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5B18
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BU of 5b18 by Molmil
Crystal Structure of a Darunavir Resistant HIV-1 Protease
分子名称: ACETATE ION, CHLORIDE ION, Protease
著者Suzuki, K, Ode, H, Nakashima, M, Sugiura, W, Watanabe, N, Suzuki, A, Iwatani, Y.
登録日2015-11-30
公開日2016-04-13
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Unique Flap Conformation in an HIV-1 Protease with High-Level Darunavir Resistance
Front Microbiol, 7, 2016
3D3T
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BU of 3d3t by Molmil
Crystal Structure of HIV-1 CRF01_AE in complex with the substrate p1-p6
分子名称: HIV-1 protease, P1-P6 SUBSTRATE PEPTIDE
著者Bandaranayake, R.M, Prabu-Jeyabalan, M, Kakizawa, J, Sugiura, W, Schiffer, C.A.
登録日2008-05-12
公開日2008-07-08
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural analysis of human immunodeficiency virus type 1 CRF01_AE protease in complex with the substrate p1-p6.
J.Virol., 82, 2008
3VM8
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BU of 3vm8 by Molmil
Crystal structure of the human APOBEC3C having HIV-1 Vif-binding interface
分子名称: Probable DNA dC->dU-editing enzyme APOBEC-3C, ZINC ION
著者Kitamura, S, Suzuki, A, Watanabe, N, Iwatani, Y.
登録日2011-12-09
公開日2012-10-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal structure of the human APOBEC3C having HIV-1 Vif-binding interface
To be Published
3LZU
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BU of 3lzu by Molmil
Crystal Structure of a Nelfinavir Resistant HIV-1 CRF01_AE Protease variant (N88S) in Complex with the Protease Inhibitor Darunavir.
分子名称: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, ACETATE ION, HIV-1 protease
著者Schiffer, C.A, Bandaranayake, R.M.
登録日2010-03-01
公開日2010-08-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.76 Å)
主引用文献The Effect of Clade-Specific Sequence Polymorphisms on HIV-1 Protease Activity and Inhibitor Resistance Pathways.
J.Virol., 84, 2010
3LZV
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BU of 3lzv by Molmil
Structure of Nelfinavir-resistant HIV-1 protease (D30N/N88D) in complex with Darunavir.
分子名称: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, ACETATE ION, HIV-1 Protease, ...
著者Schiffer, C.A, Kolli, M.
登録日2010-03-01
公開日2010-08-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献The Effect of Clade-Specific Sequence Polymorphisms on HIV-1 Protease Activity and Inhibitor Resistance Pathways.
J.Virol., 84, 2010
3VOW
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BU of 3vow by Molmil
Crystal Structure of the Human APOBEC3C having HIV-1 Vif-binding Interface
分子名称: CHLORIDE ION, Probable DNA dC->dU-editing enzyme APOBEC-3C, ZINC ION
著者Kitamura, S, Suzuki, A, Watanabe, N, Iwatani, Y.
登録日2012-02-22
公開日2012-10-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献The APOBEC3C crystal structure and the interface for HIV-1 Vif binding.
Nat.Struct.Mol.Biol., 19, 2012
3WUS
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BU of 3wus by Molmil
Crystal Structure of the Vif-Binding Domain of Human APOBEC3F
分子名称: DNA dC->dU-editing enzyme APOBEC-3F, ZINC ION
著者Nakashima, M, Kawamura, T, Ode, H, Watanabe, N, Iwatani, Y.
登録日2014-05-02
公開日2015-06-24
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.54 Å)
主引用文献Structural Insights into HIV-1 Vif-APOBEC3F Interaction.
J.Virol., 90, 2015
3LZS
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BU of 3lzs by Molmil
Crystal Structure of HIV-1 CRF01_AE Protease in Complex with Darunavir
分子名称: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, ACETATE ION, HIV-1 protease
著者Schiffer, C.A, Bandaranayake, R.M.
登録日2010-03-01
公開日2010-08-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献The Effect of Clade-Specific Sequence Polymorphisms on HIV-1 Protease Activity and Inhibitor Resistance Pathways.
J.Virol., 84, 2010

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件を2024-07-17に公開中

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