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2G15
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BU of 2g15 by Molmil
Structural Characterization of autoinhibited c-Met kinase
分子名称: activated met oncogene
著者Wang, W, Marimuthu, A, Tsai, J, Kumar, A, Krupka, H.I, Zhang, C, Powell, B, Suzuki, Y, Nguyen, H, Tabrizizad, M, Luu, C, West, B.L.
登録日2006-02-13
公開日2006-03-21
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural characterization of autoinhibited c-Met kinase produced by coexpression in bacteria with phosphatase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2G1L
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BU of 2g1l by Molmil
Crystal structure of the FHA domain of human kinesin family member C
分子名称: CHLORIDE ION, Kinesin-like protein KIF1C, NICKEL (II) ION, ...
著者Wang, J, Tempel, W, Shen, Y, Shen, L, Arrowsmith, C, Edwards, A, Sundstrom, M, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2006-02-14
公開日2006-02-28
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.602 Å)
主引用文献Crystal structure of the FHA domain of human kinesin family member C
to be published
3LV4
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BU of 3lv4 by Molmil
Crystal structure of the glycoside hydrolase, family 43 YxiA protein from Bacillus licheniformis. Northeast Structural Genomics Consortium Target BiR14.
分子名称: ACETATE ION, CALCIUM ION, Glycoside hydrolase YxiA
著者Vorobiev, S, Abashidze, M, Seetharaman, J, Belote, R.L, Ciccosanti, C, Sahdev, S, Xiao, R, Acton, T.B, Everett, J.K, Montelione, G.T, Tong, L, Hunt, J.F, Northeast Structural Genomics Consortium (NESG)
登録日2010-02-19
公開日2010-03-09
最終更新日2018-01-24
実験手法X-RAY DIFFRACTION (1.695 Å)
主引用文献Crystal structure of the glycoside hydrolase, family 43 YxiA protein from Bacillus licheniformis.
To be Published
2G1P
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BU of 2g1p by Molmil
Structure of E. coli DNA adenine methyltransferase (DAM)
分子名称: 5'-D(*TP*CP*TP*AP*GP*AP*TP*CP*TP*AP*GP*A)-3', DNA adenine methylase, GLYCEROL, ...
著者Horton, J.R, Liebert, K, Bekes, M, Jeltsch, A, Cheng, X.
登録日2006-02-14
公開日2006-11-21
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献Structure and substrate recognition of the Escherichia coli DNA adenine methyltransferase.
J.Mol.Biol., 358, 2006
8W86
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HLA-DQ2.5-B/C hordein peptide in complex with DQN0385AE02
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, DQN0385AE02 Fab heavy chain, DQN0385AE02 Fab light chain, ...
著者Irie, M, Tsushima, T, Teranishi-Ikawa, Y, Takahashi, N, Ishii, S, Okura, Y, Fukami, T.A, Torizawa, T.
登録日2023-08-31
公開日2023-11-08
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.236 Å)
主引用文献Characterizations of a neutralizing antibody broadly reactive to multiple gluten peptide:HLA-DQ2.5 complexes in the context of celiac disease.
Nat Commun, 14, 2023
8W85
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HLA-DQ2.5-gamma2 gliadin peptide in complex with DQN0385AE01
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, DQN0385AE01 Fab heavy chain, DQN0385AE01 Fab light chain, ...
著者Irie, M, Tsushima, T, Teranishi-Ikawa, Y, Takahashi, N, Ishii, S, Okura, Y, Fukami, T.A, Torizawa, T.
登録日2023-08-31
公開日2023-11-08
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.769 Å)
主引用文献Characterizations of a neutralizing antibody broadly reactive to multiple gluten peptide:HLA-DQ2.5 complexes in the context of celiac disease.
Nat Commun, 14, 2023
3LW2
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Mouse Plasminogen Activator Inhibitor-1 (PAI-1)
分子名称: Plasminogen activator inhibitor 1
著者Dewilde, M, Van De Craen, B, Compernolle, G, Madsen, J.B, Strelkov, S.V, Gils, A, Declerck, P.J.
登録日2010-02-23
公開日2010-04-07
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Subtle structural differences between human and mouse PAI-1 reveal the basis for biochemical differences.
J.Struct.Biol., 171, 2010
2FZ9
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Human Aldose Reductase complexed with inhibitor zopolrestat after six days soaking.
分子名称: 3,4-DIHYDRO-4-OXO-3-((5-TRIFLUOROMETHYL-2-BENZOTHIAZOLYL)METHYL)-1-PHTHALAZINE ACETIC ACID, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, aldose reductase
著者Steuber, H, Zentgraf, M, Gerlach, C, Sotriffer, C.A, Heine, A, Klebe, G.
登録日2006-02-09
公開日2006-10-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Expect the Unexpected or Caveat for Drug Designers: Multiple Structure Determinations Using Aldose Reductase Crystals Treated under Varying Soaking and Co-crystallisation Conditions.
