1Q5R
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![BU of 1q5r by Molmil](/molmil-images/mine/1q5r) | The Rhodococcus 20S proteasome with unprocessed pro-peptides | 分子名称: | proteasome alpha-type subunit 1, proteasome beta-type subunit 1 | 著者 | Kwon, Y.D, Nagy, I, Adams, P.D, Baumeister, W, Jap, B.K. | 登録日 | 2003-08-08 | 公開日 | 2003-12-16 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Crystal structures of the Rhodococcus proteasome with and without its pro-peptides: implications for the role of the pro-peptide in proteasome assembly. J.Mol.Biol., 335, 2004
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1Q5Q
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![BU of 1q5q by Molmil](/molmil-images/mine/1q5q) | The Rhodococcus 20S proteasome | 分子名称: | proteasome alpha-type subunit 1, proteasome beta-type subunit 1 | 著者 | Kwon, Y.D, Nagy, I, Adams, P.D, Baumeister, W, Jap, B.K. | 登録日 | 2003-08-08 | 公開日 | 2003-12-16 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structures of the Rhodococcus proteasome with and without its pro-peptides: implications for the role of the pro-peptide in proteasome assembly. J.Mol.Biol., 335, 2004
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4DVS
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![BU of 4dvs by Molmil](/molmil-images/mine/4dvs) | Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with NBD-557 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, N-(4-bromophenyl)-N'-(2,2,6,6-tetramethylpiperidin-4-yl)ethanediamide, ... | 著者 | Kwon, Y.D, Kwong, P.D. | 登録日 | 2012-02-23 | 公開日 | 2013-02-27 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site. Plos One, 9, 2014
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4DVW
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![BU of 4dvw by Molmil](/molmil-images/mine/4dvw) | Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with MAE-II-167 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, N-(4-chloro-3-fluorophenyl)-N'-[(3aS,6aS)-hexahydrocyclopenta[c]pyrrol-3a(1H)-ylmethyl]ethanediamide, ... | 著者 | Kwon, Y.D, Kwong, P.D. | 登録日 | 2012-02-23 | 公開日 | 2013-02-27 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site. Plos One, 9, 2014
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4DVR
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![BU of 4dvr by Molmil](/molmil-images/mine/4dvr) | |
4DVV
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![BU of 4dvv by Molmil](/molmil-images/mine/4dvv) | Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with AS-I-261 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, N-{[(4S,5S)-5-(aminomethyl)-2,2-dimethyl-1,3-dioxolan-4-yl]methyl}-N'-(4-chloro-3-fluorophenyl)ethanediamide, ... | 著者 | Kwon, Y.D, Kwong, P.D. | 登録日 | 2012-02-23 | 公開日 | 2013-02-27 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site. Plos One, 9, 2014
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4DVT
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![BU of 4dvt by Molmil](/molmil-images/mine/4dvt) | Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with AS-II-37 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, N-(4-chloro-3-fluorophenyl)-N'-[(1S)-1,2,3,4-tetrahydroisoquinolin-1-ylmethyl]ethanediamide, ... | 著者 | Kwon, Y.D, Kwong, P.D. | 登録日 | 2012-02-23 | 公開日 | 2013-02-27 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site. Plos One, 9, 2014
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4DVX
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![BU of 4dvx by Molmil](/molmil-images/mine/4dvx) | Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with MAE-II-188 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, N-(4-chloro-3-fluorophenyl)-N'-{[(3R)-1-cyclopropylpyrrolidin-3-yl]methyl}ethanediamide, ... | 著者 | Kwon, Y.D, Kwong, P.D. | 登録日 | 2012-02-23 | 公開日 | 2013-02-27 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site. Plos One, 9, 2014
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3TGR
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![BU of 3tgr by Molmil](/molmil-images/mine/3tgr) | |
3TGT
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![BU of 3tgt by Molmil](/molmil-images/mine/3tgt) | Crystal structure of unliganded HIV-1 clade A/E strain 93TH057 gp120 core | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, HIV-1 clade A/E 93TH057 gp120 | 著者 | Kwon, Y.D, Kwong, P.D. | 登録日 | 2011-08-17 | 公開日 | 2012-04-04 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Unliganded HIV-1 gp120 core structures assume the CD4-bound conformation with regulation by quaternary interactions and variable loops. Proc.Natl.Acad.Sci.USA, 109, 2012
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3TGQ
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![BU of 3tgq by Molmil](/molmil-images/mine/3tgq) | |
3TGS
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![BU of 3tgs by Molmil](/molmil-images/mine/3tgs) | Crystal structure of HIV-1 clade C strain C1086 gp120 core in complex with NBD-556 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, HIV-1 clade C1086 gp120 core, N-(4-chlorophenyl)-N'-(2,2,6,6-tetramethylpiperidin-4-yl)ethanediamide | 著者 | Kwon, Y.D, Kwong, P.D. | 登録日 | 2011-08-17 | 公開日 | 2012-04-04 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Unliganded HIV-1 gp120 core structures assume the CD4-bound conformation with regulation by quaternary interactions and variable loops. Proc.Natl.Acad.Sci.USA, 109, 2012
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3TIH
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![BU of 3tih by Molmil](/molmil-images/mine/3tih) | |
5WDF
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![BU of 5wdf by Molmil](/molmil-images/mine/5wdf) | |
