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7WGL
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BU of 7wgl by Molmil
X-ray structure of human PPAR delta ligand binding domain-bezafibrate co-crystals obtained by co-crystallization
Descriptor: 2-[P-[2-P-CHLOROBENZAMIDO)ETHYL]PHENOXY]-2-METHYLPROPIONIC ACID, Peroxisome proliferator-activated receptor delta, octyl beta-D-glucopyranoside
Authors:Kamata, S, Honda, A, Machida, Y, Uchii, K, Shiiyama, Y, Masuda, R, Oyama, T, Ishii, I.
Deposit date:2021-12-28
Release date:2022-05-25
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.091 Å)
Cite:Functional and Structural Insights into Human PPAR alpha / delta / gamma Subtype Selectivity of Bezafibrate, Fenofibric Acid, and Pemafibrate.
Int J Mol Sci, 23, 2022
1YXK
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BU of 1yxk by Molmil
Crystal structure of human lectin-like oxidized low-density lipoprotein receptor 1 (LOX-1) disulfide-linked dimer
Descriptor: oxidised low density lipoprotein (lectin-like) receptor 1
Authors:Ohki, I, Ishigaki, T, Oyama, T, Matsunaga, S, Xie, Q, Ohnishi-Kameyama, M, Murata, T, Tsuchiya, D, Machida, S, Morikawa, K, Tate, S.
Deposit date:2005-02-22
Release date:2005-06-14
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Crystal structure of human lectin-like, oxidized low-density lipoprotein receptor 1 ligand binding domain and its ligand recognition mode to OxLDL.
Structure, 13, 2005
1YXJ
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Crystal structure of human lectin-like oxidized low-density lipoprotein receptor 1 (LOX-1) at low pH
Descriptor: 1,2-ETHANEDIOL, oxidised low density lipoprotein (lectin-like) receptor 1
Authors:Ohki, I, Ishigaki, T, Oyama, T, Matsunaga, S, Xie, Q, Ohnishi-Kameyama, M, Murata, T, Tsuchiya, D, Machida, S, Morikawa, K, Tate, S.
Deposit date:2005-02-22
Release date:2005-06-14
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.78 Å)
Cite:Crystal structure of human lectin-like, oxidized low-density lipoprotein receptor 1 ligand binding domain and its ligand recognition mode to OxLDL.
Structure, 13, 2005
2EGK
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BU of 2egk by Molmil
Crystal Structure of Tamalin PDZ-Intrinsic Ligand Fusion Protein
Descriptor: General receptor for phosphoinositides 1-associated scaffold protein, PHOSPHATE ION
Authors:Sugi, T, Oyama, T, Muto, T, Nakanishi, S, Morikawa, K, Jingami, H.
Deposit date:2007-03-01
Release date:2007-05-08
Last modified:2021-11-10
Method:X-RAY DIFFRACTION (2.85 Å)
Cite:Crystal structures of autoinhibitory PDZ domain of Tamalin: implications for metabotropic glutamate receptor trafficking regulation
Embo J., 26, 2007
2EGO
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BU of 2ego by Molmil
Crystal Structure of Tamalin PDZ Domain
Descriptor: General receptor for phosphoinositides 1-associated scaffold protein
Authors:Sugi, T, Oyama, T, Muto, T, Nakanishi, S, Morikawa, K, Jingami, H.
Deposit date:2007-03-01
Release date:2007-05-01
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystal structures of autoinhibitory PDZ domain of Tamalin: implications for metabotropic glutamate receptor trafficking regulation
Embo J., 26, 2007
2EGN
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BU of 2egn by Molmil
Crystal Structure of Tamalin PDZ Domain in Complex with mGluR5 C-terminal Peptide
Descriptor: General receptor for phosphoinositides 1-associated scaffold protein, mGluR5 C-terminal peptide
Authors:Sugi, T, Oyama, T, Muto, T, Nakanishi, S, Morikawa, K, Jingami, H.
Deposit date:2007-03-01
Release date:2007-05-15
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Crystal structures of autoinhibitory PDZ domain of Tamalin: implications for metabotropic glutamate receptor trafficking regulation
Embo J., 26, 2007
1WDL
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BU of 1wdl by Molmil
fatty acid beta-oxidation multienzyme complex from Pseudomonas fragi, form II (native4)
Descriptor: 3,6,9,12,15-PENTAOXATRICOSAN-1-OL, 3-ketoacyl-CoA thiolase, ACETYL COENZYME *A, ...
Authors:Ishikawa, M, Tsuchiya, D, Oyama, T, Tsunaka, Y, Morikawa, K.
Deposit date:2004-05-17
Release date:2004-07-27
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.5 Å)
Cite:Structural basis for channelling mechanism of a fatty acid beta-oxidation multienzyme complex
Embo J., 23, 2004
1WDK
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fatty acid beta-oxidation multienzyme complex from Pseudomonas fragi, form I (native2)
Descriptor: 3,6,9,12,15-PENTAOXATRICOSAN-1-OL, 3-ketoacyl-CoA thiolase, ACETYL COENZYME *A, ...
