Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
3PAU
DownloadVisualize
BU of 3pau by Molmil
CueO in the resting oxidized state
分子名称: Blue copper oxidase cueO, COPPER (II) ION, CU-O-CU LINKAGE
著者Roberts, S.A, Singh, S, Montfort, W.R.
登録日2010-10-19
公開日2011-10-19
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献CueO in the resting oxidized state
To be Published
3D0Q
DownloadVisualize
BU of 3d0q by Molmil
Crystal structure of calG3 from Micromonospora echinospora determined in space group I222
分子名称: 3[N-MORPHOLINO]PROPANE SULFONIC ACID, Protein CalG3
著者Bitto, E, Singh, S, Bingman, C.A, Wesenberg, G.E, Phillips Jr, G.N.
登録日2008-05-02
公開日2008-06-24
最終更新日2017-10-25
実験手法X-RAY DIFFRACTION (2.79 Å)
主引用文献Biochemical and structural insights of the early glycosylation steps in calicheamicin biosynthesis.
Chem.Biol., 15, 2008
5ZZ0
DownloadVisualize
BU of 5zz0 by Molmil
HUMAN GELSOLIN FROM RESIDUES GLU28 TO ARG161 WITH CALCIUM
分子名称: 2-(2-METHOXYETHOXY)ETHANOL, CALCIUM ION, Gelsolin
著者Sharma, P, Badmalia, M, Yadav, S.P.S, Singh, S.
登録日2018-05-29
公開日2019-06-05
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.635 Å)
主引用文献Bonsai Gelsolin Survives Heat Induced Denaturation by Forming beta-Amyloids which Leach Out Functional Monomer.
Sci Rep, 8, 2018
4K0B
DownloadVisualize
BU of 4k0b by Molmil
Crystal structure of S-Adenosylmethionine synthetase from Sulfolobus solfataricus complexed with SAM and PPi
分子名称: DIPHOSPHATE, MAGNESIUM ION, PHOSPHATE ION, ...
著者Wang, F, Hurley, K.A, Helmich, K.E, Singh, S, Bingman, C.A, Thorson, J.S, Phillips Jr, G.N, Enzyme Discovery for Natural Product Biosynthesis (NatPro)
登録日2013-04-03
公開日2013-05-01
最終更新日2014-10-08
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献Understanding molecular recognition of promiscuity of thermophilic methionine adenosyltransferase sMAT from Sulfolobus solfataricus.
Febs J., 281, 2014
4L2Z
DownloadVisualize
BU of 4l2z by Molmil
Crystal structure of S-Adenosylmethionine synthetase from Sulfolobus solfataricus complexed with SAE and PPi
分子名称: DIPHOSPHATE, MAGNESIUM ION, PHOSPHATE ION, ...
著者Wang, F, Hurley, K.A, Helmich, K.E, Singh, S, Bingman, C.A, Thorson, J.S, Phillips Jr, G.N, Enzyme Discovery for Natural Product Biosynthesis (NatPro)
登録日2013-06-05
公開日2013-06-19
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.494 Å)
主引用文献Understanding molecular recognition of promiscuity of thermophilic methionine adenosyltransferase sMAT from Sulfolobus solfataricus.
Febs J., 281, 2014
2OA1
DownloadVisualize
BU of 2oa1 by Molmil
Crystal Structure of RebH, a FAD-dependent halogenase from Lechevalieria aerocolonigenes, the L-Tryptophan with FAD complex
分子名称: ADENOSINE, CHLORIDE ION, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Bitto, E, Bingman, C.A, Singh, S, Phillips Jr, G.N.
登録日2006-12-14
公開日2007-04-10
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献The structure of flavin-dependent tryptophan 7-halogenase RebH.
