1HJ1

RAT OESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH PURE ANTIOESTROGEN ICI164,384

Summary for 1HJ1

• Entry DOI: 10.2210/pdb1hj1/pdb
• Related: 1QKN
• Descriptor: OESTROGEN RECEPTOR BETA, N-BUTYL-11-[(7R,8R,9S,13S,14S,17S)-3,17-DIHYDROXY-13-METHYL-7,8,9,11,12,13,14,15,16,17-DECAHYDRO-6H-CYCLOPENTA[A]PHENANTHREN-7-YL]-N-METHYLUNDECANAMIDE, PARA-MERCURY-BENZENESULFONIC ACID, ... (5 entities in total)
• Functional Keywords: nuclear receptor, transcription factor, oestrogen, antagonist
• Biological source: RATTUS NORVEGICUS (NORWAY RAT)
• Total number of polymer chains: 1
• Total formula weight: 29686.95

Authors

Pike, A.C.W.,Brzozowski, A.M.,Carlquist, M. (deposition date: 2001-01-08, release date: 2002-01-04, Last modification date: 2023-12-13)

• Primary citation: Pike, A.C.W.,Brzozowski, A.M.,Walton, J.,Hubbard, R.E.,Thorsell, A.G.,Li, Y.L.,Gustafsson, J.A.,Carlquist, M.; Structural Insights Into the Mode of Action of a Pure Antiestrogen; Structure, 9:145-, 2001; PubMed: 11250199; DOI: 10.1016/S0969-2126(01)00568-8

Experimental method

X-RAY DIFFRACTION (2.3 Å)