Authors:Ishikawa, M, Tsuchiya, D, Oyama, T, Tsunaka, Y, Morikawa, K.
Deposit date:2004-05-17
Release date:2004-07-27
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structural basis for channelling mechanism of a fatty acid beta-oxidation multienzyme complex
Embo J., 23, 2004
1WDM
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BU of 1wdm by Molmil
fatty acid beta-oxidation multienzyme complex from Pseudomonas fragi, form I (native3)
Descriptor: 3-ketoacyl-CoA thiolase, ACETYL COENZYME *A, Fatty oxidation complex alpha subunit, ...
Authors:Ishikawa, M, Tsuchiya, D, Oyama, T, Tsunaka, Y, Morikawa, K.
Deposit date:2004-05-17
Release date:2004-07-27
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.8 Å)
Cite:Structural basis for channelling mechanism of a fatty acid beta-oxidation multienzyme complex
Embo J., 23, 2004
1WWJ
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BU of 1wwj by Molmil
crystal structure of KaiB from Synechocystis sp.
Descriptor: Circadian clock protein kaiB, D-MALATE, IMIDAZOLE, ...
Authors:Hitomi, K, Oyama, T, Han, S, Arvai, A.S, Tainer, J.A, Getzoff, E.D.
Deposit date:2005-01-06
Release date:2005-02-15
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Tetrameric architecture of the circadian clock protein KaiB. A novel interface for intermolecular interactions and its impact on the circadian rhythm.
J.Biol.Chem., 280, 2005
3B0C
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BU of 3b0c by Molmil
Crystal structure of the chicken CENP-T histone fold/CENP-W complex, crystal form I
Descriptor: CITRIC ACID, Centromere protein T, Centromere protein W
Authors:Nishino, T, Takeuchi, K, Gascoigne, K.E, Suzuki, A, Hori, T, Oyama, T, Morikawa, K, Cheeseman, I.M, Fukagawa, T.
Deposit date:2011-06-08
Release date:2012-03-07
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.201 Å)
Cite:CENP-T-W-S-X Forms a Unique Centromeric Chromatin Structure with a Histone-like Fold.
Cell(Cambridge,Mass.), 148, 2012
3B0B
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BU of 3b0b by Molmil
Crystal structure of the chicken CENP-S/CENP-X complex
Descriptor: Centromere protein S, Centromere protein X
Authors:Nishino, T, Takeuchi, K, Gascoigne, K.E, Suzuki, A, Hori, T, Oyama, T, Morikawa, K, Cheeseman, I.M, Fukagawa, T.
Deposit date:2011-06-08
Release date:2012-03-07
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:CENP-T-W-S-X Forms a Unique Centromeric Chromatin Structure with a Histone-like Fold.
Cell(Cambridge,Mass.), 148, 2012
3B0D
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BU of 3b0d by Molmil
Crystal structure of the chicken CENP-T histone fold/CENP-W complex, crystal form II
Descriptor: CITRIC ACID, Centromere protein T, Centromere protein W
Authors:Nishino, T, Takeuchi, K, Gascoigne, K.E, Suzuki, A, Hori, T, Oyama, T, Morikawa, K, Cheeseman, I.M, Fukagawa, T.
Deposit date:2011-06-08
Release date:2012-03-07
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.197 Å)
Cite:CENP-T-W-S-X Forms a Unique Centromeric Chromatin Structure with a Histone-like Fold.
Cell(Cambridge,Mass.), 148, 2012
2ZK1
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BU of 2zk1 by Molmil
Human peroxisome proliferator-activated receptor gamma ligand binding domain complexed with 15-deoxy-delta12,14-prostaglandin J2
Descriptor: (5E,14E)-11-oxoprosta-5,9,12,14-tetraen-1-oic acid, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Fujimoto, Y, Morikawa, K.
Deposit date:2008-03-12
Release date:2009-02-24
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.61 Å)
Cite:Structural insight into PPARgamma activation through covalent modification with endogenous fatty acids
J.Mol.Biol., 385, 2009
2ZK4
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BU of 2zk4 by Molmil
Human peroxisome proliferator-activated receptor gamma ligand binding domain complexed with 15-oxo-eicosatetraenoic acid
Descriptor: (5E,8E,11Z,13E)-15-oxoicosa-5,8,11,13-tetraenoic acid, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Fujimoto, Y, Morikawa, K.
Deposit date:2008-03-12
Release date:2009-02-24
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.57 Å)
Cite:Structural insight into PPARgamma activation through covalent modification with endogenous fatty acids
J.Mol.Biol., 385, 2009
2ZK0
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BU of 2zk0 by Molmil
Human peroxisome proliferator-activated receptor gamma ligand binding domain
Descriptor: Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Fujimoto, Y, Morikawa, K.