J.Mol.Biol., 363, 2006
8W84
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HLA-DQ2.5-alpha2 gliadin peptide in complex with DQN0344AE02
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, DQN0344AE02 Fab heavy chain, DQN0344AE02 Fab light chain, ...
著者Irie, M, Tsushima, T, Teranishi-Ikawa, Y, Takahashi, N, Ishii, S, Okura, Y, Fukami, T.A, Torizawa, T.
登録日2023-08-31
公開日2023-11-08
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.105 Å)
主引用文献Characterizations of a neutralizing antibody broadly reactive to multiple gluten peptide:HLA-DQ2.5 complexes in the context of celiac disease.
Nat Commun, 14, 2023
5AHN
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BU of 5ahn by Molmil
IMP-bound form of the D199N mutant of IMPDH from Pseudomonas aeruginosa
分子名称: INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE, INOSINIC ACID, MAGNESIUM ION
著者Labesse, G, Alexandre, T, Gelin, M, Haouz, A, Munier-Lehmann, H.
登録日2015-02-06
公開日2015-07-15
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.652 Å)
主引用文献Crystallographic Studies of Two Variants of Pseudomonas Aeruginosa Impdh with Impaired Allosteric Regulation
Acta Crystallogr.,Sect.D, 71, 2015
3VNQ
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BU of 3vnq by Molmil
Co-crystal structure of NRPS adenylation protein CytC1 with ATP from streptomyces
分子名称: ADENOSINE-5'-TRIPHOSPHATE, NRPS adenylation protein CytC1
著者Okumura, H, Ueki, M, Shiro, Y, Osada, H.
登録日2012-01-17
公開日2013-01-23
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Substrate recognition mechanism of NRPS adenylation protein from Streptomyces
To be Published
8W83
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HLA-DQ2.5-alpha1 gliadin peptide in complex with DQN0344AE02
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, DQN0344AE02 Fab heavy chain, DQN0344AE02 Fab light chain, ...
著者Irie, M, Tsushima, T, Teranishi-Ikawa, Y, Takahashi, N, Ishii, S, Okura, Y, Fukami, T.A, Torizawa, T.
登録日2023-08-31
公開日2023-11-08
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.818 Å)
主引用文献Characterizations of a neutralizing antibody broadly reactive to multiple gluten peptide:HLA-DQ2.5 complexes in the context of celiac disease.
Nat Commun, 14, 2023
5HPK
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BU of 5hpk by Molmil
System-wide modulation of HECT E3 ligases with selective ubiquitin variant probes: NEDD4L and UbV NL.1
分子名称: E3 ubiquitin-protein ligase NEDD4-like, Ubiquitin variant NL.1
著者Wu, K.-P, Mukherjee, M, Mercredi, P.Y, Schulman, B.A.
登録日2016-01-20
公開日2016-03-16
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.431 Å)
主引用文献System-Wide Modulation of HECT E3 Ligases with Selective Ubiquitin Variant Probes.
Mol.Cell, 62, 2016
3LX8
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BU of 3lx8 by Molmil
Crystal structure of GDP-bound NFeoB from S. thermophilus
分子名称: Ferrous iron uptake transporter protein B, GUANOSINE-5'-DIPHOSPHATE
著者Ash, M.R, Guilfoyle, A, Maher, M.J, Clarke, R.J, Guss, J.M, Jormakka, M.
登録日2010-02-24
公開日2010-03-09
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Potassium-activated GTPase reaction in the G Protein-coupled ferrous iron transporter B.
J.Biol.Chem., 285, 2010
3LXH
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Crystal Structure of Cytochrome P450 CYP101D1
分子名称: 1,4-DIETHYLENE DIOXIDE, Cytochrome P450, PHOSPHATE ION, ...
著者Yang, W, Bell, S.G, Wang, H, Bartlam, M, Wong, L.L, Rao, Z.
登録日2010-02-25
公開日2010-06-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Molecular characterization of a class I P450 electron transfer system from Novosphingobium aromaticivorans DSM12444
J.Biol.Chem., 285, 2010
3VY9
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Crystal structure of PorB from Neisseria meningitidis in complex with cesium ion, space group H32
分子名称: CESIUM ION, Outer membrane protein
著者Kattner, C, Zaucha, J, Jaenecke, F, Zachariae, U, Tanabe, M.
登録日2012-09-21
公開日2013-01-02
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.63 Å)
主引用文献Identification of a cation transport pathway in Neisseria meningitidis PorB.
