structural Polymorphism. J.Virol., 88, 2014
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7SH8
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![BU of 7sh8 by Molmil](/molmil-images/mine/7sh8) | Structure of the SARS-CoV-2 main protease in complex with inhibitor MPI88 | Descriptor: | 3C-like proteinase nsp5, benzyl [(2S,3R)-1-{[(2S)-1-(2-acetyl-2-{[(3S)-2-oxopyrrolidin-3-yl]methyl}hydrazinyl)-3-cyclohexyl-1-oxopropan-2-yl]amino}-3-tert-butoxy-1-oxobutan-2-yl]carbamate (non-preferred name) | Authors: | Yang, K.S, Liu, W.R. | Deposit date: | 2021-10-08 | Release date: | 2023-04-12 | Last modified: | 2023-11-15 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Structure of the SARS-CoV-2 main protease in complex with inhibitors To Be Published
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7SH9
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![BU of 7sh9 by Molmil](/molmil-images/mine/7sh9) | Structure of the SARS-CoV-2 main protease in complex with inhibitor MPI86 | Descriptor: | 3C-like proteinase nsp5, benzyl [(2S,3R)-1-({(2S)-1-[2-acetyl-2-(3-amino-3-oxopropyl)hydrazinyl]-3-cyclohexyl-1-oxopropan-2-yl}amino)-3-tert-butoxy-1-oxobutan-2-yl]carbamate (non-preferred name) | Authors: | Yang, K.S, Liu, W.R. | Deposit date: | 2021-10-08 | Release date: | 2023-04-12 | Last modified: | 2023-11-15 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Structure of the SARS-CoV-2 main protease in complex with inhibitors To Be Published
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6XQR
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![BU of 6xqr by Molmil](/molmil-images/mine/6xqr) | OXA-48 bound by Compound 2.2 | Descriptor: | Beta-lactamase, CHLORIDE ION, [1,1'-biphenyl]-4,4'-disulfonic acid | Authors: | Taylor, D.M, Hu, L, Prasad, B.V.V, Palzkill, T. | Deposit date: | 2020-07-10 | Release date: | 2021-12-15 | Last modified: | 2023-11-15 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Unique Diacidic Fragments Inhibit the OXA-48 Carbapenemase and Enhance the Killing of Escherichia coli Producing OXA-48. Acs Infect Dis., 7, 2021
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8T5W
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![BU of 8t5w by Molmil](/molmil-images/mine/8t5w) | |
4RPT
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![BU of 4rpt by Molmil](/molmil-images/mine/4rpt) | |
4RSR
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![BU of 4rsr by Molmil](/molmil-images/mine/4rsr) | ArsM arsenic(III) S-adenosylmethionine methyltransferase with trivalent phenyl arsencial derivative-Roxarsone | Descriptor: | 2,3-DIHYDROXY-1,4-DITHIOBUTANE, 4-arsanyl-2-nitrophenol, Arsenic methyltransferase, ... | Authors: | Packianathan, C, Marapakala, K, Ajees, A.A, Kandavelu, P, Rosen, B.P. | Deposit date: | 2014-11-10 | Release date: | 2014-12-10 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.25 Å) | Cite: | A disulfide-bond cascade mechanism for arsenic(III) S-adenosylmethionine methyltransferase. Acta Crystallogr.,Sect.D, 71, 2015
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4WBS
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![BU of 4wbs by Molmil](/molmil-images/mine/4wbs) | |
3L3B
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![BU of 3l3b by Molmil](/molmil-images/mine/3l3b) | |
3UKN
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![BU of 3ukn by Molmil](/molmil-images/mine/3ukn) | |
3UKT
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![BU of 3ukt by Molmil](/molmil-images/mine/3ukt) | |
3UZU
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![BU of 3uzu by Molmil](/molmil-images/mine/3uzu) | |
5JEO
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![BU of 5jeo by Molmil](/molmil-images/mine/5jeo) | Phosphorylated Rotavirus NSP1 in complex with IRF-3 | Descriptor: | Interferon regulatory factor 3, PHOSPHATE ION, Rotavirus NSP1 peptide | Authors: | Zhao, B, Li, P. | Deposit date: | 2016-04-18 | Release date: | 2016-06-15 | Last modified: | 2016-06-29 | Method: | X-RAY DIFFRACTION (1.719 Å) | Cite: | Structural basis for concerted recruitment and activation of IRF-3 by innate immune adaptor proteins. Proc.Natl.Acad.Sci.USA, 113, 2016
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4E51
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![BU of 4e51 by Molmil](/molmil-images/mine/4e51) | |
8CUX
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![BU of 8cux by Molmil](/molmil-images/mine/8cux) | |
8CUV
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![BU of 8cuv by Molmil](/molmil-images/mine/8cuv) | |
8CUU
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![BU of 8cuu by Molmil](/molmil-images/mine/8cuu) | |
8CUT
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![BU of 8cut by Molmil](/molmil-images/mine/8cut) | |
8CUS
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![BU of 8cus by Molmil](/molmil-images/mine/8cus) | |
8CWZ
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![BU of 8cwz by Molmil](/molmil-images/mine/8cwz) | |