Proteins, 70, 2008
4M60
DownloadVisualize
BU of 4m60 by Molmil
Crystal structure of macrolide glycosyltransferases OleD
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Oleandomycin glycosyltransferase, SODIUM ION
著者Olmos Jr, J.L, Martinez III, E, Wang, F, Helmich, K.E, Singh, S, Xu, W, Bingman, C.A, Thorson, J.S, Phillips Jr, G.N, Enzyme Discovery for Natural Product Biosynthesis (NatPro)
登録日2013-08-08
公開日2013-09-04
最終更新日2019-07-17
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Crystal structure of macrolide glycosyltransferases OleD
To be Published
4L7I
DownloadVisualize
BU of 4l7i by Molmil
Crystal structure of S-Adenosylmethionine synthase from Sulfolobus solfataricus complexed with SAM and PPi
分子名称: DIPHOSPHATE, MAGNESIUM ION, PHOSPHATE ION, ...
著者Wang, F, Hurley, K.A, Helmich, K.E, Singh, S, Bingman, C.A, Thorson, J.S, Phillips Jr, G.N, Enzyme Discovery for Natural Product Biosynthesis (NatPro)
登録日2013-06-13
公開日2013-07-03
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.189 Å)
主引用文献Understanding molecular recognition of promiscuity of thermophilic methionine adenosyltransferase sMAT from Sulfolobus solfataricus.
Febs J., 281, 2014
4M7P
DownloadVisualize
BU of 4m7p by Molmil
Ensemble refinement of protein crystal structure of macrolide glycosyltransferases OleD
分子名称: Oleandomycin glycosyltransferase, SODIUM ION
著者Wang, F, Helmich, K.E, Xu, W, Singh, S, Olmos Jr, J.L, Martinez iii, E, Bingman, C.A, Thorson, J.S, Phillips Jr, G.N, Enzyme Discovery for Natural Product Biosynthesis (NatPro)
登録日2013-08-12
公開日2013-09-11
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Crystal structure of macrolide glycosyltransferases OleD
To be Published
3RSC
DownloadVisualize
BU of 3rsc by Molmil
Crystal Structure of CalG2, Calicheamicin Glycosyltransferase, TDP and calicheamicin T0 bound form
分子名称: CalG2, Calicheamicin T0, PHOSPHATE ION, ...
著者Chang, A, Helmich, K.E, Singh, S, Bingman, C.A, Thorson, J.S, Phillips Jr, G.N, Center for Eukaryotic Structural Genomics (CESG), Enzyme Discovery for Natural Product Biosynthesis (NatPro)
登録日2011-05-02
公開日2011-08-10
最終更新日2017-11-08
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Complete set of glycosyltransferase structures in the calicheamicin biosynthetic pathway reveals the origin of regiospecificity.
Proc.Natl.Acad.Sci.USA, 108, 2011
3T6U
DownloadVisualize
BU of 3t6u by Molmil
Crystal Structure of Lysozyme in 40% sucrose
分子名称: CHLORIDE ION, Lysozyme, SODIUM ION, ...
著者Sharma, P, Singh, S, Ashish
登録日2011-07-29
公開日2011-08-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.213 Å)
主引用文献Crystal Structure of Lysozyme in 40% sucrose
to be published
4PIW
DownloadVisualize
BU of 4piw by Molmil
Crystal structure of sugar aminotransferase WecE from Escherichia coli K-12
分子名称: TDP-4-keto-6-deoxy-D-glucose transaminase family protein
著者Wang, F, Xu, W, Helmich, K.E, Singh, S, Yennamalli, R.M, Miller, M.D, Bingman, C.A, Thorson, J.S, Phillips Jr, G.N, Enzyme Discovery for Natural Product Biosynthesis (NatPro)
登録日2014-05-09
公開日2014-07-16
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of sugar aminotransferase WecE from Escherichia coli K-12
To Be Published
4Q31
DownloadVisualize
BU of 4q31 by Molmil
The crystal structure of cystathione gamma lyase (CalE6) from Micromonospora echinospora
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CHLORIDE ION, FORMIC ACID, ...