7TYZ
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![BU of 7tyz by Molmil](/molmil-images/mine/7tyz) | Cryo-EM structure of SARS-CoV-2 spike in complex with FSR22, an anti-SARS-CoV-2 DARPin | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, DARPin FSR22, ... | 著者 | Kwon, Y.D, Gorman, J, Kwong, P.D. | 登録日 | 2022-02-15 | 公開日 | 2022-12-07 | 最終更新日 | 2023-03-15 | 実験手法 | ELECTRON MICROSCOPY (3.51 Å) | 主引用文献 | A potent and broad neutralization of SARS-CoV-2 variants of concern by DARPins. Nat.Chem.Biol., 19, 2023
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7TZ0
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![BU of 7tz0 by Molmil](/molmil-images/mine/7tz0) | |
4RZ8
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![BU of 4rz8 by Molmil](/molmil-images/mine/4rz8) | Crystal structure of HIV-1 gp120 core in complex with NBD-11021, a small molecule CD4-antagonist | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 5-(4-chlorophenyl)-N-{(S)-[5-(hydroxymethyl)-4-methyl-1,3-thiazol-2-yl][(2R)-piperidin-2-yl]methyl}-1H-pyrrole-2-carboxamide, ... | 著者 | Kwon, Y.D, Debnath, A.K, Kwong, P.D. | 登録日 | 2014-12-18 | 公開日 | 2015-09-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-Based Design of a Small Molecule CD4-Antagonist with Broad Spectrum Anti-HIV-1 Activity. J.Med.Chem., 58, 2015
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8DW2
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![BU of 8dw2 by Molmil](/molmil-images/mine/8dw2) | Cryo-EM structure of SARS-CoV-2 RBD in complex with anti-SARS-CoV-2 DARPin,SR22, and two antibody Fabs, S309 and CR3022 | 分子名称: | Antibody CR3022 heavy chain, Antibody CR3022 light chain, Antibody S309 heavy chain, ... | 著者 | Kwon, Y.D, Gorman, J, Kwong, P.D. | 登録日 | 2022-07-30 | 公開日 | 2022-12-07 | 最終更新日 | 2023-03-15 | 実験手法 | ELECTRON MICROSCOPY (4.11 Å) | 主引用文献 | A potent and broad neutralization of SARS-CoV-2 variants of concern by DARPins. Nat.Chem.Biol., 19, 2023
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8DW3
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![BU of 8dw3 by Molmil](/molmil-images/mine/8dw3) | Cryo-EM structure of SARS-CoV-2 RBD in complex with anti-SARS-CoV-2 DARPin,SR16m, and two antibody Fabs, S309 and CR3022 | 分子名称: | Anti-SARS-CoV-2 DARPin SR16m, Antibody S309 light chain, Spike protein S1, ... | 著者 | Kwon, Y.D, Gorman, J, Kwong, P.D. | 登録日 | 2022-07-30 | 公開日 | 2022-12-07 | 最終更新日 | 2023-03-15 | 実験手法 | ELECTRON MICROSCOPY (4.26 Å) | 主引用文献 | A potent and broad neutralization of SARS-CoV-2 variants of concern by DARPins. Nat.Chem.Biol., 19, 2023
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8FA0
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![BU of 8fa0 by Molmil](/molmil-images/mine/8fa0) | |
8F9Z
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![BU of 8f9z by Molmil](/molmil-images/mine/8f9z) | Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with NBD-14204, an HIV-1 gp120 antagonist | 分子名称: | (5M)-N-{(1S)-2-amino-1-[5-(hydroxymethyl)-1,3-thiazol-2-yl]ethyl}-5-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrrole-2-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ... | 著者 | Kwon, Y.D, Kwong, P.D. | 登録日 | 2022-11-25 | 公開日 | 2023-01-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Antiviral Activity and Crystal Structures of HIV-1 gp120 Antagonists. Int J Mol Sci, 23, 2022
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2H6J
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![BU of 2h6j by Molmil](/molmil-images/mine/2h6j) | |
4JB9
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![BU of 4jb9 by Molmil](/molmil-images/mine/4jb9) | Crystal structure of antibody VRC06 in complex with HIV-1 gp120 core | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, antibody VRC06 heavy chain, antibody VRC06 light chain, ... | 著者 | Kwon, Y.D, Zhou, T, Srivatsan, S, Kwong, P.D. | 登録日 | 2013-02-19 | 公開日 | 2013-05-08 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Delineating antibody recognition in polyclonal sera from patterns of HIV-1 isolate neutralization. Science, 340, 2013
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4DKP
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![BU of 4dkp by Molmil](/molmil-images/mine/4dkp) | Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with AWS-I-50 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, N-[(1S,2S)-2-amino-2,3-dihydro-1H-inden-1-yl]-N'-(4-chloro-3-fluorophenyl)ethanediamide, ... | 著者 | Kwon, Y.D, LaLonde, J.M, Jones, D.M, Sun, A.W, Courter, J.R, Soeta, T, Kobayashi, T, Princiotto, A.M, Wu, X, Mascola, J, Schon, A, Freire, E, Sodroski, J, Madani, N, Smith III, A.B, Kwong, P.D. | 登録日 | 2012-02-03 | 公開日 | 2012-05-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.7978 Å) | 主引用文献 | Structure-Based Design, Synthesis, and Characterization of Dual Hotspot Small-Molecule HIV-1 Entry Inhibitors. J.Med.Chem., 55, 2012
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4DKR
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![BU of 4dkr by Molmil](/molmil-images/mine/4dkr) | Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with AWS-I-169 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, HIV-1 gp120 core, ... | 著者 | Kwon, Y.D, LaLonde, J.M, Jones, D.M, Sun, A.W, Courter, J.R, Soeta, T, Kobayashi, T, Princiotto, A.M, Wu, X, Mascola, J, Schon, A, Freire, E, Sodroski, J, Madani, N, Smith III, A.B, Kwong, P.D. | 登録日 | 2012-02-03 | 公開日 | 2012-05-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure-Based Design, Synthesis, and Characterization of Dual Hotspot Small-Molecule HIV-1 Entry Inhibitors. J.Med.Chem., 55, 2012
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