4JPG
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![BU of 4jpg by Molmil](/molmil-images/mine/4jpg) | 2-((1H-benzo[d]imidazol-1-yl)methyl)-4H-pyrido[1,2-a]pyrimidin-4-ones as Novel PKM2 Activators | 分子名称: | 1,6-di-O-phosphono-beta-D-fructofuranose, 2-(1H-benzimidazol-1-ylmethyl)-4H-pyrido[1,2-a]pyrimidin-4-one, Pyruvate kinase isozymes M1/M2 | 著者 | Greasley, S.E, Hickey, M, Phonephaly, H, Cronin, C. | 登録日 | 2013-03-19 | 公開日 | 2013-05-22 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | Discovery of 2-((1H-benzo[d]imidazol-1-yl)methyl)-4H-pyrido[1,2-a]pyrimidin-4-ones as novel PKM2 activators. Bioorg.Med.Chem.Lett., 23, 2013
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8K1Q
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8K1J
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8K1Z
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8K1V
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7XZO
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![BU of 7xzo by Molmil](/molmil-images/mine/7xzo) | Formate-tetrahydrofolate ligase in complex with ATP | 分子名称: | (R,R)-2,3-BUTANEDIOL, ADENOSINE-5'-TRIPHOSPHATE, Formate--tetrahydrofolate ligase, ... | 著者 | Fang, C.L, Zhang, Y. | 登録日 | 2022-06-03 | 公開日 | 2023-06-07 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Identification of FtfL as a novel target of berberine in intestinal bacteria. Bmc Biol., 21, 2023
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7XZN
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7XZP
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5VER
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![BU of 5ver by Molmil](/molmil-images/mine/5ver) | MOUSE KYNURENINE AMINOTRANSFERASE III, RE-REFINEMENT OF THE PDB STRUCTURE 3E2Z | 分子名称: | 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CALCIUM ION, ... | 著者 | Wlodawer, A, Dauter, Z, Minor, W, Stanfield, R, Porebski, P, Jaskolski, M, Pozharski, E, Weichenberger, C.X, Rupp, B. | 登録日 | 2017-04-05 | 公開日 | 2017-11-29 | 最終更新日 | 2022-04-13 | 実験手法 | X-RAY DIFFRACTION (2.81 Å) | 主引用文献 | Detect, correct, retract: How to manage incorrect structural models. FEBS J., 285, 2018
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4HJI
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1DSS
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4M5C
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![BU of 4m5c by Molmil](/molmil-images/mine/4m5c) | Crystal Structure of an Truncated Transition metal Transporter | 分子名称: | COBALT (II) ION, Cobalamin biosynthesis protein CbiM, HEXANE-1,6-DIOL | 著者 | Yu, Y, Zhou, M.Z, Gu, J.K. | 登録日 | 2013-08-08 | 公開日 | 2014-03-26 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Planar substrate-binding site dictates the specificity of ECF-type nickel/cobalt transporters Cell Res., 24, 2014
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7W1S
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![BU of 7w1s by Molmil](/molmil-images/mine/7w1s) | Crystal structure of SARS-CoV-2 spike receptor-binding domain in complex with neutralizing nanobody Nb-007 | 分子名称: | Nanobody Nb-007, Spike protein S1 | 著者 | Yang, J, Lin, S, Sun, H.L, Lu, G.W. | 登録日 | 2021-11-20 | 公開日 | 2022-06-29 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.997 Å) | 主引用文献 | A Potent Neutralizing Nanobody Targeting the Spike Receptor-Binding Domain of SARS-CoV-2 and the Structural Basis of Its Intimate Binding. Front Immunol, 13, 2022
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7XHQ
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![BU of 7xhq by Molmil](/molmil-images/mine/7xhq) | Small-molecule Allosteric Regulation Mechanism of SHP2 | 分子名称: | 2-[(3S,4R)-4-azanyl-3-methyl-2-oxa-8-azaspiro[4.5]decan-8-yl]-5-[2,3-bis(chloranyl)phenyl]-3-methyl-pyrrolo[2,1-f][1,2,4]triazin-4-one, Tyrosine-protein phosphatase non-receptor type 11 | 著者 | Luo, Y, Zhu, J, Yu, K, Liu, B. | 登録日 | 2022-04-09 | 公開日 | 2023-02-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Discovery of the SHP2 allosteric inhibitor 2-((3R,4R)-4-amino-3-methyl-2-oxa-8-azaspiro[4.5]decan-8-yl)-5-(2,3-dichlorophenyl)-3-methylpyrrolo[2,1-f][1,2,4] triazin-4(3H)-one. J Enzyme Inhib Med Chem, 38, 2023
