2W3T
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![BU of 2w3t by Molmil](/molmil-images/mine/2w3t) | Chloro complex of the Ni-Form of E.coli deformylase | 分子名称: | CHLORIDE ION, ETHANOL, NICKEL (II) ION, ... | 著者 | Ngo, Y.H.T, Palm, G.J, Hinrichs, W. | 登録日 | 2008-11-14 | 公開日 | 2009-12-15 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Structure of the Ni(II) Complex of Escherichia Coli Peptide Deformylase and Suggestions on Deformylase Activities Depending on Different Metal(II) Centres. J.Biol.Inorg.Chem., 15, 2010
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2Y6Q
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![BU of 2y6q by Molmil](/molmil-images/mine/2y6q) | Structure of the TetX monooxygenase in complex with the substrate 7- Iodtetracycline | 分子名称: | 7-IODOTETRACYCLINE, FLAVIN-ADENINE DINUCLEOTIDE, SULFATE ION, ... | 著者 | Volkers, G, Palm, G.J, Weiss, M.S, Wright, G.D, Hinrichs, W. | 登録日 | 2011-01-25 | 公開日 | 2011-03-23 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Structural Basis for a New Tetracycline Resistance Mechanism Relying on the Tetx Monooxygenase. FEBS Lett., 585, 2011
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2Y6R
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![BU of 2y6r by Molmil](/molmil-images/mine/2y6r) | Structure of the TetX monooxygenase in complex with the substrate 7- chlortetracycline | 分子名称: | 7-CHLOROTETRACYCLINE, FLAVIN-ADENINE DINUCLEOTIDE, SULFATE ION, ... | 著者 | Volkers, G, Palm, G.J, Weiss, M.S, Wright, G.D, Hinrichs, W. | 登録日 | 2011-01-25 | 公開日 | 2011-03-23 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structural Basis for a New Tetracycline Resistance Mechanism Relying on the Tetx Monooxygenase. FEBS Lett., 585, 2011
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2YH2
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![BU of 2yh2 by Molmil](/molmil-images/mine/2yh2) | |
2XRL
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![BU of 2xrl by Molmil](/molmil-images/mine/2xrl) | Tet-repressor class D T103A with doxycycline | 分子名称: | (4S,4AR,5S,5AR,6R,12AS)-4-(DIMETHYLAMINO)-3,5,10,12,12A-PENTAHYDROXY-6-METHYL-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDROTETRACENE-2-CARBOXAMIDE, CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Palm, G.J, Waack, P, Hinrichs, W. | 登録日 | 2010-09-16 | 公開日 | 2011-10-05 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Thermodynamics, cooperativity and stability of the tetracycline repressor (TetR) upon tetracycline binding. Biochim Biophys Acta Proteins Proteom, 1868, 2020
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2XYO
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![BU of 2xyo by Molmil](/molmil-images/mine/2xyo) | Structural basis for a new tetracycline resistance mechanism relying on the TetX monooxygenase | 分子名称: | FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, SULFATE ION, ... | 著者 | Volkers, G, Palm, G.J, Weiss, M.S, Hinrichs, W. | 登録日 | 2010-11-18 | 公開日 | 2011-03-23 | 最終更新日 | 2019-07-17 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural Basis for a New Tetracycline Resistance Mechanism Relying on the Tetx Monooxygenase. FEBS Lett., 585, 2011
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2X6O
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![BU of 2x6o by Molmil](/molmil-images/mine/2x6o) | Tet Repressor class D in complex with 7-chlor-2-cyano-iso- tetracycline | 分子名称: | (4S,4AS,6S,8AS)-6-[(1S)-7-CHLORO-4-HYDROXY-1-METHYL-3-OXO-1,3-DIHYDRO-2-BENZOFURAN-1-YL]-4-(DIMETHYLAMINO)-3,8A-DIHYDROXY-1,8-DIOXO-1,4,4A,5,6,7,8,8A-OCTAHYDRONAPHTHALENE-2-CARBONITRILE, CHLORIDE ION, TETRACYCLINE REPRESSOR PROTEIN CLASS D | 著者 | Volkers, G, Hinrichs, W. | 登録日 | 2010-02-18 | 公開日 | 2011-03-02 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Recognition of Drug Degradation Products by Target Proteins: Isotetracycline Binding to Tet Repressor. J.Med.Chem., 54, 2011
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2WQ5
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![BU of 2wq5 by Molmil](/molmil-images/mine/2wq5) | Non-antibiotic properties of tetracyclines: structural basis for inhibition of secretory phospholipase A2. | 分子名称: | (4S,4AS,5AR,12AS)-4,7-BIS(DIMETHYLAMINO)-3,10,12,12A-TETRAHYDROXY-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDROTETRACENE-2- CARBOXAMIDE, CALCIUM ION, PHOSPHOLIPASE A2, ... | 著者 | Dalm, D, Palm, G.J, Hinrichs, W. | 登録日 | 2009-08-13 | 公開日 | 2010-03-23 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Non-Antibiotic Properties of Tetracyclines: Structural Basis for Inhibition of Secretory Phospholipase A(2). J.Mol.Biol., 398, 2010
