2RHQ
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3GOD
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3MNR
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![BU of 3mnr by Molmil](/molmil-images/mine/3mnr) | Crystal Structure of Benzamide SNX-1321 bound to Hsp90 | 分子名称: | 2-[(3,4,5-trimethoxyphenyl)amino]-4-(2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-1-yl)benzamide, Heat shock protein HSP 90-alpha | 著者 | Veal, J.M, Fadden, P, Huang, K.H, Rice, J, Hall, S.E, Haytstead, T.A. | 登録日 | 2010-04-22 | 公開日 | 2010-08-11 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Application of Chemoproteomics to Drug Discovery: Identification of a Clinical Candidate Targeting Hsp90. Chem.Biol., 17, 2010
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5YWO
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![BU of 5ywo by Molmil](/molmil-images/mine/5ywo) | Structure of JEV-2F2 Fab complex | 分子名称: | 2F2 heavy chain, 2F2 light chain, JEV E protein, ... | 著者 | Qiu, X, Lei, Y.F, Yang, P, Gao, Q, Wang, N, Cao, L, Yuan, S, Wang, X, Xu, Z.K, Rao, Z. | 登録日 | 2017-11-29 | 公開日 | 2018-03-21 | 最終更新日 | 2018-09-12 | 実験手法 | ELECTRON MICROSCOPY (4.7 Å) | 主引用文献 | Structural basis for neutralization of Japanese encephalitis virus by two potent therapeutic antibodies Nat Microbiol, 3, 2018
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5YWP
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![BU of 5ywp by Molmil](/molmil-images/mine/5ywp) | JEV-2H4 Fab complex | 分子名称: | 2H4 heavy chain, 2H4 light chain, JEV E protein, ... | 著者 | Qiu, X.D, Lei, Y.F, Yang, P, Gao, Q, WANG, N, Cao, L, Yuan, S, Wang, X.X, Xu, Z.K, Rao, Z.H. | 登録日 | 2017-11-29 | 公開日 | 2018-05-02 | 実験手法 | ELECTRON MICROSCOPY (4.6 Å) | 主引用文献 | Structural basis for neutralization of Japanese encephalitis virus by two potent therapeutic antibodies Nat Microbiol, 3, 2018
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5YWF
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![BU of 5ywf by Molmil](/molmil-images/mine/5ywf) | Crystal structure of 2H4 Fab | 分子名称: | 2H4 heavy chain, 2H4 light chain | 著者 | Qiu, X, Lei, Y, Yang, P, Gao, Q, Wang, N, Cao, L, Wang, X, Xu, Z.K, Rao, Z. | 登録日 | 2017-11-29 | 公開日 | 2018-03-21 | 実験手法 | X-RAY DIFFRACTION (2.206 Å) | 主引用文献 | Structural basis for neutralization of Japanese encephalitis virus by two potent therapeutic antibodies Nat Microbiol, 3, 2018
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8SPB
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![BU of 8spb by Molmil](/molmil-images/mine/8spb) | Caspase-4/Pro-IL-18 complex | 分子名称: | Caspase-4 subunit p10, Caspase-4 subunit p20, Interleukin-18 | 著者 | Pascal, D, Dong, Y, Wu, H, Jon, K. | 登録日 | 2023-05-02 | 公開日 | 2023-11-22 | 最終更新日 | 2023-12-27 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structural insights into cytokine cleavage by inflammatory caspase-4. Nature, 624, 2023
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8ECM
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8U7H
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![BU of 8u7h by Molmil](/molmil-images/mine/8u7h) | Cryo-EM structure of LRRK2 bound to type I inhibitor GNE-7915 | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, [4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanone, non-specific serine/threonine protein kinase | 著者 | Zhu, H, Sun, J. | 登録日 | 2023-09-15 | 公開日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Pharmacology of LRRK2 with type I and II kinase inhibitors revealed by cryo-EM. Cell Discov, 10, 2024
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8U7L
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![BU of 8u7l by Molmil](/molmil-images/mine/8u7l) | Cryo-EM structure of LRRK2 bound to type II inhibitor GZD824 | 分子名称: | 4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-3-[(1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]benzamide, GUANOSINE-5'-DIPHOSPHATE, Leucine-rich repeat serine/threonine-protein kinase 2 | 著者 | Zhu, H, Sun, J. | 登録日 | 2023-09-15 | 公開日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Pharmacology of LRRK2 with type I and II kinase inhibitors revealed by cryo-EM. Cell Discov, 10, 2024
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8U8A
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![BU of 8u8a by Molmil](/molmil-images/mine/8u8a) | Cryo-EM structure of LRRK2 bound to type II inhibitor ponatinib | 分子名称: | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzam ide, GUANOSINE-5'-DIPHOSPHATE, Leucine-rich repeat serine/threonine-protein kinase 2 | 著者 | Zhu, H, Sun, J. | 登録日 | 2023-09-16 | 公開日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Pharmacology of LRRK2 with type I and II kinase inhibitors revealed by cryo-EM. Cell Discov, 10, 2024
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8U8B
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![BU of 8u8b by Molmil](/molmil-images/mine/8u8b) | Cryo-EM structure of LRRK2 bound to type II inhibitor rebastinib | 分子名称: | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1H-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-N-methylpyridine-2-carboxamide, GUANOSINE-5'-DIPHOSPHATE, Leucine-rich repeat serine/threonine-protein kinase 2 | 著者 | Zhu, H, Sun, J. | 登録日 | 2023-09-16 | 公開日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Pharmacology of LRRK2 with type I and II kinase inhibitors revealed by cryo-EM. Cell Discov, 10, 2024
