1EM2
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1em2 by Molmil](/molmil-images/mine/1em2) | |
1I9Z
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1i9z by Molmil](/molmil-images/mine/1i9z) | CRYSTAL STRUCTURE OF INOSITOL POLYPHOSPHATE 5-PHOSPHATASE DOMAIN (IPP5C) OF SPSYNAPTOJANIN IN COMPLEX WITH INOSITOL (1,4)-BISPHOSPHATE AND CALCIUM ION | 分子名称: | CALCIUM ION, D-MYO-INOSITOL-1,4-BISPHOSPHATE, PHOSPHATIDYLINOSITOL PHOSPHATE PHOSPHATASE | 著者 | Tsujishita, Y, Guo, S, Stolz, L, York, J.D, Hurley, J.H. | 登録日 | 2001-03-21 | 公開日 | 2001-05-16 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Specificity determinants in phosphoinositide dephosphorylation: crystal structure of an archetypal inositol polyphosphate 5-phosphatase. Cell(Cambridge,Mass.), 105, 2001
|
|
1I9Y
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1i9y by Molmil](/molmil-images/mine/1i9y) | CRYSTAL STRUCTURE OF INOSITOL POLYPHOSPHATE 5-PHOSPHATASE DOMAIN (IPP5C) OF SPSYNAPTOJANIN | 分子名称: | PHOSPHATIDYLINOSITOL PHOSPHATE PHOSPHATASE | 著者 | Tsujishita, Y, Guo, S, Stolz, L, York, J.D, Hurley, J.H. | 登録日 | 2001-03-21 | 公開日 | 2001-05-16 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Specificity determinants in phosphoinositide dephosphorylation: crystal structure of an archetypal inositol polyphosphate 5-phosphatase. Cell(Cambridge,Mass.), 105, 2001
|
|
7CMM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7cmm by Molmil](/molmil-images/mine/7cmm) | Crystal structure of TEAD1-YBD in complex with K-975 | 分子名称: | N-[3-(4-chloranylphenoxy)-4-methyl-phenyl]propanamide, Transcriptional enhancer factor TEF-1 | 著者 | Tsuji, Y, Suzuki, M, Yasunaga, M, Hamguchi, K, Saito, J. | 登録日 | 2020-07-28 | 公開日 | 2021-02-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | The novel potent TEAD inhibitor, K-975, inhibits YAP1/TAZ-TEAD protein-protein interactions and exerts an anti-tumor effect on malignant pleural mesothelioma. Am J Cancer Res, 10, 2020
|
|
1EWT
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1ewt by Molmil](/molmil-images/mine/1ewt) | CRYSTAL STRUCTURE OF METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1 LIGAND FREE FORM I | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1, SULFATE ION | 著者 | Kunishima, N, Shimada, Y, Tsuji, Y, Jingami, H, Morikawa, K. | 登録日 | 2000-04-27 | 公開日 | 2000-12-18 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.7 Å) | 主引用文献 | Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor. Nature, 407, 2000
|
|
1EWV
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1ewv by Molmil](/molmil-images/mine/1ewv) | CRYSTAL STRUCTURE OF METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1 LIGAND FREE FORM II | 分子名称: | METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1 | 著者 | Kunishima, N, Shimada, Y, Tsuji, Y, Jingami, H, Morikawa, K. | 登録日 | 2000-04-27 | 公開日 | 2000-12-18 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (4 Å) | 主引用文献 | Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor. Nature, 407, 2000
|
|
2Z6W
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2z6w by Molmil](/molmil-images/mine/2z6w) | Crystal structure of human cyclophilin D in complex with cyclosporin A | 分子名称: | CITRIC ACID, CYCLOSPORIN A, PEPTIDYL-PROLYL CIS-TRANS ISOMERASE | 著者 | Kajitani, K, Fujihashi, M, Kobayashi, Y, Shimizu, S, Tsujimoto, Y, Miki, K. | 登録日 | 2007-08-09 | 公開日 | 2008-04-29 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (0.96 Å) | 主引用文献 | Crystal Structure of Human Cyclophilin D in Complex with its Inhibitor, Cyclosporin a at 0.96-A Resolution. Proteins, 70, 2008
