2P86
| The high resolution crystal structure of rhodesain, the major cathepsin L protease from T. brucei rhodesiense, bound to inhibitor K11002 | 分子名称: | 1,2-ETHANEDIOL, 3-[[N-[MORPHOLIN-N-YL]-CARBONYL]-PHENYLALANINYL-AMINO]-5- PHENYL-PENTANE-1-SULFONYLBENZENE, Cysteine protease | 著者 | Brinen, L.S, Marion, R. | 登録日 | 2007-03-21 | 公開日 | 2008-04-01 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.16 Å) | 主引用文献 | THE high resolution structure of rhodesain, the major cathepsin L protease from trypanosoma brucei rhodesiense, illustrates the basis for differences in inhibition profiles from other papain family cysteine proteases To be Published
|
|
2O6X
| Crystal Structure of ProCathepsin L1 from Fasciola hepatica | 分子名称: | Secreted cathepsin L 1 | 著者 | Brinen, L.S, Dalton, J.P, Geiger, S, Marion, R, Stack, C.M. | 登録日 | 2006-12-08 | 公開日 | 2007-12-18 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Structural and functional relationships in the virulence-associated cathepsin L proteases of the parasitic liver fluke, Fasciola hepatica. J.Biol.Chem., 283, 2008
|
|
2P7U
| |
3BWK
| Crystal Structure of Falcipain-3 with Its inhibitor, K11017 | 分子名称: | Cysteine protease falcipain-3, N~2~-(morpholin-4-ylcarbonyl)-N-[(3S)-1-phenyl-5-(phenylsulfonyl)pentan-3-yl]-L-leucinamide, SULFATE ION | 著者 | Kerr, I, Lee, J.H, Brinen, L.S. | 登録日 | 2008-01-09 | 公開日 | 2009-01-20 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.42 Å) | 主引用文献 | Vinyl sulfones as antiparasitic agents and a structural basis for drug design. J.Biol.Chem., 284, 2009
|
|
2OZ2
| |