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7JGT
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![BU of 7jgt by Molmil](/molmil-images/mine/7jgt) | Crystal Structure of FN3tt | 分子名称: | Fibronectin type-III domain-containing protein | 著者 | Luo, J, Malia, T.J. | 登録日 | 2020-07-19 | 公開日 | 2021-07-21 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Surface salt bridges contribute to the extreme thermal stability of an FN3-like domain from a thermophilic bacterium. Proteins, 90, 2022
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7JGU
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![BU of 7jgu by Molmil](/molmil-images/mine/7jgu) | Structure of FN3tt mut | 分子名称: | Fibronectin type-III domain-containing protein, PENTAETHYLENE GLYCOL | 著者 | Luo, J, Boucher, L.E. | 登録日 | 2020-07-19 | 公開日 | 2021-07-21 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Surface salt bridges contribute to the extreme thermal stability of an FN3-like domain from a thermophilic bacterium. Proteins, 90, 2022
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8FO7
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![BU of 8fo7 by Molmil](/molmil-images/mine/8fo7) | Cryo-EM structure of LRRK2 bound to type I inhibitor LRRK2-IN-1 | 分子名称: | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one, GUANOSINE-5'-DIPHOSPHATE, Leucine-rich repeat serine/threonine-protein kinase 2 | 著者 | Zhu, H, Sun, J. | 登録日 | 2022-12-29 | 公開日 | 2024-01-17 | 最終更新日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (3.52 Å) | 主引用文献 | Pharmacology of LRRK2 with type I and II kinase inhibitors revealed by cryo-EM. Cell Discov, 10, 2024
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4PZ5
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8Z9Z
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![BU of 8z9z by Molmil](/molmil-images/mine/8z9z) | Cryo-EM structure of the insect olfactory receptor OR5-Orco heterocomplex from Acyrthosiphon pisum | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Odorant receptor, ApisOR5, ... | 著者 | Wang, Y.D, Qiu, L, Guan, Z.Y, Wang, Q, Wang, G.R, Yin, P. | 登録日 | 2024-04-24 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structural basis for odorant recognition of the insect odorant receptor OR-Orco heterocomplex. Science, 384, 2024
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8Z9A
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![BU of 8z9a by Molmil](/molmil-images/mine/8z9a) | Cryo-EM structure of the insect olfactory receptor OR5-Orco heterocomplex from Acyrthosiphon pisum bound with geranyl acetate | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Odorant receptor, ApisOR5, ... | 著者 | Wang, Y.D, Qiu, L, Guan, Z.Y, Wang, Q, Wang, G.R, Yin, P. | 登録日 | 2024-04-23 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Structural basis for odorant recognition of the insect odorant receptor OR-Orco heterocomplex. Science, 384, 2024
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7XRF
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![BU of 7xrf by Molmil](/molmil-images/mine/7xrf) | Crystal structaure of DgpB/C complex | 分子名称: | AP_endonuc_2 domain-containing protein, DgpB, MANGANESE (II) ION | 著者 | Ma, M, He, P. | 登録日 | 2022-05-10 | 公開日 | 2023-02-15 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.137 Å) | 主引用文献 | Structural mechanism of a dual-functional enzyme DgpA/B/C as both a C -glycoside cleaving enzyme and an O - to C -glycoside isomerase. Acta Pharm Sin B, 13, 2023
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7KOG
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![BU of 7kog by Molmil](/molmil-images/mine/7kog) | Lethocerus Myosin II complete coiled-coil domain resolved in its native environment | 分子名称: | Myosin heavy chain isoform Mhc_X1 | 著者 | Rahmani, H, Hu, Z, Daneshparvar, N, Taylor, D, Taylor, K.A. | 登録日 | 2020-11-09 | 公開日 | 2021-03-24 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (4.25 Å) | 主引用文献 | The myosin II coiled-coil domain atomic structure in its native environment. Proc.Natl.Acad.Sci.USA, 118, 2021
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7XVI
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7XVK
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7WQ5
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![BU of 7wq5 by Molmil](/molmil-images/mine/7wq5) | Crystal structure of Arabidopsis transcriptional factor WRINKLED1 with dsDNA | 分子名称: | AMMONIUM ION, DNA (5'-D(P*GP*TP*GP*GP*AP*CP*GP*AP*TP*GP*AP*AP*AP*CP*CP*GP*AP*GP*GP*AP*AP*GP*TP*A)-3'), DNA (5'-D(P*TP*AP*CP*TP*TP*CP*CP*TP*CP*GP*GP*TP*TP*TP*CP*AP*TP*CP*GP*TP*CP*CP*AP*C)-3'), ... | 著者 | Zhu, Q, Gao, Y.G. | 登録日 | 2022-01-24 | 公開日 | 2022-08-31 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Molecular basis of the key regulator WRINKLED1 in plant oil biosynthesis. Sci Adv, 8, 2022
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