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7Q0Z
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![BU of 7q0z by Molmil](/molmil-images/mine/7q0z) | Crystal structure of CTX-M-14 | 分子名称: | Beta-lactamase, GLYCEROL, SULFATE ION | 著者 | Werner, N, Perbandt, M, Hinrichs, W, Prester, A, Rohde, H, Aepfelbacher, M, Betzel, C. | 登録日 | 2021-10-17 | 公開日 | 2022-04-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1 Å) | 主引用文献 | Structural basis to repurpose boron-based proteasome inhibitors Bortezomib and Ixazomib as beta-lactamase inhibitors. Sci Rep, 12, 2022
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7Q11
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![BU of 7q11 by Molmil](/molmil-images/mine/7q11) | Crystal structure of CTX-M-14 in complex with Ixazomib | 分子名称: | Beta-lactamase, CHLORIDE ION, DIMETHYL SULFOXIDE, ... | 著者 | Werner, N, Perbandt, M, Hinrichs, W, Prester, A, Rohde, H, Aepfelbacher, M, Betzel, C. | 登録日 | 2021-10-17 | 公開日 | 2022-04-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.14 Å) | 主引用文献 | Structural basis to repurpose boron-based proteasome inhibitors Bortezomib and Ixazomib as beta-lactamase inhibitors. Sci Rep, 12, 2022
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7Q0Y
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![BU of 7q0y by Molmil](/molmil-images/mine/7q0y) | Crystal structure of CTX-M-14 in complex with Bortezomib | 分子名称: | ACETATE ION, Beta-lactamase, CHLORIDE ION, ... | 著者 | Werner, N, Perbandt, M, Hinrichs, W, Prester, A, Rohde, H, Aepfelbacher, M, Betzel, C. | 登録日 | 2021-10-17 | 公開日 | 2022-04-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Structural basis to repurpose boron-based proteasome inhibitors Bortezomib and Ixazomib as beta-lactamase inhibitors. Sci Rep, 12, 2022
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7PXZ
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![BU of 7pxz by Molmil](/molmil-images/mine/7pxz) | Reduced form of SARS-CoV-2 Main Protease determined by XFEL radiation | 分子名称: | 3C-like proteinase, CHLORIDE ION | 著者 | Schubert, R, Reinke, P, Galchenkova, M, Oberthuer, D, Murillo, G.E.P, Kim, C, Bean, R, Turk, D, Hinrichs, W, Middendorf, P, Round, A, Schmidt, C, Mills, G, Kirkwood, H, Han, H, Koliyadu, J, Bielecki, J, Gelisio, L, Sikorski, M, Kloos, M, Vakilii, M, Yefanov, O.N, Vagovic, P, de-Wijn, R, Letrun, R, Guenther, S, White, T.A, Sato, T, Srinivasan, V, Kim, Y, Chretien, A, Han, S, Brognaro, H, Maracke, J, Knoska, J, Seychell, B.C, Brings, L, Norton-Baker, B, Geng, T, Dore, A.S, Uetrecht, C, Redecke, L, Beck, T, Lorenzen, K, Betzel, C, Mancuso, A.P, Bajt, S, Chapman, H.N, Meents, A, Lane, T.J. | 登録日 | 2021-10-08 | 公開日 | 2023-01-18 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Reduced form of SARS-CoV-2 Main Protease determined by XFEL radiation To Be Published
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7PZQ
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![BU of 7pzq by Molmil](/molmil-images/mine/7pzq) | Oxidized form of SARS-CoV-2 Main Protease determined by XFEL radiation | 分子名称: | 3C-like proteinase, DIMETHYL SULFOXIDE | 著者 | Schubert, R, Reinke, P, Galchenkova, M, Oberthuer, D, Murillo, G.E.P, Kim, C, Bean, R, Turk, D, Hinrichs, W, Middendorf, P, Round, A, Schmidt, C, Mills, G, Kirkwood, H, Han, H, Koliyadu, J, Bielecki, J, Gelisio, L, Sikorski, M, Kloos, M, Vakilii, M, Yefanov, O.N, Vagovic, P, de-Wijn, R, Letrun, R, Guenther, S, White, T.A, Sato, T, Srinivasan, V, Kim, Y, Chretien, A, Han, S, Brognaro, H, Maracke, J, Knoska, J, Seychell, B.C, Brings, L, Norton-Baker, B, Geng, T, Dore, A.S, Uetrecht, C, Redecke, L, Beck, T, Lorenzen, K, Betzel, C, Mancuso, A.P, Bajt, S, Chapman, H.N, Meents, A, Lane, T.J. | 登録日 | 2021-10-13 | 公開日 | 2023-01-25 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Oxidized form of SARS-CoV-2 Main Protease determined by XFEL radiation To Be Published
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4CHI
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![BU of 4chi by Molmil](/molmil-images/mine/4chi) | (R)-selective amine transaminase from Aspergillus fumigatus at 1.27 A resolution | 分子名称: | BRANCHED-CHAIN AMINO ACID AMINOTRANSFERASE, CHLORIDE ION, GLYCEROL, ... | 著者 | Thomsen, M, Palm, G.J, Hinrichs, W. | 登録日 | 2013-12-02 | 公開日 | 2014-04-30 | 最終更新日 | 2017-10-18 | 実験手法 | X-RAY DIFFRACTION (1.27 Å) | 主引用文献 | Crystallographic Characterization of the (R)-Selective Amine Transaminase from Aspergillus Fumigatus. Acta Crystallogr.,Sect.D, 70, 2014