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4M5B
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3US6
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![BU of 3us6 by Molmil](/molmil-images/mine/3us6) | Crystal Structure of Histidine-containing Phosphotransfer Protein MtHPt1 from Medicago truncatula | 分子名称: | Histidine-containing Phosphotransfer Protein type 1, MtHPt1 | 著者 | Ruszkowski, M, Brzezinski, K, Jedrzejczak, R, Dauter, M, Dauter, Z, Sikorski, M, Jaskolski, M. | 登録日 | 2011-11-23 | 公開日 | 2012-01-18 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.446 Å) | 主引用文献 | Medicago truncatula histidine-containing phosphotransfer protein: Structural and biochemical insights into the cytokinin transduction pathway in plants. Febs J., 280, 2013
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1IHY
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![BU of 1ihy by Molmil](/molmil-images/mine/1ihy) | GAPDH complexed with ADP-ribose | 分子名称: | ADENOSINE-5-DIPHOSPHORIBOSE, GLYCERALDEHYDE 3-PHOSPHATE DEHYDROGENASE, SULFATE ION | 著者 | Shen, Y.-Q, Song, S.-Y, Lin, Z.-J. | 登録日 | 2001-04-20 | 公開日 | 2002-07-31 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structures of D-glyceraldehyde-3-phosphate dehydrogenase complexed with coenzyme analogues. Acta Crystallogr.,Sect.D, 58, 2002
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7WKA
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7WK9
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7WK5
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![BU of 7wk5 by Molmil](/molmil-images/mine/7wk5) | Cryo-EM structure of Omicron S-ACE2, C2 state | 分子名称: | Angiotensin-converting enzyme 2, Spike glycoprotein | 著者 | Han, W.Y, Wang, Y.F. | 登録日 | 2022-01-08 | 公開日 | 2022-02-02 | 最終更新日 | 2022-03-09 | 実験手法 | ELECTRON MICROSCOPY (3.66 Å) | 主引用文献 | Molecular basis of SARS-CoV-2 Omicron variant receptor engagement and antibody evasion and neutralization Biorxiv, 2022
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7WK4
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7WK8
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7WK6
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7Y6C
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![BU of 7y6c by Molmil](/molmil-images/mine/7y6c) | Crystal structure of the EscE/EsaG/EsaH complex | 分子名称: | EscE/YscE/SsaE family type III secretion system needle protein co-chaperone, EscG/YscG/SsaH family type III secretion system needle protein co-chaperone | 著者 | Zeng, Z.X, Xiao, S.B, Liao, L.J, Zhou, Y.Z. | 登録日 | 2022-06-18 | 公開日 | 2022-07-20 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Secreted in a Type III Secretion System-Dependent Manner, EsaH and EscE Are the Cochaperones of the T3SS Needle Protein EsaG of Edwardsiella piscicida. Mbio, 13, 2022
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7Y6B
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![BU of 7y6b by Molmil](/molmil-images/mine/7y6b) | Crystal structure of the EscE/EsaH complex | 分子名称: | EscE/YscE/SsaE family type III secretion system needle protein co-chaperone, EscG/YscG/SsaH family type III secretion system needle protein co-chaperone | 著者 | Zeng, Z.X, Xiao, S.B, Liao, L.J, Zhou, Y.Z. | 登録日 | 2022-06-18 | 公開日 | 2022-07-20 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Secreted in a Type III Secretion System-Dependent Manner, EsaH and EscE Are the Cochaperones of the T3SS Needle Protein EsaG of Edwardsiella piscicida. Mbio, 13, 2022
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