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8GB1
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BU of 8gb1 by Molmil
Crystal structure of SAMHD1 dimer bound to deoxyguanosine linked inhibitor
分子名称: 5'-O-[(R)-(3-{[(1M)-3'-bromo[1,1'-biphenyl]-3-carbonyl]amino}propoxy)(hydroxy)phosphoryl]-2'-deoxyguanosine, Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, FE (III) ION
著者Egleston, M, Dong, L, Howlader, A.H, Bhat, S, Orris, B, Bianchet, M.A, Greenberg, M.M, Stivers, J.T.
登録日2023-02-24
公開日2023-06-07
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.46 Å)
主引用文献Deoxyguanosine-Linked Bifunctional Inhibitor of SAMHD1 dNTPase Activity and Nucleic Acid Binding.
Acs Chem.Biol., 18, 2023
8GB2
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BU of 8gb2 by Molmil
Crystal structure of Apo-SAMHD1
分子名称: Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, FE (III) ION
著者Egleston, M, Dong, L, Howlader, A.H, Bhat, S, Orris, B, Bianchet, M.A, Greenberg, M.M, Stivers, J.T.
登録日2023-02-24
公開日2023-06-07
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (3.07 Å)
主引用文献Deoxyguanosine-Linked Bifunctional Inhibitor of SAMHD1 dNTPase Activity and Nucleic Acid Binding.
Acs Chem.Biol., 18, 2023
6T4D
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BU of 6t4d by Molmil
Crystal structure of Plasmodium falciparum Morn1
分子名称: Morn1, ZINC ION
著者Grishkovskaya, I, Kostan, J, Sajko, S, Morriswood, B, Djinovic-Carugo, K.
登録日2019-10-13
公開日2020-11-18
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Structures of three MORN repeat proteins and a re-evaluation of the proposed lipid-binding properties of MORN repeats.
Plos One, 15, 2020
6T6Q
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BU of 6t6q by Molmil
Crystal structure of Toxoplasma gondii Morn1 (extended conformation).
分子名称: Membrane occupation and recognition nexus protein MORN1
著者Grishkovskaya, I, Kostan, J, Sajko, S, Morriswood, B, Djinovic-Carugo, K.
登録日2019-10-18
公開日2020-11-18
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.902 Å)
主引用文献Structures of three MORN repeat proteins and a re-evaluation of the proposed lipid-binding properties of MORN repeats.
Plos One, 15, 2020
6T68
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BU of 6t68 by Molmil
Crystal structure of Trypanosoma brucei Morn1
分子名称: CHLORIDE ION, MORN repeat-containing protein 1
著者Grishkovskaya, I, Kostan, J, Sajko, S, Morriswood, B, Djinovic-Carugo, K.
登録日2019-10-17
公開日2020-11-18
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.54 Å)
主引用文献Structures of three MORN repeat proteins and a re-evaluation of the proposed lipid-binding properties of MORN repeats.
Plos One, 15, 2020
6T4R
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BU of 6t4r by Molmil
Crystal structure of Trypanosoma brucei Morn1
分子名称: MORN repeat-containing protein 1
著者Grishkovskaya, I, Kostan, J, Sajko, S, Morriswood, B, Djinovic-Carugo, K.
登録日2019-10-14
公開日2020-11-18
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.352 Å)
主引用文献Structures of three MORN repeat proteins and a re-evaluation of the proposed lipid-binding properties of MORN repeats.
Plos One, 15, 2020
6T69
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BU of 6t69 by Molmil
Crystal structure of Toxoplasma gondii Morn1(V shape)
分子名称: 1,2-ETHANEDIOL, GLYCEROL, Membrane occupation and recognition nexus protein MORN1, ...
著者Grishkovskaya, I, Kostan, J, Sajko, S, Morriswood, B, Djinovic-Carugo, K.
登録日2019-10-18
公開日2020-11-18
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structures of three MORN repeat proteins and a re-evaluation of the proposed lipid-binding properties of MORN repeats.
Plos One, 15, 2020
2MEK
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BU of 2mek by Molmil
N-terminal domain of Bilbo1 from Trypanosoma brucei
分子名称: N-TERMINAL DOMAIN OF BILBO1
著者Vidilaseris, K, Morriswood, B, Kontaxis, G, Dong, G.
登録日2013-09-24
公開日2014-01-01
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Structure and assembly mechanism of TbBILBO1, an essential flagellar pocket collar protein
To be Published
8TDW
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BU of 8tdw by Molmil
ssRNA bound SAMHD1 T open
分子名称: Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, FE (III) ION, RNA (5'-R(P*CP*CP*GP*AP*CP*C)-3'), ...
著者Sung, M, Huynh, K, Han, S.
登録日2023-07-05
公開日2023-11-22
最終更新日2023-12-20
実験手法ELECTRON MICROSCOPY (3.04 Å)
主引用文献Guanine-containing ssDNA and RNA induce dimeric and tetrameric structural forms of SAMHD1.
Nucleic Acids Res., 51, 2023
8TDV
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BU of 8tdv by Molmil
ssRNA bound SAMHD1 T closed
分子名称: Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, FE (III) ION, RNA (5'-R(P*CP*CP*GP*AP*CP*CP*C)-3'), ...
著者Sung, M, Huynh, K, Han, S.
登録日2023-07-05
公開日2023-12-20
実験手法ELECTRON MICROSCOPY (3.44 Å)
主引用文献Guanine-containing ssDNA and RNA induce dimeric and tetrameric structural forms of SAMHD1.
Nucleic Acids Res., 51, 2023
7UJN
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BU of 7ujn by Molmil
Structure of Human SAMHD1 with Non-Hydrolysable dGTP Analog
分子名称: 2'-deoxyguanosine-5'-O-(1-thiotriphosphate), Deoxynucleoside triphosphate triphosphohydrolase SAMHD1
著者Huynh, K.W, Ammirati, M, Han, S.
登録日2022-03-31
公開日2022-07-20
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (2.89 Å)
主引用文献Phosphorylation of SAMHD1 Thr592 increases C-terminal domain dynamics, tetramer dissociation and ssDNA binding kinetics.
Nucleic Acids Res., 50, 2022
1N0Z
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BU of 1n0z by Molmil
Solution structure of the first zinc-finger domain from ZNF265
分子名称: ZINC ION, ZNF265
著者Plambeck, C.A, Fairley, K, Kwan, A.H.Y, Westman, B.J, Adams, D, Morris, B, Mackay, J.P.
登録日2002-10-15
公開日2003-07-22
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献The structure of the zinc finger domain from human splicing factor ZNF265 fold
J.BIOL.CHEM., 278, 2003
5G5J
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BU of 5g5j by Molmil
Crystal structure of human CYP3A4 bound to metformin
分子名称: CYTOCHROME P450 3A4, Metformin, PROTOPORPHYRIN IX CONTAINING FE
著者Sevrioukova, I.
登録日2016-05-25
公開日2017-06-07
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Heme Binding Biguanides Target Cytochrome P450-Dependent Cancer Cell Mitochondria.
Cell Chem Biol, 24, 2017

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件を2024-07-10に公開中

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