|
|
1EWK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1ewk by Molmil](/molmil-images/mine/1ewk) | CRYSTAL STRUCTURE OF METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1 COMPLEXED WITH GLUTAMATE | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLUTAMIC ACID, ... | 著者 | Kunishima, N, Shimada, Y, Jingami, H, Morikawa, K. | 登録日 | 2000-04-26 | 公開日 | 2000-12-18 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor. Nature, 407, 2000
|
|
5ID8
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5id8 by Molmil](/molmil-images/mine/5id8) | |
5IDB
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5idb by Molmil](/molmil-images/mine/5idb) | |
5IDA
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ida by Molmil](/molmil-images/mine/5ida) | |
1ISR
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1isr by Molmil](/molmil-images/mine/1isr) | Crystal Structure of Metabotropic Glutamate Receptor Subtype 1 Complexed with Glutamate and Gadolinium Ion | 分子名称: | GADOLINIUM ATOM, GLUTAMIC ACID, Metabotropic Glutamate Receptor subtype 1 | 著者 | Tsuchiya, D, Kunishima, N, Kamiya, N, Jingami, H, Morikawa, K. | 登録日 | 2001-12-21 | 公開日 | 2002-03-13 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (4 Å) | 主引用文献 | Structural views of the ligand-binding cores of a metabotropic glutamate receptor complexed with an antagonist and both glutamate and Gd3+. Proc.Natl.Acad.Sci.USA, 99, 2002
|
|
1ISS
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1iss by Molmil](/molmil-images/mine/1iss) | Crystal Structure of Metabotropic Glutamate Receptor Subtype 1 Complexed with an antagonist | 分子名称: | (S)-(ALPHA)-METHYL-4-CARBOXYPHENYLGLYCINE, Metabotropic Glutamate Receptor subtype 1 | 著者 | Tsuchiya, D, Kunishima, N, Kamiya, N, Jingami, H, Morikawa, K. | 登録日 | 2001-12-21 | 公開日 | 2002-03-13 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.3 Å) | 主引用文献 | Structural views of the ligand-binding cores of a metabotropic glutamate receptor complexed with an antagonist and both glutamate and Gd3+. Proc.Natl.Acad.Sci.USA, 99, 2002
|
|
6AHS
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6ahs by Molmil](/molmil-images/mine/6ahs) | Mouse Kallikrein 7 in complex with imidazolinylindole derivative | 分子名称: | 1-[(2-chlorophenyl)sulfonyl]-5-methyl-3-[(4R)-2-methyl-4,5-dihydro-1H-imidazol-4-yl]-1H-indole, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ... | 著者 | Sugawara, H. | 登録日 | 2018-08-20 | 公開日 | 2019-01-02 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Discovery and structure-activity relationship of imidazolinylindole derivatives as kallikrein 7 inhibitors. Bioorg. Med. Chem. Lett., 29, 2019
|
|
2EK9
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2ek9 by Molmil](/molmil-images/mine/2ek9) | |
2EK8
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2ek8 by Molmil](/molmil-images/mine/2ek8) | |
1G5M
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1g5m by Molmil](/molmil-images/mine/1g5m) | HUMAN BCL-2, ISOFORM 1 | 分子名称: | PROTEIN (APOPTOSIS REGULATOR BCL-2 WITH PUTATIVE FLEXIBLE LOOP REPLACED WITH A PORTION OF APOPTOSIS REGULATOR BCL-X PROTEIN) | 著者 | Petros, A.M, Medek, A, Nettesheim, D.G, Kim, D.H, Yoon, H.S, Swift, K, Matayoshi, E.D, Oltersdorf, T, Fesik, S.W. | 登録日 | 2000-11-01 | 公開日 | 2001-03-21 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the antiapoptotic protein bcl-2. Proc.Natl.Acad.Sci.USA, 98, 2001
|
|