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2BJ4
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ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH A PHAGE-DISPLAY DERIVED PEPTIDE ANTAGONIST
分子名称: 4-HYDROXYTAMOXIFEN, ESTROGEN RECEPTOR, PEPTIDE ANTAGONIST
著者Kong, E, Heldring, N, Gustafsson, J.A, Treuter, E, Hubbard, R.E, Pike, A.C.W.
登録日2005-01-28
公開日2005-02-16
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Delineation of a Unique Protein-Protein Interaction Site on the Surface of the Estrogen Receptor
Proc.Natl.Acad.Sci.USA, 102, 2005
2JF9
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ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH A TAMOXIFEN-SPECIFIC PEPTIDE ANTAGONIST
分子名称: 1,2-ETHANEDIOL, 4-HYDROXYTAMOXIFEN, AB5 PEPTIDE, ...
著者Heldring, N, Pawson, T, McDonnell, D, Treuter, E, Gustafsson, J.A, Pike, A.C.W.
登録日2007-01-29
公開日2007-02-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural Insights Into Corepressor Recognition by Antagonist-Bound Estrogen Receptors.
J.Biol.Chem., 282, 2007
2JFA
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ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH AN AFFINITY-SELECTED COREPRESSOR PEPTIDE
分子名称: COREPRESSOR PEPTIDE, ESTROGEN RECEPTOR, RALOXIFENE, ...
著者Heldring, N, Pawson, T, McDonnell, D, Treuter, E, Gustafsson, J.A, Pike, A.C.W.
登録日2007-01-29
公開日2007-02-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Structural Insights Into Corepressor Recognition by Antagonist-Bound Estrogen Receptors.
J.Biol.Chem., 282, 2007
4NQA
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Crystal structure of liganded hRXR-alpha/hLXR-beta heterodimer on DNA
分子名称: (9cis)-retinoic acid, 5'-D(*TP*AP*AP*GP*GP*TP*CP*AP*CP*TP*TP*CP*AP*GP*GP*TP*CP*A)-3', 5'-D(*TP*AP*TP*GP*AP*CP*CP*TP*GP*AP*AP*GP*TP*GP*AP*CP*CP*T)-3', ...
著者Lou, X.H, Toresson, G, Benod, C, Suh, J.H, Phillips, K.J, Webb, P, Gustafsson, J.A.
登録日2013-11-24
公開日2014-02-26
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.102 Å)
主引用文献Structure of the retinoid X receptor alpha-liver X receptor beta (RXR alpha-LXR beta ) heterodimer on DNA.
Nat.Struct.Mol.Biol., 21, 2014
2GDA
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REFINED SOLUTION STRUCTURE OF THE GLUCOCORTICOID RECEPTOR DNA-BINDING DOMAIN
分子名称: GLUCOCORTICOID RECEPTOR, ZINC ION
著者Baumann, H, Paulsen, K, Kovacs, H, Berglund, H, Wright, A.P.H, Gustafsson, J.-A, Hard, T.
登録日1994-03-15
公開日1994-06-22
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Refined solution structure of the glucocorticoid receptor DNA-binding domain.
Biochemistry, 32, 1993
1GDC
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REFINED SOLUTION STRUCTURE OF THE GLUCOCORTICOID RECEPTOR DNA-BINDING DOMAIN
分子名称: GLUCOCORTICOID RECEPTOR, ZINC ION
著者Baumann, H, Paulsen, K, Kovacs, H, Berglund, H, Wright, A.P.H, Gustafsson, J.-A, Hard, T.
登録日1994-03-15
公開日1994-06-22
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Refined solution structure of the glucocorticoid receptor DNA-binding domain.
Biochemistry, 32, 1993
1UTR
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UTEROGLOBIN-PCB COMPLEX (REDUCED FORM)
分子名称: 4,4'-BIS([H]METHYLSULFONYL)-2,2',5,5'-TETRACHLOROBIPHENYL, UTEROGLOBIN
著者Hard, T, Barnes, H.J, Larsson, C, Gustafsson, J.-A, Lund, J.
登録日1995-09-01
公開日1995-12-07
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of a mammalian PCB-binding protein in complex with a PCB.
Nat.Struct.Biol., 2, 1995
1HJ1
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RAT OESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH PURE ANTIOESTROGEN ICI164,384
分子名称: N-BUTYL-11-[(7R,8R,9S,13S,14S,17S)-3,17-DIHYDROXY-13-METHYL-7,8,9,11,12,13,14,15,16,17-DECAHYDRO-6H-CYCLOPENTA[A]PHENANTHREN-7-YL]-N-METHYLUNDECANAMIDE, NICKEL (II) ION, OESTROGEN RECEPTOR BETA, ...