Proteins, 81, 2013
3LQS
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BU of 3lqs by Molmil
Complex Structure of D-Amino Acid Aminotransferase and 4-amino-4,5-dihydro-thiophenecarboxylic acid (ADTA)
分子名称: 4-[({3-HYDROXY-2-METHYL-5-[(PHOSPHONOOXY)METHYL]PYRIDIN-4-YL}METHYL)AMINO]THIOPHENE-2-CARBOXYLIC ACID, ACETIC ACID, D-alanine aminotransferase
著者Lepore, B.W, Liu, D, Peng, Y, Fu, M, Yasuda, C, Manning, J.M, Silverman, R.B, Ringe, D.
登録日2010-02-10
公開日2010-03-16
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Chiral discrimination among aminotransferases: inactivation by 4-amino-4,5-dihydrothiophenecarboxylic acid.
Biochemistry, 49, 2010
3VZT
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BU of 3vzt by Molmil
Crystal Structure of outer membrane protein PorB from Neisseria meningitidis
分子名称: CESIUM ION, outer membrane protein
著者Tanabe, M, Iverson, T.M.
登録日2012-10-15
公開日2012-11-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural basis for solute transport, nucleotide regulation, and immunological recognition of Neisseria meningitidis PorB.
Proc.Natl.Acad.Sci.USA, 107, 2010
2G64
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Structure of Caenorhabditis elegans 6-pyruvoyl tetrahydropterin synthase
分子名称: GLYCEROL, Putative 6-pyruvoyl tetrahydrobiopterin synthase, SODIUM ION, ...
著者Wengerter, B.C, Patskovsky, Y, Zhan, C, Ramagopal, U, Milstein, S, Vidal, M, Almo, S.C, Burley, S.K, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2006-02-24
公開日2006-03-14
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structure of Caenorhabditis Elegans 6-Pyruvoyl Tetrahydropterin Synthase
To be Published
3W05
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Crystal structure of Oryza sativa DWARF14 (D14) in complex with PMSF
分子名称: 1,2-ETHANEDIOL, Dwarf 88 esterase, phenylmethanesulfonic acid
著者Kagiyama, M, Hirano, Y, Mori, T, Kim, S.Y, Kyozuka, J, Seto, Y, Yamaguchi, S, Hakoshima, T.
登録日2012-10-19
公開日2013-01-23
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.58 Å)
主引用文献Structures of D14 and D14L in the strigolactone and karrikin signaling pathways
Genes Cells, 18, 2013
4ZVF
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Crystal structure of GGDEF domain of the E. coli DosC - form II (GTP-alpha-S-bound)
分子名称: 1,2-ETHANEDIOL, CALCIUM ION, Diguanylate cyclase DosC, ...
著者Tarnawski, M, Barends, T.R.M, Schlichting, I.
登録日2015-05-18
公開日2015-11-11
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Structural analysis of an oxygen-regulated diguanylate cyclase.
Acta Crystallogr.,Sect.D, 71, 2015
3W0T
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BU of 3w0t by Molmil
Human Glyoxalase I with an N-hydroxypyridone derivative inhibitor
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Lactoylglutathione lyase, N-[3-(1-hydroxy-6-oxo-4-phenyl-1,6-dihydropyridin-2-yl)phenyl]methanesulfonamide, ...
著者Fukami, T.A, Irie, M, Matsuura, T.
登録日2012-11-02
公開日2013-11-06
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.351 Å)
主引用文献N-Hydroxypyridone-based glyoxalase I inhibitors mimicking binding interactions of the substrate
To be Published
7Z3S
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CRYSTAL STRUCTURE of PheF from Geobacillus stearothermophilus
分子名称: Acetaldehyde dehydrogenase, PHOSPHATE ION
著者Driller, R, Haack, M, Brueck, T, Loll, B.
登録日2022-03-02
公開日2023-01-11
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献CRYSTAL STRUCTURE OF THE P1 trifluoroethylglycine (TfeGly) BPTI MUTANT- BOVINE CHYMOTRYPSIN COMPLEX
To Be Published
3VTW
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BU of 3vtw by Molmil
Crystal structure of T7-tagged Optineurin LIR-fused human LC3B_2-119
分子名称: Optineurin, microtubule-associated proteins 1A/1B light chain 3B, SULFATE ION
著者Suzuki, H, Kawasaki, M, Kato, R, Wakatsuki, S.
登録日2012-06-08
公開日2013-06-26
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献Structural basis for phosphorylation-triggered autophagic clearance of Salmonella
Biochem.J., 454, 2013
2G77
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Crystal Structure of Gyp1 TBC domain in complex with Rab33 GTPase bound to GDP and AlF3
分子名称: ALUMINUM FLUORIDE, GTPase-activating protein GYP1, GUANOSINE-5'-DIPHOSPHATE, ...
著者Pan, X, Eathiraj, S, Munson, M, Lambright, D.G.
登録日2006-02-27
公開日2006-07-25
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献TBC-domain GAPs for Rab GTPases accelerate GTP hydrolysis by a dual-finger mechanism.
Nature, 442, 2006

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