3KPX
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![BU of 3kpx by Molmil](/molmil-images/mine/3kpx) | Crystal Structure Analysis of photoprotein clytin | 分子名称: | Apophotoprotein clytin-3, C2-HYDROPEROXY-COELENTERAZINE, CALCIUM ION | 著者 | Titushin, M.S, Li, Y, Stepanyuk, G.A, Wang, B.-C, Lee, J, Vysotski, E.S, Liu, Z.-J. | 登録日 | 2009-11-17 | 公開日 | 2010-10-06 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.899 Å) | 主引用文献 | NMR derived topology of a GFP-photoprotein energy transfer complex J.Biol.Chem., 285, 2010
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3Q8W
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![BU of 3q8w by Molmil](/molmil-images/mine/3q8w) | A b-aminoacyl containing thiazolidine derivative and DPPIV complex | 分子名称: | Dipeptidyl peptidase 4, N-(4-{[({(2R)-3-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-1,3-thiazolidin-2-yl}carbonyl)amino]methyl}phenyl)-D-valine | 著者 | Lee, J.O, Song, D.H. | 登録日 | 2011-01-07 | 公開日 | 2011-03-16 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (3.64 Å) | 主引用文献 | Discovery of b-aminoacyl containing thiazolidine derivatives as potent and selective dipeptidyl peptidase IV inhibitors To be Published
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3EIO
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![BU of 3eio by Molmil](/molmil-images/mine/3eio) | Crystal Structure Analysis of DPPIV Inhibitor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-({4-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-1,4-diazepan-1-yl}carbonyl)benzoic acid, ... | 著者 | Ahn, J.H, Lee, J.-O. | 登録日 | 2008-09-17 | 公開日 | 2008-11-04 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Synthesis and biological evaluation of homopiperazine derivatives with beta-aminoacyl group as dipeptidyl peptidase IV inhibitors Bioorg.Med.Chem.Lett., 18, 2008
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2OLE
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![BU of 2ole by Molmil](/molmil-images/mine/2ole) | Crystal Structure Of Human Dipeptidyl Peptidase IV (DPPIV) Complex With Cyclic Hydrazine Derivatives | 分子名称: | (2R)-4-(2-BENZOYL-1,2-DIAZEPAN-1-YL)-4-OXO-1-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-AMINE, Dipeptidyl peptidase 4 | 著者 | Kim, S.S, Ahn, J.H, Lee, J.O. | 登録日 | 2007-01-19 | 公開日 | 2008-01-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Synthesis, biological evaluation and structural determination of beta-aminoacyl-containing cyclic hydrazine derivatives as dipeptidyl peptidase IV (DPP-IV) inhibitors Bioorg.Med.Chem.Lett., 17, 2007
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4GKF
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![BU of 4gkf by Molmil](/molmil-images/mine/4gkf) | Crystal structure and characterization of Cmr5 protein from Pyrococcus furiosus | 分子名称: | CRISPR system Cmr subunit Cmr5 | 著者 | Park, J, Sun, J, Park, S, Hwang, H, Park, M, Shin, M.S. | 登録日 | 2012-08-11 | 公開日 | 2013-01-23 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structure of Cmr5 from Pyrococcus furiosus and its functional implications Febs Lett., 587, 2013
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8VUW
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![BU of 8vuw by Molmil](/molmil-images/mine/8vuw) | ELIC5 with cysteamine in 2:1:1 POPC:POPE:POPG nanodisc in open conformation | 分子名称: | (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, 2-AMINO-ETHANETHIOL, Erwinia chrysanthemi ligand-gated ion channel | 著者 | Petroff II, J.T, Deng, Z, Rau, M.J, Fitzpatrick, J.A.J, Yuan, P, Cheng, W.W.L. | 登録日 | 2024-01-29 | 公開日 | 2024-02-07 | 実験手法 | ELECTRON MICROSCOPY (3.19 Å) | 主引用文献 | Open-channel structure of a pentameric ligand-gated ion channel reveals a mechanism of leaflet-specific phospholipid modulation. Nat Commun, 13, 2022
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8D64
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![BU of 8d64 by Molmil](/molmil-images/mine/8d64) | ELIC with cysteamine in POPC nanodisc | 分子名称: | 2-AMINO-ETHANETHIOL, Erwinia ligand-gated ion channel | 著者 | Petroff II, J.T, Deng, Z, Rau, M.J, Fitzpatrick, J.A.J, Yuan, P, Cheng, W.W.L. | 登録日 | 2022-06-06 | 公開日 | 2022-11-23 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.14 Å) | 主引用文献 | Open-channel structure of a pentameric ligand-gated ion channel reveals a mechanism of leaflet-specific phospholipid modulation. Nat Commun, 13, 2022
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8D67
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![BU of 8d67 by Molmil](/molmil-images/mine/8d67) | ELIC3 with cysteamine in 2:1:1 POPC:POPE:POPG nanodisc | 分子名称: | 2-AMINO-ETHANETHIOL, Erwinia ligand-gated ion channel | 著者 | Petroff II, J.T, Deng, Z, Rau, M.J, Fitzpatrick, J.A.J, Yuan, P, Cheng, W.W.L. | 登録日 | 2022-06-06 | 公開日 | 2022-11-23 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Open-channel structure of a pentameric ligand-gated ion channel reveals a mechanism of leaflet-specific phospholipid modulation. Nat Commun, 13, 2022
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8D66
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![BU of 8d66 by Molmil](/molmil-images/mine/8d66) | ELIC with cysteamine in 2:1:1 POPC:POPE:POPG nanodisc | 分子名称: | (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, 2-AMINO-ETHANETHIOL, Erwinia ligand-gated ion channel | 著者 | Petroff II, J.T, Deng, Z, Rau, M.J, Fitzpatrick, J.A.J, Yuan, P, Cheng, W.W.L. | 登録日 | 2022-06-06 | 公開日 | 2022-11-23 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.14 Å) | 主引用文献 | Open-channel structure of a pentameric ligand-gated ion channel reveals a mechanism of leaflet-specific phospholipid modulation. Nat Commun, 13, 2022
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8D65
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![BU of 8d65 by Molmil](/molmil-images/mine/8d65) | ELIC apo in 2:1:1 POPC:POPE:POPG nanodisc | 分子名称: | (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, Erwinia ligand-gated ion channel | 著者 | Petroff II, J.T, Deng, Z, Rau, M.J, Fitzpatrick, J.A.J, Yuan, P, Cheng, W.W.L. | 登録日 | 2022-06-06 | 公開日 | 2022-11-23 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.47 Å) | 主引用文献 | Open-channel structure of a pentameric ligand-gated ion channel reveals a mechanism of leaflet-specific phospholipid modulation. Nat Commun, 13, 2022
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8D63
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![BU of 8d63 by Molmil](/molmil-images/mine/8d63) | ELIC apo in POPC nanodisc | 分子名称: | 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine, Erwinia ligand-gated ion channel | 著者 | Petroff II, J.T, Deng, Z, Rau, M.J, Fitzpatrick, J.A.J, Yuan, P, Cheng, W.W.L. | 登録日 | 2022-06-06 | 公開日 | 2022-11-23 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.14 Å) | 主引用文献 | Open-channel structure of a pentameric ligand-gated ion channel reveals a mechanism of leaflet-specific phospholipid modulation. Nat Commun, 13, 2022
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