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5W6X
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BU of 5w6x by Molmil
Crystal structure of the HsNUDT16 in complex with Mg+2 and ADP-ribose
分子名称: ACETIC ACID, ADENOSINE-5-DIPHOSPHORIBOSE, DI(HYDROXYETHYL)ETHER, ...
著者Thirawatananond, P, Gabelli, S.B.
登録日2017-06-18
公開日2018-12-19
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural analyses of NudT16-ADP-ribose complexes direct rational design of mutants with improved processing of poly(ADP-ribosyl)ated proteins.
Sci Rep, 9, 2019
5VY2
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BU of 5vy2 by Molmil
Crystal structure of the F36A mutant of HsNUDT16
分子名称: SODIUM ION, U8 snoRNA-decapping enzyme
著者Thirawatananond, P, Gabelli, S.B.
登録日2017-05-24
公開日2018-11-21
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural analyses of NudT16-ADP-ribose complexes direct rational design of mutants with improved processing of poly(ADP-ribosyl)ated proteins.
Sci Rep, 9, 2019
7TDZ
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BU of 7tdz by Molmil
Cryo-EM model of protomer of the cytoplasmic ring of the nuclear pore complex from Xenopus laevis
分子名称: Nuclear pore complex protein, Nuclear pore complex protein Nup85, Nuclear pore complex protein Nup96, ...
著者Fontana, P, Wu, H.
登録日2022-01-03
公開日2022-06-22
実験手法ELECTRON MICROSCOPY (6.9 Å)
主引用文献Structure of cytoplasmic ring of nuclear pore complex by integrative cryo-EM and AlphaFold.
Science, 376, 2022
8PQQ
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BU of 8pqq by Molmil
Nucleoside 2'deoxyribosyltransferase from Chroococcidiopsis thermalis PCC 7203 E88Q Mutant bound to Clofarabine
分子名称: 2-CHLORO-9-(2-DEOXY-2-FLUORO-B -D-ARABINOFURANOSYL)-9H-PURIN-6-AMINE, MAGNESIUM ION, Nucleoside 2-deoxyribosyltransferase
著者Tang, P, Harding, C.J, Czekster, M.C.
登録日2023-07-11
公開日2024-02-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献Snapshots of the Reaction Coordinate of a Thermophilic 2'-Deoxyribonucleoside/ribonucleoside Transferase.
Acs Catalysis, 14, 2024
8QC0
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BU of 8qc0 by Molmil
Nucleoside 2'deoxyribosyltransferase from Chroococcidiopsis thermalis PCC 7203 WT ribosylated
分子名称: Nucleoside 2-deoxyribosyltransferase, ZINC ION, alpha-D-ribofuranose
著者Tang, P, Harding, C.J, Czekster, C.M.
登録日2023-08-25
公開日2024-02-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献Snapshots of the Reaction Coordinate of a Thermophilic 2'-Deoxyribonucleoside/ribonucleoside Transferase.
Acs Catalysis, 14, 2024
8RH3
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BU of 8rh3 by Molmil
Nucleoside 2'deoxyribosyltransferase from Chroococcidiopsis thermalis PCC 7203 WT bound to Gemcitabine
分子名称: (2~{R},3~{R})-4,4-bis(fluoranyl)-2-(hydroxymethyl)oxolan-3-ol, Nucleoside 2-deoxyribosyltransferase
著者Tang, P, Harding, C.J, Czekster, C.M.
登録日2023-12-14
公開日2024-02-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Snapshots of the Reaction Coordinate of a Thermophilic 2'-Deoxyribonucleoside/ribonucleoside Transferase.
Acs Catalysis, 14, 2024
8PQP
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BU of 8pqp by Molmil
Nucleoside 2'deoxyribosyltransferase from Chroococcidiopsis thermalis PCC 7203 D62N Mutant bound to ImmH-Forodesine
分子名称: 1,4-DIDEOXY-4-AZA-1-(S)-(9-DEAZAHYPOXANTHIN-9-YL)-D-RIBITOL, Nucleoside 2-deoxyribosyltransferase
著者Tang, P, Harding, C.J, Czekster, M.C.
登録日2023-07-11
公開日2024-02-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.709 Å)
主引用文献Snapshots of the Reaction Coordinate of a Thermophilic 2'-Deoxyribonucleoside/ribonucleoside Transferase.
Acs Catalysis, 14, 2024
8PQR
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Nucleoside 2'deoxyribosyltransferase from Chroococcidiopsis thermalis PCC 7203 WT bound to DAD_Immucillin-H
分子名称: 7-[[(3R,4R)-3-(hydroxymethyl)-4-oxidanyl-pyrrolidin-1-ium-1-yl]methyl]-3,5-dihydropyrrolo[3,2-d]pyrimidin-4-one, Nucleoside 2-deoxyribosyltransferase
著者Tang, P, Harding, C.J, Czekster, C.M.
登録日2023-07-11
公開日2024-02-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.586 Å)
主引用文献Snapshots of the Reaction Coordinate of a Thermophilic 2'-Deoxyribonucleoside/ribonucleoside Transferase.