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4D4F
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![BU of 4d4f by Molmil](/molmil-images/mine/4d4f) | Mutant P250A of bacterial chalcone isomerase from Eubacterium ramulus | 分子名称: | CHALCONE ISOMERASE, CHLORIDE ION, GLYCEROL | 著者 | Thomsen, M, Kratzat, H, Hinrichs, W. | 登録日 | 2014-10-28 | 公開日 | 2016-01-20 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.34 Å) | 主引用文献 | Structural Basis for (2 R ,3 R )-Taxifolin Binding and Reaction Products to the Bacterial Chalcone Isomerase of Eubacterium ramulus. Molecules, 27, 2022
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4CUO
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![BU of 4cuo by Molmil](/molmil-images/mine/4cuo) | Banyan peroxidase with glycosylation | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BANYAN PEROXIDASE, CALCIUM ION, ... | 著者 | Palm, G.J, Sharma, A, Hinrichs, W. | 登録日 | 2014-03-20 | 公開日 | 2014-07-23 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Post-Translational Modification and Extended Glycosylation Pattern of a Plant Latex Peroxidase of Native Source Characterized by X-Ray Crystallography. FEBS J., 281, 2014
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3ZPH
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![BU of 3zph by Molmil](/molmil-images/mine/3zph) | |
3ZWQ
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![BU of 3zwq by Molmil](/molmil-images/mine/3zwq) | |
3ZPX
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![BU of 3zpx by Molmil](/molmil-images/mine/3zpx) | |
4ABZ
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![BU of 4abz by Molmil](/molmil-images/mine/4abz) | |
4A5M
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![BU of 4a5m by Molmil](/molmil-images/mine/4a5m) | Redox regulator HypR in its oxidized form | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, UNCHARACTERIZED HTH-TYPE TRANSCRIPTIONAL REGULATOR YYBR | 著者 | Palm, G.J, Waack, P, Read, R.J, Hinrichs, W. | 登録日 | 2011-10-26 | 公開日 | 2012-01-11 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural Insights Into the Redox-Switch Mechanism of the Marr/Duf24-Type Regulator Hypr Nucleic Acids Res., 40, 2012
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4AL3
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![BU of 4al3 by Molmil](/molmil-images/mine/4al3) | |
4AC0
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![BU of 4ac0 by Molmil](/molmil-images/mine/4ac0) | TETR(B) IN COMPLEX WITH MINOCYCLINE AND MAGNESIUM | 分子名称: | (4S,4AS,5AR,12AS)-4,7-BIS(DIMETHYLAMINO)-3,10,12,12A-TETRAHYDROXY-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDROTETRACENE-2- CARBOXAMIDE, MAGNESIUM ION, PHOSPHATE ION, ... | 著者 | Volkers, G, Hinrichs, W. | 登録日 | 2011-12-12 | 公開日 | 2012-12-26 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Tetr(B) in Complex with Minocycline and Magnesium To be Published
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4A99
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![BU of 4a99 by Molmil](/molmil-images/mine/4a99) | STRUCTURE OF THE TETRACYCLINE DEGRADING MONOOXYGENASE TETX IN COMPLEX WITH MINOCYCLINE | 分子名称: | (4S,4AS,5AR,12AS)-4,7-BIS(DIMETHYLAMINO)-3,10,12,12A-TETRAHYDROXY-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDROTETRACENE-2- CARBOXAMIDE, FLAVIN-ADENINE DINUCLEOTIDE, SULFATE ION, ... | 著者 | Volkers, G, Palm, G.J, Weiss, M.S, Hinrichs, W. | 登録日 | 2011-11-25 | 公開日 | 2012-12-12 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | Putative Dioxygen-Binding Sites and Recognition of Tigecycline and Minocycline in the Tetracycline-Degrading Monooxygenase Tetx Acta Crystallogr.,Sect.D, 69, 2013
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4A5N
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![BU of 4a5n by Molmil](/molmil-images/mine/4a5n) | Redoxregulator HypR in its reduced form | 分子名称: | 1,2-ETHANEDIOL, BETA-MERCAPTOETHANOL, UNCHARACTERIZED HTH-TYPE TRANSCRIPTIONAL REGULATOR YYBR | 著者 | Palm, G.J, Waack, P, Read, R.J, Hinrichs, W. | 登録日 | 2011-10-26 | 公開日 | 2012-01-11 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | Structural Insights Into the Redox-Switch Mechanism of the Marr/Duf24-Type Regulator Hypr Nucleic Acids Res., 40, 2012
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