著者Pike, A.C.W, Brzozowski, A.M, Carlquist, M.
登録日2001-01-08
公開日2002-01-04
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural Insights Into the Mode of Action of a Pure Antiestrogen
Structure, 9, 2001
1GWQ
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HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE CORE AND TIF2 NRBOX2 PEPTIDE
分子名称: NUCLEAR RECEPTOR COACTIVATOR 2, OESTROGEN RECEPTOR, RALOXIFENE CORE
著者Pike, A.C.W, Brzozowski, A.M.
登録日2002-03-22
公開日2002-08-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Interaction of Transcriptional Intermediary Factor 2 Nuclear Receptor Box Peptides with the Coactivator Binding Site of Estrogen Receptor Alpha.
J.Biol.Chem., 277, 2002
1GWR
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HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 17BETA-OESTRADIOL AND TIF2 NRBOX3 PEPTIDE
分子名称: ESTRADIOL, OESTROGEN RECEPTOR, TRANSCRIPTION INTERMEDIARY FACTOR-2
著者Pike, A.C.W, Brzozowski, A.M.
登録日2002-03-22
公開日2002-08-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Interaction of Transcriptional Intermediary Factor 2 Nuclear Receptor Box Peptides with the Coactivator Binding Site of Estrogen Receptor Alpha.
J.Biol.Chem., 277, 2002
1ERR
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HUMAN ESTROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE
分子名称: ESTROGEN RECEPTOR, RALOXIFENE
著者Brzozowski, A.M, Pike, A.C.W.
登録日1997-09-08
公開日1998-09-16
最終更新日2013-05-15
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Molecular basis of agonism and antagonism in the oestrogen receptor.
Nature, 389, 1997
1ERE
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HUMAN ESTROGEN RECEPTOR LIGAND-BINDING DOMAIN IN COMPLEX WITH 17BETA-ESTRADIOL
分子名称: ESTRADIOL, ESTROGEN RECEPTOR
著者Brzozowski, A.M, Pike, A.C.W.
登録日1997-09-08
公開日1998-09-16
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Molecular basis of agonism and antagonism in the oestrogen receptor.
Nature, 389, 1997
1L2J
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Human Estrogen Receptor beta Ligand-binding Domain in Complex with (R,R)-5,11-cis-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diol
分子名称: (R,R)-5,11-CIS-DIETHYL-5,6,11,12-TETRAHYDROCHRYSENE-2,8-DIOL, ESTROGEN RECEPTOR BETA
著者Shiau, A.K, Barstad, D, Radek, J.T, Meyers, M.J, Nettles, K.W, Katzenellenbogen, B.S, Katzenellenbogen, J.A, Agard, D.A, Greene, G.L.
登録日2002-02-21
公開日2002-05-01
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism.
Nat.Struct.Biol., 9, 2002
1UVZ
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structure of human thioredoxin 2
分子名称: THIOREDOXIN
著者Smeets, A, Evrard, C, Declercq, J.P.
登録日2004-01-27
公開日2005-06-16
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Crystal Structures of Oxidized and Reduced Forms of Human Mitochondrial Thioredoxin 2.
Protein Sci., 14, 2005
1W4V
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structure of the oxidised form of human thioredoxin 2
分子名称: THIOREDOXIN, MITOCHONDRIAL
著者Smeets, A, Evrard, C, Declercq, J.P.
登録日2004-07-30
公開日2005-10-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structures of Oxidized and Reduced Forms of Human Mitochondrial Thioredoxin 2.
Protein Sci., 14, 2005
1W89
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Structure of the reduced form of human thioredoxin 2
分子名称: THIOREDOXIN
著者Smeets, A, Evrard, C, Declercq, J.P.
登録日2004-09-17
公開日2005-10-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structures of Oxidized and Reduced Forms of Human Mitochondrial Thioredoxin 2.
Protein Sci., 14, 2005
1KV6
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X-ray structure of the orphan nuclear receptor ERR3 ligand-binding domain in the constitutively active conformation
分子名称: ESTROGEN-RELATED RECEPTOR GAMMA, steroid receptor coactivator 1
著者Greschik, H, Wurtz, J.-M, Sanglier, S, Bourguet, W, van Dorsselaer, A, Moras, D, Renaud, J.-P, Structural Proteomics in Europe (SPINE)
登録日2002-01-25
公開日2003-01-25
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural and Functional Evidence for Ligand-Independent Transcriptional Activation by the Estrogen-Related Receptor 3
Mol.Cell, 9, 2002

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