Deposit date:2008-03-12
Release date:2009-02-24
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.36 Å)
Cite:Structural insight into PPARgamma activation through covalent modification with endogenous fatty acids
J.Mol.Biol., 385, 2009
2ZK6
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BU of 2zk6 by Molmil
Human peroxisome proliferator-activated receptor gamma ligand binding domain complexed with C8-BODIPY
Descriptor: Peroxisome proliferator-activated receptor gamma, difluoro(5-{2-[(5-octyl-1H-pyrrol-2-yl-kappaN)methylidene]-2H-pyrrol-5-yl-kappaN}pentanoato)boron
Authors:Waku, T, Shiraki, T, Oyama, T, Fujimoto, Y, Morikawa, K.
Deposit date:2008-03-12
Release date:2009-02-24
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.41 Å)
Cite:The nuclear receptor PPARgamma individually responds to serotonin- and fatty acid-metabolites
Embo J., 29, 2010
2ZVT
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BU of 2zvt by Molmil
Cys285Ser mutant PPARgamma ligand-binding domain complexed with 15-deoxy-delta12,14-prostaglandin J2
Descriptor: (5E,14E)-11-oxoprosta-5,9,12,14-tetraen-1-oic acid, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Oyama, T, Shiraki, T, Morikawa, K.
Deposit date:2008-11-19
Release date:2009-10-06
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Atomic structure of mutant PPARgamma LBD complexed with 15d-PGJ2: novel modulation mechanism of PPARgamma/RXRalpha function by covalently bound ligands
Febs Lett., 583, 2009
2ZK5
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BU of 2zk5 by Molmil
Human peroxisome proliferator-activated receptor gamma ligand binding domain complexed with nitro-233
Descriptor: 3-[5-(2-nitropent-1-en-1-yl)furan-2-yl]benzoic acid, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Fujimoto, Y, Morikawa, K.
Deposit date:2008-03-12
Release date:2009-02-24
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.45 Å)
Cite:Structural insight into PPARgamma activation through covalent modification with endogenous fatty acids
J.Mol.Biol., 385, 2009
3ADT
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BU of 3adt by Molmil
Human PPARgamma ligand-binding domain in complex with 5-hydroxy-indole acetate
Descriptor: (5-hydroxy-1H-indol-3-yl)acetic acid, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Morikawa, K.
Deposit date:2010-01-29
Release date:2010-12-22
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:The nuclear receptor PPARgamma individually responds to serotonin- and fatty acid-metabolites
Embo J., 29, 2010
3ADU
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BU of 3adu by Molmil
Human PPARgamma ligand-binding domain in complex with 5-methoxy-indole acetate
Descriptor: (5-methoxy-1H-indol-3-yl)acetic acid, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Morikawa, K.
Deposit date:2010-01-29
Release date:2010-12-22
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.77 Å)
Cite:The nuclear receptor PPARgamma individually responds to serotonin- and fatty acid-metabolites
Embo J., 29, 2010
2ZK3
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BU of 2zk3 by Molmil
Human peroxisome proliferator-activated receptor gamma ligand binding domain complexed with 8-oxo-eicosatetraenoic acid
Descriptor: (5E,11E,14E)-8-oxoicosa-5,9,11,14-tetraenoic acid, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Fujimoto, Y, Morikawa, K.
Deposit date:2008-03-12
Release date:2009-02-24
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.58 Å)
Cite:Structural insight into PPARgamma activation through covalent modification with endogenous fatty acids
J.Mol.Biol., 385, 2009
2ZK2
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BU of 2zk2 by Molmil
Human peroxisome proliferator-activated receptor gamma ligand binding domain complexed with glutathion conjugated 15-deoxy-delta12,14-prostaglandin J2
Descriptor: (5E,14E)-11-oxoprosta-5,9,12,14-tetraen-1-oic acid, GLUTATHIONE, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Fujimoto, Y, Morikawa, K.
Deposit date:2008-03-12
Release date:2009-02-24
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.26 Å)
Cite:Structural insight into PPARgamma activation through covalent modification with endogenous fatty acids
J.Mol.Biol., 385, 2009
3ADV
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BU of 3adv by Molmil
Human PPARgamma ligand-binding domain in complex with serotonin
Descriptor: Peroxisome proliferator-activated receptor gamma, SEROTONIN
Authors:Waku, T, Shiraki, T, Oyama, T, Morikawa, K.
Deposit date:2010-01-29
Release date:2010-12-22
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.27 Å)
Cite:The nuclear receptor PPARgamma individually responds to serotonin- and fatty acid-metabolites
Embo J., 29, 2010
3ADS
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BU of 3ads by Molmil
Human PPARgamma ligand-binding domain in complex with indomethacin
Descriptor: INDOMETHACIN, Peroxisome proliferator-activated receptor gamma
Authors:Waku, T, Shiraki, T, Oyama, T, Morikawa, K.
Deposit date:2010-01-29
Release date:2010-12-22
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:The nuclear receptor PPARgamma individually responds to serotonin- and fatty acid-metabolites
Embo J., 29, 2010

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