著者Tan, K, Bigelow, L, Jedrzejczak, R, Babnigg, G, Bingman, C.A, Yennamalli, R.M, Singh, S, Kharel, M.K, Thorson, J.S, Phillips Jr, G.N, Joachimiak, A, Midwest Center for Structural Genomics (MCSG), Enzyme Discovery for Natural Product Biosynthesis (NatPro)
登録日2014-04-10
公開日2014-05-07
最終更新日2017-03-08
実験手法X-RAY DIFFRACTION (2.099 Å)
主引用文献Structural dynamics of a methionine gamma-lyase for calicheamicin biosynthesis: Rotation of the conserved tyrosine stacking with pyridoxal phosphate.
Struct Dyn, 3, 2016
2EVN
DownloadVisualize
BU of 2evn by Molmil
NMR solution structures of At1g77540
分子名称: Protein At1g77540
著者Tyler, R.C, Singh, S, Tonelli, M, Min, M.S, Markley, J.L, Center for Eukaryotic Structural Genomics (CESG)
登録日2005-10-31
公開日2005-11-15
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structure of Arabidopsis thaliana At1g77540 Protein, a Minimal Acetyltransferase from the COG2388 Family.
Biochemistry, 45, 2006
7K6I
DownloadVisualize
BU of 7k6i by Molmil
Carbonic Anhydrase II complexed with 4-(2-(3-phenylureido)ethylsulfonamido)benzenesulfonamide
分子名称: 4-[({2-[(phenylcarbamoyl)amino]ethyl}sulfonyl)amino]benzene-1-sulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Andring, J.T, Singh, S, McKenna, R.
登録日2020-09-20
公開日2020-12-23
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.406 Å)
主引用文献Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors.
Eur.J.Med.Chem., 212, 2021
7K6U
DownloadVisualize
BU of 7k6u by Molmil
Carbonic Anhydrase IX mimic complexed with 4-(2-(3-(4-methylphenyl)ureido)ethylsulfonamido)benzenesulfonamide
分子名称: 4-{[(2-{[(4-methylphenyl)carbamoyl]amino}ethyl)sulfonyl]amino}benzene-1-sulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Andring, J.T, Singh, S, McKenna, R.
登録日2020-09-21
公開日2020-12-23
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.605 Å)
主引用文献Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors.
Eur.J.Med.Chem., 212, 2021
7K6L
DownloadVisualize
BU of 7k6l by Molmil
Carbonic Anhydrase II complexed with 4-(2-(3-(4-fluorophenyl)ureido)ethylsulfonamido)benzenesulfonamide
分子名称: 4-{[(2-{[(4-fluorophenyl)carbamoyl]amino}ethyl)sulfonyl]amino}benzene-1-sulfonamide, Carbonic anhydrase 2, ZINC ION
著者Andring, J.T, Singh, S, McKenna, R.
登録日2020-09-21
公開日2020-12-23
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.655 Å)
主引用文献Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors.
Eur.J.Med.Chem., 212, 2021
7K6X
DownloadVisualize
BU of 7k6x by Molmil
Carbonic Anhydrase IX mimic complexed with 4-(2-(3-(3,5-dimethylphenyl)ureido)ethylsulfonamido)benzenesulfonamide
分子名称: 4-{[(2-{[(3,5-dimethylphenyl)carbamoyl]amino}ethyl)sulfonyl]amino}benzene-1-sulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Andring, J.T, Singh, S, McKenna, R.
登録日2020-09-21
公開日2020-12-23
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.76 Å)
主引用文献Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors.
Eur.J.Med.Chem., 212, 2021
7K6K
DownloadVisualize
BU of 7k6k by Molmil
Carbonic Anhydrase II complexed with 4-(2-(3-(3,5-dimethylphenyl)ureido)ethylsulfonamido)benzenesulfonamide
分子名称: 4-{[(2-{[(3,5-dimethylphenyl)carbamoyl]amino}ethyl)sulfonyl]amino}benzene-1-sulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Andring, J.T, Singh, S, McKenna, R.