Acs Catalysis, 14, 2024
8PQT
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BU of 8pqt by Molmil
Nucleoside 2'deoxyribosyltransferase from Chroococcidiopsis thermalis PCC 7203 WT bound to Bis-Tris
分子名称: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Nucleoside 2-deoxyribosyltransferase
著者Tang, P, Harding, C.J, Czekster, C.M.
登録日2023-07-11
公開日2024-02-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Snapshots of the Reaction Coordinate of a Thermophilic 2'-Deoxyribonucleoside/ribonucleoside Transferase.
Acs Catalysis, 14, 2024
8PQS
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BU of 8pqs by Molmil
Nucleoside 2'deoxyribosyltransferase from Chroococcidiopsis thermalis PCC 7203 E88A Mutant
分子名称: Nucleoside 2-deoxyribosyltransferase
著者Tang, P, Harding, C.J, Czekster, C.M.
登録日2023-07-11
公開日2024-02-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Snapshots of the Reaction Coordinate of a Thermophilic 2'-Deoxyribonucleoside/ribonucleoside Transferase.
Acs Catalysis, 14, 2024
5WJI
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BU of 5wji by Molmil
Crystal structure of the F61S mutant of HsNUDT16
分子名称: ACETIC ACID, CHLORIDE ION, SULFATE ION, ...
著者Thirawatananond, P, Gabelli, S.B.
登録日2017-07-23
公開日2018-10-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural analyses of NudT16-ADP-ribose complexes direct rational design of mutants with improved processing of poly(ADP-ribosyl)ated proteins.
Sci Rep, 9, 2019
5W6Z
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BU of 5w6z by Molmil
Crystal structure of the H24W mutant of HsNUDT16
分子名称: SODIUM ION, U8 snoRNA-decapping enzyme
著者Thirawatananond, P, Gabelli, S.B.
登録日2017-06-18
公開日2018-12-19
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.61 Å)
主引用文献Structural analyses of NudT16-ADP-ribose complexes direct rational design of mutants with improved processing of poly(ADP-ribosyl)ated proteins.
Sci Rep, 9, 2019
1QHG
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BU of 1qhg by Molmil
STRUCTURE OF DNA HELICASE MUTANT WITH ADPNP
分子名称: ADENOSINE-5'-TRIPHOSPHATE, ATP-DEPENDENT HELICASE PCRA, MAGNESIUM ION
著者Soultanas, P, Dillingham, M.S, Velankar, S.S, Wigley, D.B.
登録日1999-05-14
公開日1999-07-13
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献DNA binding mediates conformational changes and metal ion coordination in the active site of PcrA helicase.
J.Mol.Biol., 290, 1999
1QHH
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BU of 1qhh by Molmil
STRUCTURE OF DNA HELICASE WITH ADPNP
分子名称: ADENOSINE-5'-TRIPHOSPHATE, PROTEIN (PCRA (SUBUNIT))
著者Soultanas, P, Dillingham, M.S, Velankar, S.S, Wigley, D.B.
登録日1999-05-14
公開日1999-07-13
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献DNA binding mediates conformational changes and metal ion coordination in the active site of PcrA helicase.
J.Mol.Biol., 290, 1999
7DJR
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BU of 7djr by Molmil
Crystal structure of SARS-CoV-2 main protease (no ligand)
分子名称: 3C-like proteinase, DIMETHYL SULFOXIDE
著者Deetanya, P, Wangkanont, K.
登録日2020-11-21
公開日2021-06-16
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Interaction of 8-anilinonaphthalene-1-sulfonate with SARS-CoV-2 main protease and its application as a fluorescent probe for inhibitor identification.
Comput Struct Biotechnol J, 19, 2021
3D4F
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BU of 3d4f by Molmil
SHV-1 beta-lactamase complex with LN1-255
分子名称: (3R)-4-{[(3,4-dihydroxyphenyl)acetyl]oxy}-N-(2-formylindolizin-3-yl)-3-sulfino-D-valine, Beta-lactamase SHV-1, CYCLOHEXYL-HEXYL-BETA-D-MALTOSIDE
著者Pattanaik, P, Bethel, C.R, Hujer, A.M, Bonomo, R.A, Buynak, J.D, van den Akker, F.
登録日2008-05-14
公開日2009-02-10
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Strategic Design of an Effective {beta}-Lactamase Inhibitor: LN-1-255, A 6-ALKYLIDENE-2'-SUBSTITUTED PENICILLIN SULFONE
J.Biol.Chem., 284, 2009
6B09
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BU of 6b09 by Molmil
Crystal structure of HsNUDT16 in complex with diADPR (soaked)
分子名称: CHLORIDE ION, MAGNESIUM ION, SODIUM ION, ...
著者Thirawatananond, P, Gabelli, S.B.
登録日2017-09-14
公開日2019-01-09
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural analyses of NudT16-ADP-ribose complexes direct rational design of mutants with improved processing of poly(ADP-ribosyl)ated proteins.
