8TRC
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8TR2
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![BU of 8tr2 by Molmil](/molmil-images/mine/8tr2) | mGluR3 in the presence of the agonist LY379268 | Descriptor: | (1S,4R,5R,6S)-4-amino-2-oxabicyclo[3.1.0]hexane-4,6-dicarboxylic acid, CALCIUM ION, Metabotropic glutamate receptor 3 | Authors: | Strauss, A, Levitz, J. | Deposit date: | 2023-08-09 | Release date: | 2024-07-31 | Method: | ELECTRON MICROSCOPY (3.5 Å) | Cite: | Structural basis of allosteric modulation of metabotropic glutamate receptor activation and desensitization. Biorxiv, 2023
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8TR0
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8TQB
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![BU of 8tqb by Molmil](/molmil-images/mine/8tqb) | mGluR3 in the presence of the agonist LY379268 and PAM VU6023326 | Descriptor: | (1R,4R,5S,6R)-4-azanyl-2-oxabicyclo[3.1.0]hexane-4,6-dicarboxylic acid, CALCIUM ION, Metabotropic glutamate receptor 3 | Authors: | Strauss, A, Levitz, J. | Deposit date: | 2023-08-06 | Release date: | 2024-07-31 | Method: | ELECTRON MICROSCOPY (3.3 Å) | Cite: | Structural basis of allosteric modulation of metabotropic glutamate receptor activation and desensitization. Biorxiv, 2023
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7LVT
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![BU of 7lvt by Molmil](/molmil-images/mine/7lvt) | Structure of full-length GluK1 with L-Glu | Descriptor: | Isoform Glur5-2 of Glutamate receptor ionotropic, kainate 1 | Authors: | Meyerson, J.R, Selvakumar, P. | Deposit date: | 2021-02-26 | Release date: | 2021-11-03 | Last modified: | 2021-11-10 | Method: | ELECTRON MICROSCOPY (4.6 Å) | Cite: | Structural and compositional diversity in the kainate receptor family. Cell Rep, 37, 2021
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3SOA
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![BU of 3soa by Molmil](/molmil-images/mine/3soa) | Full-length human CaMKII | Descriptor: | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile, Calcium/calmodulin-dependent protein kinase type II subunit alpha with a beta 7 linker | Authors: | Chao, L.H, Kuriyan, J. | Deposit date: | 2011-06-30 | Release date: | 2011-08-31 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (3.5501 Å) | Cite: | A Mechanism for Tunable Autoinhibition in the Structure of a Human Ca(2+)/Calmodulin- Dependent Kinase II Holoenzyme. Cell(Cambridge,Mass.), 146, 2011
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8THL
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8THK
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6M8S
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![BU of 6m8s by Molmil](/molmil-images/mine/6m8s) | Crystal structure of the KCTD12 H1 domain in complex with Gbeta1gamma2 subunits | Descriptor: | BTB/POZ domain-containing protein KCTD12, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 | Authors: | Zheng, S, Kruse, A.C. | Deposit date: | 2018-08-22 | Release date: | 2019-02-27 | Last modified: | 2023-10-11 | Method: | X-RAY DIFFRACTION (3.71 Å) | Cite: | Structural basis for KCTD-mediated rapid desensitization of GABABsignalling. Nature, 567, 2019
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6M8R
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8TRD
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![BU of 8trd by Molmil](/molmil-images/mine/8trd) | mGluR3 class 1 in the presence of the antagonist LY 341495 | Descriptor: | 2-[(1S,2S)-2-carboxycyclopropyl]-3-(9H-xanthen-9-yl)-D-alanine, Metabotropic glutamate receptor 3 | Authors: | Strauss, A, Levitz, J. | Deposit date: | 2023-08-09 | Release date: | 2024-07-31 | Method: | ELECTRON MICROSCOPY (3.4 Å) | Cite: | Structural basis of allosteric modulation of
metabotropic glutamate receptor activation and desensitization To be published
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