登録日2020-09-20
公開日2020-12-23
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.306 Å)
主引用文献Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors.
Eur.J.Med.Chem., 212, 2021
7K6T
DownloadVisualize
BU of 7k6t by Molmil
Carbonic Anhydrase IX mimic complexed with 4-(2-(3-phenylureido)ethylsulfonamido)benzenesulfonamide
分子名称: 4-[({2-[(phenylcarbamoyl)amino]ethyl}sulfonyl)amino]benzene-1-sulfonamide, Carbonic anhydrase 2, GLYCEROL, ...
著者Andring, J.T, Singh, S, McKenna, R.
登録日2020-09-21
公開日2020-12-23
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.759 Å)
主引用文献Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors.
Eur.J.Med.Chem., 212, 2021
7K6J
DownloadVisualize
BU of 7k6j by Molmil
Carbonic Anhydrase II complexed with 4-(2-(3-(4-methylphenyl)ureido)ethylsulfonamido)benzenesulfonamide
分子名称: 4-{[(2-{[(4-methylphenyl)carbamoyl]amino}ethyl)sulfonyl]amino}benzene-1-sulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Andring, J.T, Singh, S, McKenna, R.
登録日2020-09-20
公開日2020-12-23
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.755 Å)
主引用文献Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors.
Eur.J.Med.Chem., 212, 2021
7K6Z
DownloadVisualize
BU of 7k6z by Molmil
Carbonic Anhydrase IX mimic complexed with 4-(2-(3-(4-fluorophenyl)ureido)ethylsulfonamido)benzenesulfonamide
分子名称: 4-{[(2-{[(4-fluorophenyl)carbamoyl]amino}ethyl)sulfonyl]amino}benzene-1-sulfonamide, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ...
著者Andring, J.T, Singh, S, McKenna, R.
登録日2020-09-21
公開日2020-12-23
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.657 Å)
主引用文献Handling drug-target selectivity: A study on ureido containing Carbonic Anhydrase inhibitors.
Eur.J.Med.Chem., 212, 2021
1INF
DownloadVisualize
BU of 1inf by Molmil
INFLUENZA VIRUS B/LEE/40 NEURAMINIDASE COMPLEXED WITH BANA113 INHIBITOR
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(ACETYLAMINO)-3-GUANIDINOBENZOIC ACID, CALCIUM ION, ...
著者Jedrzejas, M.J, Luo, M.
登録日1995-07-07
公開日1996-08-17
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure-based inhibitors of influenza virus sialidase. A benzoic acid lead with novel interaction.
J.Med.Chem., 38, 1995
1INH
DownloadVisualize
BU of 1inh by Molmil
INFLUENZA A SUBTYPE N2 NEURAMINIDASE COMPLEXED WITH AROMATIC BANA111 INHIBITOR
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(ACETYLAMINO)-3-[(AMINOACETYL)AMINO]BENZOIC ACID, CALCIUM ION, ...
著者Jedrzejas, M.J, Luo, M.
登録日1995-07-07
公開日1996-08-17
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure-based inhibitors of influenza virus sialidase. A benzoic acid lead with novel interaction.
J.Med.Chem., 38, 1995
1ING
DownloadVisualize
BU of 1ing by Molmil
INFLUENZA A SUBTYPE N2 NEURAMINIDASE COMPLEXED WITH AROMATIC BANA109 INHIBITOR
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(ACETYLAMINO)-3-[(HYDROXYACETYL)AMINO]BENZOIC ACID, CALCIUM ION, ...
著者Jedrzejas, M.J, Luo, M.
登録日1995-07-07
公開日1996-08-17
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure-based inhibitors of influenza virus sialidase. A benzoic acid lead with novel interaction.
J.Med.Chem., 38, 1995

221051

件を2024-06-12に公開中

PDB statisticsPDBj update infoContact PDBjnumon