Sci Rep, 9, 2019
5I8U
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BU of 5i8u by Molmil
Crystal Structure of the RV1700 (MT ADPRASE) E142Q mutant
分子名称: ADP-ribose pyrophosphatase, DI(HYDROXYETHYL)ETHER, FORMIC ACID, ...
著者Thirawatananond, P, Kang, L.-W, Amzel, L.M, Gabelli, S.B.
登録日2016-02-19
公開日2016-10-12
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Kinetic and mutational studies of the adenosine diphosphate ribose hydrolase from Mycobacterium tuberculosis.
J. Bioenerg. Biomembr., 48, 2016
8ADK
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BU of 8adk by Molmil
Poly(ADP-ribose) glycohydrolase (PARG) from Drosophila melanogaster
分子名称: CHLORIDE ION, GLYCEROL, Poly(ADP-ribose) glycohydrolase, ...
著者Ariza, A, Fontana, P.
登録日2022-07-08
公開日2023-06-14
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.474 Å)
主引用文献Serine ADP-ribosylation in Drosophila provides insights into the evolution of reversible ADP-ribosylation signalling.
Nat Commun, 14, 2023
8ADJ
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BU of 8adj by Molmil
Poly(ADP-ribose) glycohydrolase (PARG) from Drosophila melanogaster in complex with PARG inhibitor PDD00017272
分子名称: 1-[(2,5-dimethylpyrazol-3-yl)methyl]-N-(1-methylcyclopropyl)-3-[(2-methyl-1,3-thiazol-5-yl)methyl]-2,4-bis(oxidanylidene)quinazoline-6-sulfonamide, CHLORIDE ION, GLYCEROL, ...
著者Ariza, A, Fontana, P.
登録日2022-07-08
公開日2023-06-14
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.508 Å)
主引用文献Serine ADP-ribosylation in Drosophila provides insights into the evolution of reversible ADP-ribosylation signalling.
Nat Commun, 14, 2023
4GD8
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BU of 4gd8 by Molmil
SHV-1 beta-lactamase in complex with penam sulfone SA3-53
分子名称: (2S,3R)-4-(2-aminoethylcarbamoyloxy)-2-[(2-methanoylindolizin-3-yl)amino]-3-methyl-3-sulfino-butanoic acid, Beta-lactamase SHV-1, CYCLOHEXYL-HEXYL-BETA-D-MALTOSIDE
著者Pattanaik, P, van den Akker, F.
登録日2012-07-31
公開日2013-07-31
最終更新日2013-08-07
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structures of SHV-1 beta-lactamase with penem and penam sulfone inhibitors that form cyclic intermediates stabilized by carbonyl conjugation
Plos One, 7, 2012
2JGB
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BU of 2jgb by Molmil
Structure of human eIF4E homologous protein 4EHP with m7GTP
分子名称: 7N-METHYL-8-HYDROGUANOSINE-5'-TRIPHOSPHATE, EUKARYOTIC TRANSLATION INITIATION FACTOR 4E TYPE 2, EUKARYOTIC TRANSLATION INITIATION FACTOR 4E-BINDING PROTEIN 1
著者Cameron, A.D, Rosettani, P, Knapp, S, Vismara, M.G, Rusconi, L.
登録日2007-02-12
公開日2007-02-27
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structures of the human eIF4E homologous protein, h4EHP, in its m7GTP-bound and unliganded forms.
J. Mol. Biol., 368, 2007
2JGC
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BU of 2jgc by Molmil
Structure of the human eIF4E homologous protein, 4EHP without ligand bound
分子名称: EUKARYOTIC TRANSLATION INITIATION FACTOR 4E TYPE 2, EUKARYOTIC TRANSLATION INITIATION FACTOR 4E-BINDING PROTEIN 1
著者Cameron, A.D, Rosettani, P, Knapp, S, Vismara, M.G, Rusconi, L.
登録日2007-02-12
公開日2007-02-27
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structures of the human eIF4E homologous protein, h4EHP, in its m7GTP-bound and unliganded forms.
J. Mol. Biol., 368, 2007
6CDU
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BU of 6cdu by Molmil
Crystal structure of a chimeric human alpha1GABAA receptor in complex with alphaxalone
分子名称: (3a,5a)-3-Hydroxypregnane-11,20-dione, chimeric alpha1GABAA receptor
著者Chen, Q, Arjunan, P, Cohen, A.E, Xu, Y, Tang, P.
登録日2018-02-09
公開日2018-08-22
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.45 Å)
主引用文献Structural basis of neurosteroid anesthetic action on GABAAreceptors.
Nat Commun, 9, 2018
6IZT
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BU of 6izt by Molmil
Crystal structure of Haemophilus Influenzae BamA POTRA3-5
分子名称: Outer membrane protein assembly factor BamA
著者Ma, X, Wang, Q, Li, Y, Tan, P, Wu, H, Wang, P, Dong, X, Hong, L, Meng, G.
登録日2018-12-20
公開日2019-10-30
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献How BamA recruits OMP substratesviapoly-POTRAs domain.
Faseb